DK615086A - 5,6-dialkoxy-4-imino-2(1h)quinazolinderivater - Google Patents

5,6-dialkoxy-4-imino-2(1h)quinazolinderivater

Info

Publication number
DK615086A
DK615086A DK615086A DK615086A DK615086A DK 615086 A DK615086 A DK 615086A DK 615086 A DK615086 A DK 615086A DK 615086 A DK615086 A DK 615086A DK 615086 A DK615086 A DK 615086A
Authority
DK
Denmark
Prior art keywords
dialkoxy
imino
quinazoline derivatives
quinazoline
derivatives
Prior art date
Application number
DK615086A
Other languages
English (en)
Other versions
DK615086D0 (da
Inventor
Victor T Bandurco
Stanley C Bell
Robert Falotico
Charles F Schwender
Alfonso J Tobia
Original Assignee
Ortho Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ortho Pharma Corp filed Critical Ortho Pharma Corp
Publication of DK615086D0 publication Critical patent/DK615086D0/da
Publication of DK615086A publication Critical patent/DK615086A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/95—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK615086A 1985-12-20 1986-12-18 5,6-dialkoxy-4-imino-2(1h)quinazolinderivater DK615086A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/811,238 US4668787A (en) 1985-12-20 1985-12-20 5,6-dialkoxy-4-imino-2(1H)quinazolinone derivatives

Publications (2)

Publication Number Publication Date
DK615086D0 DK615086D0 (da) 1986-12-18
DK615086A true DK615086A (da) 1987-06-21

Family

ID=25205981

Family Applications (1)

Application Number Title Priority Date Filing Date
DK615086A DK615086A (da) 1985-12-20 1986-12-18 5,6-dialkoxy-4-imino-2(1h)quinazolinderivater

Country Status (6)

Country Link
US (1) US4668787A (da)
EP (1) EP0227451A3 (da)
JP (1) JPS62187461A (da)
AU (1) AU6675386A (da)
DK (1) DK615086A (da)
ZA (1) ZA869588B (da)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2077252C (en) * 1992-08-31 2001-04-10 Khashayar Karimian Methods of making ureas and guanidines, and intermediates therefor
AU2002322720B2 (en) 2001-07-25 2008-11-13 Raptor Pharmaceutical Inc. Compositions and methods for modulating blood-brain barrier transport
CN102379684B (zh) 2005-04-28 2014-11-19 普罗透斯数字保健公司 药物信息系统
KR20090071598A (ko) 2006-09-18 2009-07-01 랩터 파마슈티컬 인코포레이티드 수용체 결합 단백질(rap)-접합체 투여에 의한 간 질환의 치료
EP2398500B1 (en) 2009-02-20 2019-03-13 2-BBB Medicines B.V. Glutathione-based drug delivery system
ES2942923T3 (es) 2009-05-06 2023-06-07 Laboratory Skin Care Inc Composiciones de administración dérmica que comprenden complejos de agente activo-partículas de fosfato de calcio y métodos de uso de las mismas
US20120077778A1 (en) 2010-09-29 2012-03-29 Andrea Bourdelais Ladder-Frame Polyether Conjugates
BR112019012045A2 (pt) 2016-12-13 2020-08-18 Beta Therapeutics Pty Ltd inibidores de heparanase e uso dos mesmos
US11787783B2 (en) 2016-12-13 2023-10-17 Beta Therapeutics Pty Ltd Heparanase inhibitors and use thereof
AU2017376818A1 (en) * 2016-12-13 2019-07-11 Beta Therapeutics Pty Ltd Heparanase inhibitors and use thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3516816A (en) * 1967-05-19 1970-06-23 United States Borax Chem Herbicidal compositions and methods utilizing alkyleneiminourea compounds
CH507917A (de) * 1969-03-12 1971-05-31 Agripat Sa Verfahren zur Herstellung neuer 2-Ureido-benzamide und deren Verwendung zur Unkrautbekämpfung
US4146717A (en) * 1972-04-07 1979-03-27 Sumitomo Chemical Company, Limited Nitroquinazolinone compounds having antiviral properties
US4287341A (en) * 1979-11-01 1981-09-01 Pfizer Inc. Alkoxy-substituted-6-chloro-quinazoline-2,4-diones
US4634769A (en) * 1984-09-25 1987-01-06 Ortho Pharmaceutical Corporation Process for the preparation of 8-halo-5,6-dialkoxyquinazoline-2,4-diones and their salts

Also Published As

Publication number Publication date
AU6675386A (en) 1987-06-25
ZA869588B (en) 1988-07-27
US4668787A (en) 1987-05-26
JPS62187461A (ja) 1987-08-15
EP0227451A3 (en) 1988-01-13
DK615086D0 (da) 1986-12-18
EP0227451A2 (en) 1987-07-01

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Legal Events

Date Code Title Description
AHB Application shelved due to non-payment