JPH11506469A5 - - Google Patents

Info

Publication number
JPH11506469A5
JPH11506469A5 JP1997502238A JP50223897A JPH11506469A5 JP H11506469 A5 JPH11506469 A5 JP H11506469A5 JP 1997502238 A JP1997502238 A JP 1997502238A JP 50223897 A JP50223897 A JP 50223897A JP H11506469 A5 JPH11506469 A5 JP H11506469A5
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
JP1997502238A
Other languages
English (en)
Japanese (ja)
Other versions
JPH11506469A (ja
Filing date
Publication date
Priority claimed from US08/485,038 external-priority patent/US6071970A/en
Application filed filed Critical
Publication of JPH11506469A publication Critical patent/JPH11506469A/ja
Publication of JPH11506469A5 publication Critical patent/JPH11506469A5/ja
Ceased legal-status Critical Current

Links

JP9502238A 1995-06-07 1996-06-07 神経障害の治療に有用な受容体作動性カルシウムチャネル上の新規部位で活性な化合物 Ceased JPH11506469A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US08/485,038 US6071970A (en) 1993-02-08 1995-06-07 Compounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders and diseases
US08/485,038 1995-06-07
PCT/US1996/010201 WO1996040097A1 (en) 1995-06-07 1996-06-07 Compounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders

Publications (2)

Publication Number Publication Date
JPH11506469A JPH11506469A (ja) 1999-06-08
JPH11506469A5 true JPH11506469A5 (2) 2004-07-29

Family

ID=23926692

Family Applications (1)

Application Number Title Priority Date Filing Date
JP9502238A Ceased JPH11506469A (ja) 1995-06-07 1996-06-07 神経障害の治療に有用な受容体作動性カルシウムチャネル上の新規部位で活性な化合物

Country Status (17)

Country Link
US (2) US6071970A (2)
EP (1) EP0831799B1 (2)
JP (1) JPH11506469A (2)
KR (1) KR100430022B1 (2)
CN (1) CN1153568C (2)
AT (1) ATE238782T1 (2)
AU (1) AU716122B2 (2)
BR (1) BR9609019A (2)
CA (1) CA2223978A1 (2)
DE (1) DE69627852T2 (2)
DK (1) DK0831799T3 (2)
ES (1) ES2197945T3 (2)
NZ (1) NZ310344A (2)
PL (1) PL185492B1 (2)
PT (1) PT831799E (2)
RU (1) RU2246300C2 (2)
WO (1) WO1996040097A1 (2)

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US7087765B2 (en) 1995-06-07 2006-08-08 Nps Pharmaceuticals, Inc. Compounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders and diseases
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KR101616246B1 (ko) 2008-01-25 2016-05-02 그뤼넨탈 게엠베하 약제학적 투여형
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CN101838235B (zh) * 2009-06-12 2013-08-07 重庆华邦制药有限公司 3-苯基-3＇-吡啶基丙烯胺类化合物及其合成方法
WO2011009602A1 (en) 2009-07-22 2011-01-27 Grünenthal GmbH Hot-melt extruded controlled release dosage form
TWI473628B (zh) 2009-07-22 2015-02-21 用於對氧化敏感之類鴉片藥劑之抗破壞劑型
CA2808219C (en) 2010-09-02 2019-05-14 Gruenenthal Gmbh Tamper resistant dosage form comprising inorganic salt
WO2012028318A1 (en) 2010-09-02 2012-03-08 Grünenthal GmbH Tamper resistant dosage form comprising an anionic polymer
AU2012289764B2 (en) 2011-07-29 2017-03-02 Grünenthal GmbH Tamper-resistant tablet providing immediate drug release
ES2648129T3 (es) 2011-07-29 2017-12-28 Grünenthal GmbH Pastilla a prueba de manipulación que proporciona una liberación inmediata de un medicamento
US20130225697A1 (en) 2012-02-28 2013-08-29 Grunenthal Gmbh Tamper-resistant dosage form comprising pharmacologically active compound and anionic polymer
PL2838512T3 (pl) 2012-04-18 2018-12-31 Grünenthal GmbH Farmaceutyczna postać dawkowania odporna na niewłaściwe użycie i odporna na uderzeniowe uwalnianie dawki
US10064945B2 (en) 2012-05-11 2018-09-04 Gruenenthal Gmbh Thermoformed, tamper-resistant pharmaceutical dosage form containing zinc
AU2014273227B2 (en) 2013-05-29 2019-08-15 Grunenthal Gmbh Tamper-resistant dosage form containing one or more particles
JP6466417B2 (ja) 2013-05-29 2019-02-06 グリュネンタール・ゲゼルシャフト・ミト・ベシュレンクテル・ハフツング 二峰性放出プロファイルを有する改変防止（ｔａｍｐｅｒ−ｒｅｓｉｓｔａｎｔ）剤形
JP6449871B2 (ja) 2013-07-12 2019-01-09 グリュネンタール・ゲゼルシャフト・ミト・ベシュレンクテル・ハフツング エチレン−酢酸ビニルポリマーを含有する改変防止剤形
EP3073994A1 (en) 2013-11-26 2016-10-05 Grünenthal GmbH Preparation of a powdery pharmaceutical composition by means of cryo-milling
EP3142646A1 (en) 2014-05-12 2017-03-22 Grünenthal GmbH Tamper resistant immediate release capsule formulation comprising tapentadol
EA201692388A1 (ru) 2014-05-26 2017-05-31 Грюненталь Гмбх Лекарственная форма в виде множества частиц, защищенная от вызываемого этанолом сброса дозы
BR112017021475A2 (pt) 2015-04-24 2018-07-10 Gruenenthal Gmbh forma de dosagem resistente à adulteração (tamper) com liberação imediata e resistência contra extração de solvente
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