IL86751A - תכשירי רוקחות המכילים ציקלוספורינים וציקלוספורינים למיניהם - Google Patents

תכשירי רוקחות המכילים ציקלוספורינים וציקלוספורינים למיניהם

Info

Publication number: IL86751A
Authority: IL; Israel
Prior art keywords: residue; cyclosporin; cyclosporins; mebmt; ciclosporin
Prior art date: 1987-06-17

Application number

IL8675188A

Other languages

English (en)

Other versions

IL86751A0 (en

Original Assignee

Sandoz Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1987-06-17

Filing date

1988-06-15

Publication date

1994-02-27

1987-06-17 Priority claimed from GB878714100A external-priority patent/GB8714100D0/en

1987-06-17 Priority claimed from GB878714119A external-priority patent/GB8714119D0/en

1987-06-17 Priority claimed from GB878714093A external-priority patent/GB8714093D0/en

1987-06-17 Priority claimed from GB878714090A external-priority patent/GB8714090D0/en

1987-06-17 Priority claimed from GB878714115A external-priority patent/GB8714115D0/en

1987-06-17 Priority claimed from GB878714118A external-priority patent/GB8714118D0/en

1987-06-17 Priority claimed from GB878714125A external-priority patent/GB8714125D0/en

1987-06-17 Priority claimed from GB878714098A external-priority patent/GB8714098D0/en

1988-06-15 Application filed by Sandoz Ag filed Critical Sandoz Ag

1988-11-30 Publication of IL86751A0 publication Critical patent/IL86751A0/xx

1994-02-27 Publication of IL86751A publication Critical patent/IL86751A/he

Links

229930182912 cyclosporin Natural products 0.000 title claims abstract description 337
108010036941 Cyclosporins Proteins 0.000 title claims abstract description 180
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229960001265 ciclosporin Drugs 0.000 claims description 251
108010036949 Cyclosporine Proteins 0.000 claims description 180
PMATZTZNYRCHOR-CGLBZJNRSA-N Cyclosporin A Chemical compound CC[C@@H]1NC(=O)[C@H]([C@H](O)[C@H](C)C\C=C\C)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)N(C)C(=O)CN(C)C1=O PMATZTZNYRCHOR-CGLBZJNRSA-N 0.000 claims description 178
229930105110 Cyclosporin A Natural products 0.000 claims description 161
125000001183 hydrocarbyl group Chemical group 0.000 claims description 27
229910052799 carbon Inorganic materials 0.000 claims description 21
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Classifications

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- C—CHEMISTRY; METALLURGY
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- C07K—PEPTIDES
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- C07K7/645—Cyclosporins; Related peptides
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Immunology (AREA)
Biochemistry (AREA)
Molecular Biology (AREA)
Genetics & Genomics (AREA)
Biophysics (AREA)
Oncology (AREA)
Bioinformatics & Cheminformatics (AREA)
Communicable Diseases (AREA)
Engineering & Computer Science (AREA)
Hematology (AREA)
Tropical Medicine & Parasitology (AREA)
Rheumatology (AREA)
Virology (AREA)
Pain & Pain Management (AREA)
Transplantation (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

IL8675188A 1987-06-17 1988-06-15 תכשירי רוקחות המכילים ציקלוספורינים וציקלוספורינים למיניהם IL86751A (he)

Applications Claiming Priority (8)

Application Number	Priority Date	Filing Date	Title
GB878714100A GB8714100D0 (en)	1987-06-17	1987-06-17	Organic compounds
GB878714119A GB8714119D0 (en)	1987-06-17	1987-06-17	Organic compounds
GB878714093A GB8714093D0 (en)	1987-06-17	1987-06-17	Organic compounds
GB878714090A GB8714090D0 (en)	1987-06-17	1987-06-17	Organic compounds
GB878714115A GB8714115D0 (en)	1987-06-17	1987-06-17	Organic compounds
GB878714118A GB8714118D0 (en)	1987-06-17	1987-06-17	Organic compounds
GB878714125A GB8714125D0 (en)	1987-06-17	1987-06-17	Organic compounds
GB878714098A GB8714098D0 (en)	1987-06-17	1987-06-17	Organic compounds

Publications (2)

Publication Number	Publication Date
IL86751A0 IL86751A0 (en)	1988-11-30
IL86751A true IL86751A (he)	1994-02-27

Family

ID=27571252

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL8675188A IL86751A (he)	1987-06-17	1988-06-15	תכשירי רוקחות המכילים ציקלוספורינים וציקלוספורינים למיניהם

Country Status (21)

Country	Link
US (1)	US5525590A (he)
EP (1)	EP0296122B1 (he)
JP (2)	JPH0832724B2 (he)
KR (1)	KR970010927B1 (he)
AT (1)	ATE95193T1 (he)
AU (1)	AU614086B2 (he)
CA (1)	CA1338728C (he)
CY (1)	CY1939A (he)
CZ (1)	CZ411791A3 (he)
DE (1)	DE3884470T2 (he)
DK (1)	DK173873B1 (he)
ES (1)	ES2059558T3 (he)
HK (1)	HK152796A (he)
HU (1)	HU211678A9 (he)
IE (1)	IE62482B1 (he)
IL (1)	IL86751A (he)
MY (1)	MY103582A (he)
NZ (1)	NZ225041A (he)
PT (1)	PT87745B (he)
SA (1)	SA97170746A (he)
SK (1)	SK411791A3 (he)

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1988
- 1988-06-14 ES ES88810403T patent/ES2059558T3/es not_active Expired - Lifetime
- 1988-06-14 DE DE88810403T patent/DE3884470T2/de not_active Expired - Lifetime
- 1988-06-14 EP EP88810403A patent/EP0296122B1/en not_active Expired - Lifetime
- 1988-06-14 AT AT88810403T patent/ATE95193T1/de not_active IP Right Cessation
- 1988-06-15 DK DK198803265A patent/DK173873B1/da not_active IP Right Cessation
- 1988-06-15 IL IL8675188A patent/IL86751A/he not_active IP Right Cessation
- 1988-06-15 CA CA000569523A patent/CA1338728C/en not_active Expired - Fee Related
- 1988-06-15 MY MYPI88000662A patent/MY103582A/en unknown
- 1988-06-15 AU AU17679/88A patent/AU614086B2/en not_active Expired
- 1988-06-15 IE IE180788A patent/IE62482B1/en not_active IP Right Cessation
- 1988-06-15 NZ NZ225041A patent/NZ225041A/en unknown
- 1988-06-16 JP JP63149227A patent/JPH0832724B2/ja not_active Expired - Lifetime
- 1988-06-16 PT PT87745A patent/PT87745B/pt not_active IP Right Cessation
- 1988-06-16 KR KR1019880007330A patent/KR970010927B1/ko not_active Expired - Fee Related
1991
- 1991-12-27 SK SK4117-91A patent/SK411791A3/sk unknown
- 1991-12-27 CZ CS914117A patent/CZ411791A3/cs unknown
1994
- 1994-11-10 US US08/337,346 patent/US5525590A/en not_active Expired - Lifetime
1995
- 1995-06-22 HU HU95P/P00332P patent/HU211678A9/hu unknown
- 1995-08-16 JP JP7208783A patent/JP2772372B2/ja not_active Expired - Lifetime
1996
- 1996-08-08 HK HK152796A patent/HK152796A/en not_active IP Right Cessation
1997
- 1997-03-25 SA SA97170746A patent/SA97170746A/ar unknown
- 1997-05-16 CY CY193997A patent/CY1939A/xx unknown

Also Published As

Publication number	Publication date
ES2059558T3 (es)	1994-11-16
IE62482B1 (en)	1995-02-08
CZ411791A3 (en)	1993-02-17
PT87745A (pt)	1988-07-01
DE3884470T2 (de)	1994-03-10
IE881807L (en)	1988-12-17
CA1338728C (en)	1996-11-19
ATE95193T1 (de)	1993-10-15
NZ225041A (en)	1991-03-26
JPS6445396A (en)	1989-02-17
DK326588A (da)	1988-12-18
SA97170746A (ar)	2005-12-03
US5525590A (en)	1996-06-11
DK326588D0 (da)	1988-06-15
DK173873B1 (da)	2002-01-21
EP0296122A2 (en)	1988-12-21
AU1767988A (en)	1988-12-22
JP2772372B2 (ja)	1998-07-02
DE3884470D1 (de)	1993-11-04
JPH0832724B2 (ja)	1996-03-29
EP0296122A3 (en)	1990-06-20
AU614086B2 (en)	1991-08-22
HU211678A9 (en)	1995-12-28
PT87745B (pt)	1992-10-30
JPH0848696A (ja)	1996-02-20
KR890000519A (ko)	1989-03-15
EP0296122B1 (en)	1993-09-29
KR970010927B1 (ko)	1997-07-02
HK152796A (en)	1996-08-16
CY1939A (en)	1997-05-16
MY103582A (en)	1993-08-28
SK411791A3 (en)	1995-07-11
IL86751A0 (en)	1988-11-30

Legal Events

Date	Code	Title
1997-11-20	HC	Change of name of proprietor(s)
1998-12-06	KB	Patent renewed
2002-08-14	KB	Patent renewed
2008-12-29	EXP	Patent expired

Publication	Publication Date	Title
CA1338728C (en)	1996-11-19	Cyclosporins and their use a pharmaceuticals
US4639434A (en)	1987-01-27	Novel cyclosporins
US4764503A (en)	1988-08-16	Novel cyclosporins
US6710029B1 (en)	2004-03-23	Dehydrodidemnin B
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