|
US6140317A
(en)
*
|
1996-01-23 |
2000-10-31 |
Novartis Ag |
Pyrrolopyrimidines and processes for their preparation
|
|
JP4471404B2
(ja)
|
1996-02-13 |
2010-06-02 |
アストラゼネカ ユーケイ リミテッド |
Vegfインヒビターとしてのキナゾリン誘導体
|
|
ATE211134T1
(de)
|
1996-03-05 |
2002-01-15 |
|
4-anilinochinazolin derivate
|
|
GB9707800D0
(en)
|
1996-05-06 |
1997-06-04 |
Zeneca Ltd |
Chemical compounds
|
|
HRP970371A2
(en)
*
|
1996-07-13 |
1998-08-31 |
Kathryn Jane Smith |
Heterocyclic compounds
|
|
GB9718972D0
(en)
|
1996-09-25 |
1997-11-12 |
Zeneca Ltd |
Chemical compounds
|
|
WO1998013350A1
(en)
|
1996-09-25 |
1998-04-02 |
Zeneca Limited |
Qinoline derivatives inhibiting the effect of growth factors such as vegf
|
|
ZA986729B
(en)
*
|
1997-07-29 |
1999-02-02 |
Warner Lambert Co |
Irreversible inhibitors of tyrosine kinases
|
|
ATE368665T1
(de)
|
1997-08-22 |
2007-08-15 |
Astrazeneca Ab |
Oxindolylchinazolinderivate als angiogenesehemmer
|
|
PA8474101A1
(es)
*
|
1998-06-19 |
2000-09-29 |
Pfizer Prod Inc |
Compuestos de pirrolo [2,3-d] pirimidina
|
|
TW505646B
(en)
|
1998-06-19 |
2002-10-11 |
Pfizer Prod Inc |
Pyrrolo [2,3-d] pyrimidine compounds
|
|
UA71945C2
(en)
*
|
1999-01-27 |
2005-01-17 |
Pfizer Prod Inc |
Substituted bicyclic derivatives being used as anticancer agents
|
|
US6794393B1
(en)
|
1999-10-19 |
2004-09-21 |
Merck & Co., Inc. |
Tyrosine kinase inhibitors
|
|
DZ3223A1
(fr)
|
1999-10-19 |
2001-04-26 |
Merck & Co Inc |
Inhibiteurs de tyrosine kinases
|
|
PL203782B1
(pl)
|
1999-11-05 |
2009-11-30 |
Astrazeneca Ab |
Pochodne chinazoliny,sposoby ich wytwarzania,ich kompozycje farmaceutyczne oraz ich zastosowania
|
|
PT1382339E
(pt)
|
1999-12-10 |
2008-02-06 |
Pfizer Prod Inc |
Composições que contêm derivados de pirrolo[2,3-d]- pirimidina
|
|
AU2728201A
(en)
|
1999-12-21 |
2001-07-03 |
Sugen, Inc. |
4-substituted 7-aza-indolin-2-ones and their use as protein kinase inhibitors
|
|
US6420382B2
(en)
|
2000-02-25 |
2002-07-16 |
Merck & Co., Inc. |
Tyrosine kinase inhibitors
|
|
US6313138B1
(en)
|
2000-02-25 |
2001-11-06 |
Merck & Co., Inc. |
Tyrosine kinase inhibitors
|
|
AU779695B2
(en)
|
2000-04-07 |
2005-02-10 |
Astrazeneca Ab |
Quinazoline compounds
|
|
US6608053B2
(en)
|
2000-04-27 |
2003-08-19 |
Yamanouchi Pharmaceutical Co., Ltd. |
Fused heteroaryl derivatives
|
|
TR200402656T4
(tr)
|
2000-06-06 |
2004-11-22 |
Pfizer Products Inc. |
Antikanser ajanları olarak faydalı tiyofen türevleri
|
|
PL359563A1
(pl)
|
2000-06-26 |
2004-08-23 |
Pfizer Products Inc. |
Związki pirolo [2,3-d] pirymidynowe jako środki immunosupresyjne
|
|
WO2002032861A2
(en)
|
2000-10-17 |
2002-04-25 |
Merck & Co., Inc. |
Orally active salts with tyrosine kinase activity
|
|
ATE419239T1
(de)
|
2000-10-20 |
2009-01-15 |
Eisai R&D Man Co Ltd |
Verfahren zur herstellung von 4-phenoxy chinolin derivaten
|
|
JP4524072B2
(ja)
|
2000-10-23 |
2010-08-11 |
グラクソスミスクライン・リミテッド・ライアビリティ・カンパニー |
新規化合物
|
|
TWI238824B
(en)
|
2001-05-14 |
2005-09-01 |
Novartis Ag |
4-amino-5-phenyl-7-cyclobutyl-pyrrolo[2,3-d]pyrimidine derivatives
|
|
US7301023B2
(en)
|
2001-05-31 |
2007-11-27 |
Pfizer Inc. |
Chiral salt resolution
|
|
US6995171B2
(en)
|
2001-06-21 |
2006-02-07 |
Agouron Pharmaceuticals, Inc. |
Bicyclic pyrimidine and pyrimidine derivatives useful as anticancer agents
|
|
GB0115393D0
(en)
*
|
2001-06-23 |
2001-08-15 |
Aventis Pharma Ltd |
Chemical compounds
|
|
AU2002361577A1
(en)
|
2001-10-30 |
2003-05-12 |
Merck And Co., Inc. |
Tyrosine kinase inhibitors
|
|
RS63204A
(sr)
|
2002-01-17 |
2006-10-27 |
Neurogen Corporation |
Supstituisani analozi hinazolin-4-ilamina kao modulatori kapsaicina
|
|
BR0308162A
(pt)
|
2002-03-01 |
2004-12-07 |
Pfizer |
Derivados de indolil-uréia de tienopiridinas úteis como agentes antiangiogênicos e métodos para o seu uso
|
|
UA77303C2
(en)
|
2002-06-14 |
2006-11-15 |
Pfizer |
Derivatives of thienopyridines substituted by benzocondensed heteroarylamide useful as therapeutic agents, pharmaceutical compositions and methods for their use
|
|
WO2004047843A1
(en)
|
2002-11-26 |
2004-06-10 |
Pfizer Products Inc. |
Method of treatment of transplant rejection
|
|
AR042461A1
(es)
*
|
2002-12-13 |
2005-06-22 |
Neurogen Corp |
Analogos 2-sustituidos de quinazolin-4-il - amina. composiciones farmaceuticas
|
|
US7329664B2
(en)
*
|
2003-07-16 |
2008-02-12 |
Neurogen Corporation |
Substituted (7-pyridyl-4-phenylamino-quinazolin-2-yl)-methanol analogues
|
|
EP1660504B1
(en)
|
2003-08-29 |
2008-10-29 |
Pfizer Inc. |
Thienopyridine-phenylacet amides and their derivatives useful as new anti-angiogenic agents
|
|
AU2004270740A1
(en)
*
|
2003-09-09 |
2005-03-17 |
Neurogen Corporation |
4 - heterobicyclyamino - substituted quinazolines and analogues therof as capsaicin - antagonists
|
|
CN101337930B
(zh)
|
2003-11-11 |
2010-09-08 |
卫材R&D管理有限公司 |
脲衍生物的制备方法
|
|
CA2546192C
(en)
*
|
2003-11-17 |
2010-04-06 |
Pfizer Products Inc. |
Pyrrolopyrimidine compounds useful in treatment of cancer
|
|
KR100807920B1
(ko)
|
2003-12-23 |
2008-02-27 |
화이자 인코포레이티드 |
신규한 퀴놀린 유도체
|
|
BRPI0511512A
(pt)
|
2004-05-27 |
2007-12-26 |
Pfizer Prod Inc |
derivados pirrolpirimidina úteis no tratamento do cáncer
|
|
CN1993362B
(zh)
*
|
2004-06-02 |
2010-12-15 |
武田药品工业株式会社 |
稠合的杂环化合物
|
|
MEP8409A
(en)
*
|
2004-06-02 |
2011-12-20 |
|
Fused heterocyclic compound
|
|
JP4834553B2
(ja)
|
2004-09-17 |
2011-12-14 |
エーザイ・アール・アンド・ディー・マネジメント株式会社 |
医薬組成物
|
|
GB0423554D0
(en)
*
|
2004-10-22 |
2004-11-24 |
Cancer Rec Tech Ltd |
Therapeutic compounds
|
|
WO2006091450A1
(en)
|
2005-02-18 |
2006-08-31 |
Lexicon Genetics Incorporated |
4-piperidin-1-yl-7h-pyrrolo[2,3-d]pyrimidine compounds
|
|
WO2006130673A1
(en)
*
|
2005-05-31 |
2006-12-07 |
Janssen Pharmaceutica, N.V. |
3-benzoimidazolyl-pyrazolopyridines useful in treating kinase disorders
|
|
EP1925676A4
(en)
|
2005-08-02 |
2010-11-10 |
Eisai R&D Man Co Ltd |
TEST METHOD FOR THE EFFECT OF A VASCULARIZATION INHIBITOR
|
|
EP2345652A1
(en)
|
2005-12-21 |
2011-07-20 |
Abbott Laboratories |
Antiviral compounds
|
|
ES2395386T3
(es)
|
2005-12-21 |
2013-02-12 |
Abbott Laboratories |
Compuestos antivirales
|
|
RU2441869C2
(ru)
|
2005-12-21 |
2012-02-10 |
Эбботт Лэборетриз |
Противовирусные соединения
|
|
RU2467007C2
(ru)
|
2005-12-21 |
2012-11-20 |
Эбботт Лэборетриз |
Производные [1,8]нафтиридина, полезные в качестве ингибиторов репликации вируса hcv
|
|
RU2441010C2
(ru)
*
|
2005-12-21 |
2012-01-27 |
Эбботт Лэборетриз |
Противовирусные соединения
|
|
TWI392676B
(zh)
*
|
2005-12-21 |
2013-04-11 |
Abbott Lab |
抗病毒化合物、其製備方法及用途
|
|
US7851468B2
(en)
*
|
2006-05-15 |
2010-12-14 |
Cephalon, Inc. |
Substituted pyrazolo[3,4-d]pyrimidines
|
|
RU2448708C3
(ru)
|
2006-05-18 |
2017-09-28 |
Эйсай Ар Энд Ди Менеджмент Ко., Лтд. |
Противоопухолевое средство против рака щитовидной железы
|
|
US8865737B2
(en)
|
2006-08-28 |
2014-10-21 |
Eisai R&D Management Co., Ltd. |
Antitumor agent for undifferentiated gastric cancer
|
|
RU2009126576A
(ru)
|
2006-12-12 |
2011-01-20 |
Такеда Фармасьютикал Компани Лимитед (Jp) |
Конденсированное гетероциклическое соединение
|
|
CA2672737A1
(en)
*
|
2006-12-20 |
2008-11-06 |
Abbott Laboratories |
Anti-viral compounds
|
|
WO2008093855A1
(ja)
|
2007-01-29 |
2008-08-07 |
Eisai R & D Management Co., Ltd. |
未分化型胃癌治療用組成物
|
|
KR101513326B1
(ko)
|
2007-11-09 |
2015-04-17 |
에자이 알앤드디 매니지먼트 가부시키가이샤 |
혈관 신생 저해 물질과 항종양성 백금 착물의 병용
|
|
MX2010005671A
(es)
*
|
2007-11-28 |
2010-06-25 |
Dana Farber Cancer Inst Inc |
Inhibidores de miristato de moleculas pequeñas contra bcr-abl y metodos de uso.
|
|
TW200944528A
(en)
|
2008-03-12 |
2009-11-01 |
Takeda Pharmaceutical |
Fused heterocyclic compound
|
|
EP2384326B1
(en)
|
2008-08-20 |
2014-04-23 |
Zoetis LLC |
Pyrrolo[2,3-d]pyrimidine compounds
|
|
WO2011018894A1
(en)
*
|
2009-08-10 |
2011-02-17 |
Raqualia Pharma Inc. |
Pyrrolopyrimidine derivatives as potassium channel modulators
|
|
TH121482A
(th)
|
2009-08-19 |
2013-02-28 |
นางสาวปัณณพัฒน์ เหลืองธาตุทอง |
องค์ประกอบทางเภสัชกรรมที่ประกอบด้วยอนุพันธ์ของควิโนลีน
|
|
AU2011270165B2
(en)
|
2010-06-25 |
2015-12-24 |
Eisai R&D Management Co., Ltd. |
Antitumor agent using compounds having kinase inhibitory effect in combination
|
|
WO2012106522A2
(en)
|
2011-02-04 |
2012-08-09 |
Duquesne University Of The Holy Spirit |
Bicyclic and tricyclic pyrimidine tyrosine kinase inhibitors with antitubulin activity and methods of treating a patient
|
|
WO2012144463A1
(ja)
|
2011-04-18 |
2012-10-26 |
エーザイ・アール・アンド・ディー・マネジメント株式会社 |
腫瘍治療剤
|
|
EP3444363B1
(en)
|
2011-06-03 |
2020-11-25 |
Eisai R&D Management Co., Ltd. |
Biomarkers for prediciting and assessing responsiveness of thyroid and kidney cancer subjects to lenvatinib compounds
|
|
EP2852595B1
(en)
|
2012-05-21 |
2016-06-22 |
Bayer Pharma Aktiengesellschaft |
Substituted benzothienopyrimidines
|
|
CN105732639A
(zh)
*
|
2012-06-29 |
2016-07-06 |
辉瑞大药厂 |
作为LRRK2抑制剂的4-(取代的氨基)-7H-吡咯并〔2,3-d〕嘧啶类
|
|
TW201412740A
(zh)
|
2012-09-20 |
2014-04-01 |
Bayer Pharma AG |
經取代之吡咯并嘧啶胺基苯并噻唑酮
|
|
CN104781260A
(zh)
|
2012-09-26 |
2015-07-15 |
拜耳制药股份公司 |
用于治疗过度增殖性障碍的取代的吲唑-吡咯并嘧啶
|
|
US20150252047A1
(en)
|
2012-09-26 |
2015-09-10 |
Bayer Pharma Aktiengesellschaft |
Substituted indazol-pyrrolopyrimidines useful in the treatment of hyperproliferative diseases
|
|
JP6290917B2
(ja)
*
|
2012-11-29 |
2018-03-07 |
メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツングMerck Patent Gesellschaft mit beschraenkter Haftung |
アザキナゾリンカルボキサミド誘導体
|
|
RU2015115397A
(ru)
|
2012-12-21 |
2017-01-25 |
Эйсай Ар Энд Ди Менеджмент Ко., Лтд. |
Аморфная форма производного хинолина и способ его получения
|
|
ES2687968T3
(es)
|
2013-05-14 |
2018-10-30 |
Eisai R&D Management Co., Ltd. |
Biomarcadores para pronosticar y evaluar la reactividad de sujetos con cáncer de endometrio a compuestos con lenvatinib
|
|
EP3083618B1
(en)
|
2013-12-17 |
2018-02-21 |
Pfizer Inc |
Novel 3,4-disubstituted-1h-pyrrolo[2,3-b]pyridines and 4,5-disubstituted-7h-pyrrolo[2,3-c]pyridazines as lrrk2 inhibitors
|
|
LT3177612T
(lt)
|
2014-08-04 |
2022-06-10 |
Nuevolution A/S |
Pirimidino dariniai, pakeisti pasirinktinai kondensuotu heterociklilu, tinkami uždegiminių, metabolinių, onkologinių ir autoimuninių ligų gydymui
|
|
KR20230043234A
(ko)
|
2014-08-28 |
2023-03-30 |
에자이 알앤드디 매니지먼트 가부시키가이샤 |
고순도의 퀴놀린 유도체 및 이를 제조하는 방법
|
|
LT3263106T
(lt)
|
2015-02-25 |
2024-01-10 |
Eisai R&D Management Co., Ltd. |
Chinolino darinių kartumo sumažinimo būdas
|
|
KR102662228B1
(ko)
|
2015-03-04 |
2024-05-02 |
머크 샤프 앤드 돔 코포레이션 |
암을 치료하기 위한 pd-1 길항제 및 vegfr/fgfr/ret 티로신 키나제 억제제의 조합
|
|
HUE047477T2
(hu)
|
2015-06-04 |
2020-04-28 |
Pfizer |
Palbociclib szilárd dózisformái
|
|
MX373231B
(es)
|
2015-06-16 |
2020-05-08 |
Eisai R&D Man Co Ltd |
Agente anticancerigeno.
|
|
CA2994925C
(en)
|
2015-08-20 |
2023-08-29 |
Eisai R&D Management Co., Ltd. |
Tumor therapeutic agent
|
|
CN108137586B
(zh)
|
2015-09-14 |
2021-04-13 |
辉瑞大药厂 |
作为LRRK2抑制剂的新颖咪唑并[4,5-c]喹啉和咪唑并[4,5-c][1,5]萘啶衍生物
|
|
GB201520499D0
(en)
|
2015-11-20 |
2016-01-06 |
Medical Res Council Technology |
Compounds
|
|
JP6563623B1
(ja)
|
2016-08-15 |
2019-08-21 |
ファイザー・インク |
ピリドピリミジノンcdk2/4/6阻害剤
|
|
US12303505B2
(en)
|
2017-02-08 |
2025-05-20 |
Eisai R&D Management Co., Ltd. |
Tumor-treating pharmaceutical composition
|
|
BR112019023064A2
(pt)
|
2017-05-16 |
2020-06-09 |
Eisai R&D Man Co Ltd |
tratamento de carcinoma hepatocelular
|
|
US11633399B2
(en)
|
2018-12-25 |
2023-04-25 |
Sol-Gel Technologies Ltd. |
Treatment of skin disorders with compositions comprising an EGFR inhibitor
|
|
NL2022471B1
(en)
|
2019-01-29 |
2020-08-18 |
Vationpharma B V |
Solid state forms of oclacitinib
|
|
AU2020315192A1
(en)
|
2019-07-17 |
2022-02-24 |
2692372 Ontario, Inc. |
Benzenesulfonamide derivatives and uses thereof
|
|
MX2022007265A
(es)
|
2019-12-20 |
2022-09-09 |
Nuevolution As |
Compuestos activos frente a receptores nucleares.
|
|
TWI872177B
(zh)
|
2019-12-20 |
2025-02-11 |
丹麥商紐韋盧森公司 |
對核受體具有活性之化合物
|
|
US11613532B2
(en)
|
2020-03-31 |
2023-03-28 |
Nuevolution A/S |
Compounds active towards nuclear receptors
|
|
US11780843B2
(en)
|
2020-03-31 |
2023-10-10 |
Nuevolution A/S |
Compounds active towards nuclear receptors
|
|
US12037346B2
(en)
|
2021-04-13 |
2024-07-16 |
Nuvalent, Inc. |
Amino-substituted heteroaryls for treating cancers with EGFR mutations
|