IL141242A0 - Substituted imidazo [1,2a] azines as selective inhibitors of cox-2 - Google Patents

Substituted imidazo [1,2a] azines as selective inhibitors of cox-2

Info

Publication number
IL141242A0
IL141242A0 IL14124299A IL14124299A IL141242A0 IL 141242 A0 IL141242 A0 IL 141242A0 IL 14124299 A IL14124299 A IL 14124299A IL 14124299 A IL14124299 A IL 14124299A IL 141242 A0 IL141242 A0 IL 141242A0
Authority
IL
Israel
Prior art keywords
azines
cox
selective inhibitors
substituted imidazo
imidazo
Prior art date
Application number
IL14124299A
Other languages
English (en)
Original Assignee
S A L V A T Lab Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by S A L V A T Lab Sa filed Critical S A L V A T Lab Sa
Publication of IL141242A0 publication Critical patent/IL141242A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL14124299A 1998-08-03 1999-07-23 Substituted imidazo [1,2a] azines as selective inhibitors of cox-2 IL141242A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ES009801652A ES2140354B1 (es) 1998-08-03 1998-08-03 Imidazo (1,2a) azinas sustituidas como inhibidores selectivos de la cox-2.
PCT/ES1999/000235 WO2000008024A1 (fr) 1998-08-03 1999-07-23 Imidazo[1,2a]azines substituees servant d'inhibiteurs selectifs de la cox-2

Publications (1)

Publication Number Publication Date
IL141242A0 true IL141242A0 (en) 2002-03-10

Family

ID=8304755

Family Applications (1)

Application Number Title Priority Date Filing Date
IL14124299A IL141242A0 (en) 1998-08-03 1999-07-23 Substituted imidazo [1,2a] azines as selective inhibitors of cox-2

Country Status (30)

Country Link
US (1) US6670365B1 (fr)
EP (1) EP1104762B1 (fr)
JP (1) JP2002522438A (fr)
KR (1) KR20010079602A (fr)
CN (1) CN1131865C (fr)
AP (1) AP2001002082A0 (fr)
AT (1) ATE224391T1 (fr)
AU (1) AU749770B2 (fr)
BG (1) BG105299A (fr)
BR (1) BR9912968A (fr)
CA (1) CA2339187A1 (fr)
CZ (1) CZ291783B6 (fr)
DE (1) DE69903046T2 (fr)
DK (1) DK1104762T3 (fr)
EA (1) EA003399B1 (fr)
ES (2) ES2140354B1 (fr)
HU (1) HUP0103004A3 (fr)
ID (1) ID28539A (fr)
IL (1) IL141242A0 (fr)
MX (1) MXPA01001332A (fr)
NO (1) NO20010568L (fr)
NZ (1) NZ510196A (fr)
OA (1) OA11592A (fr)
PL (1) PL345804A1 (fr)
PT (1) PT1104762E (fr)
SK (1) SK1662001A3 (fr)
TR (1) TR200100359T2 (fr)
WO (1) WO2000008024A1 (fr)
YU (1) YU7401A (fr)
ZA (1) ZA200101632B (fr)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE283048T1 (de) 1999-12-08 2004-12-15 Pharmacia Corp Cyclooxygenase-2 hemmer enthaltende zusammensetzungen mit schnellem wirkungseintritt
US8241622B2 (en) * 2001-07-13 2012-08-14 University Of Iowa Research Foundation Adeno-associated virus vectors with intravector heterologous terminal palindromic sequences
US20030100594A1 (en) * 2001-08-10 2003-05-29 Pharmacia Corporation Carbonic anhydrase inhibitor
DE10247271A1 (de) * 2002-10-10 2004-08-26 Grünenthal GmbH Substituierte C-Imidazo[1,2-a]pyridin-3-yle
DE10256881A1 (de) * 2002-12-05 2004-06-24 Beiersdorf Ag Neue topische Verwendung von Bis-Arylimidazo[1,2-a]thiolanderivaten
EP1745791B1 (fr) 2003-05-07 2013-06-26 Osteologix A/S Sels de strontium hydrosolubles pour le traitement d'affections de cartilage et/ou d'os
EP1660500B1 (fr) * 2003-07-30 2007-12-12 Laboratorios S.A.L.V.A.T., S.A. Imidazopyrimidines substituees pour la prevention et le traitement du cancer
WO2007034278A2 (fr) * 2005-09-19 2007-03-29 Pfizer Products Inc. Antagonistes du recepteur du c3a
CA2634670A1 (fr) * 2005-12-30 2007-07-12 University Of Iowa Research Foundation Procede d'identification de composes utiles pour le traitement de maladies degeneratives neuronales
WO2007096764A2 (fr) * 2006-02-27 2007-08-30 Glenmark Pharmaceuticals S.A. Dérivés d'hétéroaryles bicycliques en tant que modulateurs des récepteurs cannabinoïdes
RU2492170C9 (ru) * 2007-11-14 2013-12-27 Орто-Макнейл-Янссен Фармасьютикалз, Инк. Имидазо[1,2-а]пиридиновые производные и их применение в качестве положительных аллостерических модуляторов рецепторов mglur2
EP2350006A1 (fr) * 2008-10-01 2011-08-03 Synta Pharmaceuticals Corp. Composés pour des utilisations liées à une inflammation et au système immunitaire
GB201321732D0 (en) * 2013-12-09 2014-01-22 Ucb Pharma Sa Therapeutic agents
WO2017139381A1 (fr) 2016-02-08 2017-08-17 University Of Iowa Research Foundation Procédés pour produire des virus adéno-associés/bocavirus parvovirus chimériques
CA3198936A1 (fr) 2016-03-07 2017-09-14 University Of Iowa Research Foundation Expression mediee par aav utilisant un promoteur et un activateur synthetiques
US12173305B2 (en) 2016-05-26 2024-12-24 University Of Iowa Research Foundation cis and trans requirements for terminal resolution of human bocavirus 1
US11142775B2 (en) 2017-01-13 2021-10-12 University Of Iowa Research Foundation Bocaparvovirus small noncoding RNA and uses thereof
WO2022195579A1 (fr) 2021-03-15 2022-09-22 Saul Yedgar Dipalmitoyl-phosphatidyl-éthanol-amine conjuguée à l'acide hyaluronique en combinaison avec des médicaments anti-inflammatoires non stéroïdiens (ains) pour traiter ou soulager des maladies inflammatoires

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2785133A (en) * 1954-03-26 1957-03-12 Gen Aniline & Film Corp Compositions for a method of whitening fine fabrics
US3455924A (en) * 1967-02-08 1969-07-15 Upjohn Co Dianisylimidazoles
JPH06504779A (ja) * 1990-12-13 1994-06-02 スミスクライン・ビーチャム・コーポレイション 新規ｃｓａｉｄｓ
WO1993019066A1 (fr) * 1992-03-17 1993-09-30 Nippon Shinyaku Co., Ltd. Derive de l'imidazopyridine et medicament
US5620999A (en) * 1994-07-28 1997-04-15 Weier; Richard M. Benzenesulfonamide subtituted imidazolyl compounds for the treatment of inflammation
EA199700209A1 (ru) * 1995-04-04 1998-04-30 Глаксо Груп Лимитед ПРОИЗВОДНЫЕ ИМИДАЗО[1,2-a]ПИРИДИНА
UA57002C2 (uk) * 1995-10-13 2003-06-16 Мерк Фросст Кенада Енд Ко./Мерк Фросст Кенада Енд Сі. Похідне (метилсульфоніл)феніл-2-(5н)-фуранону, фармацевтична композиція та спосіб лікування

Also Published As

Publication number Publication date
CZ2001433A3 (cs) 2001-08-15
PT1104762E (pt) 2002-11-29
HUP0103004A2 (hu) 2002-01-28
WO2000008024A1 (fr) 2000-02-17
ATE224391T1 (de) 2002-10-15
ES2182546T3 (es) 2003-03-01
YU7401A (sh) 2003-10-31
CN1131865C (zh) 2003-12-24
EP1104762A1 (fr) 2001-06-06
AP2001002082A0 (en) 2001-03-31
ES2140354A1 (es) 2000-02-16
DE69903046D1 (de) 2002-10-24
NO20010568L (no) 2001-04-02
EA200100212A1 (ru) 2001-08-27
CN1321157A (zh) 2001-11-07
ID28539A (id) 2001-05-31
EA003399B1 (ru) 2003-04-24
DK1104762T3 (da) 2002-10-21
HK1037629A1 (en) 2002-02-15
US6670365B1 (en) 2003-12-30
TR200100359T2 (tr) 2001-06-21
SK1662001A3 (en) 2001-08-06
HUP0103004A3 (en) 2003-03-28
CA2339187A1 (fr) 2000-02-17
AU749770B2 (en) 2002-07-04
AU4782499A (en) 2000-02-28
DE69903046T2 (de) 2003-05-22
OA11592A (en) 2004-07-30
NO20010568D0 (no) 2001-02-02
ZA200101632B (en) 2001-08-30
PL345804A1 (en) 2002-01-02
BG105299A (en) 2001-11-30
KR20010079602A (ko) 2001-08-22
JP2002522438A (ja) 2002-07-23
EP1104762B1 (fr) 2002-09-18
ES2140354B1 (es) 2000-11-01
BR9912968A (pt) 2001-05-08
MXPA01001332A (es) 2002-11-29
NZ510196A (en) 2002-09-27
CZ291783B6 (cs) 2003-05-14

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