EP2630133A1 - Nouveaux composés hétérocycliques utilisés en tant qu'agents pour lutter contre des nuisibles - Google Patents

Nouveaux composés hétérocycliques utilisés en tant qu'agents pour lutter contre des nuisibles

Info

Publication number
EP2630133A1
EP2630133A1 EP11771129.1A EP11771129A EP2630133A1 EP 2630133 A1 EP2630133 A1 EP 2630133A1 EP 11771129 A EP11771129 A EP 11771129A EP 2630133 A1 EP2630133 A1 EP 2630133A1
Authority
EP
European Patent Office
Prior art keywords
alkyl
spp
optionally substituted
alkoxy
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
EP11771129.1A
Other languages
German (de)
English (en)
Inventor
Thomas Bretschneider
Adeline KÖHLER
Joachim Kluth
Martin FÜSSLEIN
Peter Jeschke
Reiner Fischer
Friedrich August MÜHLTHAU
Olga Malsam
Arnd Voerste
Klaus-Helmut Müller
Yoshitaka Sato
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer Intellectual Property GmbH
Original Assignee
Bayer Intellectual Property GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Intellectual Property GmbH filed Critical Bayer Intellectual Property GmbH
Priority to EP11771129.1A priority Critical patent/EP2630133A1/fr
Publication of EP2630133A1 publication Critical patent/EP2630133A1/fr
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/76—1,3-Oxazoles; Hydrogenated 1,3-oxazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/78—1,3-Thiazoles; Hydrogenated 1,3-thiazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/82—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with three ring hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Definitions

  • R 17 is a radical from the series in each case optionally substituted alkyl, alkoxy, alkenyl and alkynyl, in each case optionally substituted cycloalkyl, cycloalkylalkyl and cycloalkenyl, in which the rings are at least one heteroatom from the series sulfur, oxygen (oxygen atoms may not be immediately adjacent) and each may contain nitrogen, each optionally substituted aryl, heteroaryl, arylalkyl and heteroarylalkyl and an optionally substituted amino group,
  • R 8 and R 16 may also together with the N-atom to which they are attached form a saturated or unsaturated and optionally substituted 4- to 8-membered ring containing one or more further heteroatoms selected from the group consisting of sulfur and oxygen (where Oxygen atoms may not be immediately adjacent) and nitrogen and / or at least one carbonyl group may contain,
  • R 16 represents a radical from the group hydrogen, in each case optionally substituted by halogen, Ci-C 6 - alkoxy, Ci-C 6 haloalkoxy, Ci-C 6 alkylthio, Ci-C 6 haloalkylthio, Ci-C 6 alkylsulfinyl , Ci-C 6 haloalkylsulfinyl, Ci-C 6 alkylsulfonyl or Ci-6 haloalkylsulfonyl C substituted C 6 alkyl, Ci-C 6 alkoxy, C 2 -C 6 -alkenyl and C 2 -C 6 - alkynyl, each optionally substituted by halo gen, Ci-C ß alkyl, Ci-C ß haloalkyl, Ci-C ß alkoxy or Ci-C -haloalkoxy ß-substituted C 3 -C 6 cycloalkyl, C 3 -C 6 - Cyclo
  • the compounds of the formula (A-6) are partially known or known. can be obtained by known production methods.
  • the compounds of the formula (A-6) simultaneously represent representatives of the radicals Q, which are mentioned by way of example above.
  • helminths e.g. Ancylostoma duodenale, Ancylostoma ceylanicum, Acylostoma braziliensis, Ancylostoma spp., Ascaris lubricoides, Ascaris spp., Brugia malayi, Brugia timori, Bunostomum spp., Chabertia spp., Clonorchis spp., Cooperia spp., Dicrocoelium spp., Dictyocaulus filaria, Diphyllobothrium latum, Dracunculus medinensis, Echinococcus granulosus, Echinococcus multilocularis, Enterobius vermicularis, Faciola spp., Haemonchus spp., Heterakis spp., Hymenolepis nana, Hyostrongulus spp., Loa Loa, Ne
  • the plant parasitic nematodes include e.g. Anguina spp., Aphelenchoides spp., Belonoaimus spp., Bursaphelenchus spp., Ditylenchus dipsaci, Globodera spp., Heliocotylenchus spp., Heterodera spp., Longidorus spp., Meloidogyne spp., Pratylenchus spp., Radopholus similis, Rotylenchus spp. Trichodorus spp., Tylenchorhynchus spp., Tylenchulus spp., Tylenchulus semipenetrans, Xiphinema spp.
  • Anguina spp. Aphelenchoides spp., Belonoaimus spp., Bursaphelenchus spp., Ditylenchus dipsaci, Globodera
  • Stabilizers such as cold stabilizers, preservatives, antioxidants, light stabilizers or other chemical and / or physical stability-improving agents may also be present.
  • the formulations generally contain between 0.01 and 98% by weight of active ingredient, preferably between 0.5 and 90%.
  • the active compounds according to the invention can also be used in admixture with one or more suitable fungicides, bactericides, acaricides, nematicides, insecticides, microbicides, fertilizers, attractants, sterilants, synergists, safeners, semiochemicals and / or plant growth regulators, in order to: eg to widen the spectrum of action, to extend the duration of action, to increase the speed of action, to prevent re-exposure or to prevent the development of resistance.
  • Fiproles phenylpyrazoles
  • Ethiprole e.g. Ethiprole
  • Fipronil e.g. Fipronil
  • Pyrafluprole e.g. Pyrafluprole
  • chloride channel activators such as Avermectins / milbemycins, eg abamectin, emamectin benzoate, lepimectin and milbemectin.
  • Organotin compounds e.g. Azocyclotine, cyhexatin, fenbutatin oxide; or propargite; Tetradifon.
  • inhibitors of chitin biosynthesis type 1, such as buprofezin.
  • active compound preparation 1 part by weight of active compound is mixed with the indicated amounts of solvent and emulsifier, and the concentrate is diluted with emulsifier-containing water to the desired concentration.
  • Bean leaf discs Phaseolus vulgaris
  • etranychus urticae Bean leaf discs infected by all stages of the common spider mite (Tetranychus urticae) are sprayed with an active compound preparation of the desired concentration.

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

L'invention concerne de nouveaux composés hétérocycliques, des procédés de production desdits composés et leur utilisation pour lutter contre des animaux nuisibles parmi lesquels figurent des arthropodes et des insectes.
EP11771129.1A 2010-10-22 2011-10-17 Nouveaux composés hétérocycliques utilisés en tant qu'agents pour lutter contre des nuisibles Withdrawn EP2630133A1 (fr)

Priority Applications (1)

Application Number Priority Date Filing Date Title
EP11771129.1A EP2630133A1 (fr) 2010-10-22 2011-10-17 Nouveaux composés hétérocycliques utilisés en tant qu'agents pour lutter contre des nuisibles

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US40580210P 2010-10-22 2010-10-22
EP10188470 2010-10-22
PCT/EP2011/068129 WO2012052412A1 (fr) 2010-10-22 2011-10-17 Nouveaux composés hétérocycliques utilisés en tant qu'agents pour lutter contre des nuisibles
EP11771129.1A EP2630133A1 (fr) 2010-10-22 2011-10-17 Nouveaux composés hétérocycliques utilisés en tant qu'agents pour lutter contre des nuisibles

Publications (1)

Publication Number Publication Date
EP2630133A1 true EP2630133A1 (fr) 2013-08-28

Family

ID=43568272

Family Applications (1)

Application Number Title Priority Date Filing Date
EP11771129.1A Withdrawn EP2630133A1 (fr) 2010-10-22 2011-10-17 Nouveaux composés hétérocycliques utilisés en tant qu'agents pour lutter contre des nuisibles

Country Status (6)

Country Link
US (2) US9173396B2 (fr)
EP (1) EP2630133A1 (fr)
JP (1) JP5953308B2 (fr)
CN (1) CN103270029B (fr)
BR (1) BR112013009823A2 (fr)
WO (1) WO2012052412A1 (fr)

Families Citing this family (44)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA107791C2 (en) 2009-05-05 2015-02-25 Dow Agrosciences Llc Pesticidal compositions
BR112012027762B1 (pt) * 2010-04-28 2018-06-05 Bayer Intellectual Property Gmbh Derivados de cetoheteroarilpiperidina e - piperazina como fungicidas
RU2576316C2 (ru) 2010-11-03 2016-02-27 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи Пестицидная композиция, способ контроля вредителей, способ контроля эндопаразитов, эктопаразитов или обоих и способ усиления жизнестойкости растений
JP6027128B2 (ja) 2011-10-26 2016-11-16 ダウ アグロサイエンシィズ エルエルシー 有害生物防除組成物およびそれに関連した方法
BR122014028247A2 (pt) 2012-04-27 2019-05-07 Dow Agrosciences Llc composições pesticidas, processo para controlar praga, uso de uma molécula, processo para aumentar a saúde, rendimento, vigor, qualidade ou tolerância de uma planta e processos para produção de compostos
US9282739B2 (en) 2012-04-27 2016-03-15 Dow Agrosciences Llc Pesticidal compositions and processes related thereto
US9708288B2 (en) 2012-04-27 2017-07-18 Dow Agrosciences Llc Pesticidal compositions and processes related thereto
WO2013186089A2 (fr) 2012-06-14 2013-12-19 Basf Se Procédés pesticides utilisant des composés thiazole à substitution 3-pyridyle et leurs dérivés pour lutter contre des nuisibles
CR20190436A (es) 2012-10-02 2019-10-29 Bayer Cropscience Ag COMPUESTOS HETEROCICLICOS COMO PLAGUICIDAS (Divisional 2015-0182)
EP3057429A4 (fr) 2013-10-17 2017-08-09 Dow AgroSciences LLC Procédés de préparation de de composés pesticides
CA2925952A1 (fr) 2013-10-17 2015-04-23 Dow Agrosciences Llc Procedes de preparation de composes pesticides
MX2016004941A (es) 2013-10-17 2016-06-28 Dow Agrosciences Llc Proceso para la preparacion de compuestos plaguicidas.
CA2926095A1 (fr) 2013-10-17 2015-04-23 Dow Agrosciences Llc Procedes de preparation de composes pesticides
JP2016539092A (ja) 2013-10-17 2016-12-15 ダウ アグロサイエンシィズ エルエルシー 有害生物防除性化合物の製造方法
US9029554B1 (en) 2013-10-17 2015-05-12 Dow Agrosciences Llc Processes for the preparation of pesticidal compounds
CA2925953C (fr) 2013-10-17 2021-11-02 Dow Agrosciences Llc Procedes de preparation de composes pesticides
JP2016534073A (ja) 2013-10-22 2016-11-04 ダウ アグロサイエンシィズ エルエルシー 相乗的有害生物防除組成物および関連する方法
NZ719952A (en) 2013-10-22 2017-05-26 Dow Agrosciences Llc Pesticidal compositions and related methods
KR20160074628A (ko) 2013-10-22 2016-06-28 다우 아그로사이언시즈 엘엘씨 상승작용적 살충 조성물 및 관련 방법
AR098100A1 (es) 2013-10-22 2016-05-04 Dow Agrosciences Llc Composiciones plaguicidas y los métodos relacionados
EP3060044A4 (fr) 2013-10-22 2017-04-05 Dow AgroSciences LLC Compositions pesticides synergiques et procédés associés
MX2016005305A (es) 2013-10-22 2017-03-01 Dow Agrosciences Llc Composiciones pesticidas sinergicas y metodos relacionados.
TW201517797A (zh) 2013-10-22 2015-05-16 Dow Agrosciences Llc 協同性殺蟲組成物及相關方法（十一）
AR098099A1 (es) 2013-10-22 2016-05-04 Dow Agrosciences Llc Composiciones plaguicidas sinérgicas y los métodos relacionados
US9801383B2 (en) 2013-10-22 2017-10-31 Dow Agrosciences Llc Synergistic pesticidal compositions and related methods
NZ719776A (en) 2013-10-22 2017-06-30 Dow Agrosciences Llc Synergistic pesticidal compositions and related methods
AR098101A1 (es) 2013-10-22 2016-05-04 Dow Agrosciences Llc Composiciones plaguicidas y métodos relacionados
US9295260B2 (en) 2013-10-22 2016-03-29 Dow Agrosciences Llc Pesticidal compositions and related methods
AU2014340424B2 (en) 2013-10-22 2017-06-29 Dow Agrosciences Llc Pesticidal compositions and related methods
RU2656894C2 (ru) 2013-10-22 2018-06-07 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи Пестицидные композиции и соответствующие способы
US9282740B2 (en) 2013-10-22 2016-03-15 Dow Agrosciences Llc Synergistic pesticidal compositions and related methods
JP2016535026A (ja) 2013-10-22 2016-11-10 ダウ アグロサイエンシィズ エルエルシー 相乗的有害生物防除組成物および関連する方法
US9788545B2 (en) 2013-10-22 2017-10-17 Dow Agrosciences Llc Synergistic pesticidal compositions and related methods
TWI647222B (zh) * 2014-03-06 2019-01-11 德商拜耳作物科學股份有限公司 作為殺蟲劑之雜環化合物
AR099677A1 (es) * 2014-03-07 2016-08-10 Sumitomo Chemical Co Compuesto heterocíclico fusionado y su uso para el control de plagas
US9249122B1 (en) 2014-07-31 2016-02-02 Dow Agrosciences Llc Process for the preparation of 3-(3-chloro-1H-pyrazol-1-yl)pyridine
JP2017523168A (ja) 2014-07-31 2017-08-17 ダウ アグロサイエンシィズ エルエルシー ３−（３−クロロ−１ｈ−ピラゾール−１−イル）ピリジンの製造方法
BR112017000293A2 (pt) 2014-07-31 2017-10-31 Dow Agrosciences Llc processo para a preparação de 3-(3-cloro-1h-pirazol-1-il)piridina
JP2017525703A (ja) 2014-08-19 2017-09-07 ダウ アグロサイエンシィズ エルエルシー ３−（３−クロロ−１ｈ−ピラゾール−１−イル）ピリジンの調製方法
AR098113A1 (es) 2014-09-12 2016-05-04 Dow Agrosciences Llc Proceso para la preparación de 3-(3-cloro-1h-pirazol-1-il)piridina
BR112018014518B1 (pt) 2016-02-26 2022-06-14 Nihon Nohyaku Co., Ltd Composto heterocíclico condensado ligado ao heterociclo ou sal deste, composição inseticida agrícola e hortícola, método para utilizar a referida composição, e composição para controle de ectoparasitas
CN110325036B (zh) 2016-12-29 2021-10-26 美国陶氏益农公司 用于制备杀虫化合物的方法
JP2020503336A (ja) 2016-12-29 2020-01-30 ダウ アグロサイエンシィズ エルエルシー 殺有害生物化合物の調製方法
WO2020113094A1 (fr) 2018-11-30 2020-06-04 Nuvation Bio Inc. Composés pyrrole et pyrazole et leurs procédés d'utilisation

Family Cites Families (109)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE42938C (de) Dr. O. BRAUN in Berlin W., Lützowstr. 60 Riemgetriebe mit Spannrollen und selbstthätiger Ausrückvorrichtung bei Ueberschreitung der vorbestimmten Kraftabgabe
US2847417A (en) 1956-07-13 1958-08-12 Houdry Process Corp Preparation of imidazole compounds
BE569324A (fr) 1957-07-11
US3542798A (en) 1968-12-30 1970-11-24 Geigy Chem Corp Pyridyl-2-imidazolone derivatives
US3666765A (en) 1969-10-27 1972-05-30 Union Carbide Corp Synthesis of 2-pyridones and derivatives thereof
US4089865A (en) 1971-10-27 1978-05-16 Syntex (U.S.A.) Inc. Certain thiazole compounds
BE790569A (fr) 1971-10-27 1973-04-26 Syntex Corp Agents cardiovasculaires a base de thiazoles
BE791871A (fr) 1971-11-26 1973-03-16 Veba Chemie Ag Procede de preparation d'esters d'imido-acide cycliques, et produits obtenus
US3927008A (en) 1973-08-30 1975-12-16 Denis M Bailey 5-(3-Pyridyl)-2-furoic acid
US4144343A (en) 1978-01-04 1979-03-13 Merck & Co., Inc. Heterocycle substituted (3-loweralkylamino-2-R1 O-propoxy)pyridines
DE3474093D1 (en) 1983-01-19 1988-10-27 Ciba Geigy Ag Pesticide
GB8306351D0 (en) 1983-03-08 1983-04-13 Ici Plc Azole fungicides
US4824859A (en) 1983-05-21 1989-04-25 Fisons Plc. Pyrazoline compounds compositions and use
US4775762A (en) 1987-05-11 1988-10-04 The Dow Chemical Company Novel (1H-1,2,3-triazol-1-yl)pyridines
GB8714789D0 (en) 1987-06-24 1987-07-29 Lundbeck & Co As H Heterocyclic compounds
DE3824658A1 (de) * 1988-07-15 1990-01-18 Schering Ag N-hetaryl-imidazolderivate
EP0539588A1 (fr) 1990-07-05 1993-05-05 Nippon Soda Co., Ltd. Derive d'amine
DE4114074A1 (de) 1991-04-30 1992-11-05 Bayer Ag Substituierte triazolinone
IE922270A1 (en) 1991-07-26 1993-01-27 Akzo Nv Pyrazole derivatives
DE4128029A1 (de) 1991-08-23 1993-02-25 Bayer Ag Substituierte triazolinone
US5536720A (en) 1992-09-09 1996-07-16 Uniroyal Chemical Company, Inc. Pesticidal oxadiazines
FR2707295A1 (fr) 1993-06-07 1995-01-13 Rhone Poulenc Agrochimie Fongicides pyrazoles substitués en position 3 par un hétérocycle.
JPH0741485A (ja) 1993-07-30 1995-02-10 Katayama Seiyakushiyo:Kk セフェム誘導体およびそれを含有する抗菌剤
JPH07138258A (ja) 1993-11-16 1995-05-30 Taiho Yakuhin Kogyo Kk チアゾリジンジオン誘導体又はその塩
JP3694051B2 (ja) 1994-07-12 2005-09-14 バイエルクロップサイエンス株式会社 １−ピリジルテトラゾリノン誘導体および除草剤
GB9512961D0 (en) 1995-06-26 1995-08-30 Pfizer Ltd Antifungal agents
WO1998025912A1 (fr) 1996-12-13 1998-06-18 E.I. Du Pont De Nemours And Company Amides heterocycliques herbicides
AU7553198A (en) * 1997-06-12 1998-12-30 Sumitomo Pharmaceuticals Company, Limited Pyrazole derivatives
DE19725450A1 (de) 1997-06-16 1998-12-17 Hoechst Schering Agrevo Gmbh 4-Haloalkyl-3-heterocyclylpyridine und 4-Haloalkyl-5-heterocyclylpyrimidine, Verfahren zu ihrer Herstellung, sie enthaltende Mittel und ihre Verwendung als Schädlingsbekämpfungsmittel
FR2780973B1 (fr) 1998-07-09 2001-10-05 Hoechst Marion Roussel Inc Procede de preparation du 4-(3-pyridinyl)-1h-imidazole, et les intermediaires mis en oeuvre
IT1301968B1 (it) 1998-07-30 2000-07-20 Zambon Spa Derivati di eritromicina ad attivita' antibiotica
WO2000007446A1 (fr) 1998-08-04 2000-02-17 Ciba Specialty Chemicals Holding Inc. Substances actives microbicides
US6747023B1 (en) 1998-08-11 2004-06-08 Daiichi Pharmaceutical Co., Ltd. Sulfonyl derivatives
FR2786188B1 (fr) 1998-11-24 2002-10-31 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur applicaion comme medicaments
US6660753B2 (en) 1999-08-19 2003-12-09 Nps Pharmaceuticals, Inc. Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists
WO2001038332A1 (fr) 1999-11-24 2001-05-31 Merck & Co., Inc. Gamma-hydroxy-2-(fluoroalkylaminocarbonyl)-1-piperazinepentanamides intervenant comme inhibiteurs de la protease du vih
FI19992686A7 (fi) 1999-12-14 2001-06-15 Nokia Networks Oy Synkronitasasuuntaus
US6372752B1 (en) 2000-02-07 2002-04-16 Genzyme Corporation Inha inhibitors and methods of use thereof
RU15525U1 (ru) 2000-07-04 2000-10-20 Федеральный научно-производственный центр закрытое акционерное общество "Научно-производственный концерн (объединение) "ЭНЕРГИЯ" Электродвигатель постоянного тока
IL158693A0 (en) * 2001-05-09 2004-05-12 Sumitomo Chem Takeda Agro Co Azole compounds, process for preparation of the same and use thereof
WO2003004509A2 (fr) 2001-07-03 2003-01-16 Chiron Corporation Macrolides et cetolides d'erythromycine modifiee c12 a activite antibacterienne
JPWO2003022821A1 (ja) 2001-09-06 2004-12-24 大正製薬株式会社 ２０−ｈｅｔｅ産生酵素阻害作用を有するヘテロ環誘導体
WO2003024986A1 (fr) 2001-09-17 2003-03-27 Ortho-Mcneil Pharmaceutical, Inc. Agents antimicrobiens 6-o-carbamate-11,12-lacto-cetolide
CA2461363A1 (fr) * 2001-09-26 2003-04-03 Bayer Pharmaceuticals Corporation 3-pyridyl indoles et indazoles substitues servant d'inhibiteurs de c17,20 lyase
DE60226756D1 (de) 2001-10-04 2008-07-03 Merck & Co Inc Heteroarylsubstituierte tetrazolmodulatoren des metabotropischen glutamatrezeptors-5
NZ533282A (en) 2001-12-05 2006-09-29 Ortho Mcneil Pharm Inc 6-O-Acyl ketolide derivatives of erythromycine useful as antibacterials
DE60334781D1 (de) 2002-03-12 2010-12-16 Merck Sharp & Dohme Di-aryl-substituierte tetrazol-modulatoren des metabotropen glutamat-rezeptors-5
US20040033970A1 (en) 2002-04-30 2004-02-19 Clark Richard F. Antibacterial compounds with improved pharmacokinetic profiles
PL374970A1 (en) 2002-08-02 2005-11-14 Argenta Discovery Limited Substituted thienyl-hydroxamic acids as histone deacetylase inhibitors
CN1829721A (zh) 2003-07-08 2006-09-06 阿斯利康(瑞典)有限公司 对α7烟碱乙酰胆碱受体具有亲和力的螺[1－氮杂二环[2.2.2]辛烷－3,5’－噁唑烷]－2’－酮衍生物
UA79404C2 (en) 2003-10-02 2007-06-11 Basf Ag 2-cyanobenzenesulfonamide for controlling pests
CN1897939A (zh) 2003-10-31 2007-01-17 詹森药业有限公司 适用作过氧化物酶体增生物激活受体（ppar）双重激动剂的苯氧基乙酸衍生物
WO2005047281A1 (fr) * 2003-11-13 2005-05-26 Syngenta Participations Ag Nouveaux herbicides
TW200529860A (en) 2003-12-22 2005-09-16 Astrazeneca Ab Nicotinic acetylcholine receptor ligands
US20080188527A1 (en) 2003-12-23 2008-08-07 Cashman John R Synthetic Compounds and Derivatives as Modulators of Smoking or Nicotine Ingestion and Lung Cancer
JP2005223238A (ja) 2004-02-09 2005-08-18 Konica Minolta Holdings Inc 有機半導体材料及びそれを用いた有機薄膜トランジスタ、電界効果有機薄膜トランジスタ並びにそれらを用いたスイッチング素子
KR20100017777A (ko) 2004-02-18 2010-02-16 이시하라 산교 가부시끼가이샤 안트라닐아미드계 화합물, 그의 제조 방법 및 그것을 함유하는 유해 생물 방제제
WO2005085214A1 (fr) 2004-03-05 2005-09-15 Banyu Pharmaceutical Co., Ltd Dérivé hétérocyclique à cinq éléments substitués par un diaryle
WO2006038100A1 (fr) 2004-10-08 2006-04-13 Ranbaxy Laboratories Limited Derives d'oxazolidinone utilises comme agents antimicrobiens
WO2006043635A1 (fr) 2004-10-20 2006-04-27 Kumiai Chemical Industry Co., Ltd. Dérivé de 3-triazolylphénylsulfide et insecticide/acaricide/nématicide incluant ledit dérivé au titre de principe actif
CN101065353A (zh) 2004-11-26 2007-10-31 巴斯福股份公司 用于防治动物害虫的新型2－氰基－3－(卤代)烷氧基苯磺酰胺化合物
DE102005008021A1 (de) 2005-02-22 2006-08-24 Bayer Cropscience Ag Spiroketal-substituierte cyclische Ketoenole
MX2007010840A (es) 2005-03-24 2007-10-16 Basf Ag Compuestos de 2-cianobencenosulfonamida para el tratamiento de semillas.
TW200637559A (en) 2005-03-29 2006-11-01 Shionogi & Co 3-propenylcefem derivative
DE102005019712A1 (de) * 2005-04-28 2006-11-09 Bayer Healthcare Ag Dipyridyl-dihydropyrazolone und ihre Verwendung
TWI388282B (zh) 2005-06-01 2013-03-11 Meiji Seika Pharma Co Ltd 害蟲控制劑
US7491738B2 (en) 2005-06-01 2009-02-17 Meiji Seika Kaisha, Ltd. Pest control agents
AU2006258101A1 (en) 2005-06-09 2006-12-21 Merck Sharp & Dohme Corp. Inhibitors of checkpoint kinases
US7452892B2 (en) 2005-06-17 2008-11-18 Bristol-Myers Squibb Company Triazolopyrimidine cannabinoid receptor 1 antagonists
JP2007145806A (ja) 2005-09-27 2007-06-14 Sagami Chem Res Center オキサゾール誘導体、それらの製造方法及びそれらを用いたオキサゾリル基導入方法
KR20080066938A (ko) * 2005-10-07 2008-07-17 깃세이 야쿠힌 고교 가부시키가이샤 질소 함유 복소환 화합물 및 그것을 함유하는 의약 조성물
PT1937664E (pt) 2005-10-14 2011-07-07 Sumitomo Chemical Co Composto de hidrazida e utilização pesticida do mesmo
EP1954138A2 (fr) 2005-11-21 2008-08-13 Basf Se Procedes insecticides utilisant des derives de 3-amino-1,2-benzisothiazole
JP2009518442A (ja) 2005-12-05 2009-05-07 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 可溶性エポキシド加水分解酵素インヒビターとして有益な置換ピラゾール化合物
DE102006015468A1 (de) 2006-03-31 2007-10-04 Bayer Cropscience Ag Substituierte Enaminocarbonylverbindungen
DE102006015470A1 (de) 2006-03-31 2007-10-04 Bayer Cropscience Ag Substituierte Enaminocarbonylverbindungen
DE102006015467A1 (de) 2006-03-31 2007-10-04 Bayer Cropscience Ag Substituierte Enaminocarbonylverbindungen
TWI381811B (zh) 2006-06-23 2013-01-11 Dow Agrosciences Llc 用以防治可抵抗一般殺蟲劑之昆蟲的方法
US20080090834A1 (en) 2006-07-06 2008-04-17 Pfizer Inc Selective azole pde10a inhibitor compounds
US20100234349A1 (en) 2006-09-04 2010-09-16 Olsen Gunnar M Pharmaceutical combinations of a nicotine receptor modulator and a cognitive enhancer
EP2079734A1 (fr) * 2006-10-25 2009-07-22 NeuroSearch A/S Composes de type oxadiazole et thiadiazole et leur utilisation comme modulateurs des recepteurs nicotiniques de l'acetylcholine
CA2668210C (fr) 2006-10-31 2013-03-12 Schering Corporation Derives d'anilinopiperazine et leurs methodes d'utilisation
DE102006057036A1 (de) 2006-12-04 2008-06-05 Bayer Cropscience Ag Biphenylsubstituierte spirocyclische Ketoenole
US7795249B2 (en) 2006-12-22 2010-09-14 Millennium Pharmaceuticals, Inc. Certain pyrazoline derivatives with kinase inhibitory activity
EA200901143A1 (ru) 2007-03-01 2010-04-30 Басф Се Пестицидные активные смеси, включающие аминотиазолиновые соединения
US20080255203A1 (en) * 2007-04-12 2008-10-16 Abbott Laboratories Heterocyclic compounds and their methods of use
JP5326424B2 (ja) 2007-08-31 2013-10-30 住友化学株式会社 含フッ素有機硫黄化合物およびその有害節足動物防除剤
US8530480B2 (en) * 2007-09-04 2013-09-10 The Scripps Research Institute Substituted pyrimidinyl-amines as protein kinase inhibitors
EP2211619A1 (fr) * 2007-10-18 2010-08-04 Merck Sharp & Dohme Corp. 1,2,4-oxadiazoles substitués et leurs analogues comme modulateurs des récepteurs cb2, utiles dans le traitement de la douleur et de maladies respiratoires et non respiratoires
EP2070925A1 (fr) 2007-12-10 2009-06-17 Bayer Schering Pharma Aktiengesellschaft Nouveaux dérivés de 2-thiazol-4-amides d'acide carboxylique substitués, leur fabrication et leur utilisation en tant que médicament
WO2009105500A1 (fr) 2008-02-21 2009-08-27 Schering Corporation Composés inhibiteurs de la voie erk
GB0804685D0 (en) 2008-03-13 2008-04-16 Univ Edinburgh Therapeutic compounds and their use
WO2009129036A1 (fr) 2008-04-14 2009-10-22 Merck & Co., Inc. Composés cyclopropyliques substitués, compositions contenant de tels composés et procédés de traitement
GB0806794D0 (en) 2008-04-15 2008-05-14 Ludwig Inst Cancer Res Therapeutic compounds
CN102047061A (zh) * 2008-05-30 2011-05-04 福斯特韦勒能源股份公司 通过氧化燃料燃烧发电的方法和系统
WO2009149135A1 (fr) * 2008-06-04 2009-12-10 Abbott Laboratories Isoxazoles substitués de bis (hétéro) aryle pour utilisation comme modulateurs de récepteurs nicotiniques neuronaux
CN102089297A (zh) * 2008-06-06 2011-06-08 雅培制药有限公司 新的1,2,4-噁二唑化合物和其使用方法
WO2009149858A1 (fr) 2008-06-13 2009-12-17 Bayer Cropscience Ag Nouveaux amides et thioamides utilisés comme agents de lutte contre les parasites
WO2010005572A2 (fr) 2008-07-09 2010-01-14 The Scripps Research Institute Alpha-cétohétérocycles comme inhibiteurs de faah
EP2586311B1 (fr) 2008-07-17 2016-12-14 Bayer CropScience AG Liaisons hétérocycliques en tant que moyen de lutte contre les parasites
CA2735392A1 (fr) 2008-08-15 2010-02-18 F. Hoffmann-La Roche Ag Bi-aryle aminotetralines
BRPI0917693A2 (pt) * 2008-09-02 2016-05-17 Neurosearch As composto derivado de triazol, composição farmacêutica, e, uso de um derivado de triazol
JP2012501975A (ja) 2008-09-08 2012-01-26 メルク カナダ インコーポレイテッド ステアロイルコエンザイムＡδ−９デサチュラーゼの阻害剤としての芳香族複素環化合物
US8436008B2 (en) 2008-12-22 2013-05-07 Incyte Corporation Substituted heterocyclic compounds
WO2010075356A1 (fr) 2008-12-23 2010-07-01 Forest Laboratories Holdings Limited Nouveaux dérivés de pipérazine constituant des inhibiteurs de stéaroyl-coa désaturase
US20100168177A1 (en) 2008-12-26 2010-07-01 Dow Agrosciences, Llc Stable insecticide compositions
MX343270B (es) 2008-12-26 2016-10-31 Dow Agrosciences Llc * Composiciones de insecticida estables y metodos para producir las mismas.
CN102574833B (zh) 2009-10-12 2014-08-20 拜尔农作物科学股份公司 用作杀虫剂的酰胺和硫代酰胺
WO2011045224A1 (fr) 2009-10-12 2011-04-21 Bayer Cropscience Ag 1-(pyrid-3-yl)-pyrazole et 1-(pyrimid-5-yl)-pyrazole en tant qu'agents antiparasites

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
See references of WO2012052412A1 *

Also Published As

Publication number Publication date
BR112013009823A2 (pt) 2016-07-05
CN103270029B (zh) 2016-01-20
US20150373978A1 (en) 2015-12-31
US20130261141A1 (en) 2013-10-03
CN103270029A (zh) 2013-08-28
JP2013544792A (ja) 2013-12-19
JP5953308B2 (ja) 2016-07-20
WO2012052412A1 (fr) 2012-04-26
US9173396B2 (en) 2015-11-03

Similar Documents

Publication Publication Date Title
US9173396B2 (en) Heterocyclic compounds as pesticides
US9233951B2 (en) Heterocyclic compounds as pesticides
US9688681B2 (en) Heterocyclic compounds as pest control agents
EP2566865B1 (fr) Dérivés de thiazole utilisés comme pesticides
EP2585451B1 (fr) Composés hétérocycliques utilisés en tant qu'agents de lutte contre les parasites
EP2591674B1 (fr) Liaisons hétérocycliques en tant que moyen de lutte contre les parasites
ES2555260T3 (es) Derivados de diamida de ácido antranílico
EP2582691A1 (fr) Dérivés d'acide anthranilique
EP2582695A1 (fr) Dérivés de diamide d'acide anthranilique à chaînes latérales cycliques
EP2582693A1 (fr) Nouveaux dérivés arylamide ortho-substitués

Legal Events

Date Code Title Description
PUAI Public reference made under article 153(3) epc to a published international application that has entered the european phase

Free format text: ORIGINAL CODE: 0009012

17P Request for examination filed

Effective date: 20130522

AK Designated contracting states

Kind code of ref document: A1

Designated state(s): AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

DAX Request for extension of the european patent (deleted)
17Q First examination report despatched

Effective date: 20150825

STAA Information on the status of an ep patent application or granted ep patent

Free format text: STATUS: THE APPLICATION IS DEEMED TO BE WITHDRAWN

18D Application deemed to be withdrawn

Effective date: 20160927