ES3043807A2 - Proceso para preparar hemifumarato de 5-{2-[bencil-(1-(4-hidroxifenil)-1-metiletil)amino]-1-hidroxietil}benceno-1,3-diol - Google Patents
Proceso para preparar hemifumarato de 5-{2-[bencil-(1-(4-hidroxifenil)-1-metiletil)amino]-1-hidroxietil}benceno-1,3-diolInfo
- Publication number
- ES3043807A2 ES3043807A2 ES202590070A ES202590070A ES3043807A2 ES 3043807 A2 ES3043807 A2 ES 3043807A2 ES 202590070 A ES202590070 A ES 202590070A ES 202590070 A ES202590070 A ES 202590070A ES 3043807 A2 ES3043807 A2 ES 3043807A2
- Authority
- ES
- Spain
- Prior art keywords
- acid
- solution
- methylethyl
- hydroxyphenyl
- amino
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
- C07C213/08—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reactions not involving the formation of amino groups, hydroxy groups or etherified or esterified hydroxy groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C215/00—Compounds containing amino and hydroxy groups bound to the same carbon skeleton
- C07C215/46—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
- C07C215/56—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups linked to the six-membered aromatic ring, or to the condensed ring system containing that ring, by carbon chains further substituted by hydroxy groups
- C07C215/58—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups linked to the six-membered aromatic ring, or to the condensed ring system containing that ring, by carbon chains further substituted by hydroxy groups with hydroxy groups and the six-membered aromatic ring, or the condensed ring system containing that ring, bound to the same carbon atom of the carbon chain
- C07C215/60—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups linked to the six-membered aromatic ring, or to the condensed ring system containing that ring, by carbon chains further substituted by hydroxy groups with hydroxy groups and the six-membered aromatic ring, or the condensed ring system containing that ring, bound to the same carbon atom of the carbon chain the chain having two carbon atoms between the amino groups and the six-membered aromatic ring or the condensed ring system containing that ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C221/00—Preparation of compounds containing amino groups and doubly-bound oxygen atoms bound to the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C225/00—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones
- C07C225/02—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton
- C07C225/14—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being unsaturated
- C07C225/16—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT102023000008112A IT202300008112A1 (it) | 2023-04-26 | 2023-04-26 | Processo per la preparazione di emifumarato di 5-{2-[benzil-(1-(4-idrossifenil)-1-metiletil)ammino]-1-idrossietil}benzene-1,3-diolo |
| PCT/EP2024/060701 WO2024223428A1 (en) | 2023-04-26 | 2024-04-19 | Process for preparing 5-{2-[benzyl-(1-(4-hydroxyphenyl)-1-methylethyl)amino]-1-hydroxyethyl}benzene-1,3-diol hemifumarate |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES3043807A2 true ES3043807A2 (es) | 2025-11-25 |
Family
ID=87514228
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES202590070A Pending ES3043807A2 (es) | 2023-04-26 | 2024-04-19 | Proceso para preparar hemifumarato de 5-{2-[bencil-(1-(4-hidroxifenil)-1-metiletil)amino]-1-hidroxietil}benceno-1,3-diol |
Country Status (10)
| Country | Link |
|---|---|
| KR (1) | KR20260003013A (de) |
| CN (1) | CN121358709A (de) |
| AT (1) | AT528464A2 (de) |
| CO (1) | CO2025016166A2 (de) |
| DE (1) | DE112024001886T5 (de) |
| ES (1) | ES3043807A2 (de) |
| FR (1) | FR3148237B1 (de) |
| IT (1) | IT202300008112A1 (de) |
| PE (1) | PE20260045A1 (de) |
| WO (1) | WO2024223428A1 (de) |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL300751A (de) | 1962-11-30 | 1900-01-01 |
-
2023
- 2023-04-26 IT IT102023000008112A patent/IT202300008112A1/it unknown
-
2024
- 2024-04-19 PE PE2025002387A patent/PE20260045A1/es unknown
- 2024-04-19 DE DE112024001886.6T patent/DE112024001886T5/de active Pending
- 2024-04-19 AT ATA95011/2025A patent/AT528464A2/de unknown
- 2024-04-19 CN CN202480039489.5A patent/CN121358709A/zh active Pending
- 2024-04-19 ES ES202590070A patent/ES3043807A2/es active Pending
- 2024-04-19 KR KR1020257038826A patent/KR20260003013A/ko active Pending
- 2024-04-19 WO PCT/EP2024/060701 patent/WO2024223428A1/en not_active Ceased
- 2024-04-25 FR FR2404346A patent/FR3148237B1/fr active Active
-
2025
- 2025-11-24 CO CONC2025/0016166A patent/CO2025016166A2/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2024223428A1 (en) | 2024-10-31 |
| AT528464A2 (de) | 2025-12-15 |
| CN121358709A (zh) | 2026-01-16 |
| DE112024001886T5 (de) | 2026-02-19 |
| FR3148237A1 (fr) | 2024-11-01 |
| CO2025016166A2 (es) | 2025-12-09 |
| FR3148237B1 (fr) | 2025-10-17 |
| IT202300008112A1 (it) | 2024-10-26 |
| PE20260045A1 (es) | 2026-01-09 |
| KR20260003013A (ko) | 2026-01-06 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| BA2A | Patent application published |
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