DK3210991T3 - Krystallinsk form af levoisovalerylspiramycin ii og præparater, fremstillingsfremgangsmåder og anvendelser deraf - Google Patents

Krystallinsk form af levoisovalerylspiramycin ii og præparater, fremstillingsfremgangsmåder og anvendelser deraf Download PDF

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Publication number
DK3210991T3
DK3210991T3 DK17166118T DK17166118T DK3210991T3 DK 3210991 T3 DK3210991 T3 DK 3210991T3 DK 17166118 T DK17166118 T DK 17166118T DK 17166118 T DK17166118 T DK 17166118T DK 3210991 T3 DK3210991 T3 DK 3210991T3
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Prior art keywords
piramycine
levoisovaleryl
preparations
procedure
applications
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DK17166118T
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English (en)
Inventor
Yang Jiang
Xiaofeng Zhao
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Shenyang Fuyang Pharmaceutical Tech Co Ltd
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12NMICROORGANISMS OR ENZYMES; COMPOSITIONS THEREOF; PROPAGATING, PRESERVING, OR MAINTAINING MICROORGANISMS; MUTATION OR GENETIC ENGINEERING; CULTURE MEDIA
    • C12N9/00Enzymes; Proenzymes; Compositions thereof; Processes for preparing, activating, inhibiting, separating or purifying enzymes
    • C12N9/10Transferases (2.)
    • C12N9/1025Acyltransferases (2.3)
    • C12N9/1029Acyltransferases (2.3) transferring groups other than amino-acyl groups (2.3.1)
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P19/00Preparation of compounds containing saccharide radicals
    • C12P19/44Preparation of O-glycosides, e.g. glucosides
    • C12P19/60Preparation of O-glycosides, e.g. glucosides having an oxygen of the saccharide radical directly bound to a non-saccharide heterocyclic ring or a condensed ring system containing a non-saccharide heterocyclic ring, e.g. coumermycin, novobiocin
    • C12P19/62Preparation of O-glycosides, e.g. glucosides having an oxygen of the saccharide radical directly bound to a non-saccharide heterocyclic ring or a condensed ring system containing a non-saccharide heterocyclic ring, e.g. coumermycin, novobiocin the hetero ring having eight or more ring members and only oxygen as ring hetero atoms, e.g. erythromycin, spiramycin, nystatin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins

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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biotechnology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Microbiology (AREA)
  • General Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Public Health (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Saccharide Compounds (AREA)
DK17166118T 2010-05-25 2011-05-25 Krystallinsk form af levoisovalerylspiramycin ii og præparater, fremstillingsfremgangsmåder og anvendelser deraf DK3210991T3 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CN201010182108 2010-05-25
CN201010182109 2010-05-25
CN201010182111 2010-05-25
EP11786085.8A EP2578595B1 (en) 2010-05-25 2011-05-25 Crystalline levoisovalerylspiramycin i

Publications (1)

Publication Number Publication Date
DK3210991T3 true DK3210991T3 (da) 2019-11-11

Family

ID=45003321

Family Applications (3)

Application Number Title Priority Date Filing Date
DK17166118T DK3210991T3 (da) 2010-05-25 2011-05-25 Krystallinsk form af levoisovalerylspiramycin ii og præparater, fremstillingsfremgangsmåder og anvendelser deraf
DK11786085.8T DK2578595T3 (da) 2010-05-25 2011-05-25 Krystallinsk levoisovalerylspiramycin i
DK17166117.6T DK3210990T3 (da) 2010-05-25 2011-05-25 Levoisovalerylspiramycin iii og præparater, fremstillingsfremgangsmåder og anvendelser deraf

Family Applications After (2)

Application Number Title Priority Date Filing Date
DK11786085.8T DK2578595T3 (da) 2010-05-25 2011-05-25 Krystallinsk levoisovalerylspiramycin i
DK17166117.6T DK3210990T3 (da) 2010-05-25 2011-05-25 Levoisovalerylspiramycin iii og præparater, fremstillingsfremgangsmåder og anvendelser deraf

Country Status (16)

Country Link
US (1) US8778896B2 (da)
EP (3) EP2578595B1 (da)
JP (1) JP5945868B2 (da)
KR (2) KR101706518B1 (da)
BR (1) BR112012029913B1 (da)
CA (3) CA2915236C (da)
DK (3) DK3210991T3 (da)
ES (3) ES2754614T3 (da)
MX (1) MX340626B (da)
MY (1) MY164231A (da)
PH (1) PH12012502323A1 (da)
PL (3) PL3210990T3 (da)
PT (1) PT3210990T (da)
RU (3) RU2647237C1 (da)
WO (1) WO2011147313A1 (da)
ZA (3) ZA201209738B (da)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2800019C (en) * 2010-05-25 2015-05-26 Shenyang Tonglian Group Co., Ltd. Levocarrimycin, pharmaceutical compositions, preparation methods and uses thereof
CN105497053B (zh) * 2015-12-31 2018-02-13 沈阳福洋医药科技有限公司 可利霉素在抗结核分枝杆菌感染中的应用
RU2766176C2 (ru) * 2017-07-04 2022-02-08 Шенянг Фуянг Фармасьютекал Технолоджи Ко., Лтд. Применение изовалерил-спирамицина i, ii и/или iii при изготовлении препарата для лечения и/или профилактики опухоли и получения лекарственного препарата
CN110051845A (zh) * 2018-01-19 2019-07-26 沈阳福洋医药科技有限公司 一种mTOR抑制剂、药物组合物及其应用
MX2020007627A (es) * 2018-01-19 2020-11-24 Shenyang Fuyang Pharmaceutical Tech Co Ltd Uso de la carrimicina o de sus ingredientes activos.
KR20200144568A (ko) * 2018-04-17 2020-12-29 상하이 통리엔 파마슈티컬 컴퍼니 리미티드 통증 및/또는 발열을 예방 및/또는 치료하는 의약품, 조합 산물 및 그 응용
CN110384710B (zh) * 2018-04-17 2023-01-10 沈阳福洋医药科技有限公司 一种用于预防和/或治疗疼痛的药物、组合产品及其应用
KR20220008895A (ko) * 2019-05-16 2022-01-21 쉔양 푸양 파마슈티컬 테크놀로지 컴퍼니 리미티드 섬유증을 예방, 완화 및/또는 치료하는 약물, 복합 제품 및 이의 응용
CN112239483B (zh) * 2019-07-18 2023-10-27 沈阳福洋医药科技有限公司 一种化合物及药物组合物
US11351185B2 (en) 2020-03-11 2022-06-07 Asclea Corporation Use of isovalerylspiramycins as anti-cancer agents to inhibit metastasis

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5334788A (en) * 1976-09-11 1978-03-31 Sanraku Inc Antibiotics spiramycin derivatives
CN1058295C (zh) 1997-06-03 2000-11-08 中国医学科学院医药生物技术研究所 一种利用基因工程技术制造生技霉素的方法
CN1169947C (zh) * 2002-11-19 2004-10-06 中国医学科学院医药生物技术研究所 必特螺旋霉素的基因工程菌株螺旋霉素链霉菌wsj-195
CN1237976C (zh) 2003-12-23 2006-01-25 沈阳同联集团有限公司 必特螺旋霉素及其在抗感染性疾病中的应用
RU2007108544A (ru) * 2004-08-12 2008-09-20 Глаксосмитклайн Истраживацки Центар Загреб Д.О.О.(Hr) Применение клеточно-специфических конъюгатов для лечения воспалительных заболеваний желудочно-кишечного тракта
CN101054553A (zh) * 2007-04-09 2007-10-17 中国医学科学院医药生物技术研究所 异戊酰螺旋霉素i基因工程菌株的构建
CN101649325B (zh) * 2009-07-03 2011-09-07 中国医学科学院医药生物技术研究所 一种提高基因工程异戊酰螺旋霉素主组分含量的基因串连技术
CN101785779B (zh) 2010-03-09 2014-03-05 沈阳同联集团有限公司 异戊酰螺旋霉素ii的分离制备
CN101785778A (zh) * 2010-03-09 2010-07-28 沈阳同联集团有限公司 异戊酰螺旋霉素i的分离制备及其应用
CN101773510B (zh) * 2010-03-09 2013-06-05 沈阳同联集团有限公司 异戊酰螺旋霉素iii的分离制备
CA2800019C (en) * 2010-05-25 2015-05-26 Shenyang Tonglian Group Co., Ltd. Levocarrimycin, pharmaceutical compositions, preparation methods and uses thereof

Also Published As

Publication number Publication date
CA2800021A1 (en) 2011-12-01
CA2915222A1 (en) 2011-12-01
EP2578595A1 (en) 2013-04-10
EP3210990A1 (en) 2017-08-30
KR20130041829A (ko) 2013-04-25
CA2915236A1 (en) 2011-12-01
BR112012029913A8 (pt) 2018-01-09
PH12012502323A1 (en) 2023-03-10
RU2012156420A (ru) 2014-06-27
DK3210990T3 (da) 2020-03-23
DK2578595T3 (da) 2017-07-10
ES2781425T3 (es) 2020-09-02
CA2915236C (en) 2019-03-12
PL2578595T3 (pl) 2017-10-31
US20130065848A1 (en) 2013-03-14
PL3210991T3 (pl) 2020-03-31
RU2593498C2 (ru) 2016-08-10
EP3210991A1 (en) 2017-08-30
ZA201406382B (en) 2015-12-23
EP2578595B1 (en) 2017-04-19
US8778896B2 (en) 2014-07-15
KR20160017124A (ko) 2016-02-15
MY164231A (en) 2017-11-30
RU2647236C1 (ru) 2018-03-14
ES2754614T3 (es) 2020-04-20
MX2012013470A (es) 2013-03-18
EP3210990B1 (en) 2020-01-01
BR112012029913A2 (pt) 2017-11-28
CA2915222C (en) 2019-03-12
EP3210991B1 (en) 2019-08-07
JP2013528166A (ja) 2013-07-08
CA2800021C (en) 2016-03-22
MX340626B (es) 2016-07-18
ES2633723T3 (es) 2017-09-25
PL3210990T3 (pl) 2020-10-05
PT3210990T (pt) 2020-04-01
EP2578595A4 (en) 2013-11-06
RU2647237C1 (ru) 2018-03-14
BR112012029913B1 (pt) 2021-02-02
WO2011147313A1 (zh) 2011-12-01
ZA201209738B (en) 2015-04-29
KR101706518B1 (ko) 2017-02-14
JP5945868B2 (ja) 2016-07-13
ZA201406381B (en) 2016-08-31

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