ID28740A - SENYAWA-SENYAWA SEFEM YANG MENGANDUNG IMIDAZO [4,5-b] PIRIDINIUMMETIL YANG MEMPUNYAI SPEKTRUM ANTIBAKTERI YANG LUAS - Google Patents

SENYAWA-SENYAWA SEFEM YANG MENGANDUNG IMIDAZO [4,5-b] PIRIDINIUMMETIL YANG MEMPUNYAI SPEKTRUM ANTIBAKTERI YANG LUAS

Info

Publication number
ID28740A
ID28740A IDW00200100967A ID20010967A ID28740A ID 28740 A ID28740 A ID 28740A ID W00200100967 A IDW00200100967 A ID W00200100967A ID 20010967 A ID20010967 A ID 20010967A ID 28740 A ID28740 A ID 28740A
Authority
ID
Indonesia
Prior art keywords
hydrogen
antibacterial spectrum
pyridiniummetyl
sefem
optionally substituted
Prior art date
Application number
IDW00200100967A
Other languages
English (en)
Inventor
Yasuhiro Nishitani
Hikaru Itani
Tadashi Irie
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi & Co filed Critical Shionogi & Co
Publication of ID28740A publication Critical patent/ID28740A/id

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/48—Methylene radicals, substituted by hetero rings
    • C07D501/56—Methylene radicals, substituted by hetero rings with the 7-amino radical acylated by carboxylic acids containing hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Cephalosporin Compounds (AREA)
IDW00200100967A 1998-11-27 1999-11-25 SENYAWA-SENYAWA SEFEM YANG MENGANDUNG IMIDAZO [4,5-b] PIRIDINIUMMETIL YANG MEMPUNYAI SPEKTRUM ANTIBAKTERI YANG LUAS ID28740A (id)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP33670798 1998-11-27

Publications (1)

Publication Number Publication Date
ID28740A true ID28740A (id) 2001-06-28

Family

ID=18301969

Family Applications (1)

Application Number Title Priority Date Filing Date
IDW00200100967A ID28740A (id) 1998-11-27 1999-11-25 SENYAWA-SENYAWA SEFEM YANG MENGANDUNG IMIDAZO [4,5-b] PIRIDINIUMMETIL YANG MEMPUNYAI SPEKTRUM ANTIBAKTERI YANG LUAS

Country Status (23)

Country Link
US (2) US6518263B1 (id)
EP (1) EP1134222B1 (id)
JP (1) JP3636663B2 (id)
KR (1) KR100692169B1 (id)
CN (1) CN100436456C (id)
AT (1) ATE293114T1 (id)
AU (1) AU758662B2 (id)
BR (1) BR9915743A (id)
CA (1) CA2350905C (id)
CZ (1) CZ20011719A3 (id)
DE (1) DE69924751T2 (id)
ES (1) ES2241374T3 (id)
HU (1) HUP0200450A3 (id)
ID (1) ID28740A (id)
IL (1) IL143314A0 (id)
NO (1) NO20012554L (id)
NZ (1) NZ511619A (id)
PL (1) PL347897A1 (id)
RU (1) RU2223964C2 (id)
TR (1) TR200101507T2 (id)
TW (1) TW526202B (id)
WO (1) WO2000032606A1 (id)
ZA (1) ZA200103850B (id)

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AU2003264462A1 (en) * 2002-09-20 2004-04-08 Shionogi And Co., Ltd. Process for the preparation of cephems
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CN1922190A (zh) * 2004-03-05 2007-02-28 盐野义制药株式会社 3－吡啶甲基头胞化合物
CA2568914C (en) * 2004-06-04 2013-09-24 Affinium Pharmaceuticals, Inc. Therapeutic agents, and methods of making and using the same
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EP2687533B1 (en) 2006-07-20 2017-07-19 Debiopharm International SA Acrylamide derivatives as FAB I inhibitors
US8263613B2 (en) * 2007-02-16 2012-09-11 Affinium Pharmaceuticals, Inc. Salts, prodrugs and polymorphs of fab I inhibitors
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CN102443017B (zh) * 2010-10-13 2014-10-29 石药集团中奇制药技术（石家庄）有限公司 一种盐酸头孢唑兰的制备方法
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SMT201900411T1 (it) 2012-06-19 2019-09-09 Debiopharm Int Sa Derivati di profaramci di (e)-n-metil-n-((3-metilbenzofuran-2-il)metil -3-(7-osso-5,6,7,8-tetraidro-1,8-naftiridin-3-il)acrilammide
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US8476425B1 (en) 2012-09-27 2013-07-02 Cubist Pharmaceuticals, Inc. Tazobactam arginine compositions
HUE043853T2 (hu) 2012-10-12 2019-09-30 Broad Inst Inc GSK3 inhibitorok és eljárások azok alkalmazására
US20140274996A1 (en) 2013-03-15 2014-09-18 Cubist Pharmaceuticals, Inc. Tazobactam and ceftolozane antibiotic compositions
PE20160048A1 (es) 2013-03-15 2016-02-12 Merck Sharp & Dohme Composiciones antibioticas de ceftolozano
US9872906B2 (en) 2013-03-15 2018-01-23 Merck Sharp & Dohme Corp. Ceftolozane antibiotic compositions
WO2015035376A2 (en) 2013-09-09 2015-03-12 Calixa Therapeutics, Inc. Treating infections with ceftolozane/tazobactam in subjects having impaired renal function
US8906898B1 (en) 2013-09-27 2014-12-09 Calixa Therapeutics, Inc. Solid forms of ceftolozane
CN107787324B (zh) * 2015-06-29 2020-05-19 桑多斯股份公司 氨甲酰基氨基吡唑衍生物的制备方法
WO2017096472A1 (en) * 2015-12-10 2017-06-15 Naeja-Rgm Pharmaceuticals Inc. Cephem compounds, their production and use
BR122023021456A2 (pt) 2016-02-26 2024-02-20 Debiopharm International S.A. Uso de di-hidrogeno fosfato de {6- [(e)-3-{metil[(3-metil-1-benfofuran-2- iol)metil]amino)-3- oxopro-1-en-1-il]-2-oxo-3,4-di-hidro-1,8-naftiridin-1(2h)- il}metila para tratamento de osteomielite do pé diabético e composição farmacêutica
WO2018187630A1 (en) 2017-04-05 2018-10-11 The Broad Institute, Inc. Tricyclic compounds as glycogen synthase kinase 3 (gsk3) inhibitors and uses thereof
FI3923914T3 (fi) 2019-02-14 2023-04-27 Debiopharm Int Sa Afabisiiniformulaatio, menetelmä sen valmistamiseksi
MA56184A (fr) 2019-06-14 2022-04-20 Debiopharm Int Sa Afabicine pour utilisation dans le traitement d'infections bactériennes impliquant un biofilm

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Also Published As

Publication number Publication date
CN1333776A (zh) 2002-01-30
CN100436456C (zh) 2008-11-26
EP1134222A1 (en) 2001-09-19
HUP0200450A2 (hu) 2002-07-29
WO2000032606A1 (en) 2000-06-08
ES2241374T3 (es) 2005-10-16
KR20010086058A (ko) 2001-09-07
TW526202B (en) 2003-04-01
NO20012554L (no) 2001-07-27
US6800621B2 (en) 2004-10-05
DE69924751D1 (de) 2005-05-19
EP1134222A4 (en) 2003-01-29
ZA200103850B (en) 2002-05-13
TR200101507T2 (tr) 2001-09-21
EP1134222B1 (en) 2005-04-13
NO20012554D0 (no) 2001-05-23
NZ511619A (en) 2002-11-26
HUP0200450A3 (en) 2004-04-28
RU2223964C2 (ru) 2004-02-20
BR9915743A (pt) 2001-08-21
AU758662B2 (en) 2003-03-27
JP3636663B2 (ja) 2005-04-06
KR100692169B1 (ko) 2007-03-12
CZ20011719A3 (cs) 2001-12-12
ATE293114T1 (de) 2005-04-15
PL347897A1 (en) 2002-04-22
AU1409000A (en) 2000-06-19
DE69924751T2 (de) 2006-03-09
IL143314A0 (en) 2002-04-21
US20030149014A1 (en) 2003-08-07
US6518263B1 (en) 2003-02-11
CA2350905A1 (en) 2000-06-08
CA2350905C (en) 2007-10-23

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