ES2138668T3 - Nuevos derivados de peptidos terapeuticamente activos en la cadena de coagulacion sanguinea, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen. - Google Patents
Nuevos derivados de peptidos terapeuticamente activos en la cadena de coagulacion sanguinea, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen.Info
- Publication number
- ES2138668T3 ES2138668T3 ES94929585T ES94929585T ES2138668T3 ES 2138668 T3 ES2138668 T3 ES 2138668T3 ES 94929585 T ES94929585 T ES 94929585T ES 94929585 T ES94929585 T ES 94929585T ES 2138668 T3 ES2138668 T3 ES 2138668T3
- Authority
- ES
- Spain
- Prior art keywords
- contain
- pharmaceutical compositions
- blood coagulation
- therapeutically active
- preparation procedure
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/81—Protease inhibitors
- C07K14/815—Protease inhibitors from leeches, e.g. hirudin, eglin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Tropical Medicine & Parasitology (AREA)
- Biophysics (AREA)
- Diabetes (AREA)
- Biochemistry (AREA)
- Genetics & Genomics (AREA)
- Gastroenterology & Hepatology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Hematology (AREA)
- Molecular Biology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Abstract
LA INVENCION SE REFIERE A LOS DERIVADOS DE FORMULA (I): H-PHE, A{SUB,1}-ARG-PRO-(GLY){SUB,4}-ASN-GLY-ASP-PHE-GLU-ABO-ILE-PROGLU-GLU-A{SUB,2}-LEU-GLU-OH, EN LA QUE A{SUB,1} Y A{SUB,2} SON TAL COMO SE DEFINEN EN LA DESCRIPCION. MEDICAMENTOS.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9311942A FR2710917B1 (fr) | 1993-10-07 | 1993-10-07 | Nouveaux dérivés de peptides thérapeutiquement actifs dans la cascade de coagulation sanguine, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2138668T3 true ES2138668T3 (es) | 2000-01-16 |
Family
ID=9451616
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES94929585T Expired - Lifetime ES2138668T3 (es) | 1993-10-07 | 1994-10-06 | Nuevos derivados de peptidos terapeuticamente activos en la cadena de coagulacion sanguinea, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen. |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US5786330A (es) |
| EP (1) | EP0722460B1 (es) |
| JP (1) | JP2899415B2 (es) |
| CN (1) | CN1053451C (es) |
| AT (1) | ATE184287T1 (es) |
| AU (1) | AU680696B2 (es) |
| CA (1) | CA2173598A1 (es) |
| DE (1) | DE69420574T2 (es) |
| DK (1) | DK0722460T3 (es) |
| ES (1) | ES2138668T3 (es) |
| FI (1) | FI961505A7 (es) |
| FR (1) | FR2710917B1 (es) |
| GR (1) | GR3031254T3 (es) |
| NO (1) | NO961357L (es) |
| NZ (1) | NZ274524A (es) |
| WO (1) | WO1995009869A1 (es) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20020045589A1 (en) * | 2000-03-30 | 2002-04-18 | Gary Shen | Hirulog-like peptide and gene therapy |
| DK1737889T3 (da) | 2004-10-19 | 2011-01-03 | Lonza Ag | Fremgangsmåde til fastfase-peptidsyntese |
| US7598343B1 (en) | 2008-07-27 | 2009-10-06 | The Medicines Company | Pharmaceutical formulations of bivalirudin and processes of making the same |
| US7582727B1 (en) | 2008-07-27 | 2009-09-01 | The Medicinces Company | Pharmaceutical formulations of bivalirudin and processes of making the same |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2686086A1 (fr) * | 1992-01-15 | 1993-07-16 | Adir | Nouveaux derives de peptides et de pseudopeptides therapeutiquement actifs dans la cascade de coagulation sanguine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent. |
-
1993
- 1993-10-07 FR FR9311942A patent/FR2710917B1/fr not_active Expired - Fee Related
-
1994
- 1994-10-06 CA CA002173598A patent/CA2173598A1/fr not_active Abandoned
- 1994-10-06 AU AU78587/94A patent/AU680696B2/en not_active Ceased
- 1994-10-06 EP EP94929585A patent/EP0722460B1/fr not_active Expired - Lifetime
- 1994-10-06 ES ES94929585T patent/ES2138668T3/es not_active Expired - Lifetime
- 1994-10-06 AT AT94929585T patent/ATE184287T1/de not_active IP Right Cessation
- 1994-10-06 DE DE69420574T patent/DE69420574T2/de not_active Expired - Fee Related
- 1994-10-06 NZ NZ274524A patent/NZ274524A/en unknown
- 1994-10-06 WO PCT/FR1994/001166 patent/WO1995009869A1/fr not_active Ceased
- 1994-10-06 DK DK94929585T patent/DK0722460T3/da active
- 1994-10-06 US US08/619,683 patent/US5786330A/en not_active Expired - Fee Related
- 1994-10-06 CN CN94194052A patent/CN1053451C/zh not_active Expired - Fee Related
- 1994-10-06 FI FI961505A patent/FI961505A7/fi unknown
- 1994-10-06 JP JP7510650A patent/JP2899415B2/ja not_active Expired - Fee Related
-
1996
- 1996-04-02 NO NO961357A patent/NO961357L/no not_active Application Discontinuation
-
1999
- 1999-09-20 GR GR990402347T patent/GR3031254T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| GR3031254T3 (en) | 1999-12-31 |
| EP0722460A1 (fr) | 1996-07-24 |
| AU680696B2 (en) | 1997-08-07 |
| FR2710917B1 (fr) | 1995-11-24 |
| DK0722460T3 (da) | 2000-03-20 |
| CN1134706A (zh) | 1996-10-30 |
| CN1053451C (zh) | 2000-06-14 |
| EP0722460B1 (fr) | 1999-09-08 |
| US5786330A (en) | 1998-07-28 |
| AU7858794A (en) | 1995-05-01 |
| JPH09503221A (ja) | 1997-03-31 |
| FI961505L (fi) | 1996-04-03 |
| ATE184287T1 (de) | 1999-09-15 |
| CA2173598A1 (fr) | 1995-04-13 |
| DE69420574T2 (de) | 2000-05-04 |
| NO961357L (no) | 1996-06-06 |
| JP2899415B2 (ja) | 1999-06-02 |
| FI961505A0 (fi) | 1996-04-03 |
| WO1995009869A1 (fr) | 1995-04-13 |
| DE69420574D1 (de) | 1999-10-14 |
| NZ274524A (en) | 1996-12-20 |
| NO961357D0 (no) | 1996-04-02 |
| FI961505A7 (fi) | 1996-04-03 |
| FR2710917A1 (fr) | 1995-04-14 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| BG60102B2 (bg) | Метод за получаване на 5-флуор-2(((4-циклопропил- метокси-2-пиридинил)метил)тионил)-1н-бензимидазол | |
| ES2058411T3 (es) | Sustancia fr 901228 y su preparacion. | |
| ES2161291T3 (es) | N-(indol-2-carbonil)amidas y derivados como inhibidores de la glucogeno fosforilasa. | |
| AR003427A1 (es) | Péptidos relacionados con dolastatina, procedimiento para prepararlos, composiciones farmacéuticas que los contienen y el uso de los mismos para la preparación de dichas composiciones farmacéuticas. | |
| EA200201271A1 (ru) | Ингибиторы 11-бета-гидроксистероиддегидрогеназы типа 1 | |
| ES2084944T3 (es) | Amidas terapeuticas. | |
| ECSP034883A (es) | Amidas de acidos antranilicos con cadena lateral de heteroarilsulfonilo, procedimiento para su preparacion, su empleo como medicamento o agente de diagnostico, asi como preparados farmaceuticos que las contienen | |
| CR9879A (es) | Moduladores de ccr5 (divisional de la solicitud n° 6392) | |
| ES2076935T3 (es) | Compuesto de pirazolopiridina y procedimientos para su preparacion. | |
| UY26372A1 (es) | "imidazo-3-il-aminas bicíclicas procedimiento para su preparación y medicamentos que las contienen " | |
| ES2093440T3 (es) | Derivados en la serie de la vitamina d con modificaciones en la posicion 20, procedimiento para su preparacion, productos intermedios para este procedimiento, preparados farmaceuticos que contienen estos derivados asi como su utilizacion para la preparacion de medicamentos. | |
| ES2169147T3 (es) | Derivados de beta-carbolina agonistas de la melatonina, sus procedimientos de preparacion y su utilizacion a titulo de medicamento. | |
| AR006401A1 (es) | Compuestos de pirrolopirrolona, una composicion farmaceutica que los contiene, su uso en la fabricacion de un medicamento y en terapia, procesospara su preparación y compuestos intermediarios para dichos procesos. | |
| ES2142030T3 (es) | Nuevos compuestos espiro-heterociclicos, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen. | |
| ES2180933T3 (es) | Inhibidor de la serina-proteasa. | |
| IT1170214B (it) | Composizione farmaceutica per la cura delle arteriopatie periferiche | |
| DK0736029T3 (da) | Antikonvulsive pseudofructopyranosesulfamater | |
| ES2134237T3 (es) | Composiciones farmaceuticas que contienen acido ursodesoxicolico. | |
| ES2077559T3 (es) | Estabilizacion de proteinas terapeuticamente activas en preparados farmaceuticos. | |
| AR021086A1 (es) | Omega-amidas de n-arilsulfonil-aminoacidos, un procedimiento para su preparacion, medicamento, uso de dichos compuestos para la preparacion de un medicamento y procedimiento para la preparacion de un medicamento. | |
| CO4940448A1 (es) | Modificacion a cristal de una sustancia de medicamento | |
| ES2127263T3 (es) | Nuevos trien-derivados cromenicos, su procedimiento de preparacion y composiciones farmaceuticas que los contienen. | |
| ES2145234T3 (es) | Derivados de la diosmetina, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen. | |
| MY126358A (en) | Compositions comprising vx478 and a water soluble tocopherol derivative such as vitamin e-tpgs | |
| DK77588A (da) | Prostaglandin e1-derivater og farmaceutiske praeparater, der indeholder dem |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG2A | Definitive protection |
Ref document number: 722460 Country of ref document: ES |