ECSP066797A - Procedimientos para la preparacion de halogenuros de aril- y heteroarilalquilsulfonilo - Google Patents

Procedimientos para la preparacion de halogenuros de aril- y heteroarilalquilsulfonilo

Info

Publication number
ECSP066797A
ECSP066797A EC2006006797A ECSP066797A ECSP066797A EC SP066797 A ECSP066797 A EC SP066797A EC 2006006797 A EC2006006797 A EC 2006006797A EC SP066797 A ECSP066797 A EC SP066797A EC SP066797 A ECSP066797 A EC SP066797A
Authority
EC
Ecuador
Prior art keywords
preparation
heteroarilalquilsulfonilo
halogenures
aril
procedures
Prior art date
Application number
EC2006006797A
Other languages
English (en)
Inventor
Mousumi Ghosh
Mahmut Levent
Ronald S Mickalak
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of ECSP066797A publication Critical patent/ECSP066797A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/32—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of salts of sulfonic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/02—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof
    • C07C303/22—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof from sulfonic acids, by reactions not involving the formation of sulfo or halosulfonyl groups; from sulfonic halides by reactions not involving the formation of halosulfonyl groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

La presente invención provee procedimientos de preparación de halogenuros de arilalquilsulfonilo y halogenuros de heteroarilalquilsulfonilo de la fórmula Ar-R-SO2-X, que son útiles como intermediarios en la preparación de agentes farmacéuticos.
EC2006006797A 2004-02-25 2006-08-25 Procedimientos para la preparacion de halogenuros de aril- y heteroarilalquilsulfonilo ECSP066797A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US54760004P 2004-02-25 2004-02-25

Publications (1)

Publication Number Publication Date
ECSP066797A true ECSP066797A (es) 2006-11-16

Family

ID=34910921

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2006006797A ECSP066797A (es) 2004-02-25 2006-08-25 Procedimientos para la preparacion de halogenuros de aril- y heteroarilalquilsulfonilo

Country Status (24)

Country Link
US (1) US7321061B2 (es)
EP (1) EP1718605B1 (es)
JP (1) JP2007523954A (es)
CN (1) CN1922136A (es)
AR (1) AR048239A1 (es)
AT (1) ATE433955T1 (es)
AU (1) AU2005217619A1 (es)
BR (1) BRPI0507979A (es)
CA (1) CA2555247A1 (es)
CO (1) CO5720992A2 (es)
CR (1) CR8550A (es)
DE (1) DE602005014942D1 (es)
EC (1) ECSP066797A (es)
ES (1) ES2326746T3 (es)
GT (1) GT200500031A (es)
IL (1) IL177432A0 (es)
NO (1) NO20063611L (es)
PA (1) PA8624401A1 (es)
PE (1) PE20060018A1 (es)
RU (1) RU2006129650A (es)
SV (1) SV2005002015A (es)
TW (1) TW200602298A (es)
WO (1) WO2005082843A1 (es)
ZA (1) ZA200607097B (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1907355B1 (en) 2005-07-21 2015-08-05 Ziarco Pharma Ltd Process for the synthesis of sulfonyl halides and sulfonamides from sulfonic acid salts
BRPI0718042A2 (pt) * 2006-10-31 2013-11-12 Wyeth Corp Formulações semissólidas de inibidores de enzima fosfolipase
WO2008055136A2 (en) * 2006-10-31 2008-05-08 Wyeth Liquid formulations of phospholipase enzyme inhibitors
CN102471245A (zh) * 2009-07-30 2012-05-23 陶氏环球技术有限责任公司 用于烃的磺基氯化作用的改善方法
CN102241613B (zh) * 2011-05-09 2013-06-05 南通维立科化工有限公司 甲基磺酸钠制备高纯度甲基磺酰氯的生产方法
CN102295587A (zh) * 2011-05-26 2011-12-28 安徽丰乐农化有限责任公司 对甲基苯磺酰氯的制备新工艺
CN102976988B (zh) * 2012-12-24 2014-06-18 三门峡奥科化工有限公司 2-萘硫酚的合成工艺
KR102122111B1 (ko) * 2017-09-01 2020-06-11 주식회사 엘지화학 대체 용매의 선정 방법
CN111718286A (zh) * 2020-07-23 2020-09-29 邓博天 一种带供电基团芳烃磺酰氯的工业化生产方法

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE150313C (es) *
DE48722C (de) * Dr. E. FISCHER in Stuttgart, Schlofsstrafse 29 Verfahren zur Darstellung von O-Nitrobenzaldehyd aus O-Nitrobenzylchlorid
US2199568A (en) * 1938-06-11 1940-05-07 Gen Aniline & Film Corp Manufacture of 1-methyl-4-chloro-5-hydroxynaphthalene-11-sulphonic acid
US2507408A (en) 1948-03-05 1950-05-09 Rhone Poulenc Sa 1-alkylsulfonyl-4-alkyl piperazines
US2888486A (en) 1953-11-20 1959-05-26 Du Pont Process for producing aromatic sulfonyl halides
DE2545644A1 (de) * 1975-10-11 1977-04-14 Bayer Ag Verfahren zur herstellung von sulfonsaeuren
US4150049A (en) * 1975-11-05 1979-04-17 The Government Of The United States Esters of aromatic sulfonic acids
JPS5277030A (en) * 1975-12-23 1977-06-29 Toyo Pharma Kk Production of novel benzyl sulphonic acid derivatives
JPH09295962A (ja) * 1996-03-08 1997-11-18 Nagase & Co Ltd ２，２−ジ置換−エタンスルホン酸誘導体およびその塩
DE19838516A1 (de) * 1998-08-25 2000-03-09 Degussa Verfahren zur Herstellung von Sulfonylhalogeniden
JP2000072739A (ja) * 1998-09-01 2000-03-07 Tanabe Seiyaku Co Ltd スルホン酸類またはその塩の製法
PT1451154E (pt) 2001-12-03 2008-04-21 Wyeth Corp Inibidores de fosfolipase a2 citossólica
EP1907355B1 (en) 2005-07-21 2015-08-05 Ziarco Pharma Ltd Process for the synthesis of sulfonyl halides and sulfonamides from sulfonic acid salts

Also Published As

Publication number Publication date
IL177432A0 (en) 2006-12-10
US7321061B2 (en) 2008-01-22
PE20060018A1 (es) 2006-02-20
GT200500031A (es) 2005-09-30
EP1718605B1 (en) 2009-06-17
EP1718605A1 (en) 2006-11-08
AR048239A1 (es) 2006-04-12
CR8550A (es) 2007-02-05
CO5720992A2 (es) 2007-01-31
ES2326746T3 (es) 2009-10-19
CN1922136A (zh) 2007-02-28
BRPI0507979A (pt) 2007-07-24
DE602005014942D1 (de) 2009-07-30
NO20063611L (no) 2006-09-21
SV2005002015A (es) 2005-11-04
PA8624401A1 (es) 2006-08-03
JP2007523954A (ja) 2007-08-23
ZA200607097B (en) 2009-08-26
RU2006129650A (ru) 2008-03-27
TW200602298A (en) 2006-01-16
AU2005217619A1 (en) 2005-09-09
US20050187408A1 (en) 2005-08-25
CA2555247A1 (en) 2005-09-09
ATE433955T1 (de) 2009-07-15
WO2005082843A1 (en) 2005-09-09

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