IS6528A - Aðferð til framleiðslu á sítalóprami - Google Patents

Aðferð til framleiðslu á sítalóprami

Info

Publication number: IS6528A
Authority: IS; Iceland
Prior art keywords: producing citalopram; citalopram; producing
Prior art date: 2000-03-13

Application number

IS6528A

Other languages

English (en)

Inventor

Petersen Hans

Original Assignee

H. Lundbeck A/S

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-03-13

Filing date

2002-08-27

Publication date

2002-08-27

2002-08-27 Application filed by H. Lundbeck A/S filed Critical H. Lundbeck A/S

2002-08-27 Publication of IS6528A publication Critical patent/IS6528A/is

Links

WSEQXVZVJXJVFP-HXUWFJFHSA-N (R)-citalopram Chemical compound C1([C@@]2(C3=CC=C(C=C3CO2)C#N)CCCN(C)C)=CC=C(F)C=C1 WSEQXVZVJXJVFP-HXUWFJFHSA-N 0.000 title 1
229960001653 citalopram Drugs 0.000 title 1
238000004519 manufacturing process Methods 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
- A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Neurology (AREA)
Pain & Pain Management (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Psychiatry (AREA)
General Chemical & Material Sciences (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Steroid Compounds (AREA)
Furan Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

IS6528A 2000-03-13 2002-08-27 Aðferð til framleiðslu á sítalóprami IS6528A (is)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DKPA200000404		2000-03-13
PCT/DK2001/000149 WO2001068628A1 (en)	2000-03-13	2001-03-07	Method for the preparation of citalopram

Publications (1)

Publication Number	Publication Date
IS6528A true IS6528A (is)	2002-08-27

Family

ID=8159323

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IS6528A IS6528A (is)	2000-03-13	2002-08-27	Aðferð til framleiðslu á sítalóprami

Country Status (31)

Country	Link
US (1)	US6717000B2 (is)
EP (1)	EP1265880B1 (is)
JP (1)	JP2003527384A (is)
KR (1)	KR20020080471A (is)
CN (1)	CN1423644A (is)
AR (1)	AR029893A1 (is)
AT (1)	ATE282031T1 (is)
AU (1)	AU3920301A (is)
BE (1)	BE1011598A6 (is)
BG (1)	BG107048A (is)
BR (1)	BR0109267A (is)
CA (1)	CA2402386A1 (is)
CZ (1)	CZ20023383A3 (is)
DE (1)	DE60107061D1 (is)
EA (1)	EA200200971A1 (is)
FR (1)	FR2806085B1 (is)
HR (1)	HRP20020741A2 (is)
HU (1)	HUP0300180A2 (is)
IE (1)	IES20010206A2 (is)
IL (1)	IL151489A0 (is)
IS (1)	IS6528A (is)
IT (1)	ITMI20010487A1 (is)
MX (1)	MXPA02008872A (is)
NL (1)	NL1017500C1 (is)
NO (1)	NO20024214L (is)
NZ (1)	NZ521202A (is)
PL (1)	PL360108A1 (is)
SK (1)	SK14592002A3 (is)
TR (1)	TR200202167T2 (is)
WO (1)	WO2001068628A1 (is)
ZA (1)	ZA200206898B (is)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DK1173431T4 (da)	1999-04-14	2010-01-04	Lundbeck & Co As H	Fremgangsmåde til fremstilling af citalopram
IES20010157A2 (en)	2000-03-03	2002-03-06	Lundbeck & Co As H	Method for the preparation of citalopram
AU2001242298A1 (en)	2000-03-13	2001-09-24	H Lunbeck A/S	Method for the preparation of citalopram
KR20020080485A (ko)	2000-03-13	2002-10-23	하. 룬트벡 아크티에 셀스카브	5-치환 1-(4-플루오로페닐)-1,3-디히드로이소벤조푸란의단계적 알킬화
ES2214400T3 (es)	2000-03-14	2004-09-16	H. Lundbeck A/S	Metodo para la preparacion de citalopram.
AR032455A1 (es)	2000-05-12	2003-11-12	Lundbeck & Co As H	Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
AU2003223105A1 (en) *	2003-03-24	2004-10-18	Hetero Drugs Limited	Novel crystalline forms of (s)-citalopram oxalate
CN100569765C (zh)	2003-12-19	2009-12-16	杭州民生药业集团有限公司	西酞普兰中间体晶体碱

Family Cites Families (37)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1143703A (is)	1965-03-18
GB1526331A (en)	1976-01-14	1978-09-27	Kefalas As	Phthalanes
GB8419963D0 (en)	1984-08-06	1984-09-12	Lundbeck & Co As H	Intermediate compound and method
GB8814057D0 (en)	1988-06-14	1988-07-20	Lundbeck & Co As H	New enantiomers & their isolation
US5296507A (en)	1990-09-06	1994-03-22	H.Lundbeck A/S	Treatment of cerbrovascular disorders
DE19626659A1 (de)	1996-07-03	1998-01-08	Basf Ag	Verfahren zur Herstellung von Phthaliden
DE19627697A1 (de)	1996-07-10	1998-01-15	Basf Ag	Verfahren zur Herstellung von Phthaliden
SK283309B6 (sk)	1997-07-08	2003-05-02	H. Lundbeck A/S	Spôsob výroby citalopramu a medziprodukty
UA62985C2 (en) *	1997-11-10	2004-01-15	Lunnbeck As H	A method for the preparation of citalopram
DK1042310T3 (da)	1997-11-11	2002-12-02	Lundbeck & Co As H	Fremgangsmåde til fremstilling af citalopram
ES2189502T3 (es)	1998-10-20	2003-07-01	Lundbeck & Co As H	Metodo para la prevencion de citalopram.
IL143422A0 (en)	1998-12-23	2002-04-21	Lundbeck & Co As H	Method for the preparation of 5-cyanophthalide
AR022329A1 (es)	1999-01-29	2002-09-04	Lundbeck & Co As H	Metodo para la preparacion de 5-cianoftalida
DK1173431T4 (da)	1999-04-14	2010-01-04	Lundbeck & Co As H	Fremgangsmåde til fremstilling af citalopram
ITMI991581A1 (it)	1999-06-25	2001-01-15	Lundbeck & Co As H	Metodo per la preparazione di citalopram
ITMI991579A1 (it)	1999-06-25	2001-01-15	Lundbeck & Co As H	Metodo per la preparazione di citalopram
CH692421A5 (de)	1999-10-25	2002-06-14	Lundbeck & Co As H	Verfahren zur Herstellung von Citalopram.
US6310222B1 (en)	1999-11-01	2001-10-30	Sumika Fine Chemicals Co., Ltd.	Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
AR026063A1 (es)	1999-11-01	2002-12-26	Lundbeck & Co As H	Metodo para la preparacion de 5-carboxiftalida.
JP2003519136A (ja)	1999-12-28	2003-06-17	ハー・ルンドベック・アクチエゼルスカベット	シタロプラムの製造方法
DK1246813T3 (da)	1999-12-30	2004-03-01	Lundbeck & Co As H	Fremgangsmåde til fremstilling af Citalopram
AU3033700A (en)	2000-01-14	2001-07-24	H. Lundbeck A/S	Method for the preparation of 5-cyanophthalide
US6433196B1 (en)	2000-02-17	2002-08-13	Sumika Fine Chemicals Co., Ltd.	Production method of citalopram, intermediate therefor and production method of the intermediate
FR2805812A1 (fr)	2000-02-24	2001-09-07	Lundbeck & Co As H	Procede de preparation du citalopram
IES20010143A2 (en)	2000-02-24	2001-07-25	Lundbeck & Co As H	Method for the preparation of citalopram
IES20010157A2 (en)	2000-03-03	2002-03-06	Lundbeck & Co As H	Method for the preparation of citalopram
GB0005477D0 (en)	2000-03-07	2000-04-26	Resolution Chemicals Limited	Process for the preparation of citalopram
KR20020080485A (ko)	2000-03-13	2002-10-23	하. 룬트벡 아크티에 셀스카브	5-치환 1-(4-플루오로페닐)-1,3-디히드로이소벤조푸란의단계적 알킬화
AU2001242298A1 (en)	2000-03-13	2001-09-24	H Lunbeck A/S	Method for the preparation of citalopram
GB2357762B (en)	2000-03-13	2002-01-30	Lundbeck & Co As H	Crystalline base of citalopram
ES2214400T3 (es)	2000-03-14	2004-09-16	H. Lundbeck A/S	Metodo para la preparacion de citalopram.
DE10190485T1 (de)	2000-03-16	2002-03-21	Lundbeck & Co As H	Verfahren zur Herstellung von 5-Cyano-1-(4-fluorphenyl)-1,3-dihydroisobenzofuranen
AR032455A1 (es)	2000-05-12	2003-11-12	Lundbeck & Co As H	Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
WO2002004435A1 (en)	2000-07-06	2002-01-17	H. Lundbeck A/S	Method for the preparation of citalopram
CA2354877C (en)	2000-08-18	2006-05-02	H. Lundbeck A/S	Method for the preparation of citalopram
CA2360303C (en)	2000-12-22	2003-08-12	Marco Villa	Process for the preparation of pure citalopram
SK284418B6 (sk)	2000-12-28	2005-04-01	H. Lundbeck A/S	Spôsob výroby citalopramu

2001
- 2001-03-05 NL NL1017500A patent/NL1017500C1/nl not_active IP Right Cessation
- 2001-03-05 IE IE20010206A patent/IES20010206A2/en not_active IP Right Cessation
- 2001-03-07 CA CA002402386A patent/CA2402386A1/en not_active Abandoned
- 2001-03-07 EP EP01913728A patent/EP1265880B1/en not_active Expired - Lifetime
- 2001-03-07 TR TR2002/02167T patent/TR200202167T2/xx unknown
- 2001-03-07 IL IL15148901A patent/IL151489A0/xx unknown
- 2001-03-07 AT AT01913728T patent/ATE282031T1/de not_active IP Right Cessation
- 2001-03-07 AU AU39203/01A patent/AU3920301A/en not_active Abandoned
- 2001-03-07 DE DE60107061T patent/DE60107061D1/de not_active Expired - Lifetime
- 2001-03-07 CZ CZ20023383A patent/CZ20023383A3/cs unknown
- 2001-03-07 JP JP2001567720A patent/JP2003527384A/ja not_active Withdrawn
- 2001-03-07 KR KR1020027011671A patent/KR20020080471A/ko not_active Withdrawn
- 2001-03-07 CN CN01806481A patent/CN1423644A/zh active Pending
- 2001-03-07 SK SK1459-2002A patent/SK14592002A3/sk unknown
- 2001-03-07 PL PL36010801A patent/PL360108A1/xx not_active Application Discontinuation
- 2001-03-07 EA EA200200971A patent/EA200200971A1/ru unknown
- 2001-03-07 HU HU0300180A patent/HUP0300180A2/hu unknown
- 2001-03-07 NZ NZ521202A patent/NZ521202A/en unknown
- 2001-03-07 HR HR20020741A patent/HRP20020741A2/hr not_active Application Discontinuation
- 2001-03-07 AR ARP010101064A patent/AR029893A1/es unknown
- 2001-03-07 MX MXPA02008872A patent/MXPA02008872A/es unknown
- 2001-03-07 BR BR0109267-7A patent/BR0109267A/pt not_active IP Right Cessation
- 2001-03-07 WO PCT/DK2001/000149 patent/WO2001068628A1/en not_active Ceased
- 2001-03-08 IT IT2001MI000487A patent/ITMI20010487A1/it unknown
- 2001-03-09 FR FR0103245A patent/FR2806085B1/fr not_active Expired - Fee Related
- 2001-03-13 BE BE2001/0159A patent/BE1011598A6/fr not_active IP Right Cessation
2002
- 2002-08-27 IS IS6528A patent/IS6528A/is unknown
- 2002-08-28 ZA ZA200206898A patent/ZA200206898B/en unknown
- 2002-09-02 BG BG107048A patent/BG107048A/xx unknown
- 2002-09-04 NO NO20024214A patent/NO20024214L/no not_active Application Discontinuation
- 2002-09-09 US US10/238,843 patent/US6717000B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
ZA200206898B (en)	2004-04-20
DE60107061D1 (de)	2004-12-16
AU3920301A (en)	2001-09-24
TR200202167T2 (tr)	2002-12-23
CA2402386A1 (en)	2001-09-20
HRP20020741A2 (en)	2003-12-31
NL1017500C1 (nl)	2001-04-26
WO2001068628A1 (en)	2001-09-20
CN1423644A (zh)	2003-06-11
ATE282031T1 (de)	2004-11-15
FR2806085A1 (fr)	2001-09-14
BR0109267A (pt)	2002-12-17
KR20020080471A (ko)	2002-10-23
MXPA02008872A (es)	2003-02-10
JP2003527384A (ja)	2003-09-16
NZ521202A (en)	2004-11-26
AR029893A1 (es)	2003-07-23
PL360108A1 (en)	2004-09-06
IES20010206A2 (en)	2002-03-06
EA200200971A1 (ru)	2003-02-27
EP1265880B1 (en)	2004-11-10
IL151489A0 (en)	2003-04-10
CZ20023383A3 (cs)	2003-01-15
SK14592002A3 (sk)	2003-03-04
NO20024214D0 (no)	2002-09-04
NO20024214L (no)	2002-10-31
BE1011598A6 (fr)	2001-07-03
US6717000B2 (en)	2004-04-06
FR2806085B1 (fr)	2005-02-25
US20030069304A1 (en)	2003-04-10
BG107048A (en)	2003-05-30
HUP0300180A2 (en)	2003-05-28
ITMI20010487A1 (it)	2002-09-08
EP1265880A1 (en)	2002-12-18

Publication	Publication Date	Title
IS6091A (is)	2001-09-28	Aðferð til framleiðslu á sítalóprami
IS2120B (is)	2006-06-15	Aðferð til framleiðslu á sítalóprami
IS5862A (is)	2001-02-23	Aðferð til framleiðslu á sítalóprami
IS2343B (is)	2008-02-15	Aðferð til framleiðslu á sítalóprami
IS6512A (is)	2002-08-20	Aðferð til framleiðslu á sítalóprami
IS2256B (is)	2007-06-15	Aðferð til framleiðslu á sítalóprami
IS6487A (is)	2002-07-29	Aðferð til framleiðslu á Sítalóprami
IS5884A (is)	2002-06-28	Aðferð til framleiðslu á hreinu sítalóprami
IS5473A (is)	2000-04-26	Aðferð til framleiðslu á sítalóprami
FI109024B (fi)	2002-05-15	Menetelmä puhtaan sitalopraamin valmistamiseksi
DK1161426T3 (da)	2007-10-08	Fremgangsmåde til fremstilling af furfural
FI20002720A7 (fi)	2002-06-13	Menetelmä konversioiden suorittamiseksi
IS6526A (is)	2002-08-27	Aðferð til framleiðslu á sítalóprami
IS2586B (is)	2010-02-15	Aðferð til framleiðslu á sítalóprami
IS6529A (is)	2002-08-27	Aðferð til framleiðslu á sítalóprami
IS6293A (is)	2002-03-05	Aðferð til framleiðslu á sítalóprami
IS6716A (is)	2003-02-13	Aðferðir við að framleiða sílostasól
IS2260B (is)	2007-06-15	Aðferð til framleiðslu á sítalóprami
IS6528A (is)	2002-08-27	Aðferð til framleiðslu á sítalóprami
FI20000453L (fi)	2001-08-28	Menetelmä massan valmistamiseksi
ID30126A (id)	2001-11-08	METODE UNTUK MENGHASILKAN SIKLO-(Asp-DPhe-NMeVal-Arg-Gly)
FI20000185L (fi)	2001-07-29	Menetelmä painotuotteiden valmistamiseksi
FI20010892L (fi)	2002-10-28	Menetelmä ksylitolin valmistamiseksi
FI20000901L (fi)	2001-10-15	Menetelmä eetterin valmistamiseksi
FI20001328L (fi)	2001-12-03	Menetelmä monitoimisen entsyymin tuottamiseksi