IT8348005A0 - 3,4-diammino-1,2,5-tiadiazoli dotati di attivita' antagonista dei recettori istaminici - Google Patents

3,4-diammino-1,2,5-tiadiazoli dotati di attivita' antagonista dei recettori istaminici

Info

Publication number: IT8348005A0
Authority: IT; Italy
Prior art keywords: histamines; thiadiazoles; diamino; receptor antagonist; antagonist activity
Prior art date: 1982-03-29

Application number

IT8348005A

Other languages

English (en)

Other versions

IT1164633B (it

Inventor

Crenshaw Ronnie Ray

Algieri Aldo Antonio

Original Assignee

Bristol Myers Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1982-03-29

Filing date

1983-03-28

Publication date

1983-03-28

1983-03-28 Application filed by Bristol Myers Co filed Critical Bristol Myers Co

1983-03-28 Publication of IT8348005A0 publication Critical patent/IT8348005A0/it

1987-04-15 Application granted granted Critical

1987-04-15 Publication of IT1164633B publication Critical patent/IT1164633B/it

Links

239000002464 receptor antagonist Substances 0.000 title 1
229940044551 receptor antagonist Drugs 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/06—1,2,3-Thiadiazoles; Hydrogenated 1,2,3-thiadiazoles
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/10—1,2,5-Thiadiazoles; Hydrogenated 1,2,5-thiadiazoles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Heterocyclic Compounds Containing Sulfur Atoms (AREA)
Pyridine Compounds (AREA)
Furan Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Hydrogenated Pyridines (AREA)
Pyrrole Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

IT48005/83A 1982-03-29 1983-03-28 3,4-diammino-1,2,5-tiadiazoli dotati di attivita' antagonista dei recettori istaminici IT1164633B (it)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US36320782A	1982-03-29	1982-03-29

Publications (2)

Publication Number	Publication Date
IT8348005A0 true IT8348005A0 (it)	1983-03-28
IT1164633B IT1164633B (it)	1987-04-15

Family

ID=23429274

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IT48005/83A IT1164633B (it)	1982-03-29	1983-03-28	3,4-diammino-1,2,5-tiadiazoli dotati di attivita' antagonista dei recettori istaminici

Country Status (30)

Country	Link
JP (2)	JPS58180477A (it)
KR (1)	KR880002209B1 (it)
AT (1)	AT386599B (it)
AU (2)	AU557577B2 (it)
BE (1)	BE896291A (it)
CH (2)	CH660880A5 (it)
CS (2)	CS250229B2 (it)
DD (2)	DD219768A5 (it)
DE (1)	DE3311281A1 (it)
DK (2)	DK166677B1 (it)
ES (3)	ES520982A0 (it)
FR (2)	FR2542741B1 (it)
GB (2)	GB2117769B (it)
GR (1)	GR78524B (it)
HU (2)	HU196386B (it)
IE (1)	IE55596B1 (it)
IL (1)	IL68259A0 (it)
IT (1)	IT1164633B (it)
LU (1)	LU84716A1 (it)
MY (1)	MY8700942A (it)
NL (1)	NL8301063A (it)
NO (1)	NO163055C (it)
NZ (1)	NZ203726A (it)
OA (1)	OA07356A (it)
PT (1)	PT76459B (it)
SE (2)	SE461040B (it)
SU (2)	SU1419518A3 (it)
YU (1)	YU44849B (it)
ZA (1)	ZA832154B (it)
ZW (1)	ZW7683A1 (it)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU2222083A (en) *	1982-12-14	1984-06-21	Smith Kline & French Laboratories Limited	Pyridine derivatives
US4593039A (en) *	1984-04-02	1986-06-03	Merck & Co., Inc.	1-aryloxy-3-(substituted aminoalkylamino)-2-propanols
US4644006A (en) *	1984-06-22	1987-02-17	Bristol-Myers Company	Substituted 3,4-diamino-1,2,5-thiadiazoles having histamine H2 -receptor antagonist activity
JPH0622828B2 (ja) *	1986-06-30	1994-03-30	フアナツク株式会社	直圧式型締機構
EP4196793A1 (en)	2020-08-11	2023-06-21	Université de Strasbourg	H2 blockers targeting liver macrophages for the prevention and treatment of liver disease and cancer

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3018289A (en) *	1960-02-10	1962-01-23	Wyandotte Chemicals Corp	Process for preparing oxamidines
GB1595291A (en) *	1976-09-21	1981-08-12	Smith Kline French Lab	Pyrimidone and thiopyrimidone derivatives
DK160611C (da) *	1979-09-04	1991-09-16	Bristol Myers Squibb Co	Analogifremgangsmaade til fremstilling af 3,4-disubstituerede 1,2,5-thiadiazol-1-oxider og -1,1-dioxider
DE3175201D1 (en) *	1980-04-30	1986-10-02	Merck & Co Inc	Aminothiadiazoles as gastric secretion inhibitors
AU2222083A (en) *	1982-12-14	1984-06-21	Smith Kline & French Laboratories Limited	Pyridine derivatives

1983
- 1983-03-25 ZA ZA832154A patent/ZA832154B/xx unknown
- 1983-03-25 ZW ZW76/83A patent/ZW7683A1/xx unknown
- 1983-03-25 NL NL8301063A patent/NL8301063A/nl not_active Application Discontinuation
- 1983-03-25 ES ES520982A patent/ES520982A0/es active Granted
- 1983-03-25 FR FR838304934A patent/FR2542741B1/fr not_active Expired
- 1983-03-28 PT PT76459A patent/PT76459B/pt not_active IP Right Cessation
- 1983-03-28 IE IE686/83A patent/IE55596B1/en not_active IP Right Cessation
- 1983-03-28 GR GR70903A patent/GR78524B/el unknown
- 1983-03-28 BE BE0/210417A patent/BE896291A/fr not_active IP Right Cessation
- 1983-03-28 SE SE8301725A patent/SE461040B/sv not_active IP Right Cessation
- 1983-03-28 AU AU12907/83A patent/AU557577B2/en not_active Ceased
- 1983-03-28 IT IT48005/83A patent/IT1164633B/it active
- 1983-03-28 HU HU854071A patent/HU196386B/hu not_active IP Right Cessation
- 1983-03-28 DK DK141383A patent/DK166677B1/da not_active IP Right Cessation
- 1983-03-28 NO NO831100A patent/NO163055C/no unknown
- 1983-03-28 IL IL68259A patent/IL68259A0/xx not_active IP Right Cessation
- 1983-03-28 GB GB08308518A patent/GB2117769B/en not_active Expired
- 1983-03-28 DE DE19833311281 patent/DE3311281A1/de not_active Withdrawn
- 1983-03-28 HU HU831040A patent/HU188742B/hu not_active IP Right Cessation
- 1983-03-28 SU SU833568849A patent/SU1419518A3/ru active
- 1983-03-28 NZ NZ203726A patent/NZ203726A/en unknown
- 1983-03-28 LU LU84716A patent/LU84716A1/fr unknown
- 1983-03-29 KR KR1019830001283A patent/KR880002209B1/ko not_active Expired
- 1983-03-29 JP JP58051740A patent/JPS58180477A/ja active Granted
- 1983-03-29 CH CH575/86A patent/CH660880A5/de not_active IP Right Cessation
- 1983-03-29 DD DD83260707A patent/DD219768A5/de not_active IP Right Cessation
- 1983-03-29 CH CH1749/83A patent/CH655111A5/de not_active IP Right Cessation
- 1983-03-29 DD DD83249300A patent/DD210909A5/de not_active IP Right Cessation
- 1983-03-29 OA OA57955A patent/OA07356A/xx unknown
- 1983-03-29 CS CS832191A patent/CS250229B2/cs unknown
- 1983-03-29 AT AT0111083A patent/AT386599B/de not_active IP Right Cessation
- 1983-03-29 CS CS841958A patent/CS250240B2/cs unknown
- 1983-03-29 YU YU744/83A patent/YU44849B/xx unknown
- 1983-11-30 ES ES527685A patent/ES527685A0/es active Granted
- 1983-11-30 ES ES527686A patent/ES8505978A1/es not_active Expired
1984
- 1984-06-08 SU SU843750493A patent/SU1355123A3/ru active
- 1984-12-31 GB GB08432809A patent/GB2149406B/en not_active Expired
1986
- 1986-09-30 AU AU63272/86A patent/AU586037B2/en not_active Ceased
1987
- 1987-05-22 FR FR878707197A patent/FR2597867B1/fr not_active Expired
- 1987-11-25 SE SE8704689A patent/SE464302B/sv not_active IP Right Cessation
- 1987-12-30 MY MY942/87A patent/MY8700942A/xx unknown
1992
- 1992-06-18 DK DK92811A patent/DK81192D0/da not_active Application Discontinuation
1993
- 1993-04-16 JP JP5124585A patent/JPH06135925A/ja active Pending

Also Published As

Publication number	Publication date
ES8505977A1 (es)	1985-06-16
YU44849B (en)	1991-04-30
GB2149406A (en)	1985-06-12
JPH06135925A (ja)	1994-05-17
DK166677B1 (da)	1993-06-28
DK141383A (da)	1983-09-30
JPS58180477A (ja)	1983-10-21
NO163055C (no)	1990-03-28
IE830686L (en)	1983-09-29
OA07356A (fr)	1984-08-31
CH660880A5 (de)	1987-05-29
KR840004095A (ko)	1984-10-06
ES8404683A1 (es)	1984-05-16
GB2149406B (en)	1986-01-02
ES520982A0 (es)	1984-05-16
LU84716A1 (fr)	1983-12-05
GB8432809D0 (en)	1985-02-06
NL8301063A (nl)	1983-10-17
PT76459B (en)	1986-03-11
ES527685A0 (es)	1985-06-16
IT1164633B (it)	1987-04-15
AU586037B2 (en)	1989-06-29
FR2597867B1 (fr)	1989-12-08
HU196386B (en)	1988-11-28
HU188742B (en)	1986-05-28
CS250229B2 (en)	1987-04-16
DE3311281A1 (de)	1983-11-24
SE8301725D0 (sv)	1983-03-28
AT386599B (de)	1988-09-12
ATA111083A (de)	1988-02-15
MY8700942A (en)	1987-12-31
ZA832154B (en)	1983-12-28
SE8704689L (sv)	1987-11-25
DK81192A (da)	1992-06-18
CH655111A5 (de)	1986-03-27
SE8704689D0 (sv)	1987-11-25
NO163055B (no)	1989-12-18
ZW7683A1 (en)	1984-01-04
AU1290783A (en)	1983-10-06
NO831100L (no)	1983-09-30
DD210909A5 (de)	1984-06-27
SE8301725L (sv)	1983-11-25
CS250240B2 (en)	1987-04-16
FR2597867A1 (fr)	1987-10-30
DK141383D0 (da)	1983-03-28
AU6327286A (en)	1987-01-08
SU1419518A3 (ru)	1988-08-23
KR880002209B1 (ko)	1988-10-18
DD219768A5 (de)	1985-03-13
GB2117769A (en)	1983-10-19
GR78524B (it)	1984-09-27
ES527686A0 (es)	1985-06-16
ES8505978A1 (es)	1985-06-16
SU1355123A3 (ru)	1987-11-23
FR2542741B1 (fr)	1989-12-08
PT76459A (en)	1983-04-01
BE896291A (fr)	1983-09-28
YU74483A (en)	1986-02-28
SE464302B (sv)	1991-04-08
JPH0568472B2 (it)	1993-09-29
NZ203726A (en)	1986-05-09
IL68259A0 (en)	1983-06-15
SE461040B (sv)	1989-12-18
FR2542741A1 (fr)	1984-09-21
GB2117769B (en)	1985-08-29
IE55596B1 (en)	1990-11-21
AU557577B2 (en)	1986-12-24
DK81192D0 (da)	1992-06-18
GB8308518D0 (en)	1983-05-05

Publication	Publication Date	Title
ATE52495T1 (de)	1990-05-15	2-(2'-nitrobenzoyl)-1,3-cyclohexandionen.
TR22585A (tr)	1987-12-07	Bazi 2-(2'-alkilbenzoil)-1,3-sikloheksandion'lar
FI865263A7 (fi)	1987-06-24	Laett, elektromagnetisk transduktor med stor effekt.
DE3586192D1 (de)	1992-07-16	Roentgen-anordnung.
FI834202A0 (fi)	1983-11-16	Slangformigt livsmedelshoelje, i synnerhet korvskinn med foerbaettrad avskalbarhet
NO167168C (no)	1991-10-09	Naerhetstenner med justerbart naerhetsomraade.
MX163934B (es)	1992-07-01	Procedimiento para preparar haluros de 1-metil-3,5,7-triaza-1-azoniatriciclodecano
FI894675A7 (fi)	1990-04-05	Muskarinreceptorantagonister.
OA07356A (fr)	1984-08-31	3,4-Diamino-1,2,5-thiadiazoles substitués possedant une activité antagoniste du récepteur-H2 de l'histamine.
IT1227503B (it)	1991-04-12	Scaldabevande, specialmente per impiego domestico
IT8319192A0 (it)	1983-01-20	1,3,4-tiadiazolo [3,2-a] pirimidine sostituite e procedimento per laloro preparazione
IT1140961B (it)	1986-10-10	Procedimento di preparazione di 5-mercapto-1,2,3-triazoli
TR20096A (tr)	1980-07-08	2-(2'2'-dihalojenovinil)-ve 2(2',2',2'-trihalojenoetil)-siklomutano lar
IT8521217A0 (it)	1985-06-20	3,4-diammino-1,2,5-tiadiazoli sostituiti aventi attivita'antagonista nei confronti di h2-recettori della istamina.
RO86358A2 (ro)	1985-03-15	Procedeu pentru prepararea unor 1,2,4-triazolil-u-il-propionitrili
NO851398L (no)	1985-10-04	Taakeleggingslegeme.
ES542499A0 (es)	1986-06-16	Derivados anillados de 4h-1,4-benzotiazina
DE3576574D1 (de)	1990-04-19	Roentgenvorrichtung.
ES264437Y (es)	1983-05-16	"porta-servilletas perfeccionado".
ES546784A0 (es)	1986-01-01	Procedimiento de obtencion del 2,6-dimetil-3-metoxicarbonil-4-(2-nitrofenil)-1,4-dihidropiridina-5-carboxilato de isobu-tilo
ES295626Y (es)	1989-04-16	Bolsa mejorada para urostomia
DE3574786D1 (de)	1990-01-18	Roentgenvorrichtung.
ES264126Y (es)	1983-05-16	"asiento perfeccionado".
ES263615Y (es)	1983-10-16	"asiento".
IT8423967A0 (it)	1984-12-10	Composti eterociclici dotati di attivita' terapeutica.