DK615086A - 5,6-dialkoxy-4-imino-2(1h)quinazolinderivater - Google Patents

5,6-dialkoxy-4-imino-2(1h)quinazolinderivater

Info

Publication number
DK615086A
DK615086A DK615086A DK615086A DK615086A DK 615086 A DK615086 A DK 615086A DK 615086 A DK615086 A DK 615086A DK 615086 A DK615086 A DK 615086A DK 615086 A DK615086 A DK 615086A
Authority
DK
Denmark
Prior art keywords
dialkoxy
imino
quinazoline derivatives
quinazoline
derivatives
Prior art date
Application number
DK615086A
Other languages
English (en)
Other versions
DK615086D0 (da
Inventor
Victor T Bandurco
Stanley C Bell
Robert Falotico
Charles F Schwender
Alfonso J Tobia
Original Assignee
Ortho Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ortho Pharma Corp filed Critical Ortho Pharma Corp
Publication of DK615086D0 publication Critical patent/DK615086D0/da
Publication of DK615086A publication Critical patent/DK615086A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK615086A 1985-12-20 1986-12-18 5,6-dialkoxy-4-imino-2(1h)quinazolinderivater DK615086A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/811,238 US4668787A (en) 1985-12-20 1985-12-20 5,6-dialkoxy-4-imino-2(1H)quinazolinone derivatives

Publications (2)

Publication Number Publication Date
DK615086D0 DK615086D0 (da) 1986-12-18
DK615086A true DK615086A (da) 1987-06-21

Family

ID=25205981

Family Applications (1)

Application Number Title Priority Date Filing Date
DK615086A DK615086A (da) 1985-12-20 1986-12-18 5,6-dialkoxy-4-imino-2(1h)quinazolinderivater

Country Status (6)

Country Link
US (1) US4668787A (da)
EP (1) EP0227451A3 (da)
JP (1) JPS62187461A (da)
AU (1) AU6675386A (da)
DK (1) DK615086A (da)
ZA (1) ZA869588B (da)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2077252C (en) * 1992-08-31 2001-04-10 Khashayar Karimian Methods of making ureas and guanidines, and intermediates therefor
AU2002322720B2 (en) 2001-07-25 2008-11-13 Raptor Pharmaceutical Inc. Compositions and methods for modulating blood-brain barrier transport
CA2789262C (en) 2005-04-28 2016-10-04 Proteus Digital Health, Inc. Pharma-informatics system
EP2063905B1 (en) 2006-09-18 2014-07-30 Raptor Pharmaceutical Inc Treatment of liver disorders by administration of receptor-associated protein (rap)-conjugates
TR201908314T4 (tr) 2009-02-20 2019-06-21 2 Bbb Medicines B V Glutatyon bazlı ilaç dağıtım sistemi.
KR101909711B1 (ko) 2009-05-06 2018-12-19 라보라토리 스킨 케어, 인크. 활성제-칼슘 포스페이트 입자 복합체를 포함하는 피부 전달 조성물 및 이들을 이용하는 방법
US20120077778A1 (en) 2010-09-29 2012-03-29 Andrea Bourdelais Ladder-Frame Polyether Conjugates
EP3555071A4 (en) * 2016-12-13 2020-06-10 Beta Therapeutics Pty. Ltd. HEPARANASE INHIBITORS AND THEIR USE
US11787783B2 (en) 2016-12-13 2023-10-17 Beta Therapeutics Pty Ltd Heparanase inhibitors and use thereof
WO2018107200A1 (en) 2016-12-13 2018-06-21 Beta Therapeutics Pty Ltd Heparanase inhibitors and use thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3516816A (en) * 1967-05-19 1970-06-23 United States Borax Chem Herbicidal compositions and methods utilizing alkyleneiminourea compounds
CH507917A (de) * 1969-03-12 1971-05-31 Agripat Sa Verfahren zur Herstellung neuer 2-Ureido-benzamide und deren Verwendung zur Unkrautbekämpfung
US4146717A (en) * 1972-04-07 1979-03-27 Sumitomo Chemical Company, Limited Nitroquinazolinone compounds having antiviral properties
US4287341A (en) * 1979-11-01 1981-09-01 Pfizer Inc. Alkoxy-substituted-6-chloro-quinazoline-2,4-diones
US4634769A (en) * 1984-09-25 1987-01-06 Ortho Pharmaceutical Corporation Process for the preparation of 8-halo-5,6-dialkoxyquinazoline-2,4-diones and their salts

Also Published As

Publication number Publication date
EP0227451A2 (en) 1987-07-01
EP0227451A3 (en) 1988-01-13
DK615086D0 (da) 1986-12-18
JPS62187461A (ja) 1987-08-15
AU6675386A (en) 1987-06-25
US4668787A (en) 1987-05-26
ZA869588B (en) 1988-07-27

Similar Documents

Publication Publication Date Title
DK81091D0 (da) Imidazooe4,5-baaguinolin-2-thionderivater
FI860505L (fi) Dihydro- och tetrahydrokinolinderivat.
ATE49403T1 (de) N-aralkylpiperidinmethanol-derivate.
DE3675232D1 (de) Pyridinderivate.
DE3669876D1 (de) 3,4-dihydrobenzopyranderivate.
DE3678805D1 (de) Indolderivate.
DK615186A (da) Substituerede 5,6-dialkoxyquinazolinderivater
DE3684549D1 (de) Carboxamidderivate.
DE3664910D1 (de) Substituted 2,3,4,9-tetrahydro-1h-carbazole-1-acetic acid derivatives
FI861698L (fi) 2-pyrrolidonderivat.
DK615086A (da) 5,6-dialkoxy-4-imino-2(1h)quinazolinderivater
DE3680067D1 (de) Fluorphenylcyclohexanderivate.
ATE41655T1 (de) Phenaethanolaminderivate.
FI853859A7 (fi) Amidijohdannaisia.
DE3588103D1 (de) 5-Fluorouracil-Derivate
GB8605551D0 (en) 4-amino-6,7-dimethoxy-2-piperazin-1-ylquinazoline derivatives
FI865230L (fi) Antikonvulsiva -tiobutyrolaktonderivat.
FI872997A7 (fi) Amidijohdannaisia.
DE3664770D1 (de) Cardiotonic quinazoline derivatives
FI861951A7 (fi) 1,3-oxatianderivat.
DK212786D0 (da) 1,3-dioxanethere
DK601386A (da) 5-phenyl-1,4,5,6-tetrahydropyrimidinderivater
IT1190646B (it) 2,4-dicloro-5-nitro-tiazolo
FI860587A7 (fi) Imidazodiazepinderivat.
NO864162D0 (no) Bicyklo-substituerte fenylacetonitrilderivater.

Legal Events

Date Code Title Description
AHB Application shelved due to non-payment