ES424851A1 - Un procedimiento para preparar derivados de piperazina. - Google Patents

Un procedimiento para preparar derivados de piperazina.

Info

Publication number
ES424851A1
ES424851A1 ES424851A ES424851A ES424851A1 ES 424851 A1 ES424851 A1 ES 424851A1 ES 424851 A ES424851 A ES 424851A ES 424851 A ES424851 A ES 424851A ES 424851 A1 ES424851 A1 ES 424851A1
Authority
ES
Spain
Prior art keywords
formula
group
compound
procedure
piperazine derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES424851A
Other languages
English (en)
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sumitomo Pharma Co Ltd
Original Assignee
Dainippon Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP3845373A external-priority patent/JPS5546400B2/ja
Priority claimed from JP5654473A external-priority patent/JPS565753B2/ja
Priority claimed from JP6446473A external-priority patent/JPS565755B2/ja
Application filed by Dainippon Pharmaceutical Co Ltd filed Critical Dainippon Pharmaceutical Co Ltd
Publication of ES424851A1 publication Critical patent/ES424851A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
ES424851A 1973-04-03 1974-04-02 Un procedimiento para preparar derivados de piperazina. Expired ES424851A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP3845373A JPS5546400B2 (de) 1973-04-03 1973-04-03
JP5654473A JPS565753B2 (de) 1973-05-21 1973-05-21
JP6446473A JPS565755B2 (de) 1973-06-07 1973-06-07

Publications (1)

Publication Number Publication Date
ES424851A1 true ES424851A1 (es) 1976-06-01

Family

ID=27289838

Family Applications (1)

Application Number Title Priority Date Filing Date
ES424851A Expired ES424851A1 (es) 1973-04-03 1974-04-02 Un procedimiento para preparar derivados de piperazina.

Country Status (11)

Country Link
AR (2) AR204003A1 (de)
AT (1) AT340931B (de)
CA (1) CA1066701A (de)
CH (1) CH593281A5 (de)
ES (1) ES424851A1 (de)
FI (1) FI56011C (de)
IE (1) IE39102B1 (de)
NL (1) NL186087C (de)
NO (1) NO142221C (de)
PH (2) PH10529A (de)
SE (1) SE416051B (de)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1209163B (it) * 1979-12-21 1989-07-10 Unibios S P A Trecate Novara Procedimento per la fabbricazione di: 6-alcossicarbonil-8-etil-5-oxo-5,8diidro-aperta par. quadrata 2,3-dchiusa par. quadrata-primidine 2-sostituite ed acidi libri corrispondenti.
EP2845856A1 (de) 2009-06-29 2015-03-11 Incyte Corporation Pyrimidone als PI3K-Hemmer
WO2011075630A1 (en) 2009-12-18 2011-06-23 Incyte Corporation Substituted fused aryl and heteroaryl derivatives as pi3k inhibitors
US8759359B2 (en) 2009-12-18 2014-06-24 Incyte Corporation Substituted heteroaryl fused derivatives as PI3K inhibitors
TW201249844A (en) 2010-12-20 2012-12-16 Incyte Corp N-(1-(substituted-phenyl)ethyl)-9H-purin-6-amines as PI3K inhibitors
UA121539C2 (uk) 2011-09-02 2020-06-25 Інсайт Холдинґс Корпорейшн Гетероцикліламіни як інгібітори рі3к
AR090548A1 (es) 2012-04-02 2014-11-19 Incyte Corp Azaheterociclobencilaminas biciclicas como inhibidores de pi3k
US10077277B2 (en) 2014-06-11 2018-09-18 Incyte Corporation Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors
UA122332C2 (uk) 2015-02-27 2020-10-26 Інсайт Корпорейшн Солі інгібітора pi3k і способи їх отримання
WO2016183060A1 (en) 2015-05-11 2016-11-17 Incyte Corporation Process for the synthesis of a phosphoinositide 3-kinase inhibitor
WO2016183063A1 (en) 2015-05-11 2016-11-17 Incyte Corporation Crystalline forms of a pi3k inhibitor
MX2020012826A (es) 2018-06-01 2021-03-09 Incyte Corp Regimen de dosificacion para el tratamiento de trastornos relacionados con fosfatidilinositol 3-cinasas (pi3k).

Also Published As

Publication number Publication date
CH593281A5 (en) 1977-11-30
FI56011C (fi) 1979-11-12
NO740349L (no) 1974-10-04
CA1066701A (en) 1979-11-20
PH10984A (en) 1977-10-18
AR204003A1 (es) 1975-11-12
NL186087C (nl) 1990-09-17
NL7401509A (de) 1974-10-07
IE39102B1 (en) 1978-08-02
NO142221C (no) 1980-07-16
PH10529A (en) 1977-05-30
FI56011B (fi) 1979-07-31
AR204660A1 (es) 1976-02-20
IE39102L (en) 1974-10-03
AT340931B (de) 1978-01-10
ATA277774A (de) 1977-05-15
NO142221B (no) 1980-04-08
NL186087B (nl) 1990-04-17
SE416051B (sv) 1980-11-24

Similar Documents

Publication Publication Date Title
GB1428467A (en) Indane and tetrahydronaphthalene derivatives
ES425900A1 (es) Procedimiento para la preparacion de nuevos compuestos de isoflavona.
ES360948A1 (es) Procedimiento para la preparacion de derivados de sulfoni- lurea.
ES429871A1 (es) Procedimiento de preparacion de derivados 1, 3-benzodioxol.
ES405479A1 (es) Un procedimiento para la preparacion de derivados de benzo-diacepina.
ES462843A1 (es) Un procedimiento para la preparacion de compuestos imidazo (1,5-a) (1,4)diacepinicos.
ES412047A1 (es) Un procedimiento para la preparacion de dihidrocumarina o una alcohil-dihidrocumarina.
ES404315A1 (es) Un procedimiento de preparacion de un derivado de nitrosou-rea.
CH614940A5 (en) Process for the preparation of new terpenoaromatic amidines
ES423817A1 (es) Un procedimiento para la obtencion de 6-alquil-ergolinas d-2-sustituidas y 8-sustituidas.
ES442023A1 (es) Procedimiento para la preparacion de derivados de propanol.
ES364980A1 (es) Un metodo para preparar nuevos derivados de adamantano.
ES437041A1 (es) Un procedimiento para preparar derivados de 1-ftalazona.
ES422248A1 (es) Procedimiento para la preparacion de 7-cloro-1,2-dihidro-5-fenil - 1,4-benzodiazepin-2-onas.
ES459400A1 (es) Un procedimiento para la produccion de nuevos compuestos de 6,11-dihidrodibenzo (b.e.) tiepin-11-ona.
ES393953A1 (es) Procedimiento para la preparacion de compuestos de 1,4-ben-zodiacepina.
GB1467225A (en) 7-alkoxy-4,6-dihydroxy-quinoline derivatives and pharmaceuti cal compositions thereof
ES441003A1 (es) Un procedimiento para preparar productos intermedios utiles en la sintesis de prosglandinas.
ES385778A1 (es) Un metodo para producir derivados de benzazocina.
ES420004A1 (es) Un procedimiento para la preparacion de un derivado de ni- trosourea.
ES397454A1 (es) Un procedimiento para la preparacion de derivados de tetra-hidro-isoquinolina.
ES412799A1 (es) Un procedimiento para preparar alcoholes alcohilsulfonilme-tilbencilicos.
ES398222A1 (es) Un procedimiento para la preparacion de derivados de benzo-diazepina.
JPS51146481A (en) Process for preparing arabinofuranosylcytosine derivatives
FI762309A7 (de)