DK0835254T3 - Oxazolidinonderivater, deres fremstilling og deres terapeutiske anvendelse - Google Patents

Oxazolidinonderivater, deres fremstilling og deres terapeutiske anvendelse

Info

Publication number: DK0835254T3
Authority: DK; Denmark
Prior art keywords: preparation; therapeutic use; oxazolidinone derivatives; oxazolidinone; derivatives
Prior art date: 1995-06-02

Application number

DK96918719T

Other languages

English (en)

Inventor

Samir Jegham

Frederic Puech

Philippe Burnier

Original Assignee

Sanofi Synthelabo

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-06-02

Filing date

1996-05-28

Publication date

2000-03-27

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26232004&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK0835254(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1995-06-02 Priority claimed from FR9506564A external-priority patent/FR2734821B1/fr

1995-06-02 Priority claimed from FR9506563A external-priority patent/FR2734820B1/fr

1996-05-28 Application filed by Sanofi Synthelabo filed Critical Sanofi Synthelabo

2000-03-27 Application granted granted Critical

2000-03-27 Publication of DK0835254T3 publication Critical patent/DK0835254T3/da

Links

IZXIZTKNFFYFOF-UHFFFAOYSA-N 2-Oxazolidone Chemical class O=C1NCCO1 IZXIZTKNFFYFOF-UHFFFAOYSA-N 0.000 title 1
230000001225 therapeutic effect Effects 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Neurology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Epidemiology (AREA)
Hospice & Palliative Care (AREA)
Psychiatry (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

DK96918719T 1995-06-02 1996-05-28 Oxazolidinonderivater, deres fremstilling og deres terapeutiske anvendelse DK0835254T3 (da)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
FR9506564A FR2734821B1 (fr)	1995-06-02	1995-06-02	Derives de 5-methoxymethyl-3-(1,2-benzisoxazol-3-yl) oxazolidin-2-one, leur preparation et leur application en therapeutique
FR9506563A FR2734820B1 (fr)	1995-06-02	1995-06-02	Derives de 3-(1,2-benzisoxazol-3-yl)oxazolidin-2-one, leur preparation et leur application en therapeutique
PCT/FR1996/000792 WO1996038444A1 (fr)	1995-06-02	1996-05-28	Derives d'oxazolidinone, leur preparation et leur application en therapeutique

Publications (1)

Publication Number	Publication Date
DK0835254T3 true DK0835254T3 (da)	2000-03-27

Family

ID=26232004

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK96918719T DK0835254T3 (da)	1995-06-02	1996-05-28	Oxazolidinonderivater, deres fremstilling og deres terapeutiske anvendelse

Country Status (26)

Country	Link
US (1)	US5843975A (da)
EP (1)	EP0835254B1 (da)
JP (1)	JP3856829B2 (da)
KR (1)	KR100457502B1 (da)
CN (1)	CN1075072C (da)
AR (1)	AR006301A1 (da)
AT (1)	ATE184005T1 (da)
AU (1)	AU699367B2 (da)
BR (1)	BR9608896A (da)
CA (1)	CA2223011C (da)
CO (1)	CO4700462A1 (da)
CZ (1)	CZ378497A3 (da)
DE (1)	DE69604071T2 (da)
DK (1)	DK0835254T3 (da)
ES (1)	ES2138346T3 (da)
GR (1)	GR3031710T3 (da)
HU (1)	HU224879B1 (da)
MX (1)	MX9709410A (da)
NO (1)	NO309091B1 (da)
NZ (1)	NZ310487A (da)
PL (1)	PL183919B1 (da)
RU (1)	RU2164226C2 (da)
SK (1)	SK281934B6 (da)
TW (1)	TW360654B (da)
WO (1)	WO1996038444A1 (da)
ZA (1)	ZA964563B (da)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP1078632A1 (en) *	1999-08-16	2001-02-28	Sanofi-Synthelabo	Use of monoamine oxydase inhibitors for the manufacture of drugs intended for the treatment of obesity
EP1363638A4 (en) *	2001-01-31	2010-01-06	Lundbeck & Co As H	USE OF GAL3 RECEPTOR ANTAGONISTS FOR THE TREATMENT OF DEPRESSION AND / OR ANXIETIES AND USEFUL CONNECTIONS FOR SUCH PROCEDURES
TWI248438B (en) *	2001-04-10	2006-02-01	Sod Conseils Rech Applic	Derivatives of heterocycles with 5 members, their preparation and their use as medicaments
KR20040047869A (ko) *	2001-09-26	2004-06-05	파마시아 이탈리아 에스.피.에이.	키나제 억제제로서 활성인 아미노인다졸 유도체, 이의제조방법 및 이를 함유하는 약제학적 조성물
DE10334309A1 (de) *	2003-07-28	2005-03-03	Aventis Pharma Deutschland Gmbh	Substituierte Thiazol-Benzoisothiazoldioxidderivate, Verfahren zu deren Herstellung und deren Verwendung
EP2032565A2 (en) *	2006-02-01	2009-03-11	Pfizer Products Inc.	Benzisoxazole oxazolidinones as antibacterial agents
EP2141154A4 (en) *	2007-03-30	2011-06-01	Inst Med Molecular Design Inc	OXAZOLIDINONE DERIVATIVITY WITH HEMMETIC EFFECT ON TYPE I 11-HYDROXYSTEROIDDEHYDROGENASE
EP2123159A1 (de) *	2008-05-21	2009-11-25	Bayer CropScience AG	(1,2-Benzisothiazol-3-yl)(thio)carbamate und (1,2-Benzisothiazol-3-yl)(thio)oxamate und deren Oxidationsformen als Pestizide
AU2010330894A1 (en) *	2009-12-18	2012-07-05	Janssen Pharmaceutica Nv	Substituted aminothiazolone indazoles as estrogen related receptor-aalpha modulators
BR112012020604A2 (pt) *	2010-02-17	2019-09-24	Janssen Pharmaceutica Nv	"aminotiazolonas como moduladores do receptor alfa-relacionado ao estrôgenio"
WO2016097355A1 (en) *	2014-12-19	2016-06-23	Ge Healthcare Limited	Labelled oxazolidinone derivatives
DE102015012050A1 (de) *	2015-09-15	2017-03-16	Merck Patent Gmbh	Verbindungen als ASIC-Inhibitoren und deren Verwendungen
RU2637643C1 (ru) *	2016-09-05	2017-12-05	Федеральное государственное бюджетное научное учреждение "Научно-исследовательский институт фундаментальной и клинической иммунологии" (НИИФКИ)	Иммунодепрессант

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ES2076253T3 (es) *	1989-05-19	1995-11-01	Hoechst Roussel Pharma	N-(ariloxialquil)-heteroarilpiperidinas y -heteroarilpiperazinas, un procedimiento para su preparacion y su uso como medicamentos.
FR2653017B1 (fr) *	1989-10-17	1995-05-05	Delalande Sa	Derives d'aryl-3 oxazolidinone-2, leur procede de preparation et leur application en therapeutique.
US5196543A (en) *	1989-10-17	1993-03-23	Delalande S.A.	3-aryloxazolidinone derivatives, process for their preparation and their use in therapy
US5235063A (en) *	1989-10-17	1993-08-10	Delalande S.A.	Process of preparing by condensation certain
US5182296A (en) *	1989-10-26	1993-01-26	Tanabe Seiyaky Co., Ltd.	Naphthyloxazolidone derivatives
FR2671350A1 (fr) *	1991-01-08	1992-07-10	Adir	Nouveaux derives de benzisoxazole et de benzisothiazole, leur procede de preparation, et les compositions pharmaceutiques les renfermant.
EP0525209A4 (en) *	1991-02-20	1993-06-30	Yusaku Koda	Articulator

1996
- 1996-05-28 KR KR1019970708666A patent/KR100457502B1/ko not_active Expired - Lifetime
- 1996-05-28 PL PL96323673A patent/PL183919B1/pl unknown
- 1996-05-28 NZ NZ310487A patent/NZ310487A/xx not_active IP Right Cessation
- 1996-05-28 DK DK96918719T patent/DK0835254T3/da active
- 1996-05-28 JP JP53624596A patent/JP3856829B2/ja not_active Expired - Lifetime
- 1996-05-28 US US08/973,246 patent/US5843975A/en not_active Expired - Lifetime
- 1996-05-28 CN CN96195713A patent/CN1075072C/zh not_active Expired - Lifetime
- 1996-05-28 CZ CZ973784A patent/CZ378497A3/cs unknown
- 1996-05-28 AT AT96918719T patent/ATE184005T1/de active
- 1996-05-28 DE DE69604071T patent/DE69604071T2/de not_active Expired - Lifetime
- 1996-05-28 ES ES96918719T patent/ES2138346T3/es not_active Expired - Lifetime
- 1996-05-28 EP EP96918719A patent/EP0835254B1/fr not_active Expired - Lifetime
- 1996-05-28 AU AU61288/96A patent/AU699367B2/en not_active Expired
- 1996-05-28 SK SK1614-97A patent/SK281934B6/sk not_active IP Right Cessation
- 1996-05-28 WO PCT/FR1996/000792 patent/WO1996038444A1/fr not_active Ceased
- 1996-05-28 HU HU9901349A patent/HU224879B1/hu unknown
- 1996-05-28 RU RU98100257/04A patent/RU2164226C2/ru active
- 1996-05-28 CA CA002223011A patent/CA2223011C/en not_active Expired - Lifetime
- 1996-05-28 BR BR9608896A patent/BR9608896A/pt active IP Right Grant
- 1996-05-31 CO CO96028173A patent/CO4700462A1/es unknown
- 1996-06-01 TW TW085106564A patent/TW360654B/zh not_active IP Right Cessation
- 1996-06-03 AR ARP960102870A patent/AR006301A1/es active IP Right Grant
- 1996-06-03 ZA ZA964563A patent/ZA964563B/xx unknown
1997
- 1997-12-01 NO NO975530A patent/NO309091B1/no not_active IP Right Cessation
- 1997-12-02 MX MX9709410A patent/MX9709410A/es unknown
1999
- 1999-11-03 GR GR990402802T patent/GR3031710T3/el unknown

Also Published As

Publication number	Publication date
NZ310487A (en)	1999-05-28
CA2223011A1 (en)	1996-12-05
TW360654B (en)	1999-06-11
CN1075072C (zh)	2001-11-21
NO975530D0 (no)	1997-12-01
PL183919B1 (pl)	2002-08-30
RU2164226C2 (ru)	2001-03-20
SK161497A3 (en)	1998-05-06
PL323673A1 (en)	1998-04-14
DE69604071T2 (de)	2000-04-06
CZ378497A3 (cs)	1998-04-15
SK281934B6 (sk)	2001-09-11
CO4700462A1 (es)	1998-12-29
KR100457502B1 (ko)	2005-09-05
US5843975A (en)	1998-12-01
GR3031710T3 (en)	2000-02-29
JPH11507330A (ja)	1999-06-29
ES2138346T3 (es)	2000-01-01
AU6128896A (en)	1996-12-18
HU224879B1 (en)	2006-03-28
HUP9901349A2 (hu)	1999-08-30
EP0835254B1 (fr)	1999-09-01
AR006301A1 (es)	1999-08-25
AU699367B2 (en)	1998-12-03
ATE184005T1 (de)	1999-09-15
NO975530L (no)	1998-02-02
KR19990022187A (ko)	1999-03-25
ZA964563B (en)	1996-12-12
NO309091B1 (no)	2000-12-11
CN1191534A (zh)	1998-08-26
MX9709410A (es)	1998-07-31
DE69604071D1 (de)	1999-10-07
JP3856829B2 (ja)	2006-12-13
HUP9901349A3 (en)	2000-02-28
HK1014938A1 (en)	1999-10-08
WO1996038444A1 (fr)	1996-12-05
CA2223011C (en)	2007-01-09
EP0835254A1 (fr)	1998-04-15
BR9608896A (pt)	1999-06-29

Publication	Publication Date	Title
DK0869126T3 (da)	2002-11-18	Dithiolanderivater, deres fremstilling og deres terapeutiske virkning
NO954369D0 (no)	1995-11-01	Oksazolidindionderivater, deres fremstilling og anvendelse
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NO980720D0 (no)	1998-02-20	Pyridazin-3-on-derivater, deres anvendelse og mellomprodukter for deres fremstilling
NO961160D0 (no)	1996-03-21	Cykliske forbindelser, deres fremstilling og anvendelse
NO951095L (no)	1995-09-25	Tiazolidin- og oksazolidinderivater, deres fremstilling og medisinske bruk
NO943682D0 (no)	1994-10-03	Imidazol-4-yl-piperidin-derivater, deres fremstilling og terapeutiske anvendelse
NO924650D0 (no)	1992-12-02	Dialkoksy-pyridinyl-benzimidazolderivater, fremgangsmaate for deres fremstilling og deres farmasoeytiske anvendelse
DK1161434T3 (da)	2003-05-26	Pyridopyranoazepinderivater, deres fremstilling og terapeutiske anvendelse
NO955326D0 (no)	1995-12-28	Isokinolinderivater, fremgangsmåte for deres fremstilling og terapeutiske anvendelse
NO975020D0 (no)	1997-10-31	Azacykloalkanderivater, fremstilling derav og deres anvendelse i terapi
NO975530D0 (no)	1997-12-01	Oksazolidinon derivater, deres fremstilling og terapeutiske anvendelse
FI941068A7 (fi)	1994-09-09	Bentsoksatsiinijohdannaiset, niiden valmistus ja terapeuttinen käyttö
NO962477L (no)	1996-12-16	Benzamidderivater, deres fremstilling og deres terapautiske anvendelse
NO992676D0 (no)	1999-06-02	1,4-diazabicyklo[2,2,2]okt-2-ylmetylderivater, deres fremstilling og terapeutiske anvendelse
NO20001934D0 (no)	2000-04-13	3-Substituerte tetrahydropyridopyrimidinon-derivater, deres fremstilling og anvendelse
NO940130D0 (no)	1994-01-14	Benzimidazolderivater, fremgangsmaate for deres fremstilling og te rapeutisk anvendelse derav
NO980471L (no)	1998-04-06	Benzensulfonamidderivater, fremstilling derav og terapautiske anvendelser derav
NO921563L (no)	1992-10-26	Terapeutisk aktive aminopyrimidinderivater, fremgangsmaatefor deres fremstilling og anvendelse derav
NO20000066D0 (no)	2000-01-06	6-pyrrolidin-2-ylpyrindin-derivater, deres fremstilling og deres farmasoeytiske anvendelse
NO955242D0 (no)	1995-12-22	Piperidinderivater, fremgangsmåte for fremstilling derav og deres terapeutiske anvendelse
NO982549D0 (no)	1998-06-04	5-naftalen-1-yl-1,3-dioksan-derivater, fremstilling og terapeutisk anvendelse derav
NO950560D0 (no)	1995-02-15	Piperazinderivater, deres fremstilling og terapautiske anvendelse
NO992436D0 (no)	1999-05-20	N(imidazolylbutyl)benzensulfonamidderivater, deres fremstilling og terapeutiske anvendelse
NO951812D0 (no)	1995-05-09	Pyrrolderivater, deres fremstilling og anvendelse