DK1087986T3 - Testosteronderivat - Google Patents

Testosteronderivat

Info

Publication number: DK1087986T3
Authority: DK; Denmark
Prior art keywords: testosterone; compound; testosterone derivative; good; oxoundecyl
Prior art date: 1998-06-19

Application number

DK99929208T

Other languages

English (en)

Inventor

Dirk Leysen

Der Voort Hendrikus Adrian Van

Original Assignee

Akzo Nobel Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-06-19

Filing date

1999-06-14

Publication date

2002-06-17

1999-06-14 Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv

2002-06-17 Application granted granted Critical

2002-06-17 Publication of DK1087986T3 publication Critical patent/DK1087986T3/da

Links

150000003515 testosterones Chemical class 0.000 title abstract 2
MUMGGOZAMZWBJJ-DYKIIFRCSA-N Testostosterone Chemical compound O=C1CC[C@]2(C)[C@H]3CC[C@](C)([C@H](CC4)O)[C@@H]4[C@@H]3CCC2=C1 MUMGGOZAMZWBJJ-DYKIIFRCSA-N 0.000 abstract 2
150000001875 compounds Chemical class 0.000 abstract 2
YSGQGNQWBLYHPE-CFUSNLFHSA-N (7r,8r,9s,10r,13s,14s,17s)-17-hydroxy-7,13-dimethyl-2,6,7,8,9,10,11,12,14,15,16,17-dodecahydro-1h-cyclopenta[a]phenanthren-3-one Chemical compound C1C[C@]2(C)[C@@H](O)CC[C@H]2[C@@H]2[C@H](C)CC3=CC(=O)CC[C@@H]3[C@H]21 YSGQGNQWBLYHPE-CFUSNLFHSA-N 0.000 abstract 1
WRLOOHHQBLTCLM-QKLCDPPYSA-N [(7r,8r,9s,10r,13s,14s,17s)-7,13-dimethyl-3-oxo-2,6,7,8,9,10,11,12,14,15,16,17-dodecahydro-1h-cyclopenta[a]phenanthren-17-yl] undecanoate Chemical compound C([C@H]1C)C2=CC(=O)CC[C@@H]2[C@@H]2[C@@H]1[C@@H]1CC[C@H](OC(=O)CCCCCCCCCC)[C@@]1(C)CC2 WRLOOHHQBLTCLM-QKLCDPPYSA-N 0.000 abstract 1
239000003098 androgen Substances 0.000 abstract 1
238000002347 injection Methods 0.000 abstract 1
239000007924 injection Substances 0.000 abstract 1
229960003604 testosterone Drugs 0.000 abstract 1
ZDPHROOEEOARMN-UHFFFAOYSA-N undecanoic acid Chemical compound CCCCCCCCCCC(O)=O ZDPHROOEEOARMN-UHFFFAOYSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0066—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
- C07J1/007—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
- C07J1/0074—Esters
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/16—Masculine contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/26—Androgens

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
Engineering & Computer Science (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Bioinformatics & Cheminformatics (AREA)
General Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Endocrinology (AREA)
Diabetes (AREA)
Reproductive Health (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Steroid Compounds (AREA)
Cultivation Receptacles Or Flower-Pots, Or Pots For Seedlings (AREA)
Percussion Or Vibration Massage (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicinal Preparation (AREA)

DK99929208T 1998-06-19 1999-06-14 Testosteronderivat DK1087986T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP98202052		1998-06-19
PCT/EP1999/004102 WO1999067271A1 (en)	1998-06-19	1999-06-14	Testosterone derivative

Publications (1)

Publication Number	Publication Date
DK1087986T3 true DK1087986T3 (da)	2002-06-17

Family

ID=8233831

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK99929208T DK1087986T3 (da)	1998-06-19	1999-06-14	Testosteronderivat

Country Status (25)

Country	Link
US (3)	US6437158B1 (da)
EP (1)	EP1087986B1 (da)
JP (1)	JP2002518514A (da)
KR (1)	KR100596649B1 (da)
CN (1)	CN1172949C (da)
AT (1)	ATE215961T1 (da)
AU (1)	AU756739B2 (da)
BR (1)	BR9911344A (da)
CA (1)	CA2333985C (da)
CZ (1)	CZ293319B6 (da)
DE (1)	DE69901250T2 (da)
DK (1)	DK1087986T3 (da)
ES (1)	ES2175989T3 (da)
HU (1)	HUP0102274A3 (da)
ID (1)	ID27260A (da)
IL (1)	IL139689A (da)
NO (1)	NO316518B1 (da)
NZ (1)	NZ508299A (da)
PL (1)	PL191285B1 (da)
PT (1)	PT1087986E (da)
RU (1)	RU2216546C2 (da)
SK (1)	SK282796B6 (da)
TR (1)	TR200003743T2 (da)
WO (1)	WO1999067271A1 (da)
ZA (1)	ZA200006813B (da)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP1212345B1 (en) *	1999-04-06	2003-08-06	Akzo Nobel N.V.	Orally active 7-alpha-alkyl androgens
ATE294812T1 (de) *	2000-07-28	2005-05-15	Akzo Nobel Nv	16alpha-methyl oder ethyl substituierte oestrogene
JP3774888B2 (ja) *	2001-11-28	2006-05-17	日本化薬株式会社	ステロイド類化合物のｌｃ−ｍｓによる高感度検出法
TW200404552A (en) *	2002-05-30	2004-04-01	Akzo Nobel Nv	Self administered contraception
TW200400041A (en) *	2002-05-30	2004-01-01	Akzo Nobel Nv	Use of new etonogestrel esters
TW200403065A (en)	2002-05-30	2004-03-01	Akzo Nobel Nv	New etonogestrel esters
GB0304927D0 (en)	2003-03-04	2003-04-09	Resolution Chemicals Ltd	Process for the production of tibolone
JO2505B1 (en)	2003-03-14	2009-10-05	باير شيرنغ فارما اكتنجيسيلشافت	Pharmacy methods and formulations for obtaining acceptable serum testosterone levels
JO2492B1 (en)	2003-04-28	2009-10-05	شيرينج ايه جي	A pharmaceutical formula in the form of aqueous gel for the skin use of its active ingredients
PE20050677A1 (es)	2003-12-22	2005-10-04	Akzo Nobel Nv	Esteroides con perfil androgenico y progestagenico mixto
UA89964C2 (ru)	2004-09-08	2010-03-25	Н.В. Органон	15β-ЗАМЕЩЕННЫЕ СТЕРОИДЫ, КОТОРЫЕ ИМЕЮТ СЕЛЕКТИВНУЮ ЭСТРОГЕННУЮ АКТИВНОСТЬ
EP1879382B1 (en)	2006-07-10	2017-09-06	Samsung Electronics Co., Ltd.	Multi-screen display apparatus and method for digital broadcast receiver
WO2008101030A1 (en) *	2007-02-13	2008-08-21	The Regents Of The University Of California	Methods for amplifying steroid hormone effects
US20090017107A1 (en) *	2007-07-13	2009-01-15	Oral Delivery Technology Ltd.	Novel composition to increase libido
US20090018107A1 (en) *	2007-07-13	2009-01-15	Oral Delivery Technology Ltd.	Novel composition to increase muscle strength
US20100303937A1 (en) *	2009-06-01	2010-12-02	Michael Farber	Novel composition to increase testosterone levels
CN102558267A (zh) *	2012-01-13	2012-07-11	宜城市共同药业有限公司	庚酸睾酮的制备方法
JP6457383B2 (ja) *	2012-04-06	2019-01-23	アンタレス・ファーマ・インコーポレーテッド	テストステロン組成物の針支援式ジェット注入投与
EP4349383A3 (en) *	2013-02-11	2024-06-19	Antares Pharma, Inc.	Needle assisted jet injection device having reduced trigger force

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5342834A (en) *	1989-04-07	1994-08-30	The Population Council, Inc.	Method for androgen supplementation

1999
- 1999-06-14 DE DE69901250T patent/DE69901250T2/de not_active Expired - Fee Related
- 1999-06-14 SK SK1940-2000A patent/SK282796B6/sk not_active IP Right Cessation
- 1999-06-14 CA CA002333985A patent/CA2333985C/en not_active Expired - Fee Related
- 1999-06-14 HU HU0102274A patent/HUP0102274A3/hu unknown
- 1999-06-14 WO PCT/EP1999/004102 patent/WO1999067271A1/en not_active Ceased
- 1999-06-14 KR KR1020007014182A patent/KR100596649B1/ko not_active Expired - Fee Related
- 1999-06-14 PL PL344987A patent/PL191285B1/pl not_active IP Right Cessation
- 1999-06-14 NZ NZ508299A patent/NZ508299A/xx unknown
- 1999-06-14 EP EP99929208A patent/EP1087986B1/en not_active Expired - Lifetime
- 1999-06-14 AU AU46101/99A patent/AU756739B2/en not_active Ceased
- 1999-06-14 US US09/719,927 patent/US6437158B1/en not_active Expired - Fee Related
- 1999-06-14 TR TR2000/03743T patent/TR200003743T2/xx unknown
- 1999-06-14 CZ CZ20004779A patent/CZ293319B6/cs not_active IP Right Cessation
- 1999-06-14 JP JP2000555922A patent/JP2002518514A/ja active Pending
- 1999-06-14 IL IL13968999A patent/IL139689A/en not_active IP Right Cessation
- 1999-06-14 AT AT99929208T patent/ATE215961T1/de not_active IP Right Cessation
- 1999-06-14 DK DK99929208T patent/DK1087986T3/da active
- 1999-06-14 ID IDW20002632A patent/ID27260A/id unknown
- 1999-06-14 PT PT99929208T patent/PT1087986E/pt unknown
- 1999-06-14 ES ES99929208T patent/ES2175989T3/es not_active Expired - Lifetime
- 1999-06-14 RU RU2001101892/04A patent/RU2216546C2/ru not_active IP Right Cessation
- 1999-06-14 CN CNB998075175A patent/CN1172949C/zh not_active Expired - Fee Related
- 1999-06-14 BR BR9911344-9A patent/BR9911344A/pt not_active Application Discontinuation
2000
- 2000-11-21 ZA ZA200006813A patent/ZA200006813B/en unknown
- 2000-12-18 NO NO20006455A patent/NO316518B1/no unknown
2002
- 2002-06-21 US US10/177,989 patent/US20040033999A1/en not_active Abandoned
2004
- 2004-10-13 US US10/964,076 patent/US6989378B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
WO1999067271A1 (en)	1999-12-29
HK1034263A1 (en)	2001-10-19
PL191285B1 (pl)	2006-04-28
US20050153949A1 (en)	2005-07-14
US20040033999A1 (en)	2004-02-19
CN1305488A (zh)	2001-07-25
CN1172949C (zh)	2004-10-27
PT1087986E (pt)	2002-08-30
EP1087986B1 (en)	2002-04-10
KR20010052850A (ko)	2001-06-25
AU756739B2 (en)	2003-01-23
HUP0102274A2 (hu)	2001-12-28
EP1087986A1 (en)	2001-04-04
HUP0102274A3 (en)	2002-08-28
US6437158B1 (en)	2002-08-20
CZ293319B6 (cs)	2004-04-14
ES2175989T3 (es)	2002-11-16
BR9911344A (pt)	2001-03-13
CA2333985C (en)	2007-04-10
PL344987A1 (en)	2001-11-19
NO20006455D0 (no)	2000-12-18
IL139689A (en)	2004-09-27
DE69901250T2 (de)	2002-10-17
IL139689A0 (en)	2002-02-10
ID27260A (id)	2001-03-22
US6989378B2 (en)	2006-01-24
CA2333985A1 (en)	1999-12-29
TR200003743T2 (tr)	2001-07-23
NO20006455L (no)	2000-12-18
RU2216546C2 (ru)	2003-11-20
NO316518B1 (no)	2004-02-02
DE69901250D1 (de)	2002-05-16
JP2002518514A (ja)	2002-06-25
KR100596649B1 (ko)	2006-07-06
ATE215961T1 (de)	2002-04-15
SK19402000A3 (sk)	2001-07-10
SK282796B6 (sk)	2002-12-03
ZA200006813B (en)	2002-02-21
CZ20004779A3 (en)	2001-06-13
NZ508299A (en)	2003-04-29
AU4610199A (en)	2000-01-10

Publication	Publication Date	Title
DK1087986T3 (da)	2002-06-17	Testosteronderivat
ES2194446T3 (es)	2003-11-16	Derivados de bibiclooctano utilizados como plastificantes.
AU2002211216A1 (en)	2002-04-02	Substituted aminopropoxyaryl derivatives useful as agonists for lxr
FR2733244B1 (fr)	1999-07-30	Systeme de stabilisants a base de derives de polyalkylpiperidine
JO2654B1 (en)	2012-06-17	Multiple aryl caroxa amides are useful as lipid - lowering agents
AU2610699A (en)	1999-09-15	Derivatives of glp-1 analogs
MXPA05009985A (es)	2005-11-04	Ligandos de receptores de canabinoides.
DE69325454D1 (de)	1999-07-29	Taxol-derivate
CO5231161A1 (es)	2002-12-27	4-aminopicolinatos y su uso como herbicidas
PL378577A1 (pl)	2006-05-02	Pochodne estrogenu jako inhibitory sulfatazy steroidowej
IT1311922B1 (it)	2002-03-20	Composti farmaceutici.
ATE278661T1 (de)	2004-10-15	Anthranilsäurederivate
DE60135748D1 (de)	2008-10-23	Synthese zyklischerverbindungen
NO20025035D0 (no)	2002-10-18	Oksadiazolderivater som har anticancer-effekter
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DE69617909D1 (de)	2002-01-24	2-substituierte vitamin-d3-derivate
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TR200400293T4 (tr)	2004-04-21	9-dihidro-13-asetilbasatin III'e ait suda çözünebilir 9-dihidro-paklitaksel türevlerinin sentezi.
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BR0013100A (pt)	2002-04-30	Processo para a preparação de um composto de 2-arilvinil alquil éter
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ECSP992934A (es)	1999-06-11	Procedimiento mejorado para la preparacion de derivados de norbenzomorfano, valiosos farmaceuticamente