DK92486A - 1-0xa-1-dethiacephalosporinforbindelse - Google Patents
1-0xa-1-dethiacephalosporinforbindelse Download PDFInfo
- Publication number
- DK92486A DK92486A DK92486A DK92486A DK92486A DK 92486 A DK92486 A DK 92486A DK 92486 A DK92486 A DK 92486A DK 92486 A DK92486 A DK 92486A DK 92486 A DK92486 A DK 92486A
- Authority
- DK
- Denmark
- Prior art keywords
- sup
- group
- formula
- ethyl
- ring
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title 1
- -1 4-ethyl-2,3-dioxopiperazine-1-yl group Chemical group 0.000 abstract 2
- QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 abstract 2
- 125000002373 5 membered heterocyclic group Chemical group 0.000 abstract 1
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical compound [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 abstract 1
- 239000003242 anti bacterial agent Substances 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 125000002057 carboxymethyl group Chemical group [H]OC(=O)C([H])([H])[*] 0.000 abstract 1
- 229940124587 cephalosporin Drugs 0.000 abstract 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 abstract 1
- 125000005842 heteroatom Chemical group 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 abstract 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D505/00—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D505/02—Preparation
- C07D505/06—Preparation from compounds already containing the ring or condensed ring systems, e.g. by dehydrogenation of the ring, by introduction, elimination or modification of substituents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D505/00—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D505/00—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D505/10—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D505/12—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 substituted in position 7
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Cephalosporin Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/705,799 US4645769A (en) | 1985-03-01 | 1985-03-01 | 1-oxa-1-dethia-cephalosporin compounds and antibacterial agent comprising the same |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK92486D0 DK92486D0 (da) | 1986-02-28 |
| DK92486A true DK92486A (da) | 1986-09-02 |
Family
ID=24835001
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK92486A DK92486A (da) | 1985-03-01 | 1986-02-28 | 1-0xa-1-dethiacephalosporinforbindelse |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US4645769A (da) |
| EP (1) | EP0193858B1 (da) |
| JP (1) | JPH0633280B2 (da) |
| KR (1) | KR900003500B1 (da) |
| AT (1) | ATE69819T1 (da) |
| CA (1) | CA1268177A (da) |
| DE (1) | DE3682599D1 (da) |
| DK (1) | DK92486A (da) |
| ES (2) | ES8705450A1 (da) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK123488A (da) * | 1987-03-09 | 1988-09-10 | Otsuka Pharma Co Ltd | 2-oxa-isocephemforbindelser, praeparater indeholdende dem, og fremgangsmaader til fremstilling af dem |
| DK582788A (da) * | 1987-10-22 | 1989-04-23 | Otsuka Pharma Co Ltd | 2-oxa-isocephemforbindelser, midler der indeholder dem og fremgangsmaader til fremstilling af dem |
| US5525599A (en) * | 1993-07-21 | 1996-06-11 | Eli Lilly And Company | 7-substituted-amino-3-substituted-3-cephem-4-carboxylic acids |
| JP6377570B2 (ja) * | 2014-04-28 | 2018-08-22 | グラクソスミスクライン、インテレクチュアル、プロパティー、ディベロップメント、リミテッドＧｌａｘｏｓｍｉｔｈｋｌｉｎｅ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ Ｄｅｖｅｌｏｐｍｅｎｔ Ｌｉｍｉｔｅｄ | ２−置換セフェム化合物を含有する医薬組成物 |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4226866A (en) * | 1972-11-06 | 1980-10-07 | Merck & Co., Inc. | Novel antibiotic analogues of cephalosporins |
| JPS5331690A (en) * | 1976-09-01 | 1978-03-25 | Shionogi & Co Ltd | Oxadithiacephalosporins |
| GB1557552A (en) * | 1977-02-15 | 1979-12-12 | Shionogi & Co | 1 oxadethiacepham compounds |
| DE2714880A1 (de) * | 1977-04-02 | 1978-10-26 | Hoechst Ag | Cephemderivate und verfahren zu ihrer herstellung |
| ES486026A1 (es) * | 1978-11-17 | 1980-09-01 | Glaxo Group Ltd | Un procedimiento para la preparacion de antibioticos de ce- falosporina |
| FR2474504A1 (fr) * | 1979-05-23 | 1981-07-31 | Rhone Poulenc Ind | Nouvelles thiovinyl-3 cephalosporines, leur preparation et les medicaments qui les contiennent |
| CA1145744A (fr) * | 1979-05-23 | 1983-05-03 | Daniel Farge | Thiovinyl-3 cephalosporines, leur preparation et les compositions qui les contiennent |
| DE3137038A1 (de) * | 1981-09-17 | 1983-03-24 | Bayer Ag, 5090 Leverkusen | Ss-lactam antibiotika, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel |
| JPS5849382A (ja) * | 1981-09-18 | 1983-03-23 | Kyowa Hakko Kogyo Co Ltd | β−ラクタム化合物 |
| JPS5874680A (ja) * | 1981-10-01 | 1983-05-06 | Kyowa Hakko Kogyo Co Ltd | β−ラクタム化合物 |
| FR2516515A1 (fr) * | 1981-11-16 | 1983-05-20 | Sanofi Sa | Nouveaux derives de pyridinium thiomethyl cephalosporines, procede pour leur preparation et compositions pharmaceutiques les contenant |
| US4534898A (en) * | 1982-07-23 | 1985-08-13 | Merck & Co., Inc. | 1-Oxa-1-dethia-cephalosporin derivatives |
-
1985
- 1985-03-01 US US06/705,799 patent/US4645769A/en not_active Expired - Fee Related
-
1986
- 1986-02-19 CA CA000502142A patent/CA1268177A/en not_active Expired - Lifetime
- 1986-02-26 AT AT86102483T patent/ATE69819T1/de not_active IP Right Cessation
- 1986-02-26 DE DE8686102483T patent/DE3682599D1/de not_active Expired - Lifetime
- 1986-02-26 EP EP86102483A patent/EP0193858B1/en not_active Expired - Lifetime
- 1986-02-27 ES ES552486A patent/ES8705450A1/es not_active Expired
- 1986-02-28 KR KR1019860001452A patent/KR900003500B1/ko not_active Expired
- 1986-02-28 DK DK92486A patent/DK92486A/da not_active Application Discontinuation
- 1986-02-28 JP JP61041854A patent/JPH0633280B2/ja not_active Expired - Lifetime
- 1986-10-30 ES ES557155A patent/ES8707726A1/es not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| JPS61251685A (ja) | 1986-11-08 |
| KR860007264A (ko) | 1986-10-10 |
| ES552486A0 (es) | 1987-05-01 |
| US4645769A (en) | 1987-02-24 |
| DK92486D0 (da) | 1986-02-28 |
| ES8707726A1 (es) | 1987-08-16 |
| DE3682599D1 (de) | 1992-01-09 |
| ES8705450A1 (es) | 1987-05-01 |
| CA1268177A (en) | 1990-04-24 |
| ES557155A0 (es) | 1987-08-16 |
| ATE69819T1 (de) | 1991-12-15 |
| EP0193858A1 (en) | 1986-09-10 |
| KR900003500B1 (ko) | 1990-05-21 |
| EP0193858B1 (en) | 1991-11-27 |
| JPH0633280B2 (ja) | 1994-05-02 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHB | Application shelved due to non-payment |