ECSP077296A - Fenilaminotiazoles sustituidos y su uso - Google Patents

Fenilaminotiazoles sustituidos y su uso

Info

Publication number
ECSP077296A
ECSP077296A EC2007007296A ECSP077296A ECSP077296A EC SP077296 A ECSP077296 A EC SP077296A EC 2007007296 A EC2007007296 A EC 2007007296A EC SP077296 A ECSP077296 A EC SP077296A EC SP077296 A ECSP077296 A EC SP077296A
Authority
EC
Ecuador
Prior art keywords
phenylaminotiazols
substituted
treatment
diseases
prophylaxis
Prior art date
Application number
EC2007007296A
Other languages
English (en)
Inventor
Ulrich Rosentreter
Walter Huebsch
Nicole Diedrichs
Karl Heinz Schlemmer
Barbara Albrecht
Kerstin Henninger
Peter Nell
Dirk Brohm
Jens-Kerim Ergueden
Gunter Karig
Sabine Arndt
Andreas Knorr
Joachim Huetter
Original Assignee
Bayer Healthcare Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag
Publication of ECSP077296A publication Critical patent/ECSP077296A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

La presente solicitud se refiere a nuevos derivados de fenilaminotiazol, a procedimientos para su fabricación, a su uso para el tratamiento y/o la profilaxis de enfermedades, así como a su uso para la fabricación de medicamentos para el tratamiento y/o la profilaxis de enfermedades, preferiblemente para el tratamiento y/o la prevención de hipertensión y otras enfermedades cardiovasculares.
EC2007007296A 2004-09-03 2007-03-02 Fenilaminotiazoles sustituidos y su uso ECSP077296A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102004042607A DE102004042607A1 (de) 2004-09-03 2004-09-03 Substituierte Phenylaminothiazole und ihre Verwendung

Publications (1)

Publication Number Publication Date
ECSP077296A true ECSP077296A (es) 2007-04-26

Family

ID=35852458

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2007007296A ECSP077296A (es) 2004-09-03 2007-03-02 Fenilaminotiazoles sustituidos y su uso

Country Status (24)

Country Link
US (1) US8691850B2 (es)
EP (1) EP1812430B1 (es)
JP (1) JP4999691B2 (es)
KR (1) KR20070057235A (es)
CN (1) CN101056875A (es)
AR (1) AR050551A1 (es)
AT (1) ATE428710T1 (es)
AU (1) AU2005281941A1 (es)
BR (1) BRPI0514833A (es)
CA (1) CA2578596C (es)
DE (2) DE102004042607A1 (es)
EC (1) ECSP077296A (es)
ES (1) ES2324049T3 (es)
GT (1) GT200500238A (es)
IL (1) IL181670A0 (es)
MA (1) MA28869B1 (es)
MX (1) MX2007002470A (es)
NO (1) NO20071343L (es)
PE (1) PE20060589A1 (es)
SV (1) SV2006002218A (es)
TW (1) TW200621765A (es)
UY (1) UY29099A1 (es)
WO (1) WO2006027142A1 (es)
ZA (1) ZA200701820B (es)

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DE102006056739A1 (de) * 2006-12-01 2008-06-05 Bayer Healthcare Ag Substituierte 4-Amino-3,5-dicyano-2-thiopyridine und ihre Verwendung
DE102006056740A1 (de) 2006-12-01 2008-06-05 Bayer Healthcare Ag Cyclisch substituierte 3,5-Dicyano-2-thiopyridine und ihre Verwendung
DE102007035367A1 (de) 2007-07-27 2009-01-29 Bayer Healthcare Ag Substituierte Aryloxazole und ihre Verwendung
DE102007036076A1 (de) 2007-08-01 2009-02-05 Bayer Healthcare Aktiengesellschaft Dipeptoid-Produgs und ihre Verwendung
DE102007061763A1 (de) * 2007-12-20 2009-06-25 Bayer Healthcare Ag Substituierte azabicyclische Verbindungen und ihre Verwendung
DE102007061764A1 (de) * 2007-12-20 2009-06-25 Bayer Healthcare Ag Anellierte Cyanopyridine und ihre Verwendung
DE102008008838A1 (de) 2008-02-13 2009-08-20 Bayer Healthcare Ag Cycloalkoxy-substituierte 4-Phenyl-3,5-dicyanopyridine und ihre Verwendung
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US8791146B2 (en) * 2008-05-29 2014-07-29 Bayer Intellectual Property Gmbh 2-alkoxy-substituted dicyanopyridines and their use
DE102008062567A1 (de) * 2008-12-16 2010-06-17 Bayer Schering Pharma Aktiengesellschaft Dipeptoid-Prodrugs und ihre Verwendung
DE102009006602A1 (de) * 2009-01-29 2010-08-05 Bayer Schering Pharma Aktiengesellschaft Alkylamino-substituierte Dicyanopyridine und deren Aminosäureester-Prodrugs
DE102009022894A1 (de) * 2009-05-27 2010-12-02 Bayer Schering Pharma Aktiengesellschaft Substituierte Piperidine
DE102010030688A1 (de) 2010-06-30 2012-01-05 Bayer Schering Pharma Aktiengesellschaft Substituierte Dicyanopyridine und ihre Verwendung
KR20160042039A (ko) 2013-08-09 2016-04-18 알데릭스, 인코포레이티드 인산염 수송을 억제하기 위한 화합물 및 방법
WO2018153898A1 (de) 2017-02-22 2018-08-30 Bayer Pharma Aktiengesellschaft Selektive partielle adenosin a1 rezeptor-agonisten in kombination mit mineralocorticoid-rezeptor-antagonisten
WO2018153895A1 (de) 2017-02-22 2018-08-30 Bayer Pharma Aktiengesellschaft Selektive partielle adenosin a1 rezeptor-agonisten in kombination mit einem inhibitor der neutralen endopeptidase und/oder einem angiotensin ii rezeptor-antagonisten
WO2018153897A1 (de) 2017-02-22 2018-08-30 Bayer Pharma Aktiengesellschaft Selektive partielle adenosin a1 rezeptor-agonisten in kombination mit hcn-kanal-hemmern
WO2018153900A1 (de) 2017-02-22 2018-08-30 Bayer Aktiengesellschaft Selektive partielle adenosin a1 rezeptor-agonisten in kombination mit sglt-2-hemmern
WO2018153899A1 (de) 2017-02-22 2018-08-30 Bayer Pharma Aktiengesellschaft Selektive partielle adenosin a1 rezeptor-agonisten in kombination mit stimulatoren und/oder aktivatoren der löslichen guanylatcyclase (sgc)
JP7323913B2 (ja) * 2019-04-12 2023-08-09 国立大学法人 筑波大学 睡眠誘導剤である複素環化合物

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DE102008062567A1 (de) 2008-12-16 2010-06-17 Bayer Schering Pharma Aktiengesellschaft Dipeptoid-Prodrugs und ihre Verwendung
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Also Published As

Publication number Publication date
SV2006002218A (es) 2006-10-04
US8691850B2 (en) 2014-04-08
WO2006027142A1 (de) 2006-03-16
DE502005007106D1 (de) 2009-05-28
IL181670A0 (en) 2007-07-04
AU2005281941A1 (en) 2006-03-16
PE20060589A1 (es) 2006-08-12
JP2008511614A (ja) 2008-04-17
NO20071343L (no) 2007-05-30
CA2578596A1 (en) 2006-03-16
KR20070057235A (ko) 2007-06-04
ATE428710T1 (de) 2009-05-15
EP1812430B1 (de) 2009-04-15
ES2324049T3 (es) 2009-07-29
EP1812430A1 (de) 2007-08-01
UY29099A1 (es) 2006-04-28
BRPI0514833A (pt) 2008-06-24
GT200500238A (es) 2006-04-10
CA2578596C (en) 2012-10-23
DE102004042607A1 (de) 2006-03-09
TW200621765A (en) 2006-07-01
AR050551A1 (es) 2006-11-01
CN101056875A (zh) 2007-10-17
MX2007002470A (es) 2009-02-12
JP4999691B2 (ja) 2012-08-15
US20080269300A1 (en) 2008-10-30
MA28869B1 (fr) 2007-09-03
ZA200701820B (en) 2008-08-27

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