ES2136086T3 - Agentes antibacterianos con azaespiroquinolona. - Google Patents

Agentes antibacterianos con azaespiroquinolona.

Info

Publication number
ES2136086T3
ES2136086T3 ES92912150T ES92912150T ES2136086T3 ES 2136086 T3 ES2136086 T3 ES 2136086T3 ES 92912150 T ES92912150 T ES 92912150T ES 92912150 T ES92912150 T ES 92912150T ES 2136086 T3 ES2136086 T3 ES 2136086T3
Authority
ES
Spain
Prior art keywords
azaespiroquinolone
antibacterial agents
quinolone
alpha
antibacterial properties
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES92912150T
Other languages
English (en)
Spanish (es)
Inventor
Bingwei Vera Yang
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
PFIZER
Pfizer Inc
Original Assignee
PFIZER
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by PFIZER, Pfizer Inc filed Critical PFIZER
Application granted granted Critical
Publication of ES2136086T3 publication Critical patent/ES2136086T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicinal Preparation (AREA)
  • Materials For Medical Uses (AREA)
ES92912150T 1991-06-19 1992-05-04 Agentes antibacterianos con azaespiroquinolona. Expired - Lifetime ES2136086T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US71755291A 1991-06-19 1991-06-19

Publications (1)

Publication Number Publication Date
ES2136086T3 true ES2136086T3 (es) 1999-11-16

Family

ID=24882485

Family Applications (1)

Application Number Title Priority Date Filing Date
ES92912150T Expired - Lifetime ES2136086T3 (es) 1991-06-19 1992-05-04 Agentes antibacterianos con azaespiroquinolona.

Country Status (13)

Country Link
US (1) US5407943A (fr)
EP (1) EP0641339B1 (fr)
JP (1) JPH0678335B2 (fr)
AT (1) ATE184603T1 (fr)
CA (1) CA2111463C (fr)
DE (1) DE69230005T2 (fr)
DK (1) DK0641339T3 (fr)
ES (1) ES2136086T3 (fr)
FI (2) FI982097A0 (fr)
GR (1) GR3031701T3 (fr)
IE (1) IE921970A1 (fr)
PT (1) PT100597B (fr)
WO (1) WO1992022550A1 (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6664271B1 (en) * 1999-05-21 2003-12-16 Eli Lilly And Company Immunopotentiator agents
US7902227B2 (en) 2007-07-27 2011-03-08 Janssen Pharmaceutica Nv. C-7 isoxazolinyl quinolone / naphthyridine derivatives useful as antibacterial agents
FR2941696B1 (fr) 2009-02-05 2011-04-15 Sanofi Aventis Derives d'azaspiranyl-alkylcarbamates d'heterocycles a 5 chainons, leur preparation et leur application en therapeutique
FR2945531A1 (fr) 2009-05-12 2010-11-19 Sanofi Aventis Derives de 7-aza-spiro°3,5!nonane-7-carboxylates, leur preparation et leur application en therapeutique
WO2012047703A2 (fr) * 2010-10-04 2012-04-12 Schering Corporation Cyclopropyl-spiro-pipéridines utiles comme bloqueurs des canaux sodiques

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4571396A (en) * 1984-04-16 1986-02-18 Warner-Lambert Company Antibacterial agents
JPH0676400B2 (ja) * 1987-08-25 1994-09-28 大日本製薬株式会社 新規ピリドンカルボン酸誘導体、そのエステルおよびその塩
MY105136A (en) * 1988-04-27 1994-08-30 Daiichi Seiyaku Co Optically active pyridonecarboxylic acid derivatives.
CA1336090C (fr) * 1988-08-31 1995-06-27 Isao Hayakawa Amines cycliques a substituant spiro de derives de la quinolone
CA2012681A1 (fr) * 1989-03-31 1990-09-30 Masayasu Okuhira Derives de la quinolone, procedes de preparation et agents antibacteriens les renfermant
RU2049777C1 (ru) * 1989-08-16 1995-12-10 Пфайзер Инк. Азабицикло-хинолон-карбоновые кислоты или их фармацевтически приемлемые кислотно-аддитивные соли и промежуточные продукты для их получения

Also Published As

Publication number Publication date
DK0641339T3 (da) 1999-12-20
PT100597B (pt) 1999-07-30
US5407943A (en) 1995-04-18
CA2111463C (fr) 1997-08-26
FI935700A0 (fi) 1993-12-17
DE69230005T2 (de) 2000-01-05
FI102900B1 (fi) 1999-03-15
JPH0678335B2 (ja) 1994-10-05
PT100597A (pt) 1993-09-30
DE69230005D1 (de) 1999-10-21
FI935700L (fi) 1993-12-17
FI102900B (fi) 1999-03-15
EP0641339A1 (fr) 1995-03-08
FI982097L (fi) 1998-09-29
CA2111463A1 (fr) 1992-12-23
IE921970A1 (en) 1992-12-30
ATE184603T1 (de) 1999-10-15
GR3031701T3 (en) 2000-02-29
WO1992022550A1 (fr) 1992-12-23
FI982097A7 (fi) 1998-09-29
JPH06503355A (ja) 1994-04-14
FI982097A0 (fi) 1998-09-29
EP0641339B1 (fr) 1999-09-15

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