IS6487A - Aðferð til framleiðslu á Sítalóprami - Google Patents

Aðferð til framleiðslu á Sítalóprami

Info

Publication number: IS6487A
Authority: IS; Iceland
Prior art keywords: citalopram; production
Prior art date: 2000-02-24

Application number

IS6487A

Other languages

English (en)

Inventor

Petersen Hans

Harold Rock Michael

Ahmadian Haleh

Original Assignee

H. Lundbeck A/S

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-02-24

Filing date

2002-07-29

Publication date

2002-07-29

2002-07-29 Application filed by H. Lundbeck A/S filed Critical H. Lundbeck A/S

2002-07-29 Publication of IS6487A publication Critical patent/IS6487A/is

Links

WSEQXVZVJXJVFP-HXUWFJFHSA-N (R)-citalopram Chemical compound C1([C@@]2(C3=CC=C(C=C3CO2)C#N)CCCN(C)C)=CC=C(F)C=C1 WSEQXVZVJXJVFP-HXUWFJFHSA-N 0.000 title 1
229960001653 citalopram Drugs 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
- A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Neurology (AREA)
Engineering & Computer Science (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Bioinformatics & Cheminformatics (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Psychiatry (AREA)
Pain & Pain Management (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Steroid Compounds (AREA)

IS6487A 2000-02-24 2002-07-29 Aðferð til framleiðslu á Sítalóprami IS6487A (is)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
DKPA200000296		2000-02-24
DKPA200000401		2000-03-13
PCT/DK2001/000123 WO2001043525A2 (en)	2000-02-24	2001-02-22	Method for the preparation of citalopram

Publications (1)

Publication Number	Publication Date
IS6487A true IS6487A (is)	2002-07-29

Family

ID=26068779

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IS6487A IS6487A (is)	2000-02-24	2002-07-29	Aðferð til framleiðslu á Sítalóprami

Country Status (26)

Country	Link
US (1)	US6420574B2 (is)
EP (1)	EP1259501A2 (is)
JP (1)	JP2003523955A (is)
KR (1)	KR20020081355A (is)
CN (1)	CN1608057A (is)
AR (1)	AR029658A1 (is)
AU (1)	AU2001235358A1 (is)
BE (1)	BE1011177A6 (is)
BG (1)	BG107061A (is)
BR (1)	BR0108937A (is)
CA (1)	CA2401236A1 (is)
EA (1)	EA005315B1 (is)
FR (1)	FR2805812A1 (is)
GR (1)	GR1004073B (is)
HR (1)	HRP20020660A2 (is)
HU (1)	HUP0300212A2 (is)
IE (1)	IES20010163A2 (is)
IL (1)	IL151059A0 (is)
IS (1)	IS6487A (is)
IT (1)	ITMI20010386A1 (is)
MX (1)	MXPA02008228A (is)
NL (1)	NL1017415C1 (is)
NO (1)	NO20023928D0 (is)
PL (1)	PL363119A1 (is)
SK (1)	SK13672002A3 (is)
WO (1)	WO2001043525A2 (is)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AR022329A1 (es)	1999-01-29	2002-09-04	Lundbeck & Co As H	Metodo para la preparacion de 5-cianoftalida
NZ514671A (en) *	1999-04-14	2003-10-31	H	Method for the preparation of citalopram
ITMI991581A1 (it) *	1999-06-25	2001-01-15	Lundbeck & Co As H	Metodo per la preparazione di citalopram
EP1298124B1 (en)	1999-10-25	2007-02-28	H. Lundbeck A/S	Method For the Preparation of Citalopram
US6310222B1 (en) *	1999-11-01	2001-10-30	Sumika Fine Chemicals Co., Ltd.	Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
AR026063A1 (es)	1999-11-01	2002-12-26	Lundbeck & Co As H	Metodo para la preparacion de 5-carboxiftalida.
EA004742B1 (ru)	1999-12-28	2004-08-26	Х.Лундбекк А/С	Способ получения циталопрама
WO2001049672A1 (en)	1999-12-30	2001-07-12	H. Lundbeck A/S	Method for the preparation of citalopram
TR200201783T2 (tr) *	2000-01-14	2002-12-23	H. Lundbeck A/S	5-Siyanofatalid hazırlamak için yöntem
US6433196B1 (en) *	2000-02-17	2002-08-13	Sumika Fine Chemicals Co., Ltd.	Production method of citalopram, intermediate therefor and production method of the intermediate
NL1017417C1 (nl) *	2000-03-03	2001-03-16	Lundbeck & Co As H	Werkwijze voor de bereiding van Citalopram.
KR20020080481A (ko)	2000-03-13	2002-10-23	하. 룬트벡 아크티에 셀스카브	시탈로프람의 제조 방법
NL1017500C1 (nl)	2000-03-13	2001-04-26	Lundbeck & Co As H	Werkwijze voor de bereiding van Citalopram.
CZ20023100A3 (cs) *	2000-03-13	2003-02-12	H. Lundbeck A/S	Způsob výroby citalopramu
SK14512002A3 (sk)	2000-03-14	2003-03-04	H. Lundbeck A/S	Spôsob výroby citalopramu, medziprodukt a citalopram výrobený týmto spôsobom
EP1274699A1 (en) *	2000-03-16	2003-01-15	H. Lundbeck A/S	Method for the preparation of 5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofurans
AR032455A1 (es)	2000-05-12	2003-11-12	Lundbeck & Co As H	Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
IL144817A0 (en)	2000-08-18	2002-06-30	Lundbeck & Co As H	Method for the preparation of citalopram
JP3798982B2 (ja)	2000-12-22	2006-07-19	ハー・ルンドベック・アクチエゼルスカベット	純粋なシタロプラムの製造方法
AR034759A1 (es) *	2001-07-13	2004-03-17	Lundbeck & Co As H	Metodo para la preparacion de escitalopram
EP1446396A1 (en) *	2001-11-08	2004-08-18	Sepracor, Inc.	Methods for treating depression and other cns disorders using enantiomerically enriched desmethyl- and didesmethyl-metabolites of citalopram
AR040970A1 (es)	2002-08-12	2005-04-27	Lundbeck & Co As H	Metodo para la separacion de intermediarios que pueden ser utilizados para la preparacion de escitalopram
TR200504022T1 (tr) *	2003-03-24	2006-08-21	Hetero Drugs Limited	(S)-sitalopram oksalatın yeni sıvı kristal formları.
CA2575975A1 (en) *	2003-11-12	2005-05-26	Dr. Reddy's Laboratories, Inc.	Preparation of escitalopram
TWI339651B (en)	2004-02-12	2011-04-01	Lundbeck & Co As H	Method for the separation of intermediates which may be used for the preparation of escitalopram
GB0601286D0 (en)	2006-01-23	2006-03-01	Sandoz Ag	Asymmetric synthesis
AU2008252631B2 (en) *	2007-05-18	2012-12-20	Cipla Limited	Process for the preparation of escitalopram via desmethylcitalopram, optical resolution and methylation of the S-isomer
WO2009111031A2 (en) *	2008-03-04	2009-09-11	Intra-Cellular Therapies, Inc.	Methods of treating vasomotor symptoms

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1143703A (is)	1965-03-18
GB1526331A (en) *	1976-01-14	1978-09-27	Kefalas As	Phthalanes
GB8419963D0 (en)	1984-08-06	1984-09-12	Lundbeck & Co As H	Intermediate compound and method
US5296007A (en)	1986-11-17	1994-03-22	Ensci Inc.	Process for removing sulfur from coal
GB8814057D0 (en)	1988-06-14	1988-07-20	Lundbeck & Co As H	New enantiomers & their isolation
DE19626659A1 (de)	1996-07-03	1998-01-08	Basf Ag	Verfahren zur Herstellung von Phthaliden
DE19627697A1 (de)	1996-07-10	1998-01-15	Basf Ag	Verfahren zur Herstellung von Phthaliden
TR200000066T2 (tr)	1997-07-08	2000-11-21	H. Lundbeck A/S	Sitalopram hazırlanması için yöntem.
UA62985C2 (en) *	1997-11-10	2004-01-15	Lunnbeck As H	A method for the preparation of citalopram
ES2149734T3 (es)	1997-11-11	2003-02-16	Lundbeck & Co As H	Metodo para la preparacion de citalopram.
PL199423B1 (pl)	1998-10-20	2008-09-30	Lundbeck & Co As H	Sposób wytwarzania citalopramu
CN1149208C (zh)	1998-12-23	2004-05-12	H.隆德贝克有限公司	制备5-氰基2-苯并[c]呋喃酮的方法
AR022329A1 (es)	1999-01-29	2002-09-04	Lundbeck & Co As H	Metodo para la preparacion de 5-cianoftalida
NZ514671A (en)	1999-04-14	2003-10-31	H	Method for the preparation of citalopram
ITMI991579A1 (it)	1999-06-25	2001-01-15	Lundbeck & Co As H	Metodo per la preparazione di citalopram
ITMI991581A1 (it)	1999-06-25	2001-01-15	Lundbeck & Co As H	Metodo per la preparazione di citalopram
CH692298A5 (de)	1999-10-25	2002-04-30	Lundbeck & Co As H	Verfahren zur Herstellung von Zwischenstufen für die Citalopramsynthese sowie zur Herstellung von Escitalopram.
US6310222B1 (en)	1999-11-01	2001-10-30	Sumika Fine Chemicals Co., Ltd.	Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate

2001
- 2001-02-21 NL NL1017415A patent/NL1017415C1/nl not_active IP Right Cessation
- 2001-02-21 FR FR0102339A patent/FR2805812A1/fr active Pending
- 2001-02-22 KR KR1020027011111A patent/KR20020081355A/ko not_active Withdrawn
- 2001-02-22 HR HRP20020660 patent/HRP20020660A2/hr not_active Application Discontinuation
- 2001-02-22 MX MXPA02008228A patent/MXPA02008228A/es unknown
- 2001-02-22 EP EP01907389A patent/EP1259501A2/en not_active Withdrawn
- 2001-02-22 SK SK1367-2002A patent/SK13672002A3/sk not_active Application Discontinuation
- 2001-02-22 JP JP2001544478A patent/JP2003523955A/ja not_active Withdrawn
- 2001-02-22 IL IL15105901A patent/IL151059A0/xx unknown
- 2001-02-22 CN CNA018055567A patent/CN1608057A/zh active Pending
- 2001-02-22 EA EA200200898A patent/EA005315B1/ru not_active IP Right Cessation
- 2001-02-22 CA CA002401236A patent/CA2401236A1/en not_active Abandoned
- 2001-02-22 IE IE20010163A patent/IES20010163A2/en not_active IP Right Cessation
- 2001-02-22 AU AU2001235358A patent/AU2001235358A1/en not_active Abandoned
- 2001-02-22 HU HU0300212A patent/HUP0300212A2/hu unknown
- 2001-02-22 WO PCT/DK2001/000123 patent/WO2001043525A2/en not_active Ceased
- 2001-02-22 GR GR20010100098A patent/GR1004073B/el unknown
- 2001-02-22 BR BR0108937-4A patent/BR0108937A/pt not_active IP Right Cessation
- 2001-02-22 PL PL01363119A patent/PL363119A1/xx not_active Application Discontinuation
- 2001-02-23 BE BE2001/0126A patent/BE1011177A6/fr not_active IP Right Cessation
- 2001-02-23 AR ARP010100836A patent/AR029658A1/es not_active Application Discontinuation
- 2001-02-26 US US09/794,762 patent/US6420574B2/en not_active Expired - Lifetime
- 2001-02-26 IT IT2001MI000386A patent/ITMI20010386A1/it unknown
2002
- 2002-07-29 IS IS6487A patent/IS6487A/is unknown
- 2002-08-19 NO NO20023928A patent/NO20023928D0/no not_active Application Discontinuation
- 2002-09-04 BG BG107061A patent/BG107061A/xx unknown

Also Published As

Publication number	Publication date
JP2003523955A (ja)	2003-08-12
GR1004073B (el)	2002-11-26
US20010027256A1 (en)	2001-10-04
MXPA02008228A (es)	2004-04-05
WO2001043525A3 (en)	2002-01-31
GR20010100098A (el)	2001-10-31
BE1011177A6 (fr)	2001-07-03
BR0108937A (pt)	2003-06-17
AU2001235358A1 (en)	2001-06-25
NO20023928L (no)	2002-08-19
EP1259501A2 (en)	2002-11-27
WO2001043525A2 (en)	2001-06-21
KR20020081355A (ko)	2002-10-26
NL1017415C1 (nl)	2001-05-18
IES20010163A2 (en)	2002-03-06
EA200200898A1 (ru)	2003-02-27
US6420574B2 (en)	2002-07-16
ITMI20010386A1 (it)	2002-08-26
PL363119A1 (en)	2004-11-15
EA005315B1 (ru)	2004-12-30
SK13672002A3 (sk)	2003-03-04
NO20023928D0 (no)	2002-08-19
AR029658A1 (es)	2003-07-10
BG107061A (en)	2003-05-30
FR2805812A1 (fr)	2001-09-07
CN1608057A (zh)	2005-04-20
HRP20020660A2 (en)	2004-12-31
HUP0300212A2 (hu)	2003-06-28
CA2401236A1 (en)	2001-06-21
IL151059A0 (en)	2003-04-10

Publication	Publication Date	Title
IS5884A (is)	2002-06-28	Aðferð til framleiðslu á hreinu sítalóprami
IS6091A (is)	2001-09-28	Aðferð til framleiðslu á sítalóprami
IS5862A (is)	2001-02-23	Aðferð til framleiðslu á sítalóprami
IS5861A (is)	2001-02-23	Aðferð til framleiðslu á sítalóprami
IS2121B (is)	2006-06-15	Aðferð til framleiðslu á sítalóprami
IS6512A (is)	2002-08-20	Aðferð til framleiðslu á sítalóprami
IS2256B (is)	2007-06-15	Aðferð til framleiðslu á sítalóprami
IS5473A (is)	2000-04-26	Aðferð til framleiðslu á sítalóprami
DE60205413D1 (de)	2005-09-15	Herstellungsverfahren
IS6834A (is)	2003-05-30	Aðferð til framleiðslu á amlódipín maleati
IS2223B (is)	2007-03-15	Aðferð til framleiðslu á 5-sýanóþalíði
IS2460B (is)	2008-11-15	Aðferð til framleiðslu á fituefnablöndu
IS5952A (is)	2001-05-22	Aðferð til framleiðslu á 5-sýanóþalíði
NO20023928L (no)	2002-08-19	Fremgangsmåte ved fremstillingen av citalopram
IS7239A (is)	2004-04-29	Aðferð til framleiðslu á essítalóprami
NO20041200L (no)	2004-03-23	Fremgangsmate for fremstilling av citalopram.
IS7153A (is)	2004-02-13	Aðferð til framleiðslu á 14-hýdroxýnormorfínon afleiðu
IS6526A (is)	2002-08-27	Aðferð til framleiðslu á sítalóprami
IS6605A (is)	2002-10-31	Aðferð til framleiðslu á sítalóprami
IS6529A (is)	2002-08-27	Aðferð til framleiðslu á sítalóprami
NO20031413D0 (no)	2003-03-27	Ny fremgangsmåte for fremstilling av oksabispidiner
IS6293A (is)	2002-03-05	Aðferð til framleiðslu á sítalóprami
IS2260B (is)	2007-06-15	Aðferð til framleiðslu á sítalóprami
IS6528A (is)	2002-08-27	Aðferð til framleiðslu á sítalóprami
IS5020A (is)	1999-10-11	Aðferð til framleiðslu á fenoxýfenýlsúlfónýl halíðum