DK3500253T3 - Kombination af inverse histamin-3-receptoragonister med acetylcholinesterasehæmmere - Google Patents
Kombination af inverse histamin-3-receptoragonister med acetylcholinesterasehæmmere Download PDFInfo
- Publication number
- DK3500253T3 DK3500253T3 DK17768234.1T DK17768234T DK3500253T3 DK 3500253 T3 DK3500253 T3 DK 3500253T3 DK 17768234 T DK17768234 T DK 17768234T DK 3500253 T3 DK3500253 T3 DK 3500253T3
- Authority
- DK
- Denmark
- Prior art keywords
- histamin
- inverse
- combination
- receptor agonists
- acetylcholine esterase
- Prior art date
Links
- 229940100578 Acetylcholinesterase inhibitor Drugs 0.000 title 1
- 238000003874 inverse correlation nuclear magnetic resonance spectroscopy Methods 0.000 title 1
- 239000000018 receptor agonist Substances 0.000 title 1
- 229940044601 receptor agonist Drugs 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/27—Esters, e.g. nitroglycerine, selenocyanates of carbamic or thiocarbamic acids, meprobamate, carbachol, neostigmine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Engineering & Computer Science (AREA)
- Neurology (AREA)
- Emergency Medicine (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN201641028166 | 2016-08-18 | ||
| PCT/IB2017/054938 WO2018033847A1 (en) | 2016-08-18 | 2017-08-14 | Combination of histamine-3 receptor inverse agonists with acetylcholinesterase inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK3500253T3 true DK3500253T3 (da) | 2020-08-17 |
Family
ID=59887325
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK17768234.1T DK3500253T3 (da) | 2016-08-18 | 2017-08-14 | Kombination af inverse histamin-3-receptoragonister med acetylcholinesterasehæmmere |
Country Status (28)
| Country | Link |
|---|---|
| US (1) | US10603323B2 (da) |
| EP (1) | EP3500253B1 (da) |
| JP (1) | JP6734470B2 (da) |
| KR (1) | KR102039585B1 (da) |
| CN (1) | CN109640975B (da) |
| AU (1) | AU2017313427B2 (da) |
| CA (1) | CA3033039C (da) |
| CY (1) | CY1123238T1 (da) |
| DK (1) | DK3500253T3 (da) |
| EA (1) | EA032957B1 (da) |
| ES (1) | ES2810983T3 (da) |
| HR (1) | HRP20201262T1 (da) |
| HU (1) | HUE052003T2 (da) |
| IL (1) | IL264406B (da) |
| LT (1) | LT3500253T (da) |
| MA (1) | MA45990B1 (da) |
| MD (1) | MD3500253T2 (da) |
| ME (1) | ME03812B (da) |
| MX (1) | MX374114B (da) |
| NZ (1) | NZ750150A (da) |
| PL (1) | PL3500253T3 (da) |
| PT (1) | PT3500253T (da) |
| RS (1) | RS60669B1 (da) |
| SG (1) | SG11201900681SA (da) |
| SI (1) | SI3500253T1 (da) |
| SM (1) | SMT202000435T1 (da) |
| WO (1) | WO2018033847A1 (da) |
| ZA (1) | ZA201900467B (da) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EA202092979A1 (ru) * | 2018-05-31 | 2021-03-12 | Сувен Лайф Сайенсиз Лимитед | Способ лечения обратным агонистом гистаминового рецептора 3 типа |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SG176735A1 (en) * | 2009-06-10 | 2012-01-30 | Sunovion Pharmaceuticals Inc | Histamine h3 inverse agonists and antagonists and methods of use thereof |
| US9079888B2 (en) * | 2011-02-23 | 2015-07-14 | Suven Life Sciences Limited | Compounds as histamine H3 receptor ligands |
| FR2974729B1 (fr) * | 2011-05-02 | 2013-04-19 | Servier Lab | Nouvelle association entre le 4-{3-[cis-hexahydrocyclopenta[c]pyrrol-2(1h)-yl]propoxy}benzamide et un inhibiteur de l'acetylcholinesterase et les compositions pharmaceutiques qui la contiennent |
| HUP1300139A2 (en) * | 2013-03-06 | 2014-09-29 | Richter Gedeon Nyrt | Phenoxypiperidine h3 antagonists |
| CN105764510A (zh) | 2013-09-09 | 2016-07-13 | 赛诺菲 | H3受体拮抗剂与胆碱酶抑制剂组合用于阿尔茨海默氏病治疗中的用途 |
-
2017
- 2017-08-14 LT LTEP17768234.1T patent/LT3500253T/lt unknown
- 2017-08-14 RS RS20200949A patent/RS60669B1/sr unknown
- 2017-08-14 SI SI201730360T patent/SI3500253T1/sl unknown
- 2017-08-14 MD MDE20190714T patent/MD3500253T2/ro unknown
- 2017-08-14 NZ NZ750150A patent/NZ750150A/en unknown
- 2017-08-14 PT PT177682341T patent/PT3500253T/pt unknown
- 2017-08-14 US US16/320,949 patent/US10603323B2/en active Active
- 2017-08-14 PL PL17768234T patent/PL3500253T3/pl unknown
- 2017-08-14 SM SM20200435T patent/SMT202000435T1/it unknown
- 2017-08-14 MA MA45990A patent/MA45990B1/fr unknown
- 2017-08-14 CN CN201780049311.9A patent/CN109640975B/zh active Active
- 2017-08-14 JP JP2019506640A patent/JP6734470B2/ja active Active
- 2017-08-14 SG SG11201900681SA patent/SG11201900681SA/en unknown
- 2017-08-14 EA EA201990480A patent/EA032957B1/ru unknown
- 2017-08-14 ME MEP-2020-167A patent/ME03812B/me unknown
- 2017-08-14 HR HRP20201262TT patent/HRP20201262T1/hr unknown
- 2017-08-14 ES ES17768234T patent/ES2810983T3/es active Active
- 2017-08-14 DK DK17768234.1T patent/DK3500253T3/da active
- 2017-08-14 MX MX2019001696A patent/MX374114B/es active IP Right Grant
- 2017-08-14 KR KR1020197007056A patent/KR102039585B1/ko active Active
- 2017-08-14 AU AU2017313427A patent/AU2017313427B2/en active Active
- 2017-08-14 WO PCT/IB2017/054938 patent/WO2018033847A1/en not_active Ceased
- 2017-08-14 CA CA3033039A patent/CA3033039C/en active Active
- 2017-08-14 EP EP17768234.1A patent/EP3500253B1/en active Active
- 2017-08-14 HU HUE17768234A patent/HUE052003T2/hu unknown
-
2019
- 2019-01-22 IL IL264406A patent/IL264406B/en active IP Right Grant
- 2019-01-23 ZA ZA2019/00467A patent/ZA201900467B/en unknown
-
2020
- 2020-08-05 CY CY20201100725T patent/CY1123238T1/el unknown
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DK3419625T3 (da) | Fremgangsmåder til anvendelse af fxr-agonister | |
| DK3419624T3 (da) | Fremgangsmåder til anvendelse af fxr-agonister | |
| DK3512850T3 (da) | Inhibitorer af menin-mll-interaktionen | |
| DK3468966T3 (da) | Inhibitorer af menin-mll-interaktionen | |
| EP3541932A4 (en) | INHIBITORS OF CRISPR-CAS9 | |
| DK3528817T3 (da) | Fremgangsmåder til behandling af leverforstyrrelser eller lipidforstyrrelser med en thr-beta-agonist | |
| DK3371171T3 (da) | Inhibitorer af RET | |
| DK3102576T3 (da) | Dihydropyrrolopyridininhibitorer af ror-gamma | |
| DK3220741T3 (da) | Sammensætning og kits til hæmning af patogen mikrobiel infektion og fremgangsmåder til anvendelse af samme | |
| DK3300500T3 (da) | Triazolagonister af apj-receptoren | |
| DK3164380T3 (da) | Hæmmere af lysinspecifik demethylase-1 | |
| DK3466432T3 (da) | Fremgangsmåder til behandling af pulmonale non-tuberkuløse mykobakterielle infektioner | |
| DK3436593T3 (da) | Fremgangsmåder til varmeinaktivering af adenovirus | |
| DK3307271T3 (da) | Fremgangsmåder til anvendelse af pyruvatkinase-aktivatorer | |
| DK3512857T3 (da) | Spiro-bicykliske inhibitorer af menin-mll-interaktion | |
| DK3551625T3 (da) | Heterocykliske inhibitorer af mct4 | |
| DK3455625T3 (da) | Fremgangsmåder til forudsigelse af anvendeligheden af neo-antigener til immunterapi | |
| EP3523315A4 (en) | INHIBITORS OF THE GLUCOCORTICOID RECEPTOR | |
| DK3204352T3 (da) | Hæmmere af lysin-gingipain | |
| EP3364189A4 (en) | IMMUNOCHROMATOGRAPHIC TEST PIECE | |
| DK3227325T3 (da) | Sammensætninger med selektive hæmmere af il-6-trans-signalering | |
| EP3394078A4 (en) | INHIBITORS OF THE GLUCOCORTICIDE RECEPTOR | |
| DK3198361T3 (da) | Hardwarestyrede effektdomæner med automatisk tænd-anmodning | |
| DK3529236T3 (da) | Krystalformer af eravacyclin | |
| EP3394079A4 (en) | INHIBITORS OF GLUCOCORTICOIDREZEPTORS |