DK2336125T3 - Thiazolopyridin-2-yloxy-phenyl- og thioazolopyrazin-2-yloxy-phenyl-aminer som modulatorer af leukotrien-A4-hydrolase - Google Patents

Thiazolopyridin-2-yloxy-phenyl- og thioazolopyrazin-2-yloxy-phenyl-aminer som modulatorer af leukotrien-A4-hydrolase

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Publication number
DK2336125T3
DK2336125T3 DK11159236.6T DK11159236T DK2336125T3 DK 2336125 T3 DK2336125 T3 DK 2336125T3 DK 11159236 T DK11159236 T DK 11159236T DK 2336125 T3 DK2336125 T3 DK 2336125T3
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Prior art keywords
yloxy
thioazolopyrazin
thiazolopyridin
phenylamines
leukotriene
Prior art date
Application number
DK11159236.6T
Other languages
English (en)
Inventor
Alejandro Santillan
Kia Sepassi
Genesis M Bacani
Diego Broggini
Eugene Y Cheung
Christa C Chrovian
Xiaohu Deng
Anne M Fourine
Laurent Gomez
Cheryl A Grice
Aaron M Kearney
Adrienne M Landry-Bayle
Alice Lee-Dutra
Jimmy T Liang
Susanne Lochner
Neelakandha S Mani
Kathleen C Sappy
Virginia M Tanis
Alvah T Wickboldt
John J M Wiener
Hartmut Zinser
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
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Publication of DK2336125T3 publication Critical patent/DK2336125T3/da

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    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
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    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof

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  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Urology & Nephrology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
DK11159236.6T 2008-04-11 2009-04-09 Thiazolopyridin-2-yloxy-phenyl- og thioazolopyrazin-2-yloxy-phenyl-aminer som modulatorer af leukotrien-A4-hydrolase DK2336125T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US4434908P 2008-04-11 2008-04-11
US14912909P 2009-02-02 2009-02-02
EP09729596.8A EP2268646B9 (en) 2008-04-11 2009-04-09 Thiazolopyridin-2-yloxy-phenyl and thiazolopyrazin-2-yloxy-phenyl amines as modulators of leukotriene a4 hydrolase

Publications (1)

Publication Number Publication Date
DK2336125T3 true DK2336125T3 (da) 2013-04-08

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DK11159236.6T DK2336125T3 (da) 2008-04-11 2009-04-09 Thiazolopyridin-2-yloxy-phenyl- og thioazolopyrazin-2-yloxy-phenyl-aminer som modulatorer af leukotrien-A4-hydrolase
DK09729596.8T DK2268646T3 (da) 2008-04-11 2009-04-09 Thiazolopyridin-2-yloxy-phenyl og thiazolopyrazin-2-yloxy-phenyl-aminer som modulatorer af leukotrien-a4-hydrolase

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US (3) US7939527B2 (da)
EP (2) EP2268646B9 (da)
JP (2) JP5530423B2 (da)
KR (1) KR101228378B1 (da)
CN (1) CN102056933B (da)
AR (1) AR072353A1 (da)
AU (1) AU2009234140B2 (da)
BR (1) BRPI0911336A2 (da)
CA (1) CA2721099C (da)
CL (1) CL2009000877A1 (da)
CO (1) CO6260069A2 (da)
CY (1) CY1114628T1 (da)
DK (2) DK2336125T3 (da)
EA (1) EA018802B1 (da)
EC (1) ECSP10010558A (da)
ES (2) ES2400875T3 (da)
HN (1) HN2010002074A (da)
HR (2) HRP20131192T1 (da)
IL (2) IL208480A (da)
JO (1) JO2911B1 (da)
MX (1) MX2010011154A (da)
MY (1) MY157597A (da)
NI (1) NI201000168A (da)
NZ (2) NZ599853A (da)
PE (1) PE20091779A1 (da)
PH (1) PH12013500094B1 (da)
PL (2) PL2268646T3 (da)
PT (2) PT2336125E (da)
RS (2) RS52712B (da)
SI (2) SI2268646T1 (da)
SV (1) SV2010003694A (da)
TW (2) TWI461196B (da)
UY (1) UY31760A (da)
WO (1) WO2009126806A2 (da)
ZA (1) ZA201008054B (da)

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