DK1549652T3 - Kondenserede azolpyrimidinderivater - Google Patents

Kondenserede azolpyrimidinderivater

Info

Publication number: DK1549652T3
Authority: DK; Denmark
Prior art keywords: pyrimidine derivatives; condensed azole; condensed; azole pyrimidine; derivatives
Prior art date: 2002-09-30

Application number

DK03788908T

Other languages

English (en)

Inventor

Toshiki Murata

Kinji Fuchikami

Hideki Tsujishita

Naoki Omori

Issei Kato

Mami Miura

Klaus Urbahns

Florian Gantner

Kevin Bacon

Mitsuyuki Shimada

Original Assignee

Bayer Healthcare Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-09-30

Filing date

2003-09-18

Publication date

2009-02-23

2003-09-18 Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag

2009-02-23 Application granted granted Critical

2009-02-23 Publication of DK1549652T3 publication Critical patent/DK1549652T3/da

Links

DDWJFSYHYPDQEL-UHFFFAOYSA-N pyrimidine;1h-pyrrole Chemical class C=1C=CNC=1.C1=CN=CN=C1 DDWJFSYHYPDQEL-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/14—Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Cardiology (AREA)
Immunology (AREA)
Heart & Thoracic Surgery (AREA)
Pulmonology (AREA)
Diabetes (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Endocrinology (AREA)
Hospice & Palliative Care (AREA)
Urology & Nephrology (AREA)
Rheumatology (AREA)
Emergency Medicine (AREA)
Psychiatry (AREA)
Hematology (AREA)
Obesity (AREA)
Pain & Pain Management (AREA)
Vascular Medicine (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Otolaryngology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

DK03788908T 2002-09-30 2003-09-18 Kondenserede azolpyrimidinderivater DK1549652T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP02021861		2002-09-30
PCT/EP2003/010377 WO2004029055A1 (en)	2002-09-30	2003-09-18	Fused azole-pyrimidine derivatives

Publications (1)

Publication Number	Publication Date
DK1549652T3 true DK1549652T3 (da)	2009-02-23

Family

ID=32039115

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
DK03788908T DK1549652T3 (da)	2002-09-30	2003-09-18	Kondenserede azolpyrimidinderivater
DK08075839.4T DK2042504T3 (da)	2002-09-30	2003-09-18	Kondenseret azole-pyrimidin-derivat

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
DK08075839.4T DK2042504T3 (da)	2002-09-30	2003-09-18	Kondenseret azole-pyrimidin-derivat

Country Status (32)

Country	Link
US (2)	US7511041B2 (da)
EP (2)	EP1549652B1 (da)
JP (1)	JP4790266B2 (da)
KR (1)	KR101059652B1 (da)
CN (1)	CN100384846C (da)
AR (2)	AR041426A1 (da)
AT (2)	ATE511510T1 (da)
AU (1)	AU2003293310B2 (da)
BR (1)	BRPI0314830B8 (da)
CA (1)	CA2499134C (da)
CY (2)	CY1109790T1 (da)
DE (1)	DE60324296D1 (da)
DK (2)	DK1549652T3 (da)
EC (2)	ECSP055768A (da)
ES (2)	ES2367141T3 (da)
HR (2)	HRP20131159B1 (da)
IL (1)	IL166855A (da)
MA (1)	MA27483A1 (da)
MX (1)	MXPA05001808A (da)
MY (1)	MY140756A (da)
NO (1)	NO331457B1 (da)
NZ (1)	NZ539062A (da)
PE (1)	PE20050089A1 (da)
PL (1)	PL226562B1 (da)
PT (2)	PT1549652E (da)
RU (1)	RU2326881C9 (da)
SI (2)	SI2042504T1 (da)
TW (1)	TWI327570B (da)
UA (1)	UA82205C2 (da)
UY (1)	UY28001A1 (da)
WO (1)	WO2004029055A1 (da)
ZA (1)	ZA200503306B (da)

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Also Published As

Publication number	Publication date
JP2006508063A (ja)	2006-03-09
TWI327570B (en)	2010-07-21
PL226562B1 (pl)	2017-08-31
PE20050089A1 (es)	2005-04-20
CA2499134A1 (en)	2004-04-08
US8129386B2 (en)	2012-03-06
KR101059652B1 (ko)	2011-08-25
ES2367141T3 (es)	2011-10-28
BRPI0314830B8 (pt)	2021-05-25
CY1112174T1 (el)	2015-12-09
NO331457B1 (no)	2012-01-09
MY140756A (en)	2010-01-15
HRP20131159B1 (hr)	2019-11-01
BRPI0314830B1 (pt)	2018-03-27
ECSP11005768A (es)	2011-03-31
WO2004029055A1 (en)	2004-04-08
SI2042504T1 (sl)	2011-10-28
HRP20050375B1 (hr)	2014-03-14
MA27483A1 (fr)	2005-08-01
ATE511510T1 (de)	2011-06-15
DK2042504T3 (da)	2011-09-19
EP1549652B1 (en)	2008-10-22
BR0314830A (pt)	2005-08-16
UA82205C2 (en)	2008-03-25
US20060128732A1 (en)	2006-06-15
TW200413379A (en)	2004-08-01
CA2499134C (en)	2011-12-20
CN100384846C (zh)	2008-04-30
EP2042504B1 (en)	2011-06-01
HK1084393A1 (zh)	2006-07-28
PT2042504E (pt)	2011-09-07
HRP20050375A2 (en)	2006-05-31
AU2003293310B2 (en)	2010-04-01
US20090270388A1 (en)	2009-10-29
ZA200503306B (en)	2006-07-26
ES2312843T3 (es)	2009-03-01
RU2326881C2 (ru)	2008-06-20
EP1549652A1 (en)	2005-07-06
RU2005113165A (ru)	2005-10-10
US7511041B2 (en)	2009-03-31
SI1549652T1 (sl)	2009-04-30
PT1549652E (pt)	2008-12-15
RU2326881C9 (ru)	2009-04-10
ECSP055768A (es)	2005-08-11
ATE411996T1 (de)	2008-11-15
AR072458A2 (es)	2010-09-01
CY1109790T1 (el)	2014-09-10
KR20050067404A (ko)	2005-07-01
UY28001A1 (es)	2004-04-30
AU2003293310A1 (en)	2004-04-19
JP4790266B2 (ja)	2011-10-12
EP2042504A1 (en)	2009-04-01
CN1688582A (zh)	2005-10-26
DE60324296D1 (de)	2008-12-04
PL375935A1 (en)	2005-12-12
HRP20131159A2 (hr)	2014-05-23
NZ539062A (en)	2007-05-31
NO20052076L (no)	2005-04-27
AR041426A1 (es)	2005-05-18
IL166855A (en)	2014-05-28
MXPA05001808A (es)	2005-08-16

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ATE411996T1 (de)	2008-11-15	Kondensierte azolpyrimidinderivate
HUS1500055I1 (hu)	2016-03-29	HIV-gátló pirimidinszármazékok
DK1487805T3 (da)	2012-10-15	Pyrimidinderivater
EP1546115A4 (en)	2010-08-04	Substituted pyrimidines
ATE517888T1 (de)	2011-08-15	Indolylmaleimid-derivate
ATE478870T1 (de)	2010-09-15	Spiroindolinpiperidinderivate
ATE460418T1 (de)	2010-03-15	Heterocyclocarboxamidderivate
DE60330372D1 (de)	2010-01-14	Indol-3-schwefelderivate
ATE467631T1 (de)	2010-05-15	Chinuclidinamidderivate
ATE438644T1 (de)	2009-08-15	Chinazolinderivate
IS7720A (is)	2005-03-01	Píperidín-N-oxíð-afleiður
DK2248807T3 (da)	2013-08-26	N-Phenyl-2-pyrimidinaminderivater
ATE370120T1 (de)	2007-09-15	Substituierte 2-pyridin-cyclohexan-1,4- diaminderivate
ATE425147T1 (de)	2009-03-15	Imidazolderivate
IS7287A (is)	2004-05-26	Pýrimídín efnasambönd
DE60307512D1 (de)	2006-09-21	3h-chinazoline -4-on derivaten
ATE366242T1 (de)	2007-07-15	5-substituierte chinazolinonderivate
ATE423771T1 (de)	2009-03-15	Tetrahydrochinolinderivate
DE60228135D1 (de)	2008-09-18	Eifen
EP1570847A4 (en)	2008-10-08	PHOSPHODIESTERASE 10A HEMMER
IS7833A (is)	2005-05-02	Efnasambönd með sameinaða heteróhringi
ATE427945T1 (de)	2009-04-15	Imidazolderivate
DE50306277D1 (de)	2007-02-22	4-alkyl-/4-alkenyl-/4-alkinylmethyl/-1-arylcyclohexylamin-derivate
DK1603910T3 (da)	2009-11-23	Substituerede 2-(diazabicykloalkyl)-pyrimidon-derivater
IS7906A (is)	2005-06-22	Afleiður própargýl-tríflúorómetoxý-amínó-benzóþíazóls