ECSP21015491A - Administración prolongada de lasmiditan por la noche para la prevención de la migraña - Google Patents
Administración prolongada de lasmiditan por la noche para la prevención de la migrañaInfo
- Publication number
- ECSP21015491A ECSP21015491A ECSENADI202115491A ECDI202115491A ECSP21015491A EC SP21015491 A ECSP21015491 A EC SP21015491A EC SENADI202115491 A ECSENADI202115491 A EC SENADI202115491A EC DI202115491 A ECDI202115491 A EC DI202115491A EC SP21015491 A ECSP21015491 A EC SP21015491A
- Authority
- EC
- Ecuador
- Prior art keywords
- migraine
- prevention
- night
- meditan
- prolonged administration
- Prior art date
Links
- 230000002265 prevention Effects 0.000 title abstract 3
- 230000002035 prolonged effect Effects 0.000 title abstract 2
- 208000019695 Migraine disease Diseases 0.000 abstract 3
- 206010027599 migraine Diseases 0.000 abstract 3
- XEDHVZKDSYZQBF-UHFFFAOYSA-N lasmiditan Chemical compound C1CN(C)CCC1C(=O)C1=CC=CC(NC(=O)C=2C(=CC(F)=CC=2F)F)=N1 XEDHVZKDSYZQBF-UHFFFAOYSA-N 0.000 abstract 1
- 229950009142 lasmiditan Drugs 0.000 abstract 1
- 238000009097 single-agent therapy Methods 0.000 abstract 1
- 238000002560 therapeutic procedure Methods 0.000 abstract 1
- 238000011282 treatment Methods 0.000 abstract 1
- 238000011269 treatment regimen Methods 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Plant Substances (AREA)
- Saccharide Compounds (AREA)
Abstract
La presente invención se refiere al uso prolongado de lasmiditan por la noche para la prevención de la migraña, particularmente la migraña resistente al tratamiento que se define en el presente documento como migraña refractaria a dos o más esquemas de prevención o tratamiento previos de monoterapia y/o terapia doble.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862726585P | 2018-09-04 | 2018-09-04 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP21015491A true ECSP21015491A (es) | 2021-04-29 |
Family
ID=68051892
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSENADI202115491A ECSP21015491A (es) | 2018-09-04 | 2021-03-04 | Administración prolongada de lasmiditan por la noche para la prevención de la migraña |
Country Status (36)
| Country | Link |
|---|---|
| US (1) | US12138254B2 (es) |
| EP (2) | EP3846810B1 (es) |
| JP (2) | JP7321256B2 (es) |
| KR (1) | KR102649644B1 (es) |
| CN (1) | CN112638383A (es) |
| AU (3) | AU2019336667B2 (es) |
| BR (1) | BR112021002945A2 (es) |
| CL (1) | CL2021000529A1 (es) |
| CO (1) | CO2021002766A2 (es) |
| CR (1) | CR20210126A (es) |
| DK (1) | DK3846810T3 (es) |
| DO (1) | DOP2021000039A (es) |
| EA (1) | EA202190440A1 (es) |
| EC (1) | ECSP21015491A (es) |
| ES (1) | ES2967665T3 (es) |
| FI (1) | FI3846810T3 (es) |
| HR (1) | HRP20231587T1 (es) |
| HU (1) | HUE064519T2 (es) |
| IL (1) | IL281208B2 (es) |
| JO (1) | JOP20210033B1 (es) |
| LT (1) | LT3846810T (es) |
| MA (1) | MA53551B1 (es) |
| MD (1) | MD3846810T2 (es) |
| MX (1) | MX2021002474A (es) |
| MY (1) | MY199662A (es) |
| PE (1) | PE20211599A1 (es) |
| PH (1) | PH12021550448A1 (es) |
| PL (1) | PL3846810T3 (es) |
| PT (1) | PT3846810T (es) |
| RS (1) | RS64857B1 (es) |
| SG (1) | SG11202101530PA (es) |
| SI (1) | SI3846810T1 (es) |
| TW (1) | TWI826514B (es) |
| UA (1) | UA129587C2 (es) |
| WO (1) | WO2020051137A1 (es) |
| ZA (1) | ZA202100666B (es) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ596161A (en) | 2009-04-02 | 2013-11-29 | Colucid Pharmaceuticals Inc | Composition of 2,4,6-trifluoro-n-[6-(1-methyl-piperidin-4-carbonyl)-pyridin-2-yl]-benzamide |
| US12168004B2 (en) | 2014-02-05 | 2024-12-17 | Merck Sharp & Dohme Llc | Treatment of migraine |
| KR102448369B1 (ko) | 2014-02-05 | 2022-09-28 | 머크 샤프 앤드 돔 엘엘씨 | Cgrp-활성 화합물에 대한 정제 제제 |
| US12090148B2 (en) | 2020-07-29 | 2024-09-17 | Allergan Pharmaceuticals International Limited | Treatment of migraine |
| US12383545B1 (en) | 2018-06-08 | 2025-08-12 | Allergan Pharmaceuticals International Limited | Treatment of migraine |
| MX2023007575A (es) | 2020-12-22 | 2023-09-21 | Allergan Pharmaceuticals Int Ltd | Tratamiento de la migraña. |
| AU2022353124A1 (en) | 2021-09-27 | 2024-04-11 | Allergan Pharmaceuticals International Limited | Combination comprising atogepant for treating migraine |
Family Cites Families (45)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5023252A (en) | 1985-12-04 | 1991-06-11 | Conrex Pharmaceutical Corporation | Transdermal and trans-membrane delivery of drugs |
| US5011472A (en) | 1988-09-06 | 1991-04-30 | Brown University Research Foundation | Implantable delivery system for biological factors |
| US5385912A (en) | 1991-03-08 | 1995-01-31 | Rhone-Poulenc Rorer Pharmaceuticals Inc. | Multicyclic tertiary amine polyaromatic squalene synthase inhibitors |
| US5360735A (en) | 1992-01-08 | 1994-11-01 | Synaptic Pharmaceutical Corporation | DNA encoding a human 5-HT1F receptor, vectors, and host cells |
| US5698571A (en) * | 1994-10-05 | 1997-12-16 | Eli Lilly And Company | 5-HT1F mediated inhibition of neurogenic meningeal extravasation: a method for the treatment of migraine |
| US5521196A (en) | 1994-10-05 | 1996-05-28 | Eli Lilly And Company | 5-HT1F agonists for the treatment of migraine |
| US5521197A (en) | 1994-12-01 | 1996-05-28 | Eli Lilly And Company | 3-<1-alkylenearyl>-4-<1,2,3,6-tetrahydropyridinyl>-and 3-<1-alkylenearyl>-4-piperidinyl-1h-indoles: new 5-HT1F agonists |
| CZ288897A3 (cs) | 1995-03-20 | 1998-02-18 | Eli Lilly And Company | V poloze 5-substituovaný 3-(1,2,3,6-tetrahydropyridin-4-yl)indol a 3-(piperidin-4-yl)indol a farmaceutický prostředek, který je obsahuje |
| JPH11513666A (ja) | 1995-10-10 | 1999-11-24 | イーライ・リリー・アンド・カンパニー | N−[2−置換−3−(2−アミノエチル)−1h−インドール−5−イル]−アミド:新規5−ht▲下1f▼作動剤 |
| US5708187A (en) | 1996-06-27 | 1998-01-13 | Eli Lilly And Company | 6-substituted-1,2,3,4-tetrahydro-9H-carbazoles and 7-substituted-10H-cyclohepta 7,6-B!indoles: New 5-HT1F agonists |
| BR9711273A (pt) | 1996-08-28 | 1999-08-17 | Lilly Co Eli | 1,2,3,4- Tetraidro-2-dibenzofuranaminas substituidas e 2- aminociclohepta b benzofuranos |
| CA2268164A1 (en) | 1996-10-08 | 1998-04-16 | Yao-Chang Xu | New serotonin 5-ht1f agonists |
| ZA979961B (en) | 1996-11-15 | 1999-05-05 | Lilly Co Eli | 5-HT1F agonists |
| EP0875513A1 (en) | 1997-04-14 | 1998-11-04 | Eli Lilly And Company | Substituted heteroaromatic 5-HT 1F agonists |
| ID23053A (id) | 1997-06-04 | 2000-01-20 | Lilly Co Eli | Karboksamida yang digunakan sebagai agonis 5-ht <if> |
| US5905084A (en) | 1997-11-14 | 1999-05-18 | Eli Lilly And Company | 5-HTIF -agonists effective in treating migraine |
| US6528529B1 (en) | 1998-03-31 | 2003-03-04 | Acadia Pharmaceuticals Inc. | Compounds with activity on muscarinic receptors |
| AU4961499A (en) | 1998-06-26 | 2000-01-17 | Eli Lilly And Company | 5-HT1f agonists |
| WO2000000487A1 (en) | 1998-06-30 | 2000-01-06 | Eli Lilly And Company | 5-ht1f agonists |
| AU1937300A (en) | 1998-12-11 | 2000-06-26 | Eli Lilly And Company | Indole derivatives and their use as 5-HT1F agonists |
| WO2000047559A2 (en) | 1999-02-10 | 2000-08-17 | Eli Lilly And Company | 5-ht1f agonists |
| US6777428B1 (en) | 1999-02-10 | 2004-08-17 | Eli Lilly And Company | 5-HT1f agonist |
| HUP0200245A2 (en) | 1999-02-26 | 2002-06-29 | Lilly Co Eli | Furo[3,2-b]pyridines as 5-ht1f agonists and pharmaceutical compositions containing them and their use |
| WO2002006196A1 (en) | 2000-07-13 | 2002-01-24 | Merck Patent Gmbh | Chiral compounds i |
| US6650463B2 (en) | 2001-03-13 | 2003-11-18 | Seiko Epson Corporation | Electrophoretic display device |
| US20050080112A1 (en) | 2001-06-22 | 2005-04-14 | Madsen Lars Siim | Compounds for use in disorders associated with mast cell or basophil acitvity |
| TWI263497B (en) | 2002-03-29 | 2006-10-11 | Lilly Co Eli | Pyridinoylpiperidines as 5-HT1F agonists |
| EP1581498A2 (en) | 2002-11-22 | 2005-10-05 | Bristol-Myers Squibb Company | Pyridinyl, pyrimidinyl and pyrazinyl amides as potassium channel openers |
| GB0308186D0 (en) | 2003-04-09 | 2003-05-14 | Smithkline Beecham Corp | Novel compounds |
| ES2388547T3 (es) | 2003-04-18 | 2012-10-16 | Eli Lilly And Company | Compuestos de (piperidiniloxi)fenilo, (piperidiniloxi)piridinilo, (piperidinilsulfanil)fenilo y (piperidinilsulfanil)piridinilo como agonistas de 5-HT 1F |
| WO2004099127A1 (en) | 2003-05-07 | 2004-11-18 | Novo Nordisk A/S | Novel compounds as kinase inhibitors |
| US7915293B2 (en) | 2003-05-30 | 2011-03-29 | Rigel Pharmaceuticals, Inc. | Ubiquitin ligase inhibitors |
| UA82711C2 (en) | 2003-09-12 | 2008-05-12 | Эли Лилли Энд Компани | Substituted 2-carbonylamino-6-piperidinaminopyridines and substituted 1-carbonylamino-3-piperidinaminobenzenes as 5-ht1f agonists |
| GB0325956D0 (en) | 2003-11-06 | 2003-12-10 | Addex Pharmaceuticals Sa | Novel compounds |
| EP1809620B1 (en) | 2004-11-04 | 2010-12-29 | Addex Pharma SA | Novel tetrazole derivatives as positive allosteric modulators of metabotropic glutamate receptors |
| GB0510143D0 (en) | 2005-05-18 | 2005-06-22 | Addex Pharmaceuticals Sa | Novel compounds A1 |
| KR20070094754A (ko) | 2004-12-01 | 2007-09-21 | 데브젠 엔브이 | 이온 채널, 특히 Kv 패밀리로부터의 이온 채널과상호작용하는 5-카복사미도 치환된 티아졸 유도체 |
| KR20060067738A (ko) | 2004-12-15 | 2006-06-20 | 주식회사 대웅제약 | 바닐로이드 수용체의 길항제로서 강력한 진통효과를나타내는 신규한 n-아릴아마이드 유도체 및 이를함유하는 약제학적 조성물 |
| US20060178349A1 (en) | 2005-01-24 | 2006-08-10 | Pozen Inc. | Compositions and therapeutic methods utilizing a combination of a 5-HT1F inhibitor and an NSAID |
| DE102005016634A1 (de) | 2005-04-12 | 2006-10-19 | Merck Patent Gmbh | Neuartige Aza-Hetercyclen als Kinase-Inhibitoren |
| KR100976063B1 (ko) | 2007-03-16 | 2010-08-17 | 동아제약주식회사 | 신규한 벤즈아미드 유도체 화합물 및 그의 제조방법 |
| NZ596161A (en) | 2009-04-02 | 2013-11-29 | Colucid Pharmaceuticals Inc | Composition of 2,4,6-trifluoro-n-[6-(1-methyl-piperidin-4-carbonyl)-pyridin-2-yl]-benzamide |
| US8697876B2 (en) * | 2010-04-02 | 2014-04-15 | Colucid Pharmaceuticals, Inc. | Compositions and methods of synthesis of pyridinolypiperidine 5-HT1F agonists |
| US11053214B2 (en) | 2016-12-06 | 2021-07-06 | Colucid Pharmaceuticals, Inc. | Compositions and methods related to pyridinoylpiperidine 5-HT1F agonists |
| TWI754772B (zh) | 2017-09-06 | 2022-02-11 | 美商美國禮來大藥廠 | 用於治療偏頭痛之拉米迪坦(lasmiditan)與cgrp拮抗劑之組合療法 |
-
2019
- 2019-09-02 TW TW108131567A patent/TWI826514B/zh active
- 2019-09-03 DK DK19773583.0T patent/DK3846810T3/da active
- 2019-09-03 HR HRP20231587TT patent/HRP20231587T1/hr unknown
- 2019-09-03 WO PCT/US2019/049340 patent/WO2020051137A1/en not_active Ceased
- 2019-09-03 CR CR20210126A patent/CR20210126A/es unknown
- 2019-09-03 CN CN201980055464.3A patent/CN112638383A/zh active Pending
- 2019-09-03 BR BR112021002945-1A patent/BR112021002945A2/pt unknown
- 2019-09-03 IL IL281208A patent/IL281208B2/en unknown
- 2019-09-03 FI FIEP19773583.0T patent/FI3846810T3/fi active
- 2019-09-03 AU AU2019336667A patent/AU2019336667B2/en not_active Ceased
- 2019-09-03 EP EP19773583.0A patent/EP3846810B1/en active Active
- 2019-09-03 UA UAA202100630A patent/UA129587C2/uk unknown
- 2019-09-03 LT LTEPPCT/US2019/049340T patent/LT3846810T/lt unknown
- 2019-09-03 SI SI201930647T patent/SI3846810T1/sl unknown
- 2019-09-03 PT PT197735830T patent/PT3846810T/pt unknown
- 2019-09-03 EP EP23195738.2A patent/EP4279132A3/en active Pending
- 2019-09-03 ES ES19773583T patent/ES2967665T3/es active Active
- 2019-09-03 PE PE2021000286A patent/PE20211599A1/es unknown
- 2019-09-03 PL PL19773583.0T patent/PL3846810T3/pl unknown
- 2019-09-03 JP JP2021512380A patent/JP7321256B2/ja active Active
- 2019-09-03 EA EA202190440A patent/EA202190440A1/ru unknown
- 2019-09-03 RS RS20231107A patent/RS64857B1/sr unknown
- 2019-09-03 HU HUE19773583A patent/HUE064519T2/hu unknown
- 2019-09-03 MX MX2021002474A patent/MX2021002474A/es unknown
- 2019-09-03 MY MYPI2021001043A patent/MY199662A/en unknown
- 2019-09-03 MD MDE20210640T patent/MD3846810T2/ro unknown
- 2019-09-03 US US17/271,950 patent/US12138254B2/en active Active
- 2019-09-03 MA MA53551A patent/MA53551B1/fr unknown
- 2019-09-03 SG SG11202101530PA patent/SG11202101530PA/en unknown
- 2019-09-03 KR KR1020217005977A patent/KR102649644B1/ko active Active
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2021
- 2021-01-29 ZA ZA2021/00666A patent/ZA202100666B/en unknown
- 2021-02-25 JO JOJO/P/2021/0033A patent/JOP20210033B1/ar active
- 2021-03-01 CO CONC2021/0002766A patent/CO2021002766A2/es unknown
- 2021-03-02 PH PH12021550448A patent/PH12021550448A1/en unknown
- 2021-03-02 DO DO2021000039A patent/DOP2021000039A/es unknown
- 2021-03-03 CL CL2021000529A patent/CL2021000529A1/es unknown
- 2021-03-04 EC ECSENADI202115491A patent/ECSP21015491A/es unknown
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2022
- 2022-12-22 AU AU2022291568A patent/AU2022291568A1/en not_active Abandoned
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2023
- 2023-07-25 JP JP2023120471A patent/JP7543497B2/ja active Active
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2025
- 2025-02-28 AU AU2025201479A patent/AU2025201479A1/en not_active Abandoned
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