DK0968211T3 - Tetrazolderivater - Google Patents

Tetrazolderivater

Info

Publication number
DK0968211T3
DK0968211T3 DK98913621T DK98913621T DK0968211T3 DK 0968211 T3 DK0968211 T3 DK 0968211T3 DK 98913621 T DK98913621 T DK 98913621T DK 98913621 T DK98913621 T DK 98913621T DK 0968211 T3 DK0968211 T3 DK 0968211T3
Authority
DK
Denmark
Prior art keywords
pct
tetrazole
radical
sec
date
Prior art date
Application number
DK98913621T
Other languages
Danish (da)
English (en)
Inventor
Beate Schmidt
Hermann Amschler
Wolf-Ruediger Ulrich
Thomas Martin
Thomas Baer
Hildegard Boss
Rolf-Peter Hummel
Armin Hatzelmann
Rolf Beume
Hans-Peter Kley
Dietrich Haefner
Karl-Josef Goebel
Dieter Flockerzi
Original Assignee
Altana Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Altana Pharma Ag filed Critical Altana Pharma Ag
Application granted granted Critical
Publication of DK0968211T3 publication Critical patent/DK0968211T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Dermatology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
DK98913621T 1997-03-07 1998-03-03 Tetrazolderivater DK0968211T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19709293 1997-03-07
EP97103924 1997-03-08
PCT/EP1998/001168 WO1998040382A1 (en) 1997-03-07 1998-03-03 Novel tetrazoles

Publications (1)

Publication Number Publication Date
DK0968211T3 true DK0968211T3 (da) 2003-12-08

Family

ID=26034595

Family Applications (1)

Application Number Title Priority Date Filing Date
DK98913621T DK0968211T3 (da) 1997-03-07 1998-03-03 Tetrazolderivater

Country Status (12)

Country Link
US (1) US6143759A (de)
EP (1) EP0968211B1 (de)
JP (1) JP2001514640A (de)
AT (1) ATE248167T1 (de)
AU (1) AU6825898A (de)
CY (1) CY2502B1 (de)
DE (1) DE69817548T2 (de)
DK (1) DK0968211T3 (de)
ES (1) ES2206909T3 (de)
PT (1) PT968211E (de)
SI (1) SI0968211T1 (de)
WO (1) WO1998040382A1 (de)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR015966A1 (es) * 1997-10-17 2001-05-30 Smithkline Beecham Corp Uso de un compuesto inhibidor de pde4 para la preparacion de un medicamento util para el tratamiento de prurito
SI1109810T1 (en) * 1998-08-31 2004-12-31 Altana Pharma Ag Benzonaphthyridine-n-oxides comprising a pde3 and pde4 inhibiting activity
ATE356810T1 (de) 1999-01-15 2007-04-15 Altana Pharma Ag Polysubstituted 6-phenylphenanthridines mit pde- iv hemmender wirkung
EE05105B1 (et) 1999-01-15 2008-12-15 Byk Gulden Lomberg Chemische Fabrik Gmbh Fenlfenantridiinid, nende kasutamine ravimite valmistamiseks ning neid sisaldav ravim
EP1147103B1 (de) 1999-01-15 2005-05-04 ALTANA Pharma AG Phenantrhridin-n-oxides mit pde-iv hemmender wirkung
AU2107700A (en) 1999-01-15 2000-08-01 Byk Gulden Lomberg Chemische Fabrik Gmbh Phenanthridine-n-oxides with pde-iv inhibiting activity
PL200923B1 (pl) 1999-08-21 2009-02-27 Nycomed Gmbh Lek zawierający inhibitor PDE w połączeniu z agonistą receptoraß₂ -adrenergicznego oraz zastosowanie połączenia roflumilastu i salmeterolu
US6936622B2 (en) 2001-02-21 2005-08-30 Altana Pharma Ag 6-phenylbenzonaphthyridines
US6479493B1 (en) 2001-08-23 2002-11-12 Cell Pathways, Inc. Methods for treatment of type I diabetes
HK1085462A1 (en) * 2002-05-31 2006-08-25 Takeda Pharmaceutical Company Limited Piperidine derivative, process for producing the same, and use
AU2003263216A1 (en) * 2002-08-17 2004-03-11 Nycomed Gmbh Benzonaphthyridines with PDE 3/4 inhibiting activity
US7470704B2 (en) 2002-09-04 2008-12-30 Nycomed Gmbh Benzonaphthyridines
JP2006522151A (ja) 2003-04-01 2006-09-28 アプライド リサーチ システムズ エーアールエス ホールディング ナームロゼ フェンノートシャップ 不妊症におけるホスホジエステラーゼ阻害剤
PL2589599T4 (pl) 2004-03-03 2015-06-30 Takeda Gmbh Nowe hydroksy-6-heteroarylofenantrydyny i ich zastosowanie jako inhibitorów PDE4
EP1732925A1 (de) 2004-03-17 2006-12-20 Altana Pharma AG Neue n-(alkoxyalkyl)carbamoylsubstituierte 6-phenylbenzonaphthyridinderivate und deren verwendung als pde3/4-inhibitoren
US7589205B2 (en) * 2004-09-08 2009-09-15 Nycomed Gmbh 3-thia-10-aza-phenanthrene derivatives
DE602005027866D1 (de) * 2004-09-08 2011-06-16 Nycomed Gmbh 3-oxa-10-aza-phenanthrene als pde4- oder pde3/4-inhibitoren
ES2337083T3 (es) 2005-03-02 2010-04-20 Nycomed Gmbh (2r,4ar,10br)-6-(2,6-dimetoxipiridin-3-il)-9-exoti-8-metoxi-1,2,3,4,4a,10b-hexahidrofenantridin-2-ol, sal de hc1.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3899494A (en) * 1970-05-13 1975-08-12 Sandoz Ltd Substituted 6-phenyl benzo-naphthyridines
EP0247971A3 (de) * 1986-05-29 1990-01-17 Sandoz Ag Pharmazeutische Zusammensetzungen mit, und Verwendung von Cis-6-(4-Acetanilido)-8,9-dimethoxy-2-methyl-1,2,3,4,4a,10b-hexahydrobenzo[c][1,6]naphthyridin
MY105344A (en) * 1990-05-16 1994-09-30 Byk Gulden Lomberg Chemische Fabrik New sulphonyl compounds

Also Published As

Publication number Publication date
CY2502B1 (en) 2005-09-02
EP0968211A1 (de) 2000-01-05
DE69817548D1 (de) 2003-10-02
US6143759A (en) 2000-11-07
ATE248167T1 (de) 2003-09-15
AU6825898A (en) 1998-09-29
EP0968211B1 (de) 2003-08-27
PT968211E (pt) 2004-01-30
DE69817548T2 (de) 2004-06-17
WO1998040382A1 (en) 1998-09-17
ES2206909T3 (es) 2004-05-16
JP2001514640A (ja) 2001-09-11
SI0968211T1 (en) 2004-02-29

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