DK120783A - Fremgangsmaade til fremstilling af substituerede 1h-pyrazolo(1,5-a)pyrimidiner - Google Patents

Fremgangsmaade til fremstilling af substituerede 1h-pyrazolo(1,5-a)pyrimidiner Download PDF

Info

Publication number: DK120783A
Authority: DK; Denmark
Prior art keywords: pyrazolo; pyrimidines; preparing substituted; substituted; preparing
Prior art date: 1982-03-16

Application number

DK120783A

Other languages

English (en)

Other versions

DK120783D0 (da

Inventor

Gianfederico Doria

Carlo Passarotti

Ada Buttinoni

Original Assignee

Erba Farmitalia

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1982-03-16

Filing date

1983-03-15

Publication date

1983-09-17

1983-02-04 Priority claimed from GB838303089A external-priority patent/GB8303089D0/en

1983-03-15 Application filed by Erba Farmitalia filed Critical Erba Farmitalia

1983-03-15 Publication of DK120783D0 publication Critical patent/DK120783D0/da

1983-09-17 Publication of DK120783A publication Critical patent/DK120783A/da

Links

150000003230 pyrimidines Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

DK120783A 1982-03-16 1983-03-15 Fremgangsmaade til fremstilling af substituerede 1h-pyrazolo(1,5-a)pyrimidiner DK120783A (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB8207637		1982-03-16
GB838303089A GB8303089D0 (en)	1983-02-04	1983-02-04	Substituted 1h-pyrazolo 1,5-a pyrimidines

Publications (2)

Publication Number	Publication Date
DK120783D0 DK120783D0 (da)	1983-03-15
DK120783A true DK120783A (da)	1983-09-17

Family

ID=26282260

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK120783A DK120783A (da)	1982-03-16	1983-03-15	Fremgangsmaade til fremstilling af substituerede 1h-pyrazolo(1,5-a)pyrimidiner

Country Status (13)

Country	Link
US (1)	US4482555A (da)
AU (1)	AU557300B2 (da)
CA (1)	CA1192546A (da)
CH (1)	CH654306A5 (da)
DE (1)	DE3309432A1 (da)
DK (1)	DK120783A (da)
FI (1)	FI74469C (da)
FR (1)	FR2523582B1 (da)
IL (1)	IL68133A (da)
IT (1)	IT1194555B (da)
NL (1)	NL8300934A (da)
SE (1)	SE450573B (da)
SU (1)	SU1366060A3 (da)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
USD344263S (en)	1991-11-15	1994-02-15	Masami Seido	Plug-receiving metal fitting
RU2147584C1 (ru) *	1995-10-27	2000-04-20	Американ Цианамид Компани	Способ получения дигалоидазолопиримидинов и способ получения дигидроксиазолопиримидинов
US6245759B1 (en) *	1999-03-11	2001-06-12	Merck & Co., Inc.	Tyrosine kinase inhibitors
MY125533A (en)	1999-12-06	2006-08-30	Bristol Myers Squibb Co	Heterocyclic dihydropyrimidine compounds
EP1782859A3 (en) *	2003-04-11	2009-09-30	High Point Pharmaceuticals, LLC	Pharmaceutical use of substituted pyrazolo [1,5- a]pyrimidines
WO2004089471A2 (en) *	2003-04-11	2004-10-21	Novo Nordisk A/S	NEW PYRAZOLO[1,5-a] PYRIMIDINES DERIVATIVES AND PHARMACEUTICAL USE THEREOF
US7772232B2 (en)	2004-04-15	2010-08-10	Bristol-Myers Squibb Company	Quinazolinyl compounds as inhibitors of potassium channel function
EP1802623A1 (en) *	2004-10-12	2007-07-04	Novo Nordisk A/S	11beta-hydroxysteroid dehydrogenase type 1 active spiro compounds
KR20080069189A (ko) *	2005-11-01	2008-07-25	트랜스테크 파르마, 인크.	치환된 아미드의 약학적 사용
EA200801243A1 (ru) *	2005-11-01	2008-10-30	Транстек Фарма	Фармацевтическое применение замещенных амидов
JP2009530346A (ja) *	2006-03-21	2009-08-27	ハイポイントファーマシューティカルズ，リミティドライアビリティカンパニー	メタボリックシンドロームの治療用のアダマンタン誘導体
KR20090014347A (ko)	2006-04-07	2009-02-10	하이 포인트 파마슈티칼스, 엘엘씨	11β-히드록시스테로이드 탈수소효소 타입 1 활성 화합물
EP2038255A2 (en) *	2006-06-16	2009-03-25	High Point Pharmaceuticals, LLC	Pharmaceutical use of substituted piperidine carboxamides
EP1878721A1 (en) *	2006-07-13	2008-01-16	Novo Nordisk A/S	4-Piperidylbenzamides as 11-beta-hydroxysteroid dehydrogenase type 1 inhibitors
WO2008006702A1 (en) *	2006-07-13	2008-01-17	High Point Pharmaceuticals, Llc.	11beta-hydroxysteroid dehydrogenase type 1 active compounds
WO2008101885A1 (en) *	2007-02-23	2008-08-28	High Point Pharmaceuticals, Llc	N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase
EP2125704A1 (en) *	2007-02-23	2009-12-02	High Point Pharmaceuticals, LLC	N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase
EP2150526B1 (en)	2007-02-23	2017-09-20	vTv Therapeutics LLC	N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase
EP2129652A2 (en) *	2007-02-23	2009-12-09	High Point Pharmaceuticals, LLC	N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase
WO2008110196A1 (en) *	2007-03-09	2008-09-18	High Point Pharmaceuticals, Llc	Indole- and benzimidazole amides as hydroxysteroid dehydrogenase inhibitors
US20100056600A1 (en) *	2007-03-28	2010-03-04	Soren Ebdrup	11beta-hsd1 active compounds
CN101677562A (zh) *	2007-04-11	2010-03-24	高点制药有限责任公司	新化合物
ES2393230T3 (es) *	2007-04-24	2012-12-19	High Point Pharmaceuticals, Llc	Uso farmacéutico de amidas sustituidas

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
BE786611A (fr) *	1971-08-16	1973-01-22	Int Chem & Nuclear Corp	Nouveaux inhibiteurs de xanthine-oxydase et leur procede de preparatio
US3907799A (en) *	1971-08-16	1975-09-23	Icn Pharmaceuticals	Xanthine oxidase inhibitors
US3925385A (en) *	1972-04-20	1975-12-09	Icn Pharmaceuticals	6-Carbethoxy-3,7-disubstitutedpyrazolo{8 1,5a{9 pyrimidines
BE792533A (fr) *	1971-12-09	1973-06-08	Int Chem & Nuclear Corp	Nouvelles pyrazolo (1,5a) pyrimidines et leur procede de preparation
US4093617A (en) *	1974-11-12	1978-06-06	Icn Pharmaceuticals, Inc.	3,5,7-Trisubstituted pyrazolo[1,5-a]pyrimidines
US4048184A (en) *	1976-11-15	1977-09-13	E. R. Squibb & Sons, Inc.	6-Phenyl-2H-pyrazolo[3,4-b]pyridines
US4281000A (en) *	1979-07-09	1981-07-28	American Cyanamid Company	Substituted pyrazolo (1,5-a)pyrimidines and their use as anxiolytic agents

1983
- 1983-03-09 AU AU12304/83A patent/AU557300B2/en not_active Ceased
- 1983-03-10 US US06/474,205 patent/US4482555A/en not_active Expired - Fee Related
- 1983-03-11 CH CH1325/83A patent/CH654306A5/de not_active IP Right Cessation
- 1983-03-11 IT IT20024/83A patent/IT1194555B/it active
- 1983-03-15 NL NL8300934A patent/NL8300934A/xx active Search and Examination
- 1983-03-15 FR FR8304253A patent/FR2523582B1/fr not_active Expired
- 1983-03-15 SE SE8301412A patent/SE450573B/sv not_active IP Right Cessation
- 1983-03-15 FI FI830864A patent/FI74469C/fi not_active IP Right Cessation
- 1983-03-15 DK DK120783A patent/DK120783A/da not_active Application Discontinuation
- 1983-03-15 CA CA000423644A patent/CA1192546A/en not_active Expired
- 1983-03-15 SU SU833565748A patent/SU1366060A3/ru active
- 1983-03-15 IL IL68133A patent/IL68133A/xx unknown
- 1983-03-16 DE DE19833309432 patent/DE3309432A1/de not_active Withdrawn

Also Published As

Publication number	Publication date
CH654306A5 (de)	1986-02-14
AU1230483A (en)	1983-09-22
US4482555A (en)	1984-11-13
CA1192546A (en)	1985-08-27
FR2523582B1 (fr)	1985-12-06
SU1366060A3 (ru)	1988-01-07
AU557300B2 (en)	1986-12-18
SE8301412L (sv)	1983-09-17
IT8320024A0 (it)	1983-03-11
DE3309432A1 (de)	1983-09-22
IL68133A0 (en)	1983-06-15
NL8300934A (nl)	1983-10-17
FI74469C (fi)	1988-02-08
IL68133A (en)	1985-12-31
FR2523582A1 (fr)	1983-09-23
SE8301412D0 (sv)	1983-03-15
FI830864A0 (fi)	1983-03-15
FI830864L (fi)	1983-09-17
IT1194555B (it)	1988-09-22
FI74469B (fi)	1987-10-30
DK120783D0 (da)	1983-03-15
SE450573B (sv)	1987-07-06

Legal Events

Date	Code	Title	Description
1989-11-13	AHB	Application shelved due to non-payment

Publication	Publication Date	Title
DK120783A (da)	1983-09-17	Fremgangsmaade til fremstilling af substituerede 1h-pyrazolo(1,5-a)pyrimidiner
DK350083A (da)	1984-02-11	Fremgangsmaade til fremstilling af phenylethanolaminer
DK194783D0 (da)	1983-05-02	Fremgangsmade til fremstilling af bicycliske forbindelser
DK29183A (da)	1983-08-02	Fremgangsmaade til fremstilling af purinderivater
DK25081A (da)	1981-07-24	Fremgangsmaade til fremstilling af imidazo(1,2-a) pyridiner
DK300883D0 (da)	1983-06-29	Fremgangsmade til fremstilling af thromobolytiske midler
DK227183A (da)	1983-11-25	Fremgangsmaade til fremstilling af imidazo(1,2-c)-pyrazolo(3,4-e)pyrimidiner med den almene formel i
DK173983D0 (da)	1983-04-20	Fremgangsmade til fremstilling af imidazo (1,2-alfa)pyridiner
DK210083A (da)	1983-11-25	Fremgangsmaade til fremstilling af 6a,10a-trans-hexahydrodibenzopyranoner
DK540984A (da)	1985-05-15	Fremgangsmaade til fremstilling af 1,2,4-triazolo-(1,5-a)pyrimidin-2-sulfonylchlorider
DK133482A (da)	1982-09-26	Fremgangsmaade til fremstilling af imidazo(1,2-a)pyrimidiner
DK390583A (da)	1984-02-28	Fremgangsmaade til fremstilling af imidazo(1,2-a)pyrimidiner
FI834665A0 (fi)	1983-12-19	Imidazo(1,5-a)pyridin-derivat
DK314682A (da)	1983-01-16	Fremgangsmaade til fremstilling af substituerede thiazolo-(3,2-a)pyrimidiner
DK200280A (da)	1980-11-09	Fremgangsmaade til fremstilling af substituerede pyrido (1,2-a) pyrimidiner
FI834664A0 (fi)	1983-12-19	Substituerade imidazo(1,5-a)pyridiner
DK44383D0 (da)	1983-02-03	Fremgangsmade til fremstilling af substituerede 1,3,4-thiadiazolo(3,2-a)pyrimidiner
DK40883A (da)	1983-08-04	Fremgangsmaade til fremstilling af benzothienylallylaminer
DK424083D0 (da)	1983-09-16	Fremgangsmade til fremstilling af anthracyclinglycosider
DK133883D0 (da)	1983-03-24	Fremgangsmade til fremstilling af substituerede ethenylderivater af 1h-pyrazolo(1,5-a)pyrimidin
DK219483D0 (da)	1983-05-17	Fremgangsmade til fremstilling af anthracyclinglycosider
DK162097C (da)	1992-02-24	Fremgangsmaade til fremstilling af riboflavin
DK446683D0 (da)	1983-09-29	Fremgangsmade til fremstilling af 6-anilino-5,8-quinoxalindioner
DK186784D0 (da)	1984-04-11	Fremgangsmaade til fremstilling af pyrimidintrionderivater
DK154971C (da)	1989-07-10	Fremgangsmaade til fremstilling af phenylpyridazinforbindelser