DK1421086T3 - 2-(Aminomethyl)-tetrahydro-9-oxa-1,3-diaza-cyclopenta[a]-naphthalenyl-derivater med antipsykotisk aktivitet - Google Patents
2-(Aminomethyl)-tetrahydro-9-oxa-1,3-diaza-cyclopenta[a]-naphthalenyl-derivater med antipsykotisk aktivitetInfo
- Publication number
- DK1421086T3 DK1421086T3 DK02756528T DK02756528T DK1421086T3 DK 1421086 T3 DK1421086 T3 DK 1421086T3 DK 02756528 T DK02756528 T DK 02756528T DK 02756528 T DK02756528 T DK 02756528T DK 1421086 T3 DK1421086 T3 DK 1421086T3
- Authority
- DK
- Denmark
- Prior art keywords
- diaza
- cyclopenta
- oxa
- aminomethyl
- tetrahydro
- Prior art date
Links
- -1 2- (Aminomethyl) -tetrahydro-9-oxa-1,3-diaza-cyclopenta [a] naphthalenyl Chemical class 0.000 title 1
- 230000000561 anti-psychotic effect Effects 0.000 title 1
- VYFYYTLLBUKUHU-UHFFFAOYSA-N dopamine Chemical compound NCCC1=CC=C(O)C(O)=C1 VYFYYTLLBUKUHU-UHFFFAOYSA-N 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 208000035475 disorder Diseases 0.000 abstract 1
- 229960003638 dopamine Drugs 0.000 abstract 1
- 230000008482 dysregulation Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Neurology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Biomedical Technology (AREA)
- Medicinal Chemistry (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
- Psychology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US30693101P | 2001-07-20 | 2001-07-20 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1421086T3 true DK1421086T3 (da) | 2006-12-11 |
Family
ID=23187510
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK02756528T DK1421086T3 (da) | 2001-07-20 | 2002-07-19 | 2-(Aminomethyl)-tetrahydro-9-oxa-1,3-diaza-cyclopenta[a]-naphthalenyl-derivater med antipsykotisk aktivitet |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US6541502B1 (de) |
| EP (1) | EP1421086B1 (de) |
| JP (1) | JP2004537556A (de) |
| CN (1) | CN100369916C (de) |
| AT (1) | ATE338046T1 (de) |
| BR (1) | BR0211207A (de) |
| CA (1) | CA2454543A1 (de) |
| DE (1) | DE60214397T2 (de) |
| DK (1) | DK1421086T3 (de) |
| ES (1) | ES2271314T3 (de) |
| MX (1) | MXPA04000581A (de) |
| WO (1) | WO2003008419A1 (de) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN101120002A (zh) | 2005-02-17 | 2008-02-06 | 惠氏公司 | 环烷基稠合的吲哚、苯并噻吩、苯并呋喃和茚衍生物 |
| TW201412727A (zh) * | 2012-08-24 | 2014-04-01 | Daiichi Sankyo Co Ltd | 具有鏈狀側鏈之色酮衍生物 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE4135474A1 (de) | 1991-10-28 | 1993-04-29 | Bayer Ag | 2-aminomethyl-chromane |
| DE4140540A1 (de) | 1991-12-09 | 1993-06-17 | Bayer Ag | Neue azaheterocyclylmethyl-chromane |
| US5756532A (en) | 1995-11-06 | 1998-05-26 | American Home Products Corporation | Aminomethyl-2 3 8 9-tetrahydro-7H-1 4-dioxino 2 3-E!-indol-8-ones and derivatives |
| IL119483A (en) * | 1995-11-06 | 1999-06-20 | American Home Prod | 2-(Aminomethyl)-3,4,7,9- tetrahydro- 2H-pyrano-2[3,3-e]indol-8-ones their derivatives and pharmaceutical compositions containing them |
| US5750556A (en) | 1996-10-30 | 1998-05-12 | American Home Products Corporation | 2-(aminomethyl)-3,4,7,9-tetrahydro-2H-pyrano- 2,3-E!indol-8-ones and derivatives |
| WO1998035945A1 (en) | 1997-02-18 | 1998-08-20 | American Home Products Corporation | 4-aminoalkoxy-1h-benzimidazole derivatives, their preparation and their use as dopamine autoreceptor (d2) agonists |
-
2002
- 2002-07-18 US US10/197,797 patent/US6541502B1/en not_active Expired - Fee Related
- 2002-07-19 CN CNB028180232A patent/CN100369916C/zh not_active Expired - Fee Related
- 2002-07-19 CA CA002454543A patent/CA2454543A1/en not_active Abandoned
- 2002-07-19 ES ES02756528T patent/ES2271314T3/es not_active Expired - Lifetime
- 2002-07-19 JP JP2003513978A patent/JP2004537556A/ja active Pending
- 2002-07-19 AT AT02756528T patent/ATE338046T1/de not_active IP Right Cessation
- 2002-07-19 DK DK02756528T patent/DK1421086T3/da active
- 2002-07-19 EP EP02756528A patent/EP1421086B1/de not_active Expired - Lifetime
- 2002-07-19 BR BR0211207-8A patent/BR0211207A/pt not_active IP Right Cessation
- 2002-07-19 WO PCT/US2002/022981 patent/WO2003008419A1/en not_active Ceased
- 2002-07-19 DE DE60214397T patent/DE60214397T2/de not_active Expired - Fee Related
- 2002-07-19 MX MXPA04000581A patent/MXPA04000581A/es active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| EP1421086B1 (de) | 2006-08-30 |
| JP2004537556A (ja) | 2004-12-16 |
| ES2271314T3 (es) | 2007-04-16 |
| US6541502B1 (en) | 2003-04-01 |
| ATE338046T1 (de) | 2006-09-15 |
| DE60214397D1 (en) | 2006-10-12 |
| DE60214397T2 (de) | 2007-10-11 |
| MXPA04000581A (es) | 2004-04-20 |
| CA2454543A1 (en) | 2003-01-30 |
| EP1421086A1 (de) | 2004-05-26 |
| CN1555377A (zh) | 2004-12-15 |
| WO2003008419A1 (en) | 2003-01-30 |
| BR0211207A (pt) | 2004-07-13 |
| CN100369916C (zh) | 2008-02-20 |
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