DK0911030T3 - Antimikrobielle præparater som omfatter et vinylpyrrolidinonderivat og et carbapenemantibiotikum eller en beta-lactamaseinhibitor - Google Patents

Antimikrobielle præparater som omfatter et vinylpyrrolidinonderivat og et carbapenemantibiotikum eller en beta-lactamaseinhibitor

Info

Publication number
DK0911030T3
DK0911030T3 DK98117009T DK98117009T DK0911030T3 DK 0911030 T3 DK0911030 T3 DK 0911030T3 DK 98117009 T DK98117009 T DK 98117009T DK 98117009 T DK98117009 T DK 98117009T DK 0911030 T3 DK0911030 T3 DK 0911030T3
Authority
DK
Denmark
Prior art keywords
beta
antimicrobial compositions
lactamase inhibitor
vinyl pyrrolidinone
carbapenem antibiotic
Prior art date
Application number
DK98117009T
Other languages
English (en)
Inventor
Peter Angehrn
Ingrid Heinze-Krauss
Malcolm Page
G F Hans Richter
Original Assignee
Basilea Pharmaceutica Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basilea Pharmaceutica Ag filed Critical Basilea Pharmaceutica Ag
Application granted granted Critical
Publication of DK0911030T3 publication Critical patent/DK0911030T3/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • A61K31/546—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine containing further heterocyclic rings, e.g. cephalothin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/74—Synthetic polymeric materials
    • A61K31/785—Polymers containing nitrogen
    • A61K31/787—Polymers containing nitrogen containing heterocyclic rings having nitrogen as a ring hetero atom
    • A61K31/79—Polymers of vinyl pyrrolidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
DK98117009T 1997-09-15 1998-09-09 Antimikrobielle præparater som omfatter et vinylpyrrolidinonderivat og et carbapenemantibiotikum eller en beta-lactamaseinhibitor DK0911030T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP97115997 1997-09-15
EP98117009A EP0911030B1 (en) 1997-09-15 1998-09-09 Antimicrobial composition comprising a vinyyl pyrrolidinon derivative and a carbapenem antibiotic or a beta-lactamase inhibitor

Publications (1)

Publication Number Publication Date
DK0911030T3 true DK0911030T3 (da) 2005-08-01

Family

ID=8227350

Family Applications (1)

Application Number Title Priority Date Filing Date
DK98117009T DK0911030T3 (da) 1997-09-15 1998-09-09 Antimikrobielle præparater som omfatter et vinylpyrrolidinonderivat og et carbapenemantibiotikum eller en beta-lactamaseinhibitor

Country Status (16)

Country Link
US (1) US6150350A (da)
EP (1) EP0911030B1 (da)
JP (1) JP4621311B2 (da)
KR (1) KR100630012B1 (da)
CN (1) CN1186021C (da)
AR (1) AR013490A1 (da)
AT (1) ATE292994T1 (da)
AU (1) AU747285B2 (da)
BR (1) BR9803443A (da)
CA (1) CA2247232C (da)
DE (1) DE69829720T2 (da)
DK (1) DK0911030T3 (da)
ES (1) ES2241084T3 (da)
PT (1) PT911030E (da)
TR (1) TR199801835A2 (da)
ZA (1) ZA988399B (da)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2335288A1 (en) * 1998-06-22 1999-12-29 F. Hoffmann-La Roche Ag Propenyl cephalosporin derivatives
WO2000032605A1 (en) * 1998-12-03 2000-06-08 F. Hoffmann-La Roche Ag Bi-pyrrolidinylvinl (carba) cephalosporins
JP4583559B2 (ja) * 2000-07-24 2010-11-17 栄研化学株式会社 Mrsaスクリーニング用培地
CN100384857C (zh) * 2003-11-28 2008-04-30 浙江永宁制药厂 耐β-内酰胺酶的头孢菌素酯化合物及其盐
CN112608369A (zh) * 2020-12-30 2021-04-06 中国海洋大学 一种具有抑菌活性的细菌素及其生产方法及用途

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0347122A (ja) * 1989-02-21 1991-02-28 Banyu Pharmaceut Co Ltd 抗菌性組成物
EP0384410B1 (en) * 1989-02-21 1995-05-17 Banyu Pharmaceutical Co., Ltd. Antimicrobial composition
GB9019743D0 (en) * 1990-09-10 1990-10-24 Beecham Group Plc Novel compounds
KR100214288B1 (ko) * 1993-04-16 1999-08-02 성재갑 안개서림 방지용 내마모성 피복조성물 및 이를 도포한 합성수지 성형품
PT620225E (pt) * 1993-04-16 2003-03-31 Basilea Pharmaceutica Ag Derivados de cefalosporina
TW383308B (en) * 1993-08-24 2000-03-01 Hoffmann La Roche 2-beta-alkenyl penam sulfones as beta-lactamase inhibitors
US5464616A (en) * 1994-08-04 1995-11-07 Synphar Laboratories, Ind. 6β-substituted penicillanic acids as beta-lactamase inhibitors
TR199700859T1 (xx) * 1995-02-27 1998-02-21 F. Hoffmann-La Roche Ag 3-Pirolidiliden-2-on-sefalosporin t�revleri.
ATE354577T1 (de) * 1996-11-06 2007-03-15 Basilea Pharmaceutica Ag Vinylpyrrolidinon-cephalosporin-derivate

Also Published As

Publication number Publication date
EP0911030A3 (en) 1999-10-13
AU8425198A (en) 1999-04-01
ES2241084T3 (es) 2005-10-16
EP0911030A2 (en) 1999-04-28
TR199801835A3 (tr) 1999-04-21
ZA988399B (en) 1999-03-15
CA2247232A1 (en) 1999-03-15
CA2247232C (en) 2007-08-28
US6150350A (en) 2000-11-21
KR100630012B1 (ko) 2006-11-30
AR013490A1 (es) 2000-12-27
KR19990029769A (ko) 1999-04-26
JPH11140087A (ja) 1999-05-25
DE69829720T2 (de) 2006-03-09
BR9803443A (pt) 2000-02-08
EP0911030B1 (en) 2005-04-13
DE69829720D1 (de) 2005-05-19
AU747285B2 (en) 2002-05-16
CN1186021C (zh) 2005-01-26
CN1216246A (zh) 1999-05-12
TR199801835A2 (xx) 1999-04-21
PT911030E (pt) 2005-08-31
JP4621311B2 (ja) 2011-01-26
ATE292994T1 (de) 2005-04-15

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