JPS617432B2 - - Google Patents

Info

Publication number: JPS617432B2
Authority: JP; Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired

Application number

JP55164502A

Other languages

Japanese (ja)

Other versions

JPS5687586A (en

Inventor

Baanaado Keidein Sooru

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

PFIZER

Original Assignee

PFIZER

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1979-11-23

Filing date

1980-11-21

Publication date

1986-03-06

1980-11-21 Application filed by PFIZER filed Critical PFIZER

1981-07-16 Publication of JPS5687586A publication Critical patent/JPS5687586A/ja

1986-03-06 Publication of JPS617432B2 publication Critical patent/JPS617432B2/ja

Status Granted legal-status Critical Current

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/40—Unsubstituted amino or imino radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pulmonology (AREA)
Immunology (AREA)
Diabetes (AREA)
Hematology (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Dermatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Thiazole And Isothizaole Compounds (AREA)

JP16450280A 1979-11-23 1980-11-21 Antiallergic and antitumoral 11oxoo1hh thiazolo*3*22a*pyrimidinee22carboxamide and intermediate therefor Granted JPS5687586A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US9663179A	1979-11-23	1979-11-23

Publications (2)

Publication Number	Publication Date
JPS5687586A JPS5687586A (en)	1981-07-16
JPS617432B2 true JPS617432B2 (fr)	1986-03-06

Family

ID=22258306

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
JP16450280A Granted JPS5687586A (en)	1979-11-23	1980-11-21	Antiallergic and antitumoral 11oxoo1hh thiazolo322a*pyrimidinee22carboxamide and intermediate therefor

Country Status (35)

Country	Link
JP (1)	JPS5687586A (fr)
KR (1)	KR830004322A (fr)
AR (2)	AR228859A1 (fr)
AT (1)	AT380883B (fr)
AU (1)	AU520995B2 (fr)
BE (1)	BE886319A (fr)
CA (1)	CA1143731A (fr)
CH (1)	CH649299A5 (fr)
CS (1)	CS241476B2 (fr)
DD (1)	DD154608A5 (fr)
DE (2)	DE3050491C2 (fr)
DK (1)	DK151811C (fr)
EG (1)	EG14929A (fr)
ES (1)	ES497066A0 (fr)
FI (1)	FI67706C (fr)
FR (1)	FR2470132A1 (fr)
GB (1)	GB2063862B (fr)
GR (1)	GR72132B (fr)
GT (1)	GT198066458A (fr)
HU (1)	HU179091B (fr)
IE (1)	IE50404B1 (fr)
IL (1)	IL61535A (fr)
IN (1)	IN154926B (fr)
IT (1)	IT1209373B (fr)
LU (1)	LU82950A1 (fr)
NL (1)	NL182565C (fr)
NO (1)	NO803521L (fr)
NZ (1)	NZ195596A (fr)
PH (1)	PH16666A (fr)
PL (1)	PL132354B1 (fr)
PT (1)	PT72090B (fr)
SE (1)	SE448732B (fr)
SU (1)	SU1042620A3 (fr)
YU (1)	YU41953B (fr)
ZA (1)	ZA807293B (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8300728D0 (en) *	1983-01-12	1983-02-16	Erba Farmitalia	Substituted carboxy-thiazolo / 3 2 - a / pyrimidine derivatives
US4457932A (en) *	1983-07-22	1984-07-03	Bristol-Myers Company	Anti-ulcer agents
GB8422916D0 (en) *	1984-09-11	1984-10-17	May & Baker Ltd	Compositions of matter
JP2690742B2 (ja) *	1987-03-30	1997-12-17	第一製薬株式会社	複素環アミン誘導体
NZ228447A (en) *	1988-03-28	1990-08-28	Janssen Pharmaceutica Nv	Cosmetic or pharmaceutical composition possessing serotonin antogonistic activity
TWI500623B (zh) *	2009-10-13	2015-09-21	Torrent Pharmaceuticals Ltd	新穎稠合噻唑及噁唑嘧啶酮

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1331059A (en)	1971-04-19	1973-09-19	Lilly Industries Ltd	Pyrimidotriazinone compounds
US4041163A (en) *	1976-03-29	1977-08-09	Pfizer Inc.	N-(5-Tetrazolyl)-4-oxo-4H-pyrimido(2,1-b)benzothiazole-3-carboxamide antiallergy agents
DE2810863A1 (de) *	1978-03-13	1979-09-27	Boehringer Mannheim Gmbh	1-oxo-1h-pyrimido eckige klammer auf 6,1-b eckige klammer zu benzthiazol-derivate und verfahren zu ihrer herstellung
US4223031A (en) *	1978-05-05	1980-09-16	Mead Johnson & Company	Azolopyrimidinones

1980
- 1980-09-30 DK DK413180A patent/DK151811C/da not_active IP Right Cessation
- 1980-10-15 IN IN760/DEL/80A patent/IN154926B/en unknown
- 1980-11-17 SU SU803212053A patent/SU1042620A3/ru active
- 1980-11-18 GB GB8036904A patent/GB2063862B/en not_active Expired
- 1980-11-18 HU HU80802755A patent/HU179091B/hu not_active IP Right Cessation
- 1980-11-18 AR AR283276A patent/AR228859A1/es active
- 1980-11-18 CS CS807820A patent/CS241476B2/cs unknown
- 1980-11-19 EG EG723/80A patent/EG14929A/xx active
- 1980-11-19 CH CH8567/80A patent/CH649299A5/fr not_active IP Right Cessation
- 1980-11-20 GR GR63413A patent/GR72132B/el unknown
- 1980-11-20 NZ NZ195596A patent/NZ195596A/en unknown
- 1980-11-20 YU YU2950/80A patent/YU41953B/xx unknown
- 1980-11-21 NL NLAANVRAGE8006362,A patent/NL182565C/xx not_active IP Right Cessation
- 1980-11-21 NO NO803521A patent/NO803521L/no unknown
- 1980-11-21 ZA ZA00807293A patent/ZA807293B/xx unknown
- 1980-11-21 CA CA000365258A patent/CA1143731A/fr not_active Expired
- 1980-11-21 PT PT72090A patent/PT72090B/pt not_active IP Right Cessation
- 1980-11-21 DD DD80225391A patent/DD154608A5/de not_active IP Right Cessation
- 1980-11-21 IL IL61535A patent/IL61535A/xx unknown
- 1980-11-21 IE IE2418/80A patent/IE50404B1/en unknown
- 1980-11-21 DE DE3050491A patent/DE3050491C2/de not_active Expired
- 1980-11-21 SE SE8008189A patent/SE448732B/sv not_active IP Right Cessation
- 1980-11-21 ES ES497066A patent/ES497066A0/es active Granted
- 1980-11-21 GT GT198066458A patent/GT198066458A/es unknown
- 1980-11-21 AT AT0570780A patent/AT380883B/de not_active IP Right Cessation
- 1980-11-21 AU AU64595/80A patent/AU520995B2/en not_active Ceased
- 1980-11-21 FR FR8024822A patent/FR2470132A1/fr active Granted
- 1980-11-21 JP JP16450280A patent/JPS5687586A/ja active Granted
- 1980-11-21 LU LU82950A patent/LU82950A1/fr unknown
- 1980-11-21 FI FI803628A patent/FI67706C/fi not_active IP Right Cessation
- 1980-11-21 IT IT8026176A patent/IT1209373B/it active
- 1980-11-21 PH PH24891A patent/PH16666A/en unknown
- 1980-11-21 DE DE3043979A patent/DE3043979C2/de not_active Expired
- 1980-11-22 KR KR1019800004474A patent/KR830004322A/ko not_active Ceased
- 1980-11-22 PL PL1980228008A patent/PL132354B1/pl unknown
- 1980-11-24 BE BE0/202915A patent/BE886319A/fr not_active IP Right Cessation
1982
- 1982-09-13 AR AR290628A patent/AR231296A1/es active

Also Published As

Publication number	Publication date
LU82950A1 (fr)	1981-06-04
PL132354B1 (en)	1985-02-28
NO803521L (no)	1981-05-25
NL182565C (nl)	1988-04-05
NZ195596A (en)	1984-05-31
FI67706C (fi)	1985-05-10
IL61535A (en)	1984-06-29
GB2063862B (en)	1983-06-22
ES8203363A1 (es)	1982-04-01
PH16666A (en)	1983-12-13
CS241476B2 (en)	1986-03-13
SU1042620A3 (ru)	1983-09-15
KR830004322A (ko)	1983-07-09
CH649299A5 (fr)	1985-05-15
AR231296A1 (es)	1984-10-31
PL228008A1 (fr)	1981-12-11
DE3050491C2 (de)	1985-10-10
IN154926B (fr)	1984-12-22
DK151811B (da)	1988-01-04
AT380883B (de)	1986-07-25
IL61535A0 (en)	1980-12-31
SE8008189L (sv)	1981-05-24
DE3043979C2 (de)	1986-08-21
YU41953B (en)	1988-02-29
AU520995B2 (en)	1982-03-11
PT72090A (en)	1980-12-01
GB2063862A (en)	1981-06-10
JPS5687586A (en)	1981-07-16
FI803628L (fi)	1981-05-24
CS782080A2 (en)	1985-06-13
CA1143731A (fr)	1983-03-29
DK413180A (da)	1981-05-24
AU6459580A (en)	1981-05-28
GR72132B (fr)	1983-09-19
FI67706B (fi)	1985-01-31
PT72090B (en)	1981-09-29
AR228859A1 (es)	1983-04-29
ATA570780A (de)	1985-12-15
DK151811C (da)	1988-06-06
DE3043979A1 (de)	1981-09-03
SE448732B (sv)	1987-03-16
NL8006362A (nl)	1981-06-16
GT198066458A (es)	1982-05-15
IE802418L (en)	1981-05-23
YU295080A (en)	1983-06-30
ZA807293B (en)	1981-12-30
DD154608A5 (de)	1982-04-07
NL182565B (nl)	1987-11-02
HU179091B (en)	1982-08-28
IE50404B1 (en)	1986-04-16
ES497066A0 (es)	1982-04-01
IT1209373B (it)	1989-07-16
FR2470132A1 (fr)	1981-05-29
FR2470132B1 (fr)	1983-07-29
EG14929A (en)	1989-01-30
IT8026176A0 (it)	1980-11-21
BE886319A (fr)	1981-05-25

Publication	Publication Date	Title
FR2456145B1 (fr)	1985-03-22
FR2447656B3 (fr)	1981-06-12
FR2455808B1 (fr)	1984-06-29
FR2463877B1 (fr)	1984-12-14
FR2447326B1 (fr)	1984-02-17
DE2936318C3 (fr)	1982-03-11
FR2461006B1 (fr)	1984-03-09
FR2446474B1 (fr)	1982-04-30
FR2460278B1 (fr)	1984-12-28
FR2457169B1 (fr)	1982-10-08
FR2461599B1 (fr)	1985-03-22
FR2449141B1 (fr)	1982-12-17
FR2459239B1 (fr)	1982-09-10
FR2447785B1 (fr)	1983-11-18
FR2466252B2 (fr)	1983-08-12
FR2463003B1 (fr)	1985-01-04
FR2448559B1 (fr)	1983-12-09
FR2448463B1 (fr)	1982-10-22
FR2473075B1 (fr)	1985-01-04
FR2468734B1 (fr)	1984-09-07
FR2478483B1 (fr)	1985-01-04
FR2470132B1 (fr)	1983-07-29
FR2496642B1 (fr)	1985-11-08
FR2454424B1 (fr)	1985-01-04
FR2459270B1 (fr)	1983-12-16