DK357181A - R fremgangsmaade til fremstilling af heterocycliske forbindelse - Google Patents

R fremgangsmaade til fremstilling af heterocycliske forbindelse

Info

Publication number
DK357181A
DK357181A DK357181A DK357181A DK357181A DK 357181 A DK357181 A DK 357181A DK 357181 A DK357181 A DK 357181A DK 357181 A DK357181 A DK 357181A DK 357181 A DK357181 A DK 357181A
Authority
DK
Denmark
Prior art keywords
procedure
heterocyclic compound
preparing heterocyclic
preparing
compound
Prior art date
Application number
DK357181A
Other languages
English (en)
Other versions
DK157680B (da
DK157680C (da
Inventor
I H Coates
K Mills
C F Webb
M D Dowle
D E Bays
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of DK357181A publication Critical patent/DK357181A/da
Publication of DK157680B publication Critical patent/DK157680B/da
Application granted granted Critical
Publication of DK157680C publication Critical patent/DK157680C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C07D209/16—Tryptamines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK357181A 1980-08-12 1981-08-11 Analogifremgangsmaade til fremstilling af indolderivater DK157680C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8026288 1980-08-12
GB8026288 1980-08-12

Publications (3)

Publication Number Publication Date
DK357181A true DK357181A (da) 1982-02-13
DK157680B DK157680B (da) 1990-02-05
DK157680C DK157680C (da) 1990-07-09

Family

ID=10515412

Family Applications (1)

Application Number Title Priority Date Filing Date
DK357181A DK157680C (da) 1980-08-12 1981-08-11 Analogifremgangsmaade til fremstilling af indolderivater

Country Status (28)

Country Link
US (2) US4672067A (da)
JP (1) JPS5759864A (da)
AR (1) AR231533A1 (da)
AT (1) AT381304B (da)
AU (1) AU548270B2 (da)
BE (1) BE889930A (da)
CA (2) CA1169429A (da)
CH (1) CH651550A5 (da)
DE (1) DE3131748A1 (da)
DK (1) DK157680C (da)
ES (2) ES8300700A1 (da)
FI (1) FI812475L (da)
FR (1) FR2488605A1 (da)
GB (1) GB2081717B (da)
GR (1) GR74536B (da)
IE (1) IE51492B1 (da)
IL (1) IL63541A (da)
IT (1) IT1171451B (da)
LU (1) LU83546A1 (da)
MY (1) MY8600577A (da)
NL (1) NL8103768A (da)
NO (1) NO812722L (da)
NZ (1) NZ197997A (da)
PH (1) PH17428A (da)
PT (1) PT73503B (da)
SE (1) SE454881B (da)
ZA (1) ZA815539B (da)
ZW (1) ZW19381A1 (da)

Families Citing this family (41)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GR79215B (da) * 1982-06-07 1984-10-22 Glaxo Group Ltd
GB8332437D0 (en) * 1983-12-06 1984-01-11 Glaxo Group Ltd Chemical compounds
GB8332435D0 (en) * 1983-12-06 1984-01-11 Glaxo Group Ltd Chemical compounds
GB8332434D0 (en) * 1983-12-06 1984-01-11 Glaxo Group Ltd Production of chemical compounds
GB8419575D0 (en) * 1984-08-01 1984-09-05 Glaxo Group Ltd Chemical compounds
DE3678805D1 (de) * 1985-11-08 1991-05-23 Glaxo Group Ltd Indolderivate.
GB8530507D0 (en) * 1985-12-11 1986-01-22 Glaxo Group Plc Chemical compounds
GB8600397D0 (en) * 1986-01-08 1986-02-12 Glaxo Group Ltd Chemical compounds
GB8600398D0 (en) * 1986-01-08 1986-02-12 Glaxo Group Ltd Chemical compounds
US5270333A (en) * 1986-01-28 1993-12-14 Glaxo Group Limited Indole derivatives
GB8607824D0 (en) * 1986-03-27 1986-04-30 Glaxo Group Ltd Chemical compounds
DE3613623A1 (de) * 1986-04-23 1987-10-29 Bayer Ag N-dihydroindolylethyl-sulfonamide
GB8615599D0 (en) * 1986-06-26 1986-07-30 Glaxo Group Ltd Chemical compounds
US5225431A (en) * 1987-10-23 1993-07-06 Burroughs Wellcome Co. Therapeutic substituted indole compounds and compositions thereof
GB8819024D0 (en) * 1988-08-10 1988-09-14 Glaxo Group Ltd Chemical compounds
CA2042295A1 (fr) * 1990-05-15 1991-11-16 Jacques Chauveau Derives de mediateurs endogenes, leurs sels, procede de preparation, applications, et compositions les renfermant
SI9111010B (sl) * 1990-06-07 2005-02-28 Astrazeneca Ab 3,5-disubstituirani indolni derivati kot "5-HT1-podobni" receptorski agonisti
GB9022250D0 (en) * 1990-10-12 1990-11-28 Glaxo Group Ltd Medicaments
PL168919B1 (pl) * 1990-10-15 1996-05-31 Pfizer Sposób wytwarzania nowych pochodnych indolu PL PL PL PL
US5578612A (en) * 1990-10-15 1996-11-26 Pfizer Inc. Indole derivatives
US5559246A (en) * 1990-10-15 1996-09-24 Pfizer Inc. Indole derivatives
US5545644A (en) * 1990-10-15 1996-08-13 Pfizer Inc. Indole derivatives
US5607951A (en) * 1990-10-15 1997-03-04 Pfizer Inc Indole derivatives
US5559129A (en) * 1990-10-15 1996-09-24 Pfizer Inc Indole derivatives
SK278998B6 (sk) * 1991-02-01 1998-05-06 Merck Sharp & Dohme Limited Deriváty imidazolu, triazolu a tetrazolu, spôsob i
GB9103770D0 (en) * 1991-02-22 1991-04-10 Glaxo Group Ltd Chemical compounds
ES2033577B1 (es) * 1991-06-06 1995-01-16 Quimica Sint S A Con El 50 Procedimiento para la obtencion de la 2-carboxi-3-(2-(dimetilamino)etil)-n-metil-1h-indol-5-metanosulfonamida y sus esteres alquilicos inferiores.
ES2033578B1 (es) * 1991-06-06 1995-01-16 Quimica Sint S A Con El 50 Procedimiento para la obtencion de 3-(2-(dimetilamino)etil)-n-metil-1h-indol-5-metanosulfonamida.
GB9209882D0 (en) * 1992-05-07 1992-06-24 Glaxo Lab Sa Compositions
GB9211277D0 (en) 1992-05-28 1992-07-15 Glaxo Group Inc Pharmaceutical compositions
IL106445A (en) * 1992-07-30 1998-01-04 Merck Sharp & Dohme History of 1,2,4-Trans-Triazole 4-Transform, Preparation and Pharmaceutical Preparations Containing Them
CN1129933A (zh) * 1993-08-31 1996-08-28 辉瑞大药厂 5-芳基吲哚衍生物
US5468768A (en) * 1994-01-06 1995-11-21 Bristol-Myers Squibb Company Antimigraine derivatives of indolylcycloalkanylamines
GB9417310D0 (en) * 1994-08-27 1994-10-19 Pfizer Ltd Therapeutic agents
JPH11513666A (ja) * 1995-10-10 1999-11-24 イーライ・リリー・アンド・カンパニー Ｎ−［２−置換−３−（２−アミノエチル）−１ｈ−インドール−５−イル］−アミド：新規５−ｈｔ▲下１ｆ▼作動剤
US7189753B1 (en) 1997-11-06 2007-03-13 Cady Roger K Preemptive prophylaxis of migraine
US5994352A (en) * 1998-11-13 1999-11-30 Pfizer Inc. 5-arylindole derivatives
WO2002079153A1 (en) * 2001-03-28 2002-10-10 Biocatalytics, Inc. Method for producing tryptamine derivatives
KR20030016291A (ko) * 2001-04-13 2003-02-26 오르가노 가부시키가이샤 이온교환체
JP5833804B2 (ja) * 2005-04-13 2015-12-16 ニューラクソン，インコーポレーテッド Ｎｏｓ阻害活性を有する置換インドール化合物
KR20180052566A (ko) 2015-07-02 2018-05-18 키비타스 테라퓨틱스, 인코포레이티드. 폐 전달용 트립탄 분말

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2870162A (en) * 1954-04-28 1959-01-20 Upjohn Co Production of certain tryptamines and compounds produced in the process
BE632051A (fr) * 1963-05-08 1963-11-18 Sandoz Sa Nouveaux dérivés de l'indole et leur préparation.
CH442303A (de) * 1964-06-26 1967-08-31 Sandoz Ag Verfahren zur Herstellung von neuen Indol-Derivaten
US3472870A (en) * 1966-08-29 1969-10-14 Mead Johnson & Co Sulfonamidotryptamines
FR2334358A1 (fr) * 1975-12-12 1977-07-08 Sogeras Nouveaux medicaments derives de l'indole
US4180509A (en) * 1977-07-01 1979-12-25 Merrell Toraude Et Compagnie α-Ethynyl tryptophanes
ZA795239B (en) * 1978-10-12 1980-11-26 Glaxo Group Ltd Heterocyclic compounds

Also Published As

Publication number Publication date
IT1171451B (it) 1987-06-10
ES8404327A1 (es) 1984-04-16
IL63541A (en) 1985-08-30
ZA815539B (en) 1983-03-30
JPS5759864A (en) 1982-04-10
SE8104782L (sv) 1982-02-13
GR74536B (da) 1984-06-29
NZ197997A (en) 1985-08-16
US4636521A (en) 1987-01-13
JPH0148895B2 (da) 1989-10-20
CA1169077A (en) 1984-06-12
AU548270B2 (en) 1985-12-05
ZW19381A1 (en) 1983-03-09
CH651550A5 (fr) 1985-09-30
GB2081717A (en) 1982-02-24
SE454881B (sv) 1988-06-06
AU7399681A (en) 1982-02-18
FR2488605B1 (da) 1984-11-16
IT8149086A0 (it) 1981-08-11
NO812722L (no) 1982-02-15
ES513935A0 (es) 1984-04-16
DK157680B (da) 1990-02-05
CA1169429A (en) 1984-06-19
US4672067A (en) 1987-06-09
FI812475A7 (fi) 1982-02-13
FI812475L (fi) 1982-02-13
AT381304B (de) 1986-09-25
PT73503A (en) 1981-09-01
AR231533A1 (es) 1984-12-28
NL8103768A (nl) 1982-03-01
PH17428A (en) 1984-08-20
GB2081717B (en) 1983-09-28
DK157680C (da) 1990-07-09
DE3131748A1 (de) 1982-04-01
IT8149086A1 (it) 1983-02-11
IE811831L (en) 1982-02-12
DE3131748C2 (da) 1992-04-23
MY8600577A (en) 1986-12-31
ES504695A0 (es) 1982-11-01
ES8300700A1 (es) 1982-11-01
LU83546A1 (fr) 1983-06-08
ATA352881A (de) 1986-02-15
IE51492B1 (en) 1987-01-07
PT73503B (en) 1983-09-14
FR2488605A1 (fr) 1982-02-19
BE889930A (fr) 1982-02-11

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