JPS5287191A - Process for preparing semiisynthetic penicillin antibiotics - Google Patents

Process for preparing semiisynthetic penicillin antibiotics

Info

Publication number
JPS5287191A
JPS5287191A JP252077A JP252077A JPS5287191A JP S5287191 A JPS5287191 A JP S5287191A JP 252077 A JP252077 A JP 252077A JP 252077 A JP252077 A JP 252077A JP S5287191 A JPS5287191 A JP S5287191A
Authority
JP
Japan
Prior art keywords
semiisynthetic
preparing
penicillin antibiotics
penicillin
antibiotics
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP252077A
Other languages
English (en)
Japanese (ja)
Inventor
Kurochi Maruko
Kotsuchi Jino
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Glaxo Laboratories Ltd
Original Assignee
Glaxo Laboratories Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Laboratories Ltd filed Critical Glaxo Laboratories Ltd
Publication of JPS5287191A publication Critical patent/JPS5287191A/ja
Pending legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/44Compounds with an amino radical acylated by carboxylic acids, attached in position 6
    • C07D499/48Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
    • C07D499/58Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical
    • C07D499/64Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms
    • C07D499/68Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms with aromatic rings as additional substituents on the carbon chain
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/04Preparation
    • C07D499/10Modification of an amino radical directly attached in position 6
    • C07D499/12Acylation

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
JP252077A 1976-01-15 1977-01-14 Process for preparing semiisynthetic penicillin antibiotics Pending JPS5287191A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT47643/76A IT1053313B (it) 1976-01-15 1976-01-15 Procedimento per produrre antibiotici semisintetici

Publications (1)

Publication Number Publication Date
JPS5287191A true JPS5287191A (en) 1977-07-20

Family

ID=11261624

Family Applications (1)

Application Number Title Priority Date Filing Date
JP252077A Pending JPS5287191A (en) 1976-01-15 1977-01-14 Process for preparing semiisynthetic penicillin antibiotics

Country Status (14)

Country Link
JP (1) JPS5287191A (da)
AU (1) AU512150B2 (da)
BE (1) BE850382A (da)
CH (1) CH627182A5 (da)
DE (1) DE2701406A1 (da)
DK (1) DK13977A (da)
ES (1) ES455026A1 (da)
FR (1) FR2338279A1 (da)
GB (1) GB1569427A (da)
IT (1) IT1053313B (da)
NL (1) NL7700396A (da)
SE (1) SE437989B (da)
YU (1) YU9277A (da)
ZA (1) ZA77195B (da)

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS523093A (en) * 1975-06-26 1977-01-11 Dobfar Spa Production of 66aminopencillanic acid and 77 aminodexethoxycephalospolanic acid derivative

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB958478A (en) * 1962-03-13 1964-05-21 Beecham Res Lab Production of penicillins
FR68F (da) * 1962-10-17
US3351597A (en) * 1966-11-23 1967-11-07 Lilly Co Eli Process for acylating 7-amino cephalosporanic acid
ZA695612B (en) * 1968-08-23 1971-03-31 Lilly Co Eli Preparation of cephalosporin compounds
US3595855A (en) * 1968-12-05 1971-07-27 American Home Prod Process for producing aminopenicillins
IT1043957B (it) * 1970-12-31 1980-02-29 Lorenzini Sas Inst Biochim Processo per la preparazione della forma anidra dell acido 6, d, meno alfa aminofenilacetamido penicillanico
GB1494902A (en) * 1974-05-09 1977-12-14 Glaxo Lab Ltd Penicillins

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS523093A (en) * 1975-06-26 1977-01-11 Dobfar Spa Production of 66aminopencillanic acid and 77 aminodexethoxycephalospolanic acid derivative

Also Published As

Publication number Publication date
DK13977A (da) 1977-07-16
NL7700396A (nl) 1977-07-19
ZA77195B (en) 1977-11-30
AU512150B2 (en) 1980-09-25
SE7700393L (sv) 1977-07-16
CH627182A5 (en) 1981-12-31
SE437989B (sv) 1985-03-25
IT1053313B (it) 1981-08-31
FR2338279B1 (da) 1980-09-05
YU9277A (en) 1982-06-30
FR2338279A1 (fr) 1977-08-12
ES455026A1 (es) 1977-12-16
GB1569427A (en) 1980-06-18
AU2134077A (en) 1978-07-20
BE850382A (fr) 1977-07-14
DE2701406A1 (de) 1977-07-21

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