ES8201529A1 - Un procedimiento para la preparacion de nuevos derivados de 1-1'-bifenil-2-il-alquilamina - Google Patents

Un procedimiento para la preparacion de nuevos derivados de 1-1'-bifenil-2-il-alquilamina

Info

Publication number
ES8201529A1
ES8201529A1 ES497210A ES497210A ES8201529A1 ES 8201529 A1 ES8201529 A1 ES 8201529A1 ES 497210 A ES497210 A ES 497210A ES 497210 A ES497210 A ES 497210A ES 8201529 A1 ES8201529 A1 ES 8201529A1
Authority
ES
Spain
Prior art keywords
hydrogen
alkyl
biphenyl
alkylamine
procedure
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES497210A
Other languages
English (en)
Other versions
ES497210A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of ES497210A0 publication Critical patent/ES497210A0/es
Publication of ES8201529A1 publication Critical patent/ES8201529A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00Compounds containing amino groups bound to a carbon skeleton
    • C07C211/01Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms
    • C07C211/26Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing at least one six-membered aromatic ring
    • C07C211/27Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing at least one six-membered aromatic ring having amino groups linked to the six-membered aromatic ring by saturated carbon chains
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • C07D295/084Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/092Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings with aromatic radicals attached to the chain
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00Carboxylic acid nitriles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Cardiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Emergency Medicine (AREA)
  • Epidemiology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

PROCEDIMIENTO PARA LA OBTENCION DE DERIVADOS DE 1,1''-BIFENIL-2-IL-ALQUILAMINA, DE FORMULA (I), DONDE X ES HIDROGENO O HALOGENO; R1 Y R2 SON HIDROGENO, R3 Y R4 SON HIDROGENO, ALQUILO, CH2-ALQUENILO, FENILALQUILO O FORMAN, CON EL ATOMO DE NITROGENO ADYACENTE, UN GRUPO HETEROCICLO Y Z ES -(CH2)N-, DONDE N ES 2, 3 O 4. CONSISTE EN SOMETER A REACCION DE REDUCCION UNA OLEFINA DE FORMULA (II). SI SE DESEA SE SEPARAN LOS GRUPOS PROTECTORES Y SE FORMAN SALES DE AMONIO CUATERNARIO O DE ADICION DE ACIDO. DE APLICACION COMO AGENTES ANTIARRITMICOS.
ES497210A 1979-03-12 1980-11-27 Un procedimiento para la preparacion de nuevos derivados de 1-1'-bifenil-2-il-alquilamina Expired ES8201529A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US1953479A 1979-03-12 1979-03-12

Publications (2)

Publication Number Publication Date
ES497210A0 ES497210A0 (es) 1981-12-16
ES8201529A1 true ES8201529A1 (es) 1981-12-16

Family

ID=21793713

Family Applications (6)

Application Number Title Priority Date Filing Date
ES489469A Expired ES8105262A1 (es) 1979-03-12 1980-03-12 Un procedimiento para la preparacion de 1, 1'-bifenil-2-il- alquilamina.
ES497209A Granted ES497209A0 (es) 1979-03-12 1980-11-27 Un procedimiento para la preparacion de nuevos derivados de 1,1'-bifenil-2-il-alquilamina
ES497206A Granted ES497206A0 (es) 1979-03-12 1980-11-27 Un procedimiento para la preparacion de nuevos derivados de 1,1'-bifenil-2-il-alquilamina
ES497208A Granted ES497208A0 (es) 1979-03-12 1980-11-27 Un procedimiento para las preparaciones de nuevos derivados de 1,1'-bifenil-2-il-alquilamina
ES497210A Expired ES8201529A1 (es) 1979-03-12 1980-11-27 Un procedimiento para la preparacion de nuevos derivados de 1-1'-bifenil-2-il-alquilamina
ES497207A Granted ES497207A0 (es) 1979-03-12 1980-11-27 Un procedimiento para la preparacion de nuevos derivados de 1,1'-binefil-2-il-alquilamina

Family Applications Before (4)

Application Number Title Priority Date Filing Date
ES489469A Expired ES8105262A1 (es) 1979-03-12 1980-03-12 Un procedimiento para la preparacion de 1, 1'-bifenil-2-il- alquilamina.
ES497209A Granted ES497209A0 (es) 1979-03-12 1980-11-27 Un procedimiento para la preparacion de nuevos derivados de 1,1'-bifenil-2-il-alquilamina
ES497206A Granted ES497206A0 (es) 1979-03-12 1980-11-27 Un procedimiento para la preparacion de nuevos derivados de 1,1'-bifenil-2-il-alquilamina
ES497208A Granted ES497208A0 (es) 1979-03-12 1980-11-27 Un procedimiento para las preparaciones de nuevos derivados de 1,1'-bifenil-2-il-alquilamina

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES497207A Granted ES497207A0 (es) 1979-03-12 1980-11-27 Un procedimiento para la preparacion de nuevos derivados de 1,1'-binefil-2-il-alquilamina

Country Status (31)

Country Link
EP (1) EP0015776B1 (es)
JP (1) JPS55127347A (es)
KR (1) KR840000103B1 (es)
AR (1) AR228852A1 (es)
AT (1) AT367395B (es)
AU (1) AU528060B2 (es)
BE (1) BE882167A (es)
CA (1) CA1144926A (es)
CH (1) CH644094A5 (es)
CS (1) CS215052B2 (es)
DD (1) DD149664A5 (es)
DE (1) DE3060611D1 (es)
DK (1) DK103480A (es)
ES (6) ES8105262A1 (es)
FI (1) FI800736A7 (es)
FR (1) FR2451363A1 (es)
GB (1) GB2046256B (es)
GR (1) GR68036B (es)
HU (1) HU180334B (es)
IE (1) IE49552B1 (es)
IL (1) IL59557A (es)
IT (1) IT1140773B (es)
LU (1) LU82237A1 (es)
MX (1) MX6219E (es)
NZ (1) NZ193079A (es)
PH (1) PH14749A (es)
PL (1) PL121662B1 (es)
PT (1) PT70928A (es)
RO (1) RO79906A (es)
SU (2) SU940645A3 (es)
ZA (1) ZA801421B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100470454B1 (ko) * 2002-05-14 2005-02-05 대한민국 돼지 사료공급을 위한 자동조절급이기
AU2005265164A1 (en) * 2004-06-17 2006-01-26 Musc Foundation For Research Development Non-natural amino acids
EP2511273B8 (en) * 2011-04-15 2019-06-26 Hivih Inhibitors of viral replication, their process of preparation and their therapeutical uses
EP2821104A1 (en) 2013-07-05 2015-01-07 Laboratoire Biodim Inhibitors of viral replication, their process of preparation and their therapeutical uses

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES236010A1 (es) * 1956-06-29 1957-12-16 Lab Pharmaceutica Dr C Janssen UN PROCEDIMIENTO PARA PREPARAR NUEVOS DERIVADOS PARASIMPATICOLiTICAMENTE ACTIVOS DE ALFAS-DEFENIL PROPANO
US3433836A (en) * 1966-01-14 1969-03-18 Rexall Drug Chemical Alpha-diaryl alpha,omega-alkylene glycol-dilower-alkylamines
GB1475314A (en) * 1973-11-02 1977-06-01 Cm Ind Phenyl-propylamine derivatives
IL48319A0 (en) * 1974-10-26 1975-12-31 Merck Patent Gmbh Araliphatic nitrogen compounds and a process for their preparation
GB1523655A (en) * 1975-02-10 1978-09-06 Armour Pharma 4-(4-biphenylyl) butylamines and treatment of the animal organism therewith

Also Published As

Publication number Publication date
ES497210A0 (es) 1981-12-16
ZA801421B (en) 1981-10-28
AU528060B2 (en) 1983-04-14
PT70928A (en) 1980-04-01
ES8201526A1 (es) 1981-12-16
IT1140773B (it) 1986-10-10
CS215052B2 (en) 1982-07-30
NZ193079A (en) 1982-05-31
PL121662B1 (en) 1982-05-31
FR2451363B1 (es) 1983-01-14
DD149664A5 (de) 1981-07-22
ES8201528A1 (es) 1981-12-16
IT8020503A0 (it) 1980-03-11
ES8201525A1 (es) 1981-12-16
ES497206A0 (es) 1981-12-16
DK103480A (da) 1980-09-13
ES497207A0 (es) 1981-12-16
FI800736A7 (fi) 1981-01-01
IE800493L (en) 1980-09-12
KR840000103B1 (ko) 1984-02-11
GB2046256B (en) 1983-04-20
EP0015776B1 (en) 1982-06-30
PH14749A (en) 1981-11-20
SU940645A3 (ru) 1982-06-30
BE882167A (fr) 1980-09-11
IE49552B1 (en) 1985-10-30
ES489469A0 (es) 1981-05-16
DE3060611D1 (en) 1982-08-19
GR68036B (es) 1981-10-27
ES8105262A1 (es) 1981-05-16
AR228852A1 (es) 1983-04-29
JPS55127347A (en) 1980-10-02
EP0015776A1 (en) 1980-09-17
AU5630280A (en) 1980-09-18
GB2046256A (en) 1980-11-12
PL222601A1 (es) 1981-01-30
KR830001854A (ko) 1983-05-19
LU82237A1 (fr) 1980-06-06
ES8201527A1 (es) 1981-12-16
IL59557A0 (en) 1980-06-30
CH644094A5 (fr) 1984-07-13
ES497209A0 (es) 1981-12-16
HU180334B (en) 1983-02-28
ATA134580A (de) 1981-11-15
FR2451363A1 (fr) 1980-10-10
CA1144926A (en) 1983-04-19
MX6219E (es) 1984-12-21
ES497208A0 (es) 1981-12-16
IL59557A (en) 1983-10-31
AT367395B (de) 1982-06-25
SU1022655A3 (ru) 1983-06-07
RO79906A (ro) 1982-10-11

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