FR3713M - Pyrimido [5,4-d] pyrimidines basiquement substituées. - Google Patents

Pyrimido [5,4-d] pyrimidines basiquement substituées.

Info

Publication number
FR3713M
FR3713M FR977447A FR977447A FR3713M FR 3713 M FR3713 M FR 3713M FR 977447 A FR977447 A FR 977447A FR 977447 A FR977447 A FR 977447A FR 3713 M FR3713 M FR 3713M
Authority
FR
France
Prior art keywords
pyrimidines
basically substituted
substituted pyrimido
pyrimido
basically
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
FR977447A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim Pharma GmbH and Co KG
Original Assignee
Dr Karl Thomae GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR966678A external-priority patent/FR1543161A/fr
Application filed by Dr Karl Thomae GmbH filed Critical Dr Karl Thomae GmbH
Priority to FR977447A priority Critical patent/FR3713M/fr
Application granted granted Critical
Publication of FR3713M publication Critical patent/FR3713M/fr
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
FR977447A 1963-03-09 1964-06-08 Pyrimido [5,4-d] pyrimidines basiquement substituées. Expired FR3713M (fr)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FR977447A FR3713M (fr) 1963-03-09 1964-06-08 Pyrimido [5,4-d] pyrimidines basiquement substituées.

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DET0023605 1963-03-09
FR966678A FR1543161A (fr) 1963-03-09 1964-03-09 Procédé de fabrication de pyrimido [5, 4-d]-pyrimidines basiquement substituées
FR977447A FR3713M (fr) 1963-03-09 1964-06-08 Pyrimido [5,4-d] pyrimidines basiquement substituées.

Publications (1)

Publication Number Publication Date
FR3713M true FR3713M (fr) 1965-11-29

Family

ID=7551073

Family Applications (1)

Application Number Title Priority Date Filing Date
FR977447A Expired FR3713M (fr) 1963-03-09 1964-06-08 Pyrimido [5,4-d] pyrimidines basiquement substituées.

Country Status (5)

Country Link
CH (1) CH438344A (fr)
DE (1) DE1470341C3 (fr)
FR (1) FR3713M (fr)
GB (1) GB1051218A (fr)
IT (1) IT7950418A0 (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US12037346B2 (en) 2021-04-13 2024-07-16 Nuvalent, Inc. Amino-substituted heteroaryls for treating cancers with EGFR mutations

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2004201A1 (de) * 1970-01-30 1971-08-05 Thomae Gmbh Dr K Neue 2,6-Bis(dialkanolamino)-pyrimido-[5,4-d]pyrimidine und Verfahren zu ihrer Herstellung
DE3049207A1 (de) * 1980-12-27 1982-07-29 Dr. Karl Thomae Gmbh, 7950 Biberach Neue trisubstituierte pyrimido (5,4-d) pyrimidine, ihre herstellung und ihre verwendung als arzneimittel
US7772188B2 (en) 2003-01-28 2010-08-10 Ironwood Pharmaceuticals, Inc. Methods and compositions for the treatment of gastrointestinal disorders
RU2005136383A (ru) 2003-04-24 2007-06-10 БЕРИНГЕР ИНГЕЛЬХАЙМ ИНТЕРНАЦИОНАЛЬ ГмбХ (DE) Применение дипиридамола или мопидамола для лечения и предупреждения тромбоэмболических заболеваний и нарушений, вызываемыхизбыточным образованием и/или повышенным уровнем экспрессии тромбиновых рецепторов
US8969514B2 (en) 2007-06-04 2015-03-03 Synergy Pharmaceuticals, Inc. Agonists of guanylate cyclase useful for the treatment of hypercholesterolemia, atherosclerosis, coronary heart disease, gallstone, obesity and other cardiovascular diseases
MX354786B (es) 2007-06-04 2018-03-21 Synergy Pharmaceuticals Inc Agonistas de guanilato ciclasa utiles para el tratamiento de trastornos gastrointestinales, inflamacion, cancer y otros trastornos.
CA2726917C (fr) 2008-06-04 2018-06-26 Synergy Pharmaceuticals Inc. Agonistes de guanylate cyclase utile dans le traitement de troubles gastro-intestinaux, d'une inflammation, d'un cancer et d'autres troubles
EP2321341B1 (fr) 2008-07-16 2017-02-22 Synergy Pharmaceuticals Inc. Agonistes de guanylate cyclase utiles pour le traitement de troubles gastro-intestinaux, inflammatoires, cancéreux et autres
US9616097B2 (en) 2010-09-15 2017-04-11 Synergy Pharmaceuticals, Inc. Formulations of guanylate cyclase C agonists and methods of use
EA201391254A1 (ru) 2011-03-01 2014-02-28 Синерджи Фармасьютикалз Инк. Способ получения агонистов гуанилатциклазы c
JP6499591B2 (ja) 2013-02-25 2019-04-10 シナジー ファーマシューティカルズ インコーポレイテッド 結腸洗浄において用いるためのグアニル酸シクラーゼ受容体アゴニスト
WO2014151200A2 (fr) 2013-03-15 2014-09-25 Synergy Pharmaceuticals Inc. Compositions utiles pour le traitement de troubles gastro-intestinaux
JP2016514671A (ja) 2013-03-15 2016-05-23 シナジー ファーマシューティカルズ インコーポレイテッド グアニル酸シクラーゼのアゴニストおよびその使用
CN105764916B (zh) 2013-06-05 2021-05-18 博士医疗爱尔兰有限公司 鸟苷酸环化酶c的超纯激动剂、制备和使用所述激动剂的方法
EP3492106B1 (fr) 2013-08-09 2021-02-17 Ardelyx, Inc. Composés et procédés d'inhibition du transport de phosphate
EP3972599B1 (fr) 2019-05-21 2025-10-22 Ardelyx, Inc. Combinaison pour baisser le phosphate sérique chez un patient

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US12037346B2 (en) 2021-04-13 2024-07-16 Nuvalent, Inc. Amino-substituted heteroaryls for treating cancers with EGFR mutations

Also Published As

Publication number Publication date
DE1470341C3 (de) 1974-07-04
DE1470341B2 (de) 1973-12-06
CH438344A (de) 1967-06-30
DE1470341A1 (de) 1969-07-03
IT7950418A0 (it) 1979-10-01
GB1051218A (fr)

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