IS8322A - Tálmar Akt virkni - Google Patents

Tálmar Akt virkni

Info

Publication number
IS8322A
IS8322A IS8322A IS8322A IS8322A IS 8322 A IS8322 A IS 8322A IS 8322 A IS8322 A IS 8322A IS 8322 A IS8322 A IS 8322A IS 8322 A IS8322 A IS 8322A
Authority
IS
Iceland
Prior art keywords
impairs
akt activity
akt
activity
impairs akt
Prior art date
Application number
IS8322A
Other languages
English (en)
Inventor
A. Heerding Dirk
J. Clark Tammy
H. Drewry David
Dale Leber Jack
Safonov Igor
S. Yamashita Dennis
Original Assignee
Smithkline Beecham Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Corporation filed Critical Smithkline Beecham Corporation
Publication of IS8322A publication Critical patent/IS8322A/is

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965Non-condensed pyrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IS8322A 2003-07-29 2006-02-22 Tálmar Akt virkni IS8322A (is)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US49085103P 2003-07-29 2003-07-29
US49105503P 2003-07-30 2003-07-30
US49310103P 2003-08-06 2003-08-06
US49475203P 2003-08-13 2003-08-13
US50701403P 2003-09-29 2003-09-29
US53084703P 2003-12-18 2003-12-18
PCT/US2004/024340 WO2005011700A1 (en) 2003-07-29 2004-07-28 INHIBITORS OF Akt ACTIVITY

Publications (1)

Publication Number Publication Date
IS8322A true IS8322A (is) 2006-02-22

Family

ID=34120170

Family Applications (1)

Application Number Title Priority Date Filing Date
IS8322A IS8322A (is) 2003-07-29 2006-02-22 Tálmar Akt virkni

Country Status (16)

Country Link
US (1) US20080255143A1 (is)
EP (1) EP1653961A4 (is)
JP (1) JP2007500709A (is)
KR (1) KR20060066714A (is)
AR (1) AR045134A1 (is)
AU (1) AU2004261214A1 (is)
BR (1) BRPI0412993A (is)
CA (1) CA2534038A1 (is)
CO (1) CO5640140A2 (is)
IL (1) IL173174A0 (is)
IS (1) IS8322A (is)
MA (1) MA27933A1 (is)
MX (1) MXPA06001134A (is)
NO (1) NO20060985L (is)
TW (1) TW200523262A (is)
WO (1) WO2005011700A1 (is)

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JP2007507547A (ja) * 2003-10-06 2007-03-29 グラクソ グループ リミテッド キナーゼ阻害剤としての1,7−二置換アザベンゾイミダゾールの調製
JP2007510667A (ja) * 2003-11-07 2007-04-26 スミスクライン ビーチャム (コーク) リミテッド 癌の治療法

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KR20060066714A (ko) 2006-06-16
WO2005011700A1 (en) 2005-02-10
EP1653961A1 (en) 2006-05-10
US20080255143A1 (en) 2008-10-16
CA2534038A1 (en) 2005-02-10
MXPA06001134A (es) 2006-04-11
NO20060985L (no) 2006-04-19
IL173174A0 (en) 2006-06-11
AU2004261214A1 (en) 2005-02-10
CO5640140A2 (es) 2006-05-31
BRPI0412993A (pt) 2006-10-03
AR045134A1 (es) 2005-10-19
MA27933A1 (fr) 2006-06-01
EP1653961A4 (en) 2009-04-01
JP2007500709A (ja) 2007-01-18

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