HRP930227A2 - Indoles - Google Patents

Indoles Download PDF

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Publication number
HRP930227A2
HRP930227A2 HR9204365.2A HRP930227A HRP930227A2 HR P930227 A2 HRP930227 A2 HR P930227A2 HR P930227 A HRP930227 A HR P930227A HR P930227 A2 HRP930227 A2 HR P930227A2
Authority
HR
Croatia
Prior art keywords
formula
compound
alkyl
image
phenyl
Prior art date
Application number
HR9204365.2A
Other languages
English (en)
Croatian (hr)
Inventor
Julian Blagg
Colin William Greengrass
Paul William Finn
Graham Nigel Maw
Original Assignee
Julian Blagg
Colin William Greengrass
Paul William Finn
Graham Nigel Maw
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Julian Blagg, Colin William Greengrass, Paul William Finn, Graham Nigel Maw filed Critical Julian Blagg
Publication of HRP930227A2 publication Critical patent/HRP930227A2/hr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Steroid Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
HR9204365.2A 1992-02-28 1993-02-24 Indoles HRP930227A2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB929204365A GB9204365D0 (en) 1992-02-28 1992-02-28 Indoles

Publications (1)

Publication Number Publication Date
HRP930227A2 true HRP930227A2 (en) 1996-10-31

Family

ID=10711259

Family Applications (1)

Application Number Title Priority Date Filing Date
HR9204365.2A HRP930227A2 (en) 1992-02-28 1993-02-24 Indoles

Country Status (24)

Country Link
US (1) US5767139A (da)
EP (1) EP0628040B1 (da)
JP (1) JP2540016B2 (da)
KR (1) KR950700287A (da)
CN (1) CN1079465A (da)
AT (1) ATE164376T1 (da)
AU (1) AU3497793A (da)
BR (1) BR9305991A (da)
CA (1) CA2117610C (da)
CZ (1) CZ207794A3 (da)
DE (1) DE69317651T2 (da)
DK (1) DK0628040T3 (da)
ES (1) ES2115053T3 (da)
FI (2) FI943931A0 (da)
GB (1) GB9204365D0 (da)
HR (1) HRP930227A2 (da)
HU (1) HUT71126A (da)
IL (1) IL104816A0 (da)
MX (1) MX9301112A (da)
NO (1) NO943187L (da)
RU (1) RU94042391A (da)
SK (1) SK100894A3 (da)
WO (1) WO1993017014A1 (da)
ZA (1) ZA931383B (da)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL109728A0 (en) * 1993-05-28 1994-08-26 Pfizer Res & Dev Indoles
ES2099007B1 (es) * 1993-07-16 1997-12-01 Pfizer Res & Dev Derivados de indol.
GB9317096D0 (en) * 1993-08-17 1993-09-29 Pfizer Ltd Indoles
GB9403516D0 (en) * 1994-02-24 1994-04-13 Pfizer Ltd Indoles
GB9409583D0 (en) * 1994-05-13 1994-07-06 Pfizer Ltd Indoles
EP0820441B1 (en) * 1995-04-10 2002-06-26 Fujisawa Pharmaceutical Co., Ltd. INDOLE DERIVATIVES AS cGMP-PDE INHIBITORS
CA2338855A1 (en) 1998-08-03 2000-02-17 Eli Lilly And Company Indole spla2 inhibitors
FR2796274B1 (fr) * 1999-07-16 2001-09-21 Oreal Utilisation de l'acide 4,6-dimethoxy-indole 2-carboxylique ou de ses derives pour stimuler ou induire la pousse des cheveux et/ou stopper leur chute
FR2796279B1 (fr) 1999-07-16 2001-09-21 Oreal Utilisation de l'acide 4,6-dimethoxy-indole 2-carboxylique ou de ses derives pour le traitement de la seborrhee
UA79504C2 (en) * 2002-11-07 2007-06-25 Organon Nv Indols for treating diseases associated with androgen receptors
HRP20050396A2 (en) * 2002-11-07 2005-06-30 Akzo Nobel N.V. Indoles useful in the treatment of androgen-receptor related diseases
TW200602317A (en) 2004-04-23 2006-01-16 Akzo Nobel Nv Novel androgens
GB201102913D0 (en) 2011-02-18 2011-04-06 Univ Birmingham Novel therapeutic

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3557142A (en) * 1968-02-20 1971-01-19 Sterling Drug Inc 4,5,6,7-tetrahydro-indole-lower-alkanoic acids and esters
PH23498A (en) * 1984-08-06 1989-08-16 Sterling Drug Inc 3-carbonyl-1-aminoalkyl-1h-indoles,composition and use thereof
CA2036307C (en) * 1990-03-08 2002-07-09 Susan Jean Ward 3-arylcarbonyl-1-aminoalkyl-1h-indole-containing antiglaucoma compositions and method
GB9011335D0 (en) * 1990-05-21 1990-07-11 Fujisawa Pharmaceutical Co Indolebutyric acid derivatives and process for preparation thereof
IL109728A0 (en) * 1993-05-28 1994-08-26 Pfizer Res & Dev Indoles

Also Published As

Publication number Publication date
NO943187L (no) 1994-09-13
FI20001771A7 (fi) 2000-08-09
KR950700287A (ko) 1995-01-16
EP0628040A1 (en) 1994-12-14
AU3497793A (en) 1993-09-13
BR9305991A (pt) 1997-10-21
CZ207794A3 (en) 1995-01-18
CA2117610C (en) 2000-07-18
WO1993017014A1 (en) 1993-09-02
JP2540016B2 (ja) 1996-10-02
ATE164376T1 (de) 1998-04-15
US5767139A (en) 1998-06-16
ES2115053T3 (es) 1998-06-16
FI943931A7 (fi) 1994-08-26
GB9204365D0 (en) 1992-04-08
MX9301112A (es) 1994-07-29
DE69317651D1 (en) 1998-04-30
NO943187D0 (no) 1994-08-29
CN1079465A (zh) 1993-12-15
EP0628040B1 (en) 1998-03-25
RU94042391A (ru) 1996-08-10
DE69317651T2 (de) 1998-07-09
DK0628040T3 (da) 1998-04-27
HU9402466D0 (en) 1994-10-28
FI943931A0 (fi) 1994-08-26
ZA931383B (en) 1994-08-26
JPH07500347A (ja) 1995-01-12
HUT71126A (en) 1995-11-28
CA2117610A1 (en) 1993-09-02
IL104816A0 (en) 1993-06-10
SK100894A3 (en) 1995-04-12

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Legal Events

Date Code Title Description
A1OB Publication of a patent application
AIPI Request for the grant of a patent on the basis of a substantive examination of a patent application
OBST Application withdrawn