FR3713M - Pyrimido [5,4-d] pyrimidines basiquement substituées. - Google Patents
Pyrimido [5,4-d] pyrimidines basiquement substituées.Info
- Publication number
- FR3713M FR3713M FR977447A FR977447A FR3713M FR 3713 M FR3713 M FR 3713M FR 977447 A FR977447 A FR 977447A FR 977447 A FR977447 A FR 977447A FR 3713 M FR3713 M FR 3713M
- Authority
- FR
- France
- Prior art keywords
- pyrimidines
- basically substituted
- substituted pyrimido
- pyrimido
- basically
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- JOZPEVMCAKXSEY-UHFFFAOYSA-N pyrimido[5,4-d]pyrimidine Chemical class N1=CN=CC2=NC=NC=C21 JOZPEVMCAKXSEY-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR977447A FR3713M (fr) | 1963-03-09 | 1964-06-08 | Pyrimido [5,4-d] pyrimidines basiquement substituées. |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DET0023605 | 1963-03-09 | ||
| FR966678A FR1543161A (fr) | 1963-03-09 | 1964-03-09 | Procédé de fabrication de pyrimido [5, 4-d]-pyrimidines basiquement substituées |
| FR977447A FR3713M (fr) | 1963-03-09 | 1964-06-08 | Pyrimido [5,4-d] pyrimidines basiquement substituées. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| FR3713M true FR3713M (fr) | 1965-11-29 |
Family
ID=7551073
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR977447A Expired FR3713M (fr) | 1963-03-09 | 1964-06-08 | Pyrimido [5,4-d] pyrimidines basiquement substituées. |
Country Status (5)
| Country | Link |
|---|---|
| CH (1) | CH438344A (fr) |
| DE (1) | DE1470341C3 (fr) |
| FR (1) | FR3713M (fr) |
| GB (1) | GB1051218A (fr) |
| IT (1) | IT7950418A0 (fr) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US12037346B2 (en) | 2021-04-13 | 2024-07-16 | Nuvalent, Inc. | Amino-substituted heteroaryls for treating cancers with EGFR mutations |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2004201A1 (de) * | 1970-01-30 | 1971-08-05 | Thomae Gmbh Dr K | Neue 2,6-Bis(dialkanolamino)-pyrimido-[5,4-d]pyrimidine und Verfahren zu ihrer Herstellung |
| DE3049207A1 (de) * | 1980-12-27 | 1982-07-29 | Dr. Karl Thomae Gmbh, 7950 Biberach | Neue trisubstituierte pyrimido (5,4-d) pyrimidine, ihre herstellung und ihre verwendung als arzneimittel |
| US7772188B2 (en) | 2003-01-28 | 2010-08-10 | Ironwood Pharmaceuticals, Inc. | Methods and compositions for the treatment of gastrointestinal disorders |
| RU2005136383A (ru) | 2003-04-24 | 2007-06-10 | БЕРИНГЕР ИНГЕЛЬХАЙМ ИНТЕРНАЦИОНАЛЬ ГмбХ (DE) | Применение дипиридамола или мопидамола для лечения и предупреждения тромбоэмболических заболеваний и нарушений, вызываемыхизбыточным образованием и/или повышенным уровнем экспрессии тромбиновых рецепторов |
| US8969514B2 (en) | 2007-06-04 | 2015-03-03 | Synergy Pharmaceuticals, Inc. | Agonists of guanylate cyclase useful for the treatment of hypercholesterolemia, atherosclerosis, coronary heart disease, gallstone, obesity and other cardiovascular diseases |
| MX354786B (es) | 2007-06-04 | 2018-03-21 | Synergy Pharmaceuticals Inc | Agonistas de guanilato ciclasa utiles para el tratamiento de trastornos gastrointestinales, inflamacion, cancer y otros trastornos. |
| CA2726917C (fr) | 2008-06-04 | 2018-06-26 | Synergy Pharmaceuticals Inc. | Agonistes de guanylate cyclase utile dans le traitement de troubles gastro-intestinaux, d'une inflammation, d'un cancer et d'autres troubles |
| EP2321341B1 (fr) | 2008-07-16 | 2017-02-22 | Synergy Pharmaceuticals Inc. | Agonistes de guanylate cyclase utiles pour le traitement de troubles gastro-intestinaux, inflammatoires, cancéreux et autres |
| US9616097B2 (en) | 2010-09-15 | 2017-04-11 | Synergy Pharmaceuticals, Inc. | Formulations of guanylate cyclase C agonists and methods of use |
| EA201391254A1 (ru) | 2011-03-01 | 2014-02-28 | Синерджи Фармасьютикалз Инк. | Способ получения агонистов гуанилатциклазы c |
| JP6499591B2 (ja) | 2013-02-25 | 2019-04-10 | シナジー ファーマシューティカルズ インコーポレイテッド | 結腸洗浄において用いるためのグアニル酸シクラーゼ受容体アゴニスト |
| WO2014151200A2 (fr) | 2013-03-15 | 2014-09-25 | Synergy Pharmaceuticals Inc. | Compositions utiles pour le traitement de troubles gastro-intestinaux |
| JP2016514671A (ja) | 2013-03-15 | 2016-05-23 | シナジー ファーマシューティカルズ インコーポレイテッド | グアニル酸シクラーゼのアゴニストおよびその使用 |
| CN105764916B (zh) | 2013-06-05 | 2021-05-18 | 博士医疗爱尔兰有限公司 | 鸟苷酸环化酶c的超纯激动剂、制备和使用所述激动剂的方法 |
| EP3492106B1 (fr) | 2013-08-09 | 2021-02-17 | Ardelyx, Inc. | Composés et procédés d'inhibition du transport de phosphate |
| EP3972599B1 (fr) | 2019-05-21 | 2025-10-22 | Ardelyx, Inc. | Combinaison pour baisser le phosphate sérique chez un patient |
-
0
- GB GB1051218D patent/GB1051218A/en active Active
-
1963
- 1963-03-09 DE DE1470341A patent/DE1470341C3/de not_active Expired
-
1964
- 1964-02-28 CH CH247764A patent/CH438344A/de unknown
- 1964-06-08 FR FR977447A patent/FR3713M/fr not_active Expired
-
1979
- 1979-10-01 IT IT7950418A patent/IT7950418A0/it unknown
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US12037346B2 (en) | 2021-04-13 | 2024-07-16 | Nuvalent, Inc. | Amino-substituted heteroaryls for treating cancers with EGFR mutations |
Also Published As
| Publication number | Publication date |
|---|---|
| DE1470341C3 (de) | 1974-07-04 |
| DE1470341B2 (de) | 1973-12-06 |
| CH438344A (de) | 1967-06-30 |
| DE1470341A1 (de) | 1969-07-03 |
| IT7950418A0 (it) | 1979-10-01 |
| GB1051218A (fr) |
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