DK1265860T3 - Amidinoforbindelse og salte deraf, der er nyttige som nitrogenoxidsyntaseinhibitorer - Google Patents

Amidinoforbindelse og salte deraf, der er nyttige som nitrogenoxidsyntaseinhibitorer

Info

Publication number: DK1265860T3
Authority: DK; Denmark
Prior art keywords: nitric oxide; oxide synthase; synthase inhibitors; salts useful; amidino compound
Prior art date: 2000-03-24

Application number

DK01922636T

Other languages

English (en)

Inventor

W Gary Phillips

Gopichand Yalamanchili

Donald W Hansen

Michelle A Promo

Ronald Keith Webber

Alok K Awasthi

Arija A Bergmanis

Richard C Durley

Timothy J Hagen

Brian S Hickory

Alan E Moormann

Barnett S Pitzele

Mahima Trivedi

Embse Richard Vonder

Scott S Ganser

Ann E Hallinan

Richard R Schartman

Jeffrey S Snyder

Sofya Tsymbalov

Original Assignee

Pharmacia Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-03-24

Filing date

2001-03-23

Publication date

2005-07-11

2001-03-23 Application filed by Pharmacia Corp filed Critical Pharmacia Corp

2005-07-11 Application granted granted Critical

2005-07-11 Publication of DK1265860T3 publication Critical patent/DK1265860T3/da

Links

-1 Amidino compound Chemical class 0.000 title 1
239000000236 nitric oxide synthase inhibitor Substances 0.000 title 1
CSYSULGPHGCBQD-UHFFFAOYSA-N s-ethylisothiouronium diethylphosphate Chemical compound CCSC(N)=N.CCOP(O)(=O)OCC CSYSULGPHGCBQD-UHFFFAOYSA-N 0.000 title 1
150000003839 salts Chemical class 0.000 title 1

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- C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
- C07D271/07—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
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DK01922636T 2000-03-24 2001-03-23 Amidinoforbindelse og salte deraf, der er nyttige som nitrogenoxidsyntaseinhibitorer DK1265860T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US19192300P	2000-03-24	2000-03-24
PCT/US2001/009433 WO2001072703A1 (en)	2000-03-24	2001-03-23	Amidino compound and salts thereof useful as nitric oxide synthase inhibitors

Publications (1)

Publication Number	Publication Date
DK1265860T3 true DK1265860T3 (da)	2005-07-11

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Application Number	Title	Priority Date	Filing Date
DK01922636T DK1265860T3 (da)	2000-03-24	2001-03-23	Amidinoforbindelse og salte deraf, der er nyttige som nitrogenoxidsyntaseinhibitorer
DK01920718T DK1265859T3 (da)	2000-03-24	2001-03-23	Amidinoforbindelser der er nyttige som nitrogenoxidsyntaseinhibitorer

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Application Number	Title	Priority Date	Filing Date
DK01920718T DK1265859T3 (da)	2000-03-24	2001-03-23	Amidinoforbindelser der er nyttige som nitrogenoxidsyntaseinhibitorer

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US (5)	US6586474B2 (da)
EP (2)	EP1265860B1 (da)
JP (2)	JP4205340B2 (da)
KR (1)	KR100835265B1 (da)
CN (1)	CN1294117C (da)
AR (1)	AR033359A1 (da)
AT (2)	ATE313525T1 (da)
AU (4)	AU4774501A (da)
BR (1)	BR0109386A (da)
CA (2)	CA2402199C (da)
DE (2)	DE60116067T2 (da)
DK (2)	DK1265860T3 (da)
ES (2)	ES2256223T3 (da)
GE (1)	GEP20094625B (da)
MX (1)	MXPA02009282A (da)
MY (1)	MY135721A (da)
NZ (4)	NZ532073A (da)
PT (1)	PT1265860E (da)
TW (1)	TWI294417B (da)
WO (2)	WO2001072702A2 (da)
ZA (2)	ZA200206459B (da)

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- 2001-03-23 JP JP2001570616A patent/JP4205340B2/ja not_active Expired - Fee Related
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Also Published As

Publication number	Publication date
CN1294117C (zh)	2007-01-10
DE60116067T2 (de)	2006-08-31
AU4941501A (en)	2001-10-08
WO2001072702A3 (en)	2002-09-19
CA2402436A1 (en)	2001-10-04
CA2402199C (en)	2010-08-03
DE60110902D1 (de)	2005-06-23
DE60116067D1 (de)	2006-01-26
DE60110902T2 (de)	2006-04-27
EP1265860A1 (en)	2002-12-18
JP2003528852A (ja)	2003-09-30
WO2001072703A1 (en)	2001-10-04
MXPA02009282A (es)	2004-06-18
NZ520812A (en)	2004-04-30
AU2001249415B8 (en)	2001-10-08
CA2402199A1 (en)	2001-10-04
US20020019563A1 (en)	2002-02-14
ATE313525T1 (de)	2006-01-15
WO2001072702A2 (en)	2001-10-04
TWI294417B (en)	2008-03-11
ES2240445T3 (es)	2005-10-16
JP2003528853A (ja)	2003-09-30
HK1056161A1 (en)	2004-02-06
CN1419539A (zh)	2003-05-21
ZA200206455B (en)	2003-08-13
AU2001247745B2 (en)	2006-08-31
NZ520813A (en)	2004-05-28
AR033359A1 (es)	2003-12-17
US6914158B2 (en)	2005-07-05
HK1050521A1 (en)	2003-06-27
ES2256223T3 (es)	2006-07-16
GEP20094625B (en)	2009-03-10
AU4774501A (en)	2001-10-08
AU2001249415B2 (en)	2007-01-04
JP4205340B2 (ja)	2009-01-07
EP1265860B1 (en)	2005-05-18
EP1265859A2 (en)	2002-12-18
EP1265859B1 (en)	2005-12-21
JP4216502B2 (ja)	2009-01-28
US7196118B2 (en)	2007-03-27
BR0109386A (pt)	2003-04-15
US20030199701A1 (en)	2003-10-23
KR100835265B1 (ko)	2008-06-09
US20040186178A1 (en)	2004-09-23
MY135721A (en)	2008-06-30
US20050165106A1 (en)	2005-07-28
US6586474B2 (en)	2003-07-01
CA2402436C (en)	2010-02-16
DK1265859T3 (da)	2006-05-01
US7102013B2 (en)	2006-09-05
PT1265860E (pt)	2005-10-31
NZ542734A (en)	2007-06-29
US6403830B2 (en)	2002-06-11
KR20020091138A (ko)	2002-12-05
ATE295832T1 (de)	2005-06-15
ZA200206459B (en)	2003-08-13
US20020111493A1 (en)	2002-08-15
NZ532073A (en)	2005-12-23

Publication	Publication Date	Title
DK1265860T3 (da)	2005-07-11	Amidinoforbindelse og salte deraf, der er nyttige som nitrogenoxidsyntaseinhibitorer
DK1318980T3 (da)	2008-02-11	Hydroxamatderivater, der kan anvendes som deacetylaseinhibitorer
IS5723A (is)	2000-11-21	Nituroxíðs efnasmíða latar (Synthase Inhibitors)
NO20031139L (no)	2003-05-09	2-amino-2-alkyl-4-heksen- og heksynsyrederivater som er anvendbare som nitrogenoksidsyntaseinhibitorer
DK1317421T3 (da)	2005-06-27	2-amino-2-alkyl-5-heptensyre- og heptynsyrederivater der er nyttige som nitrogenoxidsynthaseinhibitorer
NO20032835L (no)	2003-08-15	Nitrogenoksyd-syntase-inhibitor-fosfatsalt
DK1581532T3 (da)	2010-08-16	Pyrazolo-3,4-B pyridinforbindelser og deres anvendelse som phosphodiesterase inhibitorer
DK1220831T3 (da)	2005-08-29	Biaryletherderivater, der er nyttige som monoamingenoptagelsesinhibitorer
NO20031450D0 (no)	2003-03-28	Fumarsyrederivater som NF-kappa B inhibitorer
NO20032830D0 (no)	2003-06-20	Tetrahydropyridinderivater, fremstilling derav og anvendelse som celle-proliferasjonsinhibitorer
NO20031482L (no)	2003-04-01	Nye tiadiazoler og oksadiazoler, og anvendelse derav som fosfodiesterase-7inhibitorer
NO20030135L (no)	2003-02-19	Piperidinforbindelser for anvendelse som CCR-3-inhibitorer
NO20004531D0 (no)	2000-09-11	Halogenerte amidinoaminosyre-derivater anvendbare som nitrogenoksid syntase inhibitorer
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