DK0792879T3 - Fremgangsmåde til fremstilling af 3-[2-[4-(3-chlor-2-methylphenyl)-1-piperzinyl]ethyl]-5,6-dimethoxy-1-(4-imidazolylmethyl) - Google Patents

Fremgangsmåde til fremstilling af 3-[2-[4-(3-chlor-2-methylphenyl)-1-piperzinyl]ethyl]-5,6-dimethoxy-1-(4-imidazolylmethyl)

Info

Publication number
DK0792879T3
DK0792879T3 DK95936786T DK95936786T DK0792879T3 DK 0792879 T3 DK0792879 T3 DK 0792879T3 DK 95936786 T DK95936786 T DK 95936786T DK 95936786 T DK95936786 T DK 95936786T DK 0792879 T3 DK0792879 T3 DK 0792879T3
Authority
DK
Denmark
Prior art keywords
imidazolylmethyl
dimethoxy
methylphenyl
chloro
piperzinyl
Prior art date
Application number
DK95936786T
Other languages
Danish (da)
English (en)
Inventor
Kenjiro
Akihiko
Hiroaki
Original Assignee
Daiichi Seiyaku Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Seiyaku Co filed Critical Daiichi Seiyaku Co
Application granted granted Critical
Publication of DK0792879T3 publication Critical patent/DK0792879T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Materials For Medical Uses (AREA)
  • Medicinal Preparation (AREA)
DK95936786T 1994-11-14 1995-11-14 Fremgangsmåde til fremstilling af 3-[2-[4-(3-chlor-2-methylphenyl)-1-piperzinyl]ethyl]-5,6-dimethoxy-1-(4-imidazolylmethyl) DK0792879T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP27820494 1994-11-14
PCT/JP1995/002317 WO1996015124A1 (en) 1994-11-14 1995-11-14 Hydrate for medicinal use

Publications (1)

Publication Number Publication Date
DK0792879T3 true DK0792879T3 (da) 2001-03-26

Family

ID=17594052

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95936786T DK0792879T3 (da) 1994-11-14 1995-11-14 Fremgangsmåde til fremstilling af 3-[2-[4-(3-chlor-2-methylphenyl)-1-piperzinyl]ethyl]-5,6-dimethoxy-1-(4-imidazolylmethyl)

Country Status (16)

Country Link
US (1) US5948913A (de)
EP (1) EP0792879B1 (de)
KR (1) KR100372188B1 (de)
CN (1) CN1067998C (de)
AT (1) ATE199375T1 (de)
AU (1) AU698464B2 (de)
CA (1) CA2205206A1 (de)
DE (1) DE69520225T2 (de)
DK (1) DK0792879T3 (de)
ES (1) ES2156605T3 (de)
FI (1) FI972035L (de)
GR (1) GR3035820T3 (de)
NO (1) NO972190L (de)
PT (1) PT792879E (de)
RU (1) RU2152941C1 (de)
WO (1) WO1996015124A1 (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE510650C2 (sv) 1997-05-30 1999-06-14 Astra Ab Ny förening
WO1999024432A1 (fr) 1997-11-12 1999-05-20 Mitsubishi Chemical Corporation Derives de purine et medicament les renfermant en tant qu'ingredient actif
ES2206227T3 (es) * 1999-05-11 2004-05-16 Mitsubishi Chemical Corporation Dihidrato de un derivado de purina, farmacos que lo contienen como ingrediente activo, e intermedio en su preparacion.

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3362956A (en) * 1965-08-19 1968-01-09 Sterling Drug Inc 1-[(heterocyclyl)-lower-alkyl]-4-substituted-piperazines
JPH07507271A (ja) * 1992-03-03 1995-08-10 藤沢薬品工業株式会社 アンジオテンシン11拮抗剤としてのベンズイミダゾール誘導体
AU672047B2 (en) * 1992-10-06 1996-09-19 Ciba-Geigy Ag Novel thiosemicarbazonethiones
US5681954A (en) * 1993-05-14 1997-10-28 Daiichi Pharmaceutical Co., Ltd. Piperazine derivatives
RU2124511C1 (ru) * 1993-05-14 1999-01-10 Фармасьютикал Ко., Лтд Производные пиперазина
JPH0741431A (ja) * 1993-05-25 1995-02-10 Dai Ichi Seiyaku Co Ltd 脳保護薬
FI942400L (fi) * 1993-05-25 1994-11-26 Daiichi Seiyaku Co Lääkeaine hermosairauksia vastaan

Also Published As

Publication number Publication date
AU698464B2 (en) 1998-10-29
CA2205206A1 (en) 1996-05-23
RU2152941C1 (ru) 2000-07-20
WO1996015124A1 (en) 1996-05-23
FI972035A0 (fi) 1997-05-13
GR3035820T3 (en) 2001-07-31
EP0792879A4 (de) 1998-02-25
ES2156605T3 (es) 2001-07-01
DE69520225T2 (de) 2001-10-11
FI972035A7 (fi) 1997-07-11
AU3856595A (en) 1996-06-06
KR100372188B1 (ko) 2003-05-12
US5948913A (en) 1999-09-07
FI972035L (fi) 1997-07-11
NO972190D0 (no) 1997-05-13
KR970707118A (ko) 1997-12-01
DE69520225D1 (de) 2001-04-05
ATE199375T1 (de) 2001-03-15
PT792879E (pt) 2001-08-30
NO972190L (no) 1997-07-14
EP0792879A1 (de) 1997-09-03
CN1067998C (zh) 2001-07-04
EP0792879B1 (de) 2001-02-28
CN1171786A (zh) 1998-01-28

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