JPH04210632A - 血管拡張剤および免疫抑制薬２−イソプロピル−２−フェニルアミノバレロニトリルの使用方法 - Google Patents

血管拡張剤および免疫抑制薬２−イソプロピル−２−フェニルアミノバレロニトリルの使用方法

Info

Publication number: JPH04210632A
Authority: JP; Japan
Prior art keywords: formulas; formula; chemical; tables; following structural
Prior art date: 1989-12-21
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Withdrawn

Application number

JP2419052A

Other languages

English (en)

Japanese (ja)

Inventor

Liang Chi-Dean

チ　−　ディーン　リアング

Richard August Mueller

リチャード　オーガスト　ミューラー

Kearn John P Mc

ジョン　ピー．マックカーン

Terry B Strom

テリー　ピー．ストロム

Kenneth J Wieder

ケネス　ジェイ．ウィーダー

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

GD Searle LLC

Original Assignee

GD Searle LLC

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1989-12-21

Filing date

1990-12-21

Publication date

1992-07-31

1990-12-21 Application filed by GD Searle LLC filed Critical GD Searle LLC

1992-07-31 Publication of JPH04210632A publication Critical patent/JPH04210632A/ja

Status Withdrawn legal-status Critical Current

Links

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Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
- C07C255/01—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
- C07C255/32—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring
- C07C255/42—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by singly-bound nitrogen atoms, not being further bound to other hetero atoms
- C07C255/43—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by singly-bound nitrogen atoms, not being further bound to other hetero atoms the carbon skeleton being further substituted by singly-bound oxygen atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Immunology (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Urology & Nephrology (AREA)
Biomedical Technology (AREA)
Psychiatry (AREA)
Hospice & Palliative Care (AREA)
Transplantation (AREA)
Vascular Medicine (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

JP2419052A 1989-12-21 1990-12-21 血管拡張剤および免疫抑制薬２−イソプロピル−２−フェニルアミノバレロニトリルの使用方法 Withdrawn JPH04210632A (ja)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US45600789A	1989-12-21	1989-12-21
US456007		1989-12-21

Publications (1)

Publication Number	Publication Date
JPH04210632A true JPH04210632A (ja)	1992-07-31

Family

ID=23811068

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
JP2419052A Withdrawn JPH04210632A (ja)	1989-12-21	1990-12-21	血管拡張剤および免疫抑制薬２−イソプロピル−２−フェニルアミノバレロニトリルの使用方法

Country Status (10)

Country	Link
EP (1)	EP0434094B1 (de)
JP (1)	JPH04210632A (de)
AT (1)	ATE87614T1 (de)
CA (1)	CA2033038A1 (de)
DE (1)	DE69001240T2 (de)
DK (1)	DK0434094T3 (de)
ES (1)	ES2054207T3 (de)
GR (1)	GR3008320T3 (de)
IE (1)	IE64870B1 (de)
PT (1)	PT96283A (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
PT2170050E (pt)	2007-06-20	2014-09-04	Milestone Pharmaceuticals Inc	Bloqueadores de canais de cálcio de fenilalquilamina de atuação curta e suas utilizações

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3642331A1 (de) *	1986-12-11	1988-06-23	Basf Ag	Basisch substituierte phenylacetonitrile, ihre herstellung und diese enthaltende arzneimittel

1990
- 1990-12-20 IE IE462790A patent/IE64870B1/en not_active IP Right Cessation
- 1990-12-20 PT PT96283A patent/PT96283A/pt not_active Application Discontinuation
- 1990-12-21 DK DK90125244.5T patent/DK0434094T3/da active
- 1990-12-21 JP JP2419052A patent/JPH04210632A/ja not_active Withdrawn
- 1990-12-21 AT AT90125244T patent/ATE87614T1/de not_active IP Right Cessation
- 1990-12-21 EP EP90125244A patent/EP0434094B1/de not_active Expired - Lifetime
- 1990-12-21 ES ES90125244T patent/ES2054207T3/es not_active Expired - Lifetime
- 1990-12-21 DE DE9090125244T patent/DE69001240T2/de not_active Expired - Fee Related
- 1990-12-21 CA CA002033038A patent/CA2033038A1/en not_active Abandoned
1993
- 1993-06-30 GR GR930400669T patent/GR3008320T3/el unknown

Also Published As

Publication number	Publication date
IE64870B1 (en)	1995-09-20
DE69001240D1 (de)	1993-05-06
ATE87614T1 (de)	1993-04-15
PT96283A (pt)	1991-09-30
DE69001240T2 (de)	1993-08-05
GR3008320T3 (de)	1993-09-30
EP0434094B1 (de)	1993-03-31
IE904627A1 (en)	1991-07-17
ES2054207T3 (es)	1994-08-01
EP0434094A1 (de)	1991-06-26
CA2033038A1 (en)	1991-06-22
DK0434094T3 (da)	1993-08-16

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1998-03-10

A300

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Effective date: 19980312

Publication	Publication Date	Title
JP4151765B2 (ja)	2008-09-17	免疫調節活性を有する新規な置換プリニル誘導体
PT1438966E (pt)	2007-05-31	Uso de depsipéptidos e seus congéneres como imunosupressores para tratamento de doenças infecciosas, como uma doença autoimune, reacções alérgicas ou doença hiperproliferativa da pele.
CA2218606A1 (en)	1996-10-24	Novel peptide derivatives
JPS60215700A (ja)	1985-10-29	新規シクロスポリン類
CN104768968B (zh)	2019-04-05	环状缩酚肽化合物及其用途
CA2486872A1 (en)	2003-12-11	Nf-kb inhibitors and uses thereof
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JPH04210632A (ja)	1992-07-31	血管拡張剤および免疫抑制薬２−イソプロピル−２−フェニルアミノバレロニトリルの使用方法
WO2012170792A1 (en)	2012-12-13	Atazanavir metabolite derivatives
CA2294011A1 (en)	1998-12-23	Use of draflazine-analogues for treating pain
US6197793B1 (en)	2001-03-06	Hemoregulatory compounds
JP2002515864A (ja)	2002-05-28	造血性細胞増殖のペプチド阻害剤
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