ECSP088417A - Procedimientos para la preparacion de derivados de ciclopropilamida - Google Patents

Procedimientos para la preparacion de derivados de ciclopropilamida

Info

Publication number
ECSP088417A
ECSP088417A EC2008008417A ECSP088417A ECSP088417A EC SP088417 A ECSP088417 A EC SP088417A EC 2008008417 A EC2008008417 A EC 2008008417A EC SP088417 A ECSP088417 A EC SP088417A EC SP088417 A ECSP088417 A EC SP088417A
Authority
EC
Ecuador
Prior art keywords
preparation
derivatives
ciclopropilamide
procedures
cyclopropyl
Prior art date
Application number
EC2008008417A
Other languages
English (en)
Inventor
Sergio Cesco-Cancian
Neelakandha Mani
David C Palmer
Tong Xiao
Chennagiri R Pandit
Mayra B Reyes
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of ECSP088417A publication Critical patent/ECSP088417A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182—Radicals derived from carboxylic acids
    • C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invención se refiere a procedimientos novedosos para la preparación de derivados de ciclopropil-amida, útiles para el tratamiento de trastornos y condiciones mediados por el receptor de histamina.
EC2008008417A 2005-10-31 2008-04-30 Procedimientos para la preparacion de derivados de ciclopropilamida ECSP088417A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US73172505P 2005-10-31 2005-10-31

Publications (1)

Publication Number Publication Date
ECSP088417A true ECSP088417A (es) 2008-05-30

Family

ID=38001898

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2008008417A ECSP088417A (es) 2005-10-31 2008-04-30 Procedimientos para la preparacion de derivados de ciclopropilamida

Country Status (28)

Country Link
EP (1) EP1951699B1 (es)
JP (1) JP5185822B2 (es)
KR (1) KR20080067362A (es)
CN (2) CN101300242B (es)
AR (2) AR058171A1 (es)
AU (1) AU2006309124B2 (es)
BR (1) BRPI0618076A2 (es)
CA (2) CA2628187C (es)
CR (1) CR10036A (es)
DK (1) DK1951699T3 (es)
EA (2) EA201001872A1 (es)
EC (1) ECSP088417A (es)
ES (1) ES2395049T3 (es)
HR (1) HRP20121025T1 (es)
IL (2) IL190965A (es)
MX (1) MX367916B (es)
MY (2) MY151028A (es)
NO (1) NO340950B1 (es)
NZ (2) NZ592864A (es)
PL (1) PL1951699T3 (es)
PT (1) PT1951699E (es)
RS (1) RS52569B (es)
SG (1) SG166803A1 (es)
SI (1) SI1951699T1 (es)
TW (1) TWI377201B (es)
UA (1) UA93892C2 (es)
WO (1) WO2007053386A2 (es)
ZA (1) ZA200804730B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0324159D0 (en) 2003-10-15 2003-11-19 Glaxo Group Ltd Novel compounds
CN101835750B (zh) 2007-08-22 2013-07-17 阿斯利康(瑞典)有限公司 环丙基酰胺衍生物
US20090170869A1 (en) 2007-09-06 2009-07-02 Desmond John Best Piperazine derivative having affinity for the histamine h3 receptor
TW201039825A (en) 2009-02-20 2010-11-16 Astrazeneca Ab Cyclopropyl amide derivatives 983
US20110201623A1 (en) 2010-02-18 2011-08-18 Uczynski Michael A Crystalline Form Of A Cyclopropyl Benzamide Derivative
FR2962729B1 (fr) 2010-07-13 2012-09-21 Arkema France Molecules porteuses de groupes associatifs
US11491148B2 (en) * 2019-05-06 2022-11-08 Janssen Sciences Ireland Unlimited Company Amide derivatives useful in the treatment of HBV infection or HBV-induced diseases

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SK5202000A3 (en) * 2000-04-07 2001-12-03 Slovakofarma As Method for the preparation of (e)-n-(6,6-dimethyl-2-hepten-4- inyl)-n-methyl-1-naphthalenemethylamine (terbinaphin)
IL153414A0 (en) * 2000-07-05 2003-07-06 Basf Ag Method for the production of trioxime derivatives
US20040010746A1 (en) 2002-07-10 2004-01-15 Lucas L. Victor Forward error correction system for wireless communications
DE60330269D1 (de) * 2002-10-23 2010-01-07 Janssen Pharmaceutica Nv Piperazinyl- und diazapanylbenzamide und-benzothioamide
JP2007503440A (ja) * 2003-08-27 2007-02-22 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ アリールピペリジンアミド
PL1948607T3 (pl) * 2005-09-16 2010-09-30 Janssen Pharmaceutica Nv Cyklopropyloaminy jako modulatory receptora histaminowego H3

Also Published As

Publication number Publication date
EP1951699A2 (en) 2008-08-06
EA201001872A1 (ru) 2011-04-29
AR114493A2 (es) 2020-09-09
IL190965A (en) 2014-04-30
NO340950B1 (no) 2017-07-24
MY151028A (en) 2014-03-31
AR058171A1 (es) 2008-01-23
SG166803A1 (en) 2010-12-29
MX367916B (es) 2019-09-11
WO2007053386A3 (en) 2007-11-01
CA2628187A1 (en) 2007-05-10
CN102659718B (zh) 2015-11-25
HK1119676A1 (en) 2009-03-13
CA2628187C (en) 2015-01-27
EA014935B1 (ru) 2011-04-29
HRP20121025T1 (hr) 2013-01-31
CR10036A (es) 2009-02-23
BRPI0618076A2 (pt) 2011-08-16
JP5185822B2 (ja) 2013-04-17
MY174411A (en) 2020-04-16
NZ592864A (en) 2012-09-28
TW200736240A (en) 2007-10-01
ZA200804730B (en) 2009-10-28
PT1951699E (pt) 2012-12-26
CN101300242A (zh) 2008-11-05
EP1951699B1 (en) 2012-10-10
IL213474A (en) 2014-05-28
TWI377201B (en) 2012-11-21
IL190965A0 (en) 2008-12-29
EA200801240A1 (ru) 2008-08-29
AU2006309124A1 (en) 2007-05-10
NZ567359A (en) 2011-07-29
PL1951699T3 (pl) 2013-03-29
NO20082458L (no) 2008-07-18
CA2869539C (en) 2017-06-27
CN101300242B (zh) 2012-07-11
IL213474A0 (en) 2011-07-31
WO2007053386A2 (en) 2007-05-10
UA93892C2 (ru) 2011-03-25
SI1951699T1 (sl) 2013-01-31
ES2395049T3 (es) 2013-02-07
AU2006309124B2 (en) 2013-02-14
DK1951699T3 (da) 2013-01-14
RS52569B (sr) 2013-04-30
KR20080067362A (ko) 2008-07-18
CA2869539A1 (en) 2007-05-10
CN102659718A (zh) 2012-09-12
JP2009513701A (ja) 2009-04-02

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