CR8550A - Procedimientos para la preparacion de halogenuros de aryl- y- heteroarilalquilsulfonilo - Google Patents

Procedimientos para la preparacion de halogenuros de aryl- y- heteroarilalquilsulfonilo

Info

Publication number
CR8550A
CR8550A CR8550A CR8550A CR8550A CR 8550 A CR8550 A CR 8550A CR 8550 A CR8550 A CR 8550A CR 8550 A CR8550 A CR 8550A CR 8550 A CR8550 A CR 8550A
Authority
CR
Costa Rica
Prior art keywords
preparation
heteroarilalquilsulfonilo
halogenuros
aryl
procedures
Prior art date
Application number
CR8550A
Other languages
English (en)
Inventor
S Michalak Ronald
Ghosh Mousumi
Levent Mahmut
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of CR8550A publication Critical patent/CR8550A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/32Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of salts of sulfonic acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/02Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof
    • C07C303/22Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof from sulfonic acids, by reactions not involving the formation of sulfo or halosulfonyl groups; from sulfonic halides by reactions not involving the formation of halosulfonyl groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

La presente invencion provee procedimientos de preparacion de halogenuros de arilalquilsulfonilo y halogenuros de heteroarilalquilsulfonilo de la formula Ar-R-SO2-X, que son utiles como intermediarios en la preparacion de agentes farmaceuticos.
CR8550A 2004-02-25 2006-08-08 Procedimientos para la preparacion de halogenuros de aryl- y- heteroarilalquilsulfonilo CR8550A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US54760004P 2004-02-25 2004-02-25

Publications (1)

Publication Number Publication Date
CR8550A true CR8550A (es) 2007-02-05

Family

ID=34910921

Family Applications (1)

Application Number Title Priority Date Filing Date
CR8550A CR8550A (es) 2004-02-25 2006-08-08 Procedimientos para la preparacion de halogenuros de aryl- y- heteroarilalquilsulfonilo

Country Status (24)

Country Link
US (1) US7321061B2 (es)
EP (1) EP1718605B1 (es)
JP (1) JP2007523954A (es)
CN (1) CN1922136A (es)
AR (1) AR048239A1 (es)
AT (1) ATE433955T1 (es)
AU (1) AU2005217619A1 (es)
BR (1) BRPI0507979A (es)
CA (1) CA2555247A1 (es)
CO (1) CO5720992A2 (es)
CR (1) CR8550A (es)
DE (1) DE602005014942D1 (es)
EC (1) ECSP066797A (es)
ES (1) ES2326746T3 (es)
GT (1) GT200500031A (es)
IL (1) IL177432A0 (es)
NO (1) NO20063611L (es)
PA (1) PA8624401A1 (es)
PE (1) PE20060018A1 (es)
RU (1) RU2006129650A (es)
SV (1) SV2005002015A (es)
TW (1) TW200602298A (es)
WO (1) WO2005082843A1 (es)
ZA (1) ZA200607097B (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG163550A1 (en) * 2005-07-21 2010-08-30 Wyeth Corp Process for the synthesis of sulfonyl halides and sulfonamides from sulfonic acid salts
BRPI0718042A2 (pt) * 2006-10-31 2013-11-12 Wyeth Corp Formulações semissólidas de inibidores de enzima fosfolipase
CL2007003143A1 (es) * 2006-10-31 2008-01-25 Wyeth Corp Composicion farmaceutica que comprende un compuesto derivado de indol y un sistema portador que comprende 10-50% de un primer solubilizante, 5-50% de un segundo solubilizante, 10-30% de un primer diluyente y 1-15% de un segundo diluyente; proceso de prepracion; y forma de dosificacion.
US20120116121A1 (en) * 2009-07-30 2012-05-10 Dow Global Technologies Llc Process for the sulfochlorination of hydrocarbons
CN102241613B (zh) * 2011-05-09 2013-06-05 南通维立科化工有限公司 甲基磺酸钠制备高纯度甲基磺酰氯的生产方法
CN102295587A (zh) * 2011-05-26 2011-12-28 安徽丰乐农化有限责任公司 对甲基苯磺酰氯的制备新工艺
CN102976988B (zh) * 2012-12-24 2014-06-18 三门峡奥科化工有限公司 2-萘硫酚的合成工艺
KR102122111B1 (ko) * 2017-09-01 2020-06-11 주식회사 엘지화학 대체 용매의 선정 방법
CN111718286A (zh) * 2020-07-23 2020-09-29 邓博天 一种带供电基团芳烃磺酰氯的工业化生产方法

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE150313C (es)
DE48722C (de) Dr. E. FISCHER in Stuttgart, Schlofsstrafse 29 Verfahren zur Darstellung von O-Nitrobenzaldehyd aus O-Nitrobenzylchlorid
US2199568A (en) 1938-06-11 1940-05-07 Gen Aniline & Film Corp Manufacture of 1-methyl-4-chloro-5-hydroxynaphthalene-11-sulphonic acid
US2507408A (en) 1948-03-05 1950-05-09 Rhone Poulenc Sa 1-alkylsulfonyl-4-alkyl piperazines
US2888486A (en) 1953-11-20 1959-05-26 Du Pont Process for producing aromatic sulfonyl halides
DE2545644A1 (de) * 1975-10-11 1977-04-14 Bayer Ag Verfahren zur herstellung von sulfonsaeuren
US4150049A (en) * 1975-11-05 1979-04-17 The Government Of The United States Esters of aromatic sulfonic acids
JPS5277030A (en) * 1975-12-23 1977-06-29 Toyo Pharma Kk Production of novel benzyl sulphonic acid derivatives
JPH09295962A (ja) * 1996-03-08 1997-11-18 Nagase & Co Ltd 2,2−ジ置換−エタンスルホン酸誘導体およびその塩
DE19838516A1 (de) * 1998-08-25 2000-03-09 Degussa Verfahren zur Herstellung von Sulfonylhalogeniden
JP2000072739A (ja) * 1998-09-01 2000-03-07 Tanabe Seiyaku Co Ltd スルホン酸類またはその塩の製法
DK1451154T3 (da) 2001-12-03 2008-05-19 Wyeth Corp Inhibitorer af cytosolisk phospholipase A2
SG163550A1 (en) 2005-07-21 2010-08-30 Wyeth Corp Process for the synthesis of sulfonyl halides and sulfonamides from sulfonic acid salts

Also Published As

Publication number Publication date
AU2005217619A1 (en) 2005-09-09
BRPI0507979A (pt) 2007-07-24
IL177432A0 (en) 2006-12-10
CN1922136A (zh) 2007-02-28
TW200602298A (en) 2006-01-16
US20050187408A1 (en) 2005-08-25
JP2007523954A (ja) 2007-08-23
ATE433955T1 (de) 2009-07-15
CO5720992A2 (es) 2007-01-31
US7321061B2 (en) 2008-01-22
ES2326746T3 (es) 2009-10-19
ZA200607097B (en) 2009-08-26
EP1718605A1 (en) 2006-11-08
GT200500031A (es) 2005-09-30
AR048239A1 (es) 2006-04-12
PA8624401A1 (es) 2006-08-03
RU2006129650A (ru) 2008-03-27
WO2005082843A1 (en) 2005-09-09
PE20060018A1 (es) 2006-02-20
DE602005014942D1 (de) 2009-07-30
ECSP066797A (es) 2006-11-16
NO20063611L (no) 2006-09-21
SV2005002015A (es) 2005-11-04
EP1718605B1 (en) 2009-06-17
CA2555247A1 (en) 2005-09-09

Similar Documents

Publication Publication Date Title
CR9223A (es) 18-metil-19-nor-17-pregn-4-en-21, 17-carbolactonas,asi como preparaciones farmaceuticas que las contienen
CR8919A (es) Analogos de tetrapeptidos
SE0302811D0 (sv) Novel compounds
CR10072A (es) Derivados de pirimidinil-aril-urea que son inhibidores de fgf
CR8773A (es) Nuevo fluoroglicosido derivado de pirazoles, medicamentos contenidos en estos compuestos y sus usos
TW200716647A (en) Synthesis of (R)-N-methylnaltrexone
HN2008000311A (es) Formas cristalinas de 4-metil-n-[3-(4-metil-imidazol-1-il)-5-trifluorometil-fenil]-3-(4-piridin-3-il-pirimidin-2-ilamino)-benzamida
CR9786A (es) Compuestos de bencimidazol-tiofeno
NO20090376L (no) Fremgangsmate for fremstilling av (1R,2R)-3-(3-dimetylamino-1-etyl-2-metyl-propyl)-fenol
PA8660301A1 (es) Pirazolo piridinas sustituidas, composiciones que las contienen, procedimiento de fabricacion y utilizacion
CY1122416T1 (el) Φαρμακα τα οποια περιεχουν κρυσταλλικες τροποποιησεις (1r,2r)-3-(3-δimeθyλamino-1-αιθυλο-2-μεθυλο-προπυλο)-φαινολης
SE0401762D0 (sv) Novel compounds
UY33276A (es) Compuestos de amino-oxazinas y amino-dihidrotiazina como moduladores de beta-secretasa y métodos de uso
BRPI0607309A2 (pt) processos para a preparação de fenilpirazol uréias substituìdas
HN2003000080A (es) Indolil-urea derivados de tienopiridinas utiles como agentes antiangiogenicos y procedimientos para su uso
PA8667201A1 (es) Nuevos compuestos farmaceuticos
CR7195A (es) Nuevos derivados de oxazolidinonas como antibacterianos
UY29767A1 (es) Derivados de benzotiazolonas, procesos para su preparación, composiciones farmacéuticas que los contienen y aplicaciones
CR8550A (es) Procedimientos para la preparacion de halogenuros de aryl- y- heteroarilalquilsulfonilo
CL2007003223A1 (es) Compuestos derivados de piperidinil 4-arilsulfonamidas n-sustituidas, que actuan como moduladores de la proteina sfrp-1; proceso para preparar los compuestos; co mposicion farmaceutica que comprende a dichos copmpuestos y uso de los compuestos para preparar medicamentos para el tratamiento de enfermedades.
DOP2006000087A (es) Compuestos heteroaromaticos acilaminobiciclicos y sus usos
MX367327B (es) Formulaciones, sales y polimorfos de transnorsertralina y usos de los mismos.
SV2006002290A (es) Nonadepsipeptidos acilados ii ref. bhc041327-sv
UY28754A1 (es) Proceso quimico
UY29999A1 (es) "n-pirazinil-fenilsulfonamidas, procedimientos y compuestos intemedios utilizados en su preparacion, composiciones farmaceuticas que las contienen y aplicaciones"

Legal Events

Date Code Title Description
FA Abandonment or withdrawal (granting procedure)