IS2722B - 1, 2, 3, 4- Tetrasetin indól til meðhöndlunar á öndunarfærasjúkdómum - Google Patents

1, 2, 3, 4- Tetrasetin indól til meðhöndlunar á öndunarfærasjúkdómum

Info

Publication number: IS2722B
Authority: IS; Iceland
Prior art keywords: tetrasetin; indole; treatment; respiratory diseases; respiratory
Prior art date: 2003-05-27

Application number

IS8189A

Other languages

English (en)

Other versions

IS8189A (is

Inventor

Roger Bonnert

Rukhsana Rasul

Original Assignee

Astrazeneca Ab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-05-27

Filing date

2005-12-20

Publication date

2011-03-15

2005-12-20 Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab

2005-12-20 Publication of IS8189A publication Critical patent/IS8189A/is

2011-03-15 Publication of IS2722B publication Critical patent/IS2722B/is

Links

SIKJAQJRHWYJAI-UHFFFAOYSA-N Indole Chemical compound C1=CC=C2NC=CC2=C1 SIKJAQJRHWYJAI-UHFFFAOYSA-N 0.000 title 2
PZOUSPYUWWUPPK-UHFFFAOYSA-N indole Natural products CC1=CC=CC2=C1C=CN2 PZOUSPYUWWUPPK-UHFFFAOYSA-N 0.000 title 1
RKJUIXBNRJVNHR-UHFFFAOYSA-N indolenine Natural products C1=CC=C2CC=NC2=C1 RKJUIXBNRJVNHR-UHFFFAOYSA-N 0.000 title 1
208000023504 respiratory system disease Diseases 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/16—Central respiratory analeptics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Pulmonology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Virology (AREA)
Pain & Pain Management (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Molecular Biology (AREA)
Rheumatology (AREA)
Otolaryngology (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Indole Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

IS8189A 2003-05-27 2005-12-20 1, 2, 3, 4- Tetrasetin indól til meðhöndlunar á öndunarfærasjúkdómum IS2722B (is)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
SE0301569A SE0301569D0 (sv)	2003-05-27	2003-05-27	Novel compounds
SE0302305A SE0302305D0 (sv)	2003-05-27	2003-08-27	Novel Compounds
PCT/SE2004/000808 WO2004106302A1 (en)	2003-05-27	2004-05-25	Novel substituted 3-sulfur indoles

Publications (2)

Publication Number	Publication Date
IS8189A IS8189A (is)	2005-12-20
IS2722B true IS2722B (is)	2011-03-15

Family

ID=33492578

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
IS8189A IS2722B (is)	2003-05-27	2005-12-20	1, 2, 3, 4- Tetrasetin indól til meðhöndlunar á öndunarfærasjúkdómum
IS8920A IS8920A (is)	2003-05-27	2010-08-09	3-(Fenýl eða kínólyl)þíó- 1H-idnól-1-ediksýru afleður sem mótarar á virkni CRTh2 vitaka.

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
IS8920A IS8920A (is)	2003-05-27	2010-08-09	3-(Fenýl eða kínólyl)þíó- 1H-idnól-1-ediksýru afleður sem mótarar á virkni CRTh2 vitaka.

Country Status (30)

Country	Link
US (4)	US7687535B2 (is)
EP (3)	EP1656346B1 (is)
JP (2)	JP4541361B2 (is)
KR (3)	KR101067586B1 (is)
CN (2)	CN102391171A (is)
AR (1)	AR044552A1 (is)
AT (3)	ATE425965T1 (is)
AU (1)	AU2004242624B2 (is)
BR (1)	BRPI0410711B8 (is)
CA (1)	CA2526866C (is)
CO (1)	CO5630030A2 (is)
CY (3)	CY1109104T1 (is)
DE (2)	DE602004031894D1 (is)
DK (3)	DK1656346T3 (is)
ES (3)	ES2322650T3 (is)
HR (3)	HRP20090281T1 (is)
IL (4)	IL171928A (is)
IS (2)	IS2722B (is)
MX (1)	MXPA05012680A (is)
MY (1)	MY144483A (is)
NO (1)	NO20056130L (is)
NZ (1)	NZ543722A (is)
PL (3)	PL2025670T3 (is)
PT (3)	PT2281815E (is)
RU (1)	RU2361860C2 (is)
SE (2)	SE0301569D0 (is)
SI (3)	SI2281815T1 (is)
TW (2)	TW201024261A (is)
WO (1)	WO2004106302A1 (is)
ZA (1)	ZA200509598B (is)

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- 2003-05-27 SE SE0301569A patent/SE0301569D0/xx unknown
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2004
- 2004-05-19 TW TW099109193A patent/TW201024261A/zh unknown
- 2004-05-19 TW TW093114113A patent/TWI328004B/zh not_active IP Right Cessation
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Also Published As

Publication number	Publication date
JP4541361B2 (ja)	2010-09-08
PL1656346T3 (pl)	2009-07-31
BRPI0410711A (pt)	2006-06-13
HRP20110359T1 (hr)	2011-06-30
NO20056130L (no)	2006-02-27
CA2526866A1 (en)	2004-12-09
IL194872A0 (en)	2011-08-01
JP2010155862A (ja)	2010-07-15
DK1656346T3 (da)	2009-06-15
EP2281815B1 (en)	2012-04-04
DK2281815T3 (da)	2012-06-18
IL171928A (en)	2011-06-30
NZ543722A (en)	2007-05-31
EP2025670A1 (en)	2009-02-18
IL171928A0 (en)	2006-04-10
EP2025670B1 (en)	2011-03-16
BRPI0410711B8 (pt)	2021-05-25
ZA200509598B (en)	2006-12-27
KR20110050754A (ko)	2011-05-16
MY144483A (en)	2011-09-30
HK1126773A1 (en)	2009-09-11
ATE502010T1 (de)	2011-04-15
SE0302305D0 (sv)	2003-08-27
PT2281815E (pt)	2012-05-24
HRP20090281T1 (hr)	2009-06-30
CO5630030A2 (es)	2006-04-28
MXPA05012680A (es)	2006-02-08
CY1109104T1 (el)	2014-07-02
CY1112853T1 (el)	2016-02-10
EP2281815A1 (en)	2011-02-09
KR101067586B1 (ko)	2011-09-27
AU2004242624A1 (en)	2004-12-09
RU2005137403A (ru)	2006-05-27
IL212265A0 (en)	2011-06-30
US20080249110A1 (en)	2008-10-09
TW201024261A (en)	2010-07-01
SI2281815T1 (sl)	2012-06-29
TW200510301A (en)	2005-03-16
SE0301569D0 (sv)	2003-05-27
US7687535B2 (en)	2010-03-30
DE602004031894D1 (de)	2011-04-28
ATE425965T1 (de)	2009-04-15
ATE552243T1 (de)	2012-04-15
HK1090635A1 (zh)	2006-12-29
SI1656346T1 (sl)	2009-08-31
AR044552A1 (es)	2005-09-21
KR101067535B1 (ko)	2011-09-27
US20110263614A1 (en)	2011-10-27
KR20060015303A (ko)	2006-02-16
ES2361485T3 (es)	2011-06-17
ES2382606T3 (es)	2012-06-11
CN1795174A (zh)	2006-06-28
DE602004020072D1 (de)	2009-04-30
HRP20120390T1 (hr)	2012-06-30
IS8189A (is)	2005-12-20
PT2025670E (pt)	2011-05-24
US20090163518A1 (en)	2009-06-25
WO2004106302A1 (en)	2004-12-09
PT1656346E (pt)	2009-05-20
RU2361860C2 (ru)	2009-07-20
HK1149563A1 (en)	2011-10-07
IS8920A (is)	2010-08-09
CA2526866C (en)	2012-10-16
AU2004242624B2 (en)	2008-03-13
TWI328004B (en)	2010-08-01
EP1656346A1 (en)	2006-05-17
CN102391171A (zh)	2012-03-28
CN1795174B (zh)	2011-09-28
IL212371A0 (en)	2011-06-30
BRPI0410711B1 (pt)	2018-09-25
CY1111469T1 (el)	2015-08-05
PL2025670T3 (pl)	2011-07-29
SI2025670T1 (sl)	2011-06-30
EP1656346B1 (en)	2009-03-18
JP2007501269A (ja)	2007-01-25
US20120178764A1 (en)	2012-07-12
PL2281815T3 (pl)	2012-08-31
DK2025670T3 (da)	2011-06-06
ES2322650T3 (es)	2009-06-24
KR20110051297A (ko)	2011-05-17

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