IS8119A - Þétt N-heteróhringlaga efnasambönd og notkun þeirra sem CRF viðtakamótlyfja - Google Patents

Þétt N-heteróhringlaga efnasambönd og notkun þeirra sem CRF viðtakamótlyfja

Info

Publication number
IS8119A
IS8119A IS8119A IS8119A IS8119A IS 8119 A IS8119 A IS 8119A IS 8119 A IS8119 A IS 8119A IS 8119 A IS8119 A IS 8119A IS 8119 A IS8119 A IS 8119A
Authority
IS
Iceland
Prior art keywords
dense
receptor antagonists
heterocyclic compounds
crf receptor
crf
Prior art date
Application number
IS8119A
Other languages
English (en)
Inventor
Andreotti Daniele
Bernasconi Giovanni
Castiglioni Emiliano
Anne Contini Stefania
Di Fabio Romano
Fazzolari Elettra
Feriani Aldo
Gentile Gabriella
Mattioli Mario
Mingardi Anna
Maria Sabbatini Fabio
St-Denis Yves
Original Assignee
Sb Pharmco Puerto Rico Inc.
Neurocrine Biosciences Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sb Pharmco Puerto Rico Inc., Neurocrine Biosciences Inc. filed Critical Sb Pharmco Puerto Rico Inc.
Publication of IS8119A publication Critical patent/IS8119A/is

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • C07D487/04—Ortho-condensed systems

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Virology (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Otolaryngology (AREA)
  • Reproductive Health (AREA)
  • Communicable Diseases (AREA)
  • Urology & Nephrology (AREA)
  • Oncology (AREA)
  • Hospice & Palliative Care (AREA)
  • Molecular Biology (AREA)
  • Emergency Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
IS8119A 2003-04-09 2005-11-08 Þétt N-heteróhringlaga efnasambönd og notkun þeirra sem CRF viðtakamótlyfja IS8119A (is)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0308208.8A GB0308208D0 (en) 2003-04-09 2003-04-09 Chemical compounds
US48532203P 2003-07-07 2003-07-07
PCT/IB2004/001350 WO2004094420A1 (en) 2003-04-09 2004-04-07 Condensed n-heterocyclic compounds and their use as crf receptor antagonists

Publications (1)

Publication Number Publication Date
IS8119A true IS8119A (is) 2005-11-08

Family

ID=33312357

Family Applications (1)

Application Number Title Priority Date Filing Date
IS8119A IS8119A (is) 2003-04-09 2005-11-08 Þétt N-heteróhringlaga efnasambönd og notkun þeirra sem CRF viðtakamótlyfja

Country Status (21)

Country Link
US (2) US7427630B2 (is)
EP (3) EP2186813A1 (is)
JP (2) JP4866722B2 (is)
KR (1) KR20060021826A (is)
CN (1) CN1805958A (is)
AR (1) AR044005A1 (is)
AT (2) ATE473226T1 (is)
AU (1) AU2004232551C1 (is)
BR (1) BRPI0409117A (is)
CA (1) CA2521929C (is)
DE (2) DE602004027998D1 (is)
GB (1) GB0308208D0 (is)
IS (1) IS8119A (is)
MA (1) MA27796A1 (is)
MX (1) MXPA05010874A (is)
NO (1) NO20055238L (is)
NZ (1) NZ542780A (is)
PL (1) PL378755A1 (is)
RU (1) RU2382785C2 (is)
TW (1) TW200508232A (is)
WO (2) WO2004094420A1 (is)

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GB0117396D0 (en) 2001-07-17 2001-09-05 Glaxo Group Ltd Chemical compounds
MXPA06003150A (es) 2003-09-17 2006-08-31 Johnson & Johnson Compuestos heterociclicos fusionados.
AR046967A1 (es) * 2003-12-22 2006-01-04 Sb Pharmco Inc Compuesto de pirazol[1,5-a]pirimidina, composicion farmaceutica que lo comprende y su uso para preparar dicha composicion
WO2005103690A2 (en) * 2004-04-24 2005-11-03 Bayer Healthcare Ag Diagnostics and therapeutics for diseases associated with corticotropin releasing hormone receptor 2 (crhr2)
DE602005014375D1 (de) * 2004-10-19 2009-06-18 Neurocrine Biosciences Inc Crf-rezeptor-antagonisten und zugehörige verfahren
GB0519957D0 (en) * 2005-09-30 2005-11-09 Sb Pharmco Inc Chemical compound
GB0507198D0 (en) * 2005-04-08 2005-05-18 Sb Pharmco Inc Process for preparing bicyclic compounds
GB0507195D0 (en) * 2005-04-08 2005-05-18 Sb Pharmco Inc Process for preparing bicyclic compounds
US7598255B2 (en) 2005-08-04 2009-10-06 Janssen Pharmaceutica Nv Pyrimidine compounds as serotonin receptor modulators
US8088779B2 (en) * 2005-09-30 2012-01-03 Smithkline Beecham (Cork) Limited Pyrazolo [1,5-alpha] pyrimidinyl derivatives useful as corticotropin-releasing factor (CRF) receptor antagonists
DE602007011628D1 (de) 2006-07-06 2011-02-10 Array Biopharma Inc Dihydrofuropyrimidine als akt-proteinkinaseinhibitoren
US8063050B2 (en) 2006-07-06 2011-11-22 Array Biopharma Inc. Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors
EP2054418B1 (en) 2006-07-06 2011-11-09 Array Biopharma Inc. Dihydrothieno pyrimidines as akt protein kinase inhibitors
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