ID19406A - Keaktifan anti bakterial yang memiliki ketolida 6-0-tersubstitusi - Google Patents

Keaktifan anti bakterial yang memiliki ketolida 6-0-tersubstitusi

Info

Publication number: ID19406A
Authority: ID; Indonesia
Prior art keywords: alkyl; substituted; heteroaryl; aryl; optionally substituted
Prior art date: 1996-09-04

Application number

IDP973095A

Other languages

English (en)

Indonesian (id)

Inventor

Yat Sun Or

Daniel T Chu

Zhenkun Ma

Jacob J Plattner

Richard F Clark

Original Assignee

Abbott Lab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-09-04

Filing date

1997-09-04

Publication date

1998-07-09

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27107953&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ID19406(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1997-07-03 Priority claimed from US08/888,350 external-priority patent/US5866549A/en

1997-09-04 Application filed by Abbott Lab filed Critical Abbott Lab

1998-07-09 Publication of ID19406A publication Critical patent/ID19406A/id

Links

230000000844 anti-bacterial effect Effects 0.000 title 1
125000000217 alkyl group Chemical group 0.000 abstract 18
125000001072 heteroaryl group Chemical group 0.000 abstract 8
125000003118 aryl group Chemical group 0.000 abstract 4
125000003107 substituted aryl group Chemical group 0.000 abstract 4
125000000753 cycloalkyl group Chemical group 0.000 abstract 3
-1 CO2R10 Inorganic materials 0.000 abstract 2
125000003342 alkenyl group Chemical group 0.000 abstract 2
125000006367 bivalent amino carbonyl group Chemical group [H]N([*:1])C([*:2])=O 0.000 abstract 2
125000006297 carbonyl amino group Chemical group [H]N([*:2])C([*:1])=O 0.000 abstract 2
HCUOEKSZWPGJIM-YBRHCDHNSA-N (e,2e)-2-hydroxyimino-6-methoxy-4-methyl-5-nitrohex-3-enamide Chemical compound COCC([N+]([O-])=O)\C(C)=C\C(=N/O)\C(N)=O HCUOEKSZWPGJIM-YBRHCDHNSA-N 0.000 abstract 1
101100134929 Gallus gallus COR9 gene Proteins 0.000 abstract 1
101001109689 Homo sapiens Nuclear receptor subfamily 4 group A member 3 Proteins 0.000 abstract 1
101000598778 Homo sapiens Protein OSCP1 Proteins 0.000 abstract 1
101001067395 Mus musculus Phospholipid scramblase 1 Proteins 0.000 abstract 1
102100022673 Nuclear receptor subfamily 4 group A member 3 Human genes 0.000 abstract 1
125000000304 alkynyl group Chemical group 0.000 abstract 1
125000004429 atom Chemical group 0.000 abstract 1
150000002148 esters Chemical class 0.000 abstract 1
125000001475 halogen functional group Chemical group 0.000 abstract 1
125000000592 heterocycloalkyl group Chemical group 0.000 abstract 1
125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
239000003835 ketolide antibiotic agent Substances 0.000 abstract 1
125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
229940002612 prodrug Drugs 0.000 abstract 1
239000000651 prodrug Substances 0.000 abstract 1
125000006239 protecting group Chemical group 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1
125000001424 substituent group Chemical group 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H1/00—Processes for the preparation of sugar derivatives
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Molecular Biology (AREA)
Genetics & Genomics (AREA)
Biotechnology (AREA)
Biochemistry (AREA)
Engineering & Computer Science (AREA)
Veterinary Medicine (AREA)
Communicable Diseases (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Medicinal Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Oncology (AREA)
Animal Behavior & Ethology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Saccharide Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Cephalosporin Compounds (AREA)
Food Preservation Except Freezing, Refrigeration, And Drying (AREA)
Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Plural Heterocyclic Compounds (AREA)

IDP973095A 1996-09-04 1997-09-04 Keaktifan anti bakterial yang memiliki ketolida 6-0-tersubstitusi ID19406A (id)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US70777696A	1996-09-04	1996-09-04
US08/888,350 US5866549A (en)	1996-09-04	1997-07-03	6-O-substituted ketolides having antibacterial activity

Publications (1)

Publication Number	Publication Date
ID19406A true ID19406A (id)	1998-07-09

Family

ID=27107953

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IDP973095A ID19406A (id)	1996-09-04	1997-09-04	Keaktifan anti bakterial yang memiliki ketolida 6-0-tersubstitusi

Country Status (27)

Country	Link
US (4)	US6147197A (es)
EP (5)	EP1291352B1 (es)
JP (1)	JP4597274B2 (es)
KR (5)	KR20050044816A (es)
CN (4)	CN100460415C (es)
AT (5)	ATE296832T1 (es)
BG (1)	BG63547B1 (es)
BR (1)	BR9711661A (es)
CA (1)	CA2263972C (es)
CZ (1)	CZ300106B6 (es)
DE (5)	DE69733723T2 (es)
DK (5)	DK0929563T3 (es)
ES (5)	ES2242813T3 (es)
HR (5)	HRP970473B1 (es)
HU (1)	HU230166B1 (es)
ID (1)	ID19406A (es)
IL (1)	IL128681A0 (es)
NO (1)	NO314230B1 (es)
NZ (1)	NZ334274A (es)
PL (1)	PL188173B1 (es)
PT (5)	PT1291350E (es)
RO (1)	RO121473B1 (es)
RU (1)	RU2192427C2 (es)
SI (1)	SI20023B (es)
SK (5)	SK285533B6 (es)
TR (1)	TR199901127T2 (es)
WO (1)	WO1998009978A1 (es)

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US6171807B1 (en) *	1996-11-13	2001-01-09	Associates Of Cape Cod, Inc.	Detection and quantitation of endotoxin by fluorescence polarization

1997
- 1997-09-02 DE DE69733723T patent/DE69733723T2/de not_active Expired - Lifetime
- 1997-09-02 TR TR1999/01127T patent/TR199901127T2/xx unknown
- 1997-09-02 CN CNB2005100674132A patent/CN100460415C/zh not_active Expired - Lifetime
- 1997-09-02 ES ES02024560T patent/ES2242813T3/es not_active Expired - Lifetime
- 1997-09-02 AT AT02024560T patent/ATE296832T1/de active
- 1997-09-02 EP EP02024559A patent/EP1291352B1/en not_active Expired - Lifetime
- 1997-09-02 SK SK286-99A patent/SK285533B6/sk not_active IP Right Cessation
- 1997-09-02 PL PL97332009A patent/PL188173B1/pl unknown
- 1997-09-02 ES ES97939765T patent/ES2242983T3/es not_active Expired - Lifetime
- 1997-09-02 BR BR9711661A patent/BR9711661A/pt not_active IP Right Cessation
- 1997-09-02 DK DK97939765T patent/DK0929563T3/da active
- 1997-09-02 CA CA002263972A patent/CA2263972C/en not_active Expired - Lifetime
- 1997-09-02 EP EP02024560A patent/EP1291353B1/en not_active Expired - Lifetime
- 1997-09-02 PT PT02024557T patent/PT1291350E/pt unknown
- 1997-09-02 PT PT02024559T patent/PT1291352E/pt unknown
- 1997-09-02 DE DE69733370T patent/DE69733370T2/de not_active Expired - Lifetime
- 1997-09-02 NZ NZ334274A patent/NZ334274A/en not_active IP Right Cessation
- 1997-09-02 KR KR1020057007118A patent/KR20050044816A/ko not_active Ceased
- 1997-09-02 WO PCT/US1997/015506 patent/WO1998009978A1/en not_active Ceased
- 1997-09-02 DE DE69733369T patent/DE69733369T2/de not_active Expired - Lifetime
- 1997-09-02 ES ES02024559T patent/ES2242812T3/es not_active Expired - Lifetime
- 1997-09-02 HU HU9902869A patent/HU230166B1/hu unknown
- 1997-09-02 SK SK5085-2006A patent/SK285536B6/sk not_active IP Right Cessation
- 1997-09-02 EP EP97939765A patent/EP0929563B1/en not_active Expired - Lifetime
- 1997-09-02 CZ CZ0068599A patent/CZ300106B6/cs not_active IP Right Cessation
- 1997-09-02 AT AT02024559T patent/ATE296308T1/de active
- 1997-09-02 AT AT97939765T patent/ATE296831T1/de active
- 1997-09-02 RU RU99106778/04A patent/RU2192427C2/ru active
- 1997-09-02 SK SK5083-2006A patent/SK285534B6/sk not_active IP Right Cessation
- 1997-09-02 SK SK5086-2006A patent/SK286181B6/sk not_active IP Right Cessation
- 1997-09-02 CN CNA2005100674147A patent/CN1680419A/zh active Pending
- 1997-09-02 DK DK02024558T patent/DK1291351T3/da active
- 1997-09-02 KR KR1020057007119A patent/KR100610043B1/ko not_active Expired - Lifetime
- 1997-09-02 ES ES02024557T patent/ES2242811T3/es not_active Expired - Lifetime
- 1997-09-02 CN CNB971993343A patent/CN1273475C/zh not_active Expired - Lifetime
- 1997-09-02 CN CNB2005100674151A patent/CN100441591C/zh not_active Expired - Lifetime
- 1997-09-02 PT PT02024560T patent/PT1291353E/pt unknown
- 1997-09-02 AT AT02024558T patent/ATE299508T1/de active
- 1997-09-02 DE DE69733422T patent/DE69733422T2/de not_active Expired - Lifetime
- 1997-09-02 EP EP02024558A patent/EP1291351B1/en not_active Expired - Lifetime
- 1997-09-02 IL IL12868197A patent/IL128681A0/xx not_active IP Right Cessation
- 1997-09-02 AT AT02024557T patent/ATE296307T1/de active
- 1997-09-02 DK DK02024560T patent/DK1291353T3/da active
- 1997-09-02 PT PT97939765T patent/PT929563E/pt unknown
- 1997-09-02 ES ES02024558T patent/ES2244716T3/es not_active Expired - Lifetime
- 1997-09-02 KR KR1020057007115A patent/KR100568455B1/ko not_active Expired - Lifetime
- 1997-09-02 RO RO99-00228A patent/RO121473B1/ro unknown
- 1997-09-02 PT PT02024558T patent/PT1291351E/pt unknown
- 1997-09-02 DE DE69733439T patent/DE69733439T2/de not_active Expired - Lifetime
- 1997-09-02 SI SI9720062A patent/SI20023B/sl unknown
- 1997-09-02 DK DK02024557T patent/DK1291350T3/da active
- 1997-09-02 JP JP51285898A patent/JP4597274B2/ja not_active Expired - Lifetime
- 1997-09-02 DK DK02024559T patent/DK1291352T3/da active
- 1997-09-02 EP EP02024557A patent/EP1291350B1/en not_active Expired - Lifetime
- 1997-09-02 KR KR1020057007117A patent/KR100576988B1/ko not_active Expired - Lifetime
- 1997-09-02 KR KR10-1999-7001803A patent/KR100523679B1/ko not_active Expired - Lifetime
- 1997-09-02 SK SK5084-2006A patent/SK285535B6/sk not_active IP Right Cessation
- 1997-09-03 HR HR970473A patent/HRP970473B1/xx not_active IP Right Cessation
- 1997-09-04 ID IDP973095A patent/ID19406A/id unknown
1998
- 1998-11-04 US US09/185,903 patent/US6147197A/en not_active Expired - Lifetime
- 1998-11-04 US US09/186,395 patent/US6028181A/en not_active Expired - Lifetime
- 1998-11-04 US US09/185,883 patent/US6075133A/en not_active Expired - Lifetime
1999
- 1999-03-02 NO NO19991022A patent/NO314230B1/no not_active IP Right Cessation
- 1999-03-26 BG BG103292A patent/BG63547B1/bg unknown
2004
- 2004-01-06 US US10/752,483 patent/USRE39591E1/en not_active Expired - Lifetime
2006
- 2006-08-11 HR HRP20060277AA patent/HRP20060277B1/hr not_active IP Right Cessation
- 2006-08-11 HR HRP20060278AA patent/HRP20060278B1/hr not_active IP Right Cessation
- 2006-08-11 HR HRP20060275AA patent/HRP20060275B1/hr not_active IP Right Cessation
- 2006-08-11 HR HRP20060276AA patent/HRP20060276B1/hr not_active IP Right Cessation

Also Published As

Publication number	Publication date
AU4178097A (en)	1998-03-26
HK1021537A1 (en)	2000-06-16
EP1291351A1 (en)	2003-03-12
BG103292A (en)	1999-12-30
EP1291352A1 (en)	2003-03-12
CZ68599A3 (cs)	1999-08-11
HUP9902869A3 (en)	2001-04-28
SK28699A3 (en)	2000-03-13
DK1291352T3 (da)	2005-09-19
EP1291351B1 (en)	2005-07-13
DE69733422T2 (de)	2006-05-04
AU729348B2 (en)	2001-02-01
CN1273475C (zh)	2006-09-06
EP1291353A1 (en)	2003-03-12
RO121473B1 (ro)	2007-06-29
US6147197A (en)	2000-11-14
BG63547B1 (bg)	2002-04-30
CN1237183A (zh)	1999-12-01
ES2242813T3 (es)	2005-11-16
KR100576988B1 (ko)	2006-05-10
PL332009A1 (en)	1999-08-16
HU230166B1 (hu)	2015-09-28
CA2263972A1 (en)	1998-03-12
HRP20060277B1 (hr)	2014-04-11
DE69733439D1 (de)	2005-07-07
NO314230B1 (no)	2003-02-17
JP4597274B2 (ja)	2010-12-15
PL188173B1 (pl)	2004-12-31
US6075133A (en)	2000-06-13
HRP970473B1 (en)	2007-02-28
NO991022L (no)	1999-05-03
HRP20060277A2 (en)	2007-10-31
WO1998009978A1 (en)	1998-03-12
PT1291351E (pt)	2005-11-30
TR199901127T2 (xx)	1999-07-21
EP1291353B1 (en)	2005-06-01
DK1291351T3 (da)	2005-10-24
SI20023A (sl)	2000-02-29
ATE296307T1 (de)	2005-06-15
CN100460415C (zh)	2009-02-11
KR20050044816A (ko)	2005-05-12
EP1291350B1 (en)	2005-05-25
HRP20060276B1 (hr)	2014-04-25
HRP20060278A2 (en)	2007-10-31
PT1291350E (pt)	2005-09-30
CN1680420A (zh)	2005-10-12
PT929563E (pt)	2005-10-31
SI20023B (en)	2001-02-28
DE69733422D1 (de)	2005-07-07
CN1680418A (zh)	2005-10-12
ATE296308T1 (de)	2005-06-15
ATE296832T1 (de)	2005-06-15
HRP20060276A2 (en)	2007-10-31
ES2244716T3 (es)	2005-12-16
CN100441591C (zh)	2008-12-10
DE69733369D1 (de)	2005-06-30
SK285535B6 (sk)	2007-03-01
KR20050043994A (ko)	2005-05-11
EP1291350A1 (en)	2003-03-12
KR100610043B1 (ko)	2006-08-08
ATE299508T1 (de)	2005-07-15
PT1291352E (pt)	2005-09-30
CZ300106B6 (cs)	2009-02-11
EP0929563B1 (en)	2005-06-01
HRP20060275B1 (hr)	2014-04-11
ES2242811T3 (es)	2005-11-16
DE69733439T2 (de)	2006-05-04
KR20050044815A (ko)	2005-05-12
KR100523679B1 (ko)	2005-10-26
KR100568455B1 (ko)	2006-04-07
NZ334274A (en)	2001-02-23
EP0929563A1 (en)	1999-07-21
DK1291350T3 (da)	2005-09-26
US6028181A (en)	2000-02-22
KR20000068435A (ko)	2000-11-25
USRE39591E1 (en)	2007-04-24
DE69733369T2 (de)	2006-01-26
SK285536B6 (sk)	2007-03-01
SK285534B6 (sk)	2007-03-01
SK285533B6 (sk)	2007-03-01
IL128681A0 (en)	2000-01-31
DK1291353T3 (da)	2005-10-03
CA2263972C (en)	2008-01-29
JP2001500855A (ja)	2001-01-23
HRP970473A2 (en)	1998-08-31
BR9711661A (pt)	1999-08-24
DE69733723T2 (de)	2006-04-20
RU2192427C2 (ru)	2002-11-10
CN1680419A (zh)	2005-10-12
DE69733370D1 (de)	2005-06-30
NO991022D0 (no)	1999-03-02
KR20050043993A (ko)	2005-05-11
ATE296831T1 (de)	2005-06-15
ES2242983T3 (es)	2005-11-16
DE69733370T2 (de)	2006-02-02
ES2242812T3 (es)	2005-11-16
HRP20060275A2 (en)	2007-10-31
PT1291353E (pt)	2005-10-31
HUP9902869A2 (hu)	2000-02-28
DE69733723D1 (de)	2005-08-18
EP1291352B1 (en)	2005-05-25
HRP20060278B1 (hr)	2014-04-11
DK0929563T3 (da)	2005-10-03
SK286181B6 (sk)	2008-04-07

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