DK1989196T3 - Piperidinoylpyrrolidiner som melanocortin-type 4-receptoragonister - Google Patents

Piperidinoylpyrrolidiner som melanocortin-type 4-receptoragonister

Info

Publication number
DK1989196T3
DK1989196T3 DK07705650.5T DK07705650T DK1989196T3 DK 1989196 T3 DK1989196 T3 DK 1989196T3 DK 07705650 T DK07705650 T DK 07705650T DK 1989196 T3 DK1989196 T3 DK 1989196T3
Authority
DK
Denmark
Prior art keywords
piperidinoylpyrrolidines
receptor agonists
melanocortin type
melanocortin
type
Prior art date
Application number
DK07705650.5T
Other languages
English (en)
Inventor
Mark David Andrews
Alan Daniel Brown
Mark Ian Lansdell
Nicholas William Summerhill
Original Assignee
Pfizer Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Ltd filed Critical Pfizer Ltd
Application granted granted Critical
Publication of DK1989196T3 publication Critical patent/DK1989196T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK07705650.5T 2006-02-23 2007-02-19 Piperidinoylpyrrolidiner som melanocortin-type 4-receptoragonister DK1989196T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US77629506P 2006-02-23 2006-02-23
US88784007P 2007-02-02 2007-02-02
PCT/IB2007/000456 WO2007096763A2 (en) 2006-02-23 2007-02-19 Melanocortin type 4 receptor agonist piperidinoylpyrrolidines

Publications (1)

Publication Number Publication Date
DK1989196T3 true DK1989196T3 (da) 2013-04-15

Family

ID=38169450

Family Applications (1)

Application Number Title Priority Date Filing Date
DK07705650.5T DK1989196T3 (da) 2006-02-23 2007-02-19 Piperidinoylpyrrolidiner som melanocortin-type 4-receptoragonister

Country Status (21)

Country Link
US (1) US8138188B2 (da)
EP (1) EP1989196B1 (da)
KR (1) KR101036981B1 (da)
AP (1) AP2008004602A0 (da)
AU (1) AU2007219236B2 (da)
BR (1) BRPI0708264A2 (da)
CA (1) CA2642922C (da)
CR (1) CR10219A (da)
DK (1) DK1989196T3 (da)
EA (1) EA200801738A1 (da)
EC (1) ECSP088688A (da)
ES (1) ES2402581T3 (da)
IL (1) IL193279A (da)
MA (1) MA30228B1 (da)
ME (1) MEP6808A (da)
MX (1) MX2008010899A (da)
NO (1) NO20083480L (da)
RS (1) RS20080371A (da)
SG (1) SG185849A1 (da)
TN (1) TNSN08337A1 (da)
WO (1) WO2007096763A2 (da)

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US8828994B2 (en) 2011-03-08 2014-09-09 Sanofi Di- and tri-substituted oxathiazine derivatives, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof
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EP2683699B1 (de) 2011-03-08 2015-06-24 Sanofi Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
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US20210393621A1 (en) 2018-10-26 2021-12-23 The Research Foundation For The State University Of New York Combination serotonin specific reuptake inhibitor and serotonin 1a receptor partial agonist for reducing l-dopa-induced dyskinesia
JP7288554B1 (ja) 2020-06-09 2023-06-07 ファイザー・インク メラノコルチン４受容体アンタゴニストとしてのスピロ化合物およびそれらの使用
JP2024544021A (ja) 2021-12-06 2024-11-26 ファイザー・インク メラノコルチン４受容体アンタゴニストおよびそれらの使用
US20250333414A1 (en) 2024-04-30 2025-10-30 Boehringer Ingelheim International Gmbh Hetaryl substituted indazoles and benzimidazoles as sting antagonists and the use thereof as medicament
WO2025228900A1 (en) 2024-04-30 2025-11-06 Boehringer Ingelheim International Gmbh Arylamide substituted indazoles and the use thereof as medicament
US20250333398A1 (en) 2024-04-30 2025-10-30 Boehringer Ingelheim International Gmbh Monoaryl and hetaryl substituted indazoles and benzimidazoles as sting antagonists and the use thereof as medicament
WO2025228902A1 (en) 2024-04-30 2025-11-06 Boehringer Ingelheim International Gmbh Heterocyclic acids as sting antagonists and the use thereof as medicament
WO2025228889A1 (en) 2024-04-30 2025-11-06 Boehringer Ingelheim International Gmbh Monoarylic heterocyclic compounds as sting antagonists and the use thereof as medicament
WO2025228899A1 (en) 2024-04-30 2025-11-06 Boehringer Ingelheim International Gmbh Further heterocyclic compounds as sting antagonists and the use thereof as medicament
US12605394B2 (en) 2024-07-25 2026-04-21 Visionary Assets, Llc Compositions containing cannabinoid nanoparticles

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Also Published As

Publication number Publication date
AU2007219236A1 (en) 2007-08-30
MA30228B1 (fr) 2009-02-02
AP2008004602A0 (en) 2008-10-31
US20090036459A1 (en) 2009-02-05
EA200801738A1 (ru) 2008-12-30
AU2007219236B2 (en) 2012-06-21
CR10219A (es) 2008-09-23
EP1989196B1 (en) 2013-02-13
IL193279A0 (en) 2009-02-11
KR101036981B1 (ko) 2011-05-25
CA2642922C (en) 2011-08-02
MEP6808A (xx) 2010-02-10
US8138188B2 (en) 2012-03-20
BRPI0708264A2 (pt) 2011-05-24
MX2008010899A (es) 2008-11-27
RS20080371A (sr) 2009-07-15
IL193279A (en) 2012-12-31
EP1989196A2 (en) 2008-11-12
TNSN08337A1 (fr) 2009-12-29
KR20080095918A (ko) 2008-10-29
ES2402581T3 (es) 2013-05-06
HK1126489A1 (en) 2009-09-04
WO2007096763A3 (en) 2007-10-18
ECSP088688A (es) 2008-10-31
NO20083480L (no) 2008-09-10
SG185849A1 (en) 2012-12-28
WO2007096763A2 (en) 2007-08-30
CA2642922A1 (en) 2007-08-30

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