ES2062043T3 - Formulaciones topicas y sistemas de suministro transdermico que contienen 1-isobutil-1h-imidazo(4,5-c)-quinolein-4-amina. - Google Patents

Formulaciones topicas y sistemas de suministro transdermico que contienen 1-isobutil-1h-imidazo(4,5-c)-quinolein-4-amina.

Info

Publication number
ES2062043T3
ES2062043T3 ES89312885T ES89312885T ES2062043T3 ES 2062043 T3 ES2062043 T3 ES 2062043T3 ES 89312885 T ES89312885 T ES 89312885T ES 89312885 T ES89312885 T ES 89312885T ES 2062043 T3 ES2062043 T3 ES 2062043T3
Authority
ES
Spain
Prior art keywords
imidazo
quinolein
transdermic
isobutyl
amine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES89312885T
Other languages
English (en)
Inventor
Steven M C O Riker Labora Wick
Helen Jensen C O Riker Schultz
Gregory R C O Riker Lab Nelson
Amit K C O Riker Laborat Mitra
Stephen M C O Riker Labo Berge
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Riker Laboratories Inc
Original Assignee
Riker Laboratories Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Riker Laboratories Inc filed Critical Riker Laboratories Inc
Application granted granted Critical
Publication of ES2062043T3 publication Critical patent/ES2062043T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/74—Synthetic polymeric materials
    • A61K31/765—Polymers containing oxygen
    • A61K31/78—Polymers containing oxygen of acrylic acid or derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
    • A61K9/7053—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
    • A61K9/7061—Polyacrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/12—Carboxylic acids; Salts or anhydrides thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0014—Skin, i.e. galenical aspects of topical compositions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Dermatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

FORMULACIONES FARMACEUTICAS Y MATERIALES EN FORMA DE LAMINA REVESTIDOS CON ADHESIVO PARA LA LIBERACION TOPICA Y/O TRANSCUTANEA DE 1- IGOBUTIL-1H-IMIDAZO (A,S-C) QUINOLINA-4-AMIDA, INCLUYENDO CREMAS, UNGUENTOS Y COMPOSICIONES ADHESIVAS SENSIBLES A LA PRESION O METODOS FARMACOLOGICOS DE USO DE LAS FORMULACIONES Y LOS MATERIALES EN FORMA DE LAMINAS REVESTIDAS DE ADHESIVO DEL INVENTO EN EL TRATAMIENTO DE INFECCIONES VIRICAS.
ES89312885T 1988-12-15 1989-12-11 Formulaciones topicas y sistemas de suministro transdermico que contienen 1-isobutil-1h-imidazo(4,5-c)-quinolein-4-amina. Expired - Lifetime ES2062043T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US28493388A 1988-12-15 1988-12-15

Publications (1)

Publication Number Publication Date
ES2062043T3 true ES2062043T3 (es) 1994-12-16

Family

ID=23092090

Family Applications (1)

Application Number Title Priority Date Filing Date
ES89312885T Expired - Lifetime ES2062043T3 (es) 1988-12-15 1989-12-11 Formulaciones topicas y sistemas de suministro transdermico que contienen 1-isobutil-1h-imidazo(4,5-c)-quinolein-4-amina.

Country Status (13)

Country Link
EP (1) EP0376534B1 (es)
JP (1) JP2915034B2 (es)
KR (1) KR0150445B1 (es)
AU (1) AU631585B2 (es)
CA (1) CA2004597C (es)
DE (2) DE68911499T2 (es)
DK (1) DK176121B1 (es)
ES (1) ES2062043T3 (es)
IE (1) IE62569B1 (es)
IL (1) IL92537A (es)
NL (1) NL980042I1 (es)
NZ (1) NZ231655A (es)
ZA (1) ZA899450B (es)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ232740A (en) * 1989-04-20 1992-06-25 Riker Laboratories Inc Solution for parenteral administration comprising a 1h-imidazo(4,5-c) quinolin-4-amine derivative, an acid and a tonicity adjuster
IL105325A (en) * 1992-04-16 1996-11-14 Minnesota Mining & Mfg Immunogen/vaccine adjuvant composition
WO1995004551A1 (en) * 1993-08-10 1995-02-16 Fujisawa Pharmaceutical Co., Ltd. Percutaneously absorbable preparation
DE4434775A1 (de) * 1994-09-29 1996-04-04 Beiersdorf Ag Dermatologische Zubereitungen mit einem Gehalt an Fettsäureglyceriden gegen Superinfektionen
US5939090A (en) * 1996-12-03 1999-08-17 3M Innovative Properties Company Gel formulations for topical drug delivery
IT1294748B1 (it) 1997-09-17 1999-04-12 Permatec Tech Ag Formulazione per un dispositivo transdermico
CA2361936C (en) * 1999-01-08 2009-06-16 3M Innovative Properties Company Formulations comprising imiquimod or other immune response modifiers for treating mucosal conditions
US7658938B2 (en) 1999-02-22 2010-02-09 Merrion Reasearch III Limited Solid oral dosage form containing an enhancer
US8119159B2 (en) 1999-02-22 2012-02-21 Merrion Research Iii Limited Solid oral dosage form containing an enhancer
EP1390024A4 (en) * 2001-05-11 2010-02-17 Merrion Res Iii Ltd ISOSTEARIC ACID SALTS AS PERMEATION IMPROVERS
WO2002092069A1 (en) 2001-05-11 2002-11-21 Elan Corporation, Plc Permeation enhancers
CN1292751C (zh) * 2002-04-23 2007-01-03 四川大学 皮肤局部用咪喹莫特或其衍生物脂质体及其制备方法和用途
KR20050109562A (ko) * 2003-03-13 2005-11-21 쓰리엠 이노베이티브 프로퍼티즈 컴파니 피부의 질을 개선시키는 방법
CN105232482A (zh) 2006-04-07 2016-01-13 默里昂研究Iii有限公司 包含增强剂的固体口服剂型
EP2046121B1 (en) 2006-07-14 2012-08-22 Stiefel Research Australia Pty Ltd Fatty acid pharmaceutical foam
AU2007275815A1 (en) * 2006-07-18 2008-01-24 Wirra Ip Pty. Ltd. Immune response modifier formulations
AU2009244799B2 (en) 2008-05-07 2014-11-20 Merrion Research Iii Limited Compositions of GnRH related compounds and processes of preparation
US9089484B2 (en) 2010-03-26 2015-07-28 Merrion Research Iii Limited Pharmaceutical compositions of selective factor Xa inhibitors for oral administration
AU2012204213A1 (en) 2011-01-07 2013-06-13 Merrion Research Iii Limited Pharmaceutical compositions of iron for oral administration
US10265384B2 (en) 2015-01-29 2019-04-23 Novo Nordisk A/S Tablets comprising GLP-1 agonist and enteric coating
ES2940736B2 (es) 2021-11-09 2023-09-19 Ntd Labs S L U Uso combinado de imiquimod y de un hidrolizado de caseina para el tratamiento de condilomas

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL73534A (en) * 1983-11-18 1990-12-23 Riker Laboratories Inc 1h-imidazo(4,5-c)quinoline-4-amines,their preparation and pharmaceutical compositions containing certain such compounds
CA1272445A (en) * 1985-02-25 1990-08-07 Yie W. Chien Transdermal pharmaceutical absorption dosage unit and process of pharmaceutical administration
CA1288698C (en) * 1985-08-30 1991-09-10 Rutgers, The State University Of New Jersey Transdermal anti-anginal pharmaceutical dosage

Also Published As

Publication number Publication date
DE68911499D1 (de) 1994-01-27
DE19975026I2 (de) 2010-07-08
AU631585B2 (en) 1992-12-03
AU4670689A (en) 1990-06-21
IL92537A0 (en) 1990-08-31
EP0376534A1 (en) 1990-07-04
IE893888L (en) 1990-06-15
HK1006275A1 (en) 1999-02-19
NL980042I1 (nl) 1999-02-01
DK613889D0 (da) 1989-12-06
KR900009084A (ko) 1990-07-02
DK613889A (da) 1990-06-16
JPH02282327A (ja) 1990-11-19
CA2004597C (en) 2000-02-08
EP0376534B1 (en) 1993-12-15
NZ231655A (en) 1992-06-25
JP2915034B2 (ja) 1999-07-05
CA2004597A1 (en) 1990-06-15
IE62569B1 (en) 1995-02-08
KR0150445B1 (ko) 1998-10-15
DK176121B1 (da) 2006-09-11
IL92537A (en) 1994-04-12
ZA899450B (en) 1990-09-26
DE68911499T2 (de) 1994-06-30

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