JPS56122384A - 7alpha-methoxycephalosporin derivative, its preparation and antifungal agent comprising it - Google Patents

7alpha-methoxycephalosporin derivative, its preparation and antifungal agent comprising it

Info

Publication number: JPS56122384A
Authority: JP; Japan
Prior art keywords: formula; compound shown; 7alpha; preparation; bacteria
Prior art date: 1980-03-04
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Pending

Application number

JP2611280A

Other languages

English (en)

Japanese (ja)

Inventor

Yoshimasa Machida

Isao Saito

Seiichiro Nomoto

Shigeto Negi

Hironori Ikuta

Kyosuke Kito

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Eisai Co Ltd

Original Assignee

Eisai Co Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1980-03-04

Filing date

1980-03-04

Publication date

1981-09-25

1980-03-04 Application filed by Eisai Co Ltd filed Critical Eisai Co Ltd

1980-03-04 Priority to JP2611280A priority Critical patent/JPS56122384A/ja

1980-12-22 Priority to SE8009049A priority patent/SE8009049L/xx

1980-12-22 Priority to DK548380A priority patent/DK548380A/da

1980-12-23 Priority to DE19803048657 priority patent/DE3048657A1/de

1980-12-23 Priority to HU803106A priority patent/HU183276B/hu

1980-12-23 Priority to GB8041201A priority patent/GB2070589B/en

1980-12-23 Priority to NL8007011A priority patent/NL8007011A/nl

1980-12-23 Priority to AT0630780A priority patent/AT373895B/de

1980-12-24 Priority to FR8027482A priority patent/FR2477548A1/fr

1980-12-24 Priority to CH959380A priority patent/CH643850A5/de

1980-12-24 Priority to AU65830/80A priority patent/AU540042B2/en

1980-12-24 Priority to BE0/203321A priority patent/BE886864A/fr

1980-12-24 Priority to CA000367539A priority patent/CA1165759A/fr

1980-12-24 Priority to ES498145A priority patent/ES498145A0/es

1980-12-24 Priority to IT8026965A priority patent/IT8026965A0/it

1980-12-26 Priority to KR1019800004944A priority patent/KR840002162B1/ko

1980-12-29 Priority to US06/220,723 priority patent/US4344944A/en

1981-01-01 Priority to PH25066A priority patent/PH17794A/en

1981-01-07 Priority to SU813226153A priority patent/SU1095879A3/ru

1981-05-28 Priority to SU813288703A priority patent/SU1130569A1/ru

1981-09-25 Publication of JPS56122384A publication Critical patent/JPS56122384A/ja

1982-01-14 Priority to ES508723A priority patent/ES8300773A1/es

1982-02-18 Priority to US06/349,983 priority patent/US4415567A/en

1982-05-17 Priority to SU823436637A priority patent/SU1105117A3/ru

1982-10-28 Priority to AT0396182A priority patent/AT375376B/de

Status Pending legal-status Critical Current

Links

229940121375 antifungal agent Drugs 0.000 title 1
239000003429 antifungal agent Substances 0.000 title 1
241000894006 Bacteria Species 0.000 abstract 3
150000001875 compounds Chemical class 0.000 abstract 3
125000004423 acyloxy group Chemical group 0.000 abstract 2
IKWLIQXIPRUIDU-ZCFIWIBFSA-N (6r)-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid Chemical compound OC(=O)C1=CCS[C@@H]2CC(=O)N12 IKWLIQXIPRUIDU-ZCFIWIBFSA-N 0.000 abstract 1
108090000204 Dipeptidase 1 Proteins 0.000 abstract 1
241000588772 Morganella morganii Species 0.000 abstract 1
JCXJVPUVTGWSNB-UHFFFAOYSA-N Nitrogen dioxide Chemical compound O=[N]=O JCXJVPUVTGWSNB-UHFFFAOYSA-N 0.000 abstract 1
241000589517 Pseudomonas aeruginosa Species 0.000 abstract 1
125000000066 S-methyl group Chemical group [H]C([H])([H])S* 0.000 abstract 1
239000003242 anti bacterial agent Substances 0.000 abstract 1
230000000844 anti-bacterial effect Effects 0.000 abstract 1
125000002102 aryl alkyloxo group Chemical group 0.000 abstract 1
102000006635 beta-lactamase Human genes 0.000 abstract 1
239000000463 material Substances 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
- C07D311/22—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Cephalosporin Compounds (AREA)

JP2611280A 1980-03-04 1980-03-04 7alpha-methoxycephalosporin derivative, its preparation and antifungal agent comprising it Pending JPS56122384A (en)

Priority Applications (24)

Application Number	Priority Date	Filing Date	Title
JP2611280A JPS56122384A (en)	1980-03-04	1980-03-04	7alpha-methoxycephalosporin derivative, its preparation and antifungal agent comprising it
SE8009049A SE8009049L (sv)	1980-03-04	1980-12-22	7alfa-metoxicefalosporinderivat, sett for framstellning derav och antibakteriella lekemedel innehallande dessa foreningar
DK548380A DK548380A (da)	1980-03-04	1980-12-22	7alfa-methoxycephalsporinderivater og fremgangsmaade til fremstilling deraf
DE19803048657 DE3048657A1 (de)	1980-03-04	1980-12-23	7(alpha)-methoxycephalosporinderivate, verfahren zu deren herstellung und antibakterielle arzneimittel, welche diese derivate enthalten
HU803106A HU183276B (en)	1980-03-04	1980-12-23	Process for producing 7-alpha-metoxy-ceph-3-eme-4-carboxylic acid derivatives and for producing pharmaceutical compositions containing them as active agents
GB8041201A GB2070589B (en)	1980-03-04	1980-12-23	7a1methoxycephalospin derivatives
NL8007011A NL8007011A (nl)	1980-03-04	1980-12-23	7alfa-methoxycefalosporine-derivaten, werkwijze voor de bereiding daarvan en antibacteriele geneesmiddelen, die deze derivaten bevatten.
AT0630780A AT373895B (de)	1980-03-04	1980-12-23	Verfahren zur herstellung von neuen 7alpha -methoxycephalosporinderivaten
BE0/203321A BE886864A (fr)	1980-03-04	1980-12-24	Derives de 7-alpha-methoxycephalosporine, leur procede de preparation et leur application en therapeutique
CH959380A CH643850A5 (de)	1980-03-04	1980-12-24	7-alpha-methoxycephalosporinderivate, verfahren fuer die herstellung derselben und antibakteriell wirkende praeparate, welche diese verbindungen enthalten.
AU65830/80A AU540042B2 (en)	1980-03-04	1980-12-24	7-alpha methoxy cephalosporanic acids
FR8027482A FR2477548A1 (fr)	1980-03-04	1980-12-24	Derives de 7a-methoxycephalosporine, leur procede de preparation et leur application en therapeutique
CA000367539A CA1165759A (fr)	1980-03-04	1980-12-24	PROCEDE D'OBTENTION DE DERIVES DE LA 7.alpha.- METHOXYCEPHALOSPORINE ET REMEDES A PROPRIETES ANTIBACTERIENNES
ES498145A ES498145A0 (es)	1980-03-04	1980-12-24	Un procedimiento para la preparacion de derivados de metoxi-cefalosporinas
IT8026965A IT8026965A0 (it)	1980-03-04	1980-12-24	Derivati della 7-metossicefalosporina; procedimento per la loro preparazione; e farmaco antibatterico contenente tali derivati.
KR1019800004944A KR840002162B1 (ko)	1980-03-04	1980-12-26	7α-메톡시세팔로스포린 유도체의 제조방법
US06/220,723 US4344944A (en)	1980-03-04	1980-12-29	7-α-methoxycephalosporin derivatives, and antibacterial drugs onctaining the same
PH25066A PH17794A (en)	1980-03-04	1981-01-01	7 alpha-methoxy cephalosporin derivatives and antibacterial compositions containing them
SU813226153A SU1095879A3 (ru)	1980-03-04	1981-01-07	Способ получени производных цефалоспорина или их фармацевтически приемлемых солей
SU813288703A SU1130569A1 (ru)	1980-03-04	1981-05-28	Производные 7 @ -метоксицефалоспорина или их натриевые соли,обладающие противомикробной активностью
ES508723A ES8300773A1 (es)	1980-03-04	1982-01-14	"un procedimiento para la preparacion de derivados de metoxicefalosporinas".
US06/349,983 US4415567A (en)	1980-03-04	1982-02-18	7α-Methoxycephalosporin derivatives, and antibacterial drugs containing the same
SU823436637A SU1105117A3 (ru)	1980-03-04	1982-05-17	Способ получени производных 7 @ -метоксицефалоспорина или их солей с щелочными металлами
AT0396182A AT375376B (de)	1980-03-04	1982-10-28	Verfahren zur herstellung von neuen 7alphamethoxycephalosporinderivaten

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
JP2611280A JPS56122384A (en)	1980-03-04	1980-03-04	7alpha-methoxycephalosporin derivative, its preparation and antifungal agent comprising it

Publications (1)

Publication Number	Publication Date
JPS56122384A true JPS56122384A (en)	1981-09-25

Family

ID=12184494

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
JP2611280A Pending JPS56122384A (en)	1980-03-04	1980-03-04	7alpha-methoxycephalosporin derivative, its preparation and antifungal agent comprising it

Country Status (2)

Country	Link
JP (1)	JPS56122384A (fr)
BE (1)	BE886864A (fr)

1980
- 1980-03-04 JP JP2611280A patent/JPS56122384A/ja active Pending
- 1980-12-24 BE BE0/203321A patent/BE886864A/fr not_active IP Right Cessation

Also Published As

Publication number	Publication date
BE886864A (fr)	1981-06-24

Publication	Publication Date	Title
JPS57167992A (en)	1982-10-16	Novel cephalosporin compound
JPS565487A (en)	1981-01-20	Cephalosporin compound, its preparation, and antimicrobial comprising it
JPS5573686A (en)	1980-06-03	Novel penicillin
JPS5799592A (en)	1982-06-21	Novel cephalosporins
JPS56122384A (en)	1981-09-25	7alpha-methoxycephalosporin derivative, its preparation and antifungal agent comprising it
JPS5799591A (en)	1982-06-21	7alpha-methoxy-3-cephem derivative, its preparation and antibacterial agent comprising it
JPS5446836A (en)	1979-04-13	Antibacterial composition
JPS5718689A (en)	1982-01-30	7alpha-methoxycephem derivative
JPS54135767A (en)	1979-10-22	Penicillanic acid derivative
JPS5673087A (en)	1981-06-17	Cephalosporin derivative, its preparation and antimicrobial agent consisting of the same
JPS5764698A (en)	1982-04-19	Cephem derivative, its preparation, and antibacterial agent composed of said derivative
JPS56147790A (en)	1981-11-16	Cephalosporin type compound, its preparation, and antimicrobial agent comprising it
JPS57200394A (en)	1982-12-08	Novel 2-penem compound
JPS55136292A (en)	1980-10-23	Cephalosporin derivative, its preparation, and antibacterial comprising it
JPS57165389A (en)	1982-10-12	Novel penicillin and cephalosporin compound
JPS5718687A (en)	1982-01-30	Penicillin derivative and its salt
JPS5572196A (en)	1980-05-30	Penicillanic acid derivative
JPS54103889A (en)	1979-08-15	Novel 7alpha-methoxycephalosporin
JPS55111489A (en)	1980-08-28	Penicillin derivative, its preparation, and antibacterial agent comprising it
JPS5579394A (en)	1980-06-14	Novel 7-methoxycephalosporin derivative
JPS565484A (en)	1981-01-20	Cephalosporin derivative and its salt
JPS5791990A (en)	1982-06-08	7alpha-methoxycephem derivative, its preparation and antimicrobial agent consisting of the same
JPS56123988A (en)	1981-09-29	Novel 7- n-acylamino-alpha-arylacetamide -3- 1-substituted tetrazole-5-ylthiomethyl cephalosporins
JPS57106682A (en)	1982-07-02	Novel penicillins and their preparation
JPS57167993A (en)	1982-10-16	Novel 3-((4-carboxy-3-hydroxyisothiazole-5-yl) thiomethyl)-delta3-cephem derivative