DK1015466T3 - Derivater af 9-hydrazon og 9-azinerythromycin og en fremgangsmåde til fremstilling af samme - Google Patents

Derivater af 9-hydrazon og 9-azinerythromycin og en fremgangsmåde til fremstilling af samme

Info

Publication number: DK1015466T3
Authority: DK; Denmark
Prior art keywords: hydrazone; derivatives; same; azinerythromycin; preparing
Prior art date: 1997-09-10

Application number

DK98944641T

Other languages

English (en)

Inventor

David R Hill

Original Assignee

Abbott Lab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-09-10

Filing date

1998-09-01

Publication date

2003-09-01

1998-09-01 Application filed by Abbott Lab filed Critical Abbott Lab

2003-09-01 Application granted granted Critical

2003-09-01 Publication of DK1015466T3 publication Critical patent/DK1015466T3/da

Links

238000004519 manufacturing process Methods 0.000 title 1
ULGZDMOVFRHVEP-RWJQBGPGSA-N Erythromycin Chemical compound O([C@@H]1[C@@H](C)C(=O)O[C@@H]([C@@]([C@H](O)[C@@H](C)C(=O)[C@H](C)C[C@@](C)(O)[C@H](O[C@H]2[C@@H]([C@H](C[C@@H](C)O2)N(C)C)O)[C@H]1C)(C)O)CC)[C@H]1C[C@@](C)(OC)[C@@H](O)[C@H](C)O1 ULGZDMOVFRHVEP-RWJQBGPGSA-N 0.000 abstract 4
229960003276 erythromycin Drugs 0.000 abstract 3
150000001875 compounds Chemical class 0.000 abstract 2
238000000034 method Methods 0.000 abstract 2
238000006243 chemical reaction Methods 0.000 abstract 1
239000000543 intermediate Substances 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H1/00—Processes for the preparation of sugar derivatives

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Molecular Biology (AREA)
Life Sciences & Earth Sciences (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
General Health & Medical Sciences (AREA)
Genetics & Genomics (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Saccharide Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Solid Thermionic Cathode (AREA)
Analysing Materials By The Use Of Radiation (AREA)
Diaphragms For Electromechanical Transducers (AREA)

DK98944641T 1997-09-10 1998-09-01 Derivater af 9-hydrazon og 9-azinerythromycin og en fremgangsmåde til fremstilling af samme DK1015466T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US08/927,057 US5929219A (en)	1997-09-10	1997-09-10	9-hydrazone and 9-azine erythromycin derivatives and a process of making the same
PCT/US1998/018115 WO1999012946A1 (en)	1997-09-10	1998-09-01	9-hydrazone and 9-azine erythromycin derivatives and a process of making the same

Publications (1)

Publication Number	Publication Date
DK1015466T3 true DK1015466T3 (da)	2003-09-01

Family

ID=25454102

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK98944641T DK1015466T3 (da)	1997-09-10	1998-09-01	Derivater af 9-hydrazon og 9-azinerythromycin og en fremgangsmåde til fremstilling af samme

Country Status (13)

Country	Link
US (2)	US5929219A (da)
EP (1)	EP1015466B1 (da)
JP (1)	JP2001515914A (da)
KR (1)	KR100553468B1 (da)
AT (1)	ATE239751T1 (da)
AU (1)	AU9213698A (da)
CA (1)	CA2301639C (da)
DE (1)	DE69814422T2 (da)
DK (1)	DK1015466T3 (da)
ES (1)	ES2198745T3 (da)
IL (2)	IL134468A0 (da)
PT (1)	PT1015466E (da)
WO (1)	WO1999012946A1 (da)

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IL125372A0 (en) *	1998-07-15	1999-03-12	Chemagis Ltd	Erythromycin derivatives and methods for the preparation thereof
KR100317907B1 (ko) *	1998-11-24	2001-12-24	김 완 주	신규한 중간체, 이를 이용한 마크로라이드계 항생제의제조방법
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US6605707B1 (en)	2000-03-23	2003-08-12	Abbott Laboratories	Process for the preparation of 6-O-propargyl erythromycin derivatives
US6541014B2 (en)	2000-10-13	2003-04-01	Advancis Pharmaceutical Corp.	Antiviral product, use and formulation thereof
US20020068078A1 (en)	2000-10-13	2002-06-06	Rudnic Edward M.	Antifungal product, use and formulation thereof
US7435805B2 (en)	2003-05-30	2008-10-14	Glaxpsmithkline Istrazivacki	O-alkyl macrolide and azalide derivatives and regioselective process for their preparation
CA2533178C (en)	2003-07-21	2014-03-11	Advancis Pharmaceutical Corporation	Antibiotic product, use and formulation thereof
JP2006528185A (ja)	2003-07-21	2006-12-14	アドバンシスファーマスーティカルコーポレイション	抗生物質製剤、その使用法及び作成方法
JP2006528190A (ja)	2003-07-21	2006-12-14	アドバンシスファーマスーティカルコーポレイション	抗生物質製剤、その使用法及び作成方法
WO2005016311A1 (en)	2003-08-11	2005-02-24	Advancis Pharmaceutical Corporation	Robust pellet
AU2004264356B2 (en)	2003-08-12	2011-01-27	Shionogi, Inc.	Antibiotic product, use and formulation thereof
JP5686494B2 (ja)	2003-08-29	2015-03-18	シオノギインコーポレイテッド	抗生物質製剤、その使用法及び作成方法
EP1663169A4 (en)	2003-09-15	2010-11-24	Middlebrook Pharmaceuticals In	ANTIBIOTICS, ITS USE AND FORMULATION
WO2006014427A1 (en)	2004-07-02	2006-02-09	Advancis Pharmaceutical Corporation	Tablet for pulsed delivery
FI117133B (fi) *	2004-10-19	2006-06-30	Auramo Oy	Menetelmä ja pihtilaite kuormien käsittelemiseksi
ES2261090B1 (es) *	2005-04-25	2007-06-16	Ercros Industrial, S.A.	Procedimiento de obtencion de derivados de eritromicina a y compuestos obtenidos.
US8357394B2 (en)	2005-12-08	2013-01-22	Shionogi Inc.	Compositions and methods for improved efficacy of penicillin-type antibiotics
US8778924B2 (en)	2006-12-04	2014-07-15	Shionogi Inc.	Modified release amoxicillin products
JP5126685B2 (ja) *	2006-05-01	2013-01-23	大正製薬株式会社	マクロライド誘導体
US8299052B2 (en)	2006-05-05	2012-10-30	Shionogi Inc.	Pharmaceutical compositions and methods for improved bacterial eradication
US20090054634A1 (en) *	2007-08-09	2009-02-26	Vinod Kumar Kansal	Process for the preparation of clarithromycin
CN102382157B (zh) *	2010-09-03	2015-04-08	上海医药工业研究院	一种红霉素a衍生物及其制备方法

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BE759252A (fr)	1969-11-21	1971-05-21	Lilly Co Eli	Erytromycyl b amine
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JPS61103890A (ja) *	1984-10-26	1986-05-22	Taisho Pharmaceut Co Ltd	６−０−メチルエリスロマイシンａ誘導体
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EP0201166B1 (en)	1985-03-12	1990-02-07	Beecham Group Plc	Erythromycin derivatives
US4670549A (en) *	1985-03-18	1987-06-02	Taisho Pharmaceutical Co., Ltd.	Method for selective methylation of erythromycin a derivatives
JPS61229895A (ja) *	1985-04-03	1986-10-14	Nippon Zeon Co Ltd	保護化デス−ｎ−メチルエリスロマイシン誘導体
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JPS63107994A (ja)	1986-05-02	1988-05-12	Taisho Pharmaceut Co Ltd	エリスロマイシン誘導体
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KR960000434B1 (ko) *	1986-12-17	1996-01-06	다이쇼 세이야꾸 가부시끼가이샤	에리스로마이신 a유도체 및 그의 제조 방법
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1997
- 1997-09-10 US US08/927,057 patent/US5929219A/en not_active Ceased
1998
- 1998-09-01 DE DE69814422T patent/DE69814422T2/de not_active Expired - Fee Related
- 1998-09-01 CA CA002301639A patent/CA2301639C/en not_active Expired - Fee Related
- 1998-09-01 AT AT98944641T patent/ATE239751T1/de not_active IP Right Cessation
- 1998-09-01 PT PT98944641T patent/PT1015466E/pt unknown
- 1998-09-01 KR KR1020007002435A patent/KR100553468B1/ko not_active Expired - Fee Related
- 1998-09-01 JP JP2000510752A patent/JP2001515914A/ja active Pending
- 1998-09-01 AU AU92136/98A patent/AU9213698A/en not_active Abandoned
- 1998-09-01 WO PCT/US1998/018115 patent/WO1999012946A1/en not_active Ceased
- 1998-09-01 IL IL13446898A patent/IL134468A0/xx unknown
- 1998-09-01 ES ES98944641T patent/ES2198745T3/es not_active Expired - Lifetime
- 1998-09-01 DK DK98944641T patent/DK1015466T3/da active
- 1998-09-01 EP EP98944641A patent/EP1015466B1/en not_active Expired - Lifetime
2000
- 2000-02-09 IL IL134468A patent/IL134468A/en not_active IP Right Cessation
2004
- 2004-03-05 US US10/794,595 patent/USRE39531E1/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
CA2301639C (en)	2007-06-26
ES2198745T3 (es)	2004-02-01
EP1015466A1 (en)	2000-07-05
ATE239751T1 (de)	2003-05-15
EP1015466B1 (en)	2003-05-07
WO1999012946A1 (en)	1999-03-18
KR100553468B1 (ko)	2006-02-22
IL134468A0 (en)	2001-04-30
US5929219A (en)	1999-07-27
KR20010023778A (ko)	2001-03-26
DE69814422D1 (de)	2003-06-12
PT1015466E (pt)	2003-09-30
IL134468A (en)	2009-09-01
AU9213698A (en)	1999-03-29
JP2001515914A (ja)	2001-09-25
USRE39531E1 (en)	2007-03-27
CA2301639A1 (en)	1999-03-18
DE69814422T2 (de)	2004-05-06

Publication	Publication Date	Title
IL134468A0 (en)	2001-04-30	9-hydrazone and 9-azine erythromycin derivatives and a process of making the same
DK1040107T3 (da)	2003-05-05	6-O-alkyl-derivater af erythronolid B
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FI974435A7 (fi)	1997-12-05	Menetelmä 2,4-diklooripyridiinien muuttamiseksi 2-aryylioksi-4-kloorip yridiineiksi
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ATE196292T1 (de)	2000-09-15	Zwischenprodukte um 2-imidazolin-5onederivate herzustellen.
IS1853B (is)	2003-02-21	Ný aðferð til að búa til 3-N,N-dísýklóbútýlamínó-8-flúor-3,4-díhýdró-2H-1-bensópýran-5-karboxamíð
DK0977867T3 (da)	2007-06-18	Fremgangsmåde til fremstilling af biotin
DK1018546T3 (da)	2005-07-25	Mikroorganismer, der producerer 5-aminolevulinsyre, og fremgangsmåder til fremstilling af 5-aminolevulinsyre ved anvendelse heraf
EP0648717A3 (en)	1996-04-10	Reaction sintered ceramics and process for their manufacture.
DK1032580T3 (da)	2004-08-02	Fremgangsmåde til N-desmethylering af erythromyciner og derivater deraf