DK1389193T3 - Fremgangsmåde til fremstilling af biperiden I - Google Patents
Fremgangsmåde til fremstilling af biperiden IInfo
- Publication number
- DK1389193T3 DK1389193T3 DK02750945T DK02750945T DK1389193T3 DK 1389193 T3 DK1389193 T3 DK 1389193T3 DK 02750945 T DK02750945 T DK 02750945T DK 02750945 T DK02750945 T DK 02750945T DK 1389193 T3 DK1389193 T3 DK 1389193T3
- Authority
- DK
- Denmark
- Prior art keywords
- biperiden
- preparation
- exo
- endo
- isomer
- Prior art date
Links
- YSXKPIUOCJLQIE-UHFFFAOYSA-N biperiden Chemical compound C1C(C=C2)CC2C1C(C=1C=CC=CC=1)(O)CCN1CCCCC1 YSXKPIUOCJLQIE-UHFFFAOYSA-N 0.000 title abstract 4
- 229960003003 biperiden Drugs 0.000 title abstract 4
- 239000000203 mixture Substances 0.000 abstract 2
- KRQADKCTBWUTRW-UHFFFAOYSA-N 1-(5-bicyclo[2.2.1]hept-2-enyl)-3-piperidin-1-ylpropan-1-one Chemical compound C1C(C=C2)CC2C1C(=O)CCN1CCCCC1 KRQADKCTBWUTRW-UHFFFAOYSA-N 0.000 abstract 1
- WRYKIHMRDIOPSI-UHFFFAOYSA-N magnesium;benzene Chemical compound [Mg+2].C1=CC=[C-]C=C1.C1=CC=[C-]C=C1 WRYKIHMRDIOPSI-UHFFFAOYSA-N 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
- C07D295/084—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
- C07D295/088—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/10—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by doubly bound oxygen or sulphur atoms
- C07D295/104—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by doubly bound oxygen or sulphur atoms with the ring nitrogen atoms and the doubly bound oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
- C07D295/108—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by doubly bound oxygen or sulphur atoms with the ring nitrogen atoms and the doubly bound oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Hydrogenated Pyridines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Steroid Compounds (AREA)
- Cephalosporin Compounds (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE2001124450 DE10124450A1 (de) | 2001-05-18 | 2001-05-18 | Verfahren zur Herstellung von Biperiden |
| DE2001124452 DE10124452A1 (de) | 2001-05-18 | 2001-05-18 | Verfahren zur Herstellung von Biperiden |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1389193T3 true DK1389193T3 (da) | 2006-03-06 |
Family
ID=26009342
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK02750945T DK1389193T3 (da) | 2001-05-18 | 2002-05-17 | Fremgangsmåde til fremstilling af biperiden I |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US7034158B2 (da) |
| EP (1) | EP1389193B1 (da) |
| JP (1) | JP4338979B2 (da) |
| KR (1) | KR100896836B1 (da) |
| CN (1) | CN1281594C (da) |
| AT (1) | ATE307124T1 (da) |
| BR (1) | BRPI0209850B8 (da) |
| DE (1) | DE50204608D1 (da) |
| DK (1) | DK1389193T3 (da) |
| ES (1) | ES2250678T3 (da) |
| IL (2) | IL158932A0 (da) |
| WO (1) | WO2002094801A1 (da) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5861884B2 (ja) * | 2012-03-29 | 2016-02-16 | 荒川化学工業株式会社 | エキソ型ノルボルネン化合物の製造方法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1005067B (de) * | 1953-03-14 | 1957-03-28 | Knoll Ag | Verfahren zur Herstellung von bicyclisch substituierten Aminopropanolen |
| US2789110A (en) | 1953-03-14 | 1957-04-16 | Knoll Ag | Amino alcohols substituted by bicycloalkyl residues and a process of making same |
| JPH11189729A (ja) | 1997-12-26 | 1999-07-13 | Chemiprokasei Kaisha Ltd | 色素兼紫外線安定剤およびそれを含む高分子組成物 |
| DE10124451A1 (de) | 2001-05-18 | 2002-11-21 | Abbott Gmbh & Co Kg | Verfahren zur Herstellung von Biperiden |
| DE10124449A1 (de) * | 2001-05-18 | 2002-11-21 | Abbott Gmbh & Co Kg | Verfahren zur Herstellung von Biperiden |
-
2002
- 2002-05-17 KR KR1020037015032A patent/KR100896836B1/ko not_active Expired - Lifetime
- 2002-05-17 DE DE50204608T patent/DE50204608D1/de not_active Expired - Lifetime
- 2002-05-17 DK DK02750945T patent/DK1389193T3/da active
- 2002-05-17 WO PCT/EP2002/005498 patent/WO2002094801A1/de not_active Ceased
- 2002-05-17 ES ES02750945T patent/ES2250678T3/es not_active Expired - Lifetime
- 2002-05-17 BR BRPI0209850-4 patent/BRPI0209850B8/pt not_active IP Right Cessation
- 2002-05-17 AT AT02750945T patent/ATE307124T1/de active
- 2002-05-17 US US10/477,767 patent/US7034158B2/en not_active Expired - Lifetime
- 2002-05-17 JP JP2002591474A patent/JP4338979B2/ja not_active Expired - Lifetime
- 2002-05-17 IL IL15893202A patent/IL158932A0/xx unknown
- 2002-05-17 EP EP02750945A patent/EP1389193B1/de not_active Expired - Lifetime
- 2002-05-17 CN CNB02813740XA patent/CN1281594C/zh not_active Expired - Lifetime
-
2003
- 2003-11-18 IL IL158932A patent/IL158932A/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| WO2002094801A1 (de) | 2002-11-28 |
| ES2250678T3 (es) | 2006-04-16 |
| IL158932A0 (en) | 2004-05-12 |
| BR0209850A (pt) | 2004-06-15 |
| EP1389193B1 (de) | 2005-10-19 |
| IL158932A (en) | 2009-12-24 |
| US7034158B2 (en) | 2006-04-25 |
| EP1389193A1 (de) | 2004-02-18 |
| ATE307124T1 (de) | 2005-11-15 |
| JP4338979B2 (ja) | 2009-10-07 |
| JP2004536068A (ja) | 2004-12-02 |
| BRPI0209850B8 (pt) | 2021-05-25 |
| CN1525963A (zh) | 2004-09-01 |
| KR20040007578A (ko) | 2004-01-24 |
| KR100896836B1 (ko) | 2009-05-12 |
| US20050176963A1 (en) | 2005-08-11 |
| DE50204608D1 (de) | 2006-03-02 |
| CN1281594C (zh) | 2006-10-25 |
| BRPI0209850B1 (pt) | 2018-05-15 |
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