KR890000764B1 - 페닐 치환된 피리도[1,4]벤조디아제핀 및 이의 제조방법 - Google Patents

페닐 치환된 피리도[1,4]벤조디아제핀 및 이의 제조방법 Download PDF

Info

Publication number: KR890000764B1
Authority: KR; South Korea
Prior art keywords: pyrido; phenyl; benzodiazepine; amino; compound
Prior art date: 1981-09-24
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired

Application number

KR8200420A

Other languages

English (en)

Korean (ko)

Other versions

KR830009058A (ko

Inventor

로이 테일러 2세 챈들러

Original Assignee

알.피.울프

에이 에이취 로빈스 캄파니 인코포레이티드

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1981-09-24

Filing date

1982-02-02

Publication date

1989-04-05

1982-02-02 Application filed by 알.피.울프, 에이 에이취 로빈스 캄파니 인코포레이티드 filed Critical 알.피.울프

1983-12-17 Publication of KR830009058A publication Critical patent/KR830009058A/ko

1989-04-05 Application granted granted Critical

1989-04-05 Publication of KR890000764B1 publication Critical patent/KR890000764B1/ko

Status Expired legal-status Critical Current

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Psychiatry (AREA)
Veterinary Medicine (AREA)
Bioinformatics & Cheminformatics (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Pain & Pain Management (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pyridine Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

KR8200420A 1981-09-24 1982-02-02 페닐 치환된 피리도[1,4]벤조디아제핀 및 이의 제조방법 Expired KR890000764B1 (ko)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date
US30508081A	1981-09-24	1981-09-24
US305,080		1981-09-24
US305080		1981-09-24

Publications (2)

Publication Number	Publication Date
KR830009058A KR830009058A (ko)	1983-12-17
KR890000764B1 true KR890000764B1 (ko)	1989-04-05

Family

ID=23179241

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
KR8200420A Expired KR890000764B1 (ko)	1981-09-24	1982-02-02	페닐 치환된 피리도[1,4]벤조디아제핀 및 이의 제조방법

Country Status (27)

Country	Link
JP (1)	JPS5865290A (fr)
KR (1)	KR890000764B1 (fr)
BE (1)	BE891666A (fr)
CA (1)	CA1199324A (fr)
CH (1)	CH651833A5 (fr)
DE (1)	DE3150522A1 (fr)
DK (3)	DK186282A (fr)
EG (1)	EG15904A (fr)
ES (6)	ES507971A0 (fr)
FI (1)	FI71935C (fr)
FR (1)	FR2515183B1 (fr)
GR (1)	GR78473B (fr)
HU (2)	HU187393B (fr)
IE (1)	IE52493B1 (fr)
IL (1)	IL64284A (fr)
IN (1)	IN156080B (fr)
IT (1)	IT1146728B (fr)
LU (1)	LU83865A1 (fr)
NL (1)	NL8200549A (fr)
NO (1)	NO157700C (fr)
NZ (1)	NZ198999A (fr)
PH (2)	PH17847A (fr)
PL (6)	PL143596B1 (fr)
PT (1)	PT74286B (fr)
SE (2)	SE448629B (fr)
YU (1)	YU46128B (fr)
ZA (1)	ZA817866B (fr)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3825549A (en) *	1972-10-24	1974-07-23	Squibb & Sons Inc	Certain dihydropyrido(2,1-b)(1,3)benzodi-azepines and benzodiazocines
DE2424811C3 (de) *	1974-05-22	1981-08-20	Dr. Karl Thomae Gmbh, 7950 Biberach	Pyrido-benzodiazepinone, Verfahren zu ihrer Herstellung und diese enthaltende Arzneimittel
SE422799B (sv) *	1975-05-28	1982-03-29	Merck & Co Inc	Analogiforfarande for framstellning av 1,3-dihydroimidazo (4,5-b)pyridin-2-oner

1981
- 1981-11-05 SE SE8106573A patent/SE448629B/sv not_active IP Right Cessation
- 1981-11-12 ZA ZA817866A patent/ZA817866B/xx unknown
- 1981-11-12 NO NO813839A patent/NO157700C/no unknown
- 1981-11-13 IL IL64284A patent/IL64284A/xx unknown
- 1981-11-13 IN IN1261/CAL/81A patent/IN156080B/en unknown
- 1981-11-17 GR GR66553A patent/GR78473B/el unknown
- 1981-11-18 PH PH26507A patent/PH17847A/en unknown
- 1981-11-25 IE IE2769/81A patent/IE52493B1/en unknown
- 1981-12-09 IT IT68605/81A patent/IT1146728B/it active
- 1981-12-10 FI FI813976A patent/FI71935C/fi not_active IP Right Cessation
- 1981-12-15 HU HU813777A patent/HU187393B/hu not_active IP Right Cessation
- 1981-12-15 HU HU843212A patent/HU189426B/hu not_active IP Right Cessation
- 1981-12-15 ES ES507971A patent/ES507971A0/es active Granted
- 1981-12-21 DE DE19813150522 patent/DE3150522A1/de not_active Withdrawn
- 1981-12-23 FR FR8124111A patent/FR2515183B1/fr not_active Expired
- 1981-12-23 PL PL1981253538A patent/PL143596B1/pl unknown
- 1981-12-23 PL PL1981241409A patent/PL139381B1/pl unknown
- 1981-12-23 PL PL1981241410A patent/PL137068B1/pl unknown
- 1981-12-23 PL PL1981234426A patent/PL138859B1/pl unknown
- 1981-12-23 PL PL1981253539A patent/PL143597B1/pl unknown
- 1981-12-23 PL PL1981253540A patent/PL143322B1/pl unknown
- 1981-12-30 BE BE0/206969A patent/BE891666A/fr not_active IP Right Cessation
1982
- 1982-01-05 LU LU83865A patent/LU83865A1/fr unknown
- 1982-01-12 EG EG11/82A patent/EG15904A/xx active
- 1982-01-14 JP JP57004813A patent/JPS5865290A/ja active Pending
- 1982-01-15 PT PT74286A patent/PT74286B/pt unknown
- 1982-01-18 CA CA000394367A patent/CA1199324A/fr not_active Expired
- 1982-02-02 KR KR8200420A patent/KR890000764B1/ko not_active Expired
- 1982-02-12 NL NL8200549A patent/NL8200549A/nl not_active Application Discontinuation
- 1982-02-18 NZ NZ198999A patent/NZ198999A/en unknown
- 1982-03-23 YU YU62582A patent/YU46128B/sh unknown
- 1982-04-15 CH CH2288/82A patent/CH651833A5/fr not_active IP Right Cessation
- 1982-04-26 DK DK186282A patent/DK186282A/da not_active Application Discontinuation
- 1982-09-29 ES ES516052A patent/ES8402295A1/es not_active Expired
- 1982-09-29 ES ES516051A patent/ES8308563A1/es not_active Expired
1983
- 1983-10-19 ES ES526562A patent/ES8504148A1/es not_active Expired
- 1983-10-19 ES ES526563A patent/ES8604531A1/es not_active Expired
1984
- 1984-08-17 PH PH31120A patent/PH20536A/en unknown
1985
- 1985-05-21 ES ES543328A patent/ES8607726A1/es not_active Expired
1986
- 1986-02-17 SE SE8600688A patent/SE455305B/sv not_active IP Right Cessation
1987
- 1987-08-03 DK DK403487A patent/DK403487A/da not_active Application Discontinuation
- 1987-08-03 DK DK403387A patent/DK403387A/da not_active Application Discontinuation

Also Published As

Publication number	Publication date
HU189426B (en)	1986-07-28
DK186282A (da)	1983-03-25
ZA817866B (en)	1982-10-27
PL241409A1 (en)	1984-05-21
FI71935B (fi)	1986-11-28
IN156080B (fr)	1985-05-11
ES8604531A1 (es)	1986-02-01
FI71935C (fi)	1987-03-09
DK403387D0 (da)	1987-08-03
PL143597B1 (en)	1988-02-29
IT1146728B (it)	1986-11-19
ES526562A0 (es)	1985-04-01
IE52493B1 (en)	1987-11-25
PL241410A1 (en)	1984-01-02
CA1199324A (fr)	1986-01-14
GR78473B (fr)	1984-09-27
ES516052A0 (es)	1984-01-16
IT8168605A0 (it)	1981-12-09
EG15904A (en)	1987-03-30
PL137068B1 (en)	1986-04-30
KR830009058A (ko)	1983-12-17
PT74286A (en)	1982-02-01
PH20536A (en)	1987-02-09
ES516051A0 (es)	1983-09-16
PL138859B1 (en)	1986-11-29
PL139381B1 (en)	1987-01-31
PL143596B1 (en)	1988-02-29
ES543328A0 (es)	1986-06-01
DE3150522A1 (de)	1983-04-07
ES8308563A1 (es)	1983-09-16
CH651833A5 (fr)	1985-10-15
DK403487D0 (da)	1987-08-03
FR2515183A1 (fr)	1983-04-29
NO813839L (no)	1983-03-25
PH17847A (en)	1985-01-09
IL64284A (en)	1986-12-31
BE891666A (fr)	1982-04-16
ES8504148A1 (es)	1985-04-01
NZ198999A (en)	1987-07-31
IL64284A0 (en)	1982-02-28
ES8402295A1 (es)	1984-01-16
JPS5865290A (ja)	1983-04-18
NO157700C (no)	1988-05-04
SE8600688L (sv)	1986-02-17
FR2515183B1 (fr)	1986-11-14
ES8607726A1 (es)	1986-06-01
NO157700B (no)	1988-01-25
LU83865A1 (fr)	1983-09-02
PL143322B1 (en)	1988-02-29
HUT34732A (en)	1985-04-28
ES526563A0 (es)	1986-02-01
NL8200549A (nl)	1983-04-18
SE8106573L (sv)	1983-03-25
SE455305B (sv)	1988-07-04
ES8303348A1 (es)	1983-02-01
ES507971A0 (es)	1983-02-01
IE812769L (en)	1983-03-24
PT74286B (en)	1983-06-27
PL234426A1 (en)	1984-01-02
YU62582A (en)	1986-04-30
YU46128B (sh)	1993-05-28
DK403387A (da)	1987-08-03
SE448629B (sv)	1987-03-09
FI813976L (fi)	1983-03-25
HU187393B (en)	1985-12-28
SE8600688D0 (sv)	1986-02-17
DK403487A (da)	1987-08-03

Legal Events

Date	Code	Title	Description
1982-02-02	PA0109	Patent application	St.27 status event code: A-0-1-A10-A12-nap-PA0109
1982-02-02	R17-X000	Change to representative recorded	St.27 status event code: A-3-3-R10-R17-oth-X000
1983-12-17	PG1501	Laying open of application	St.27 status event code: A-1-1-Q10-Q12-nap-PG1501
1987-01-28	R17-X000	Change to representative recorded	St.27 status event code: A-3-3-R10-R17-oth-X000
1987-02-02	P11-X000	Amendment of application requested	St.27 status event code: A-2-2-P10-P11-nap-X000
1987-02-02	P13-X000	Application amended	St.27 status event code: A-2-2-P10-P13-nap-X000
1987-02-02	PA0201	Request for examination	St.27 status event code: A-1-2-D10-D11-exm-PA0201
1987-07-02	P11-X000	Amendment of application requested	St.27 status event code: A-2-2-P10-P11-nap-X000
1987-07-02	P13-X000	Application amended	St.27 status event code: A-2-2-P10-P13-nap-X000
1988-08-20	PE0902	Notice of grounds for rejection	St.27 status event code: A-1-2-D10-D21-exm-PE0902
1988-10-20	P11-X000	Amendment of application requested	St.27 status event code: A-2-2-P10-P11-nap-X000
1988-10-20	P13-X000	Application amended	St.27 status event code: A-2-2-P10-P13-nap-X000
1989-04-05	PG1605	Publication of application before grant of patent	St.27 status event code: A-2-2-Q10-Q13-nap-PG1605
1989-06-30	PE0701	Decision of registration	St.27 status event code: A-1-2-D10-D22-exm-PE0701
1989-07-12	PR0701	Registration of establishment	St.27 status event code: A-2-4-F10-F11-exm-PR0701
1989-07-12	PR1002	Payment of registration fee	St.27 status event code: A-2-2-U10-U11-oth-PR1002 Fee payment year number: 1
1992-04-06	PC1903	Unpaid annual fee	St.27 status event code: A-4-4-U10-U13-oth-PC1903 Not in force date: 19920406 Payment event data comment text: Termination Category : DEFAULT_OF_REGISTRATION_FEE
1994-10-08	PC1903	Unpaid annual fee	St.27 status event code: N-4-6-H10-H13-oth-PC1903 Ip right cessation event data comment text: Termination Category : DEFAULT_OF_REGISTRATION_FEE Not in force date: 19920406

Publication	Publication Date	Title
US4675319A (en)	1987-06-23	Antianaphylactic and antibronchospastic piperazinyl-(N-substituted phenyl)carboxamides, compositions and use
US4002623A (en)	1977-01-11	Anti-inflammatory 1-[3-(dialkylamino)propyl]-2-acylaminobenzimidazoles and 2-acylamino-3-[3-(dialkylamino)-propyl]imidazo[4,5-b]pyridines
EP1446399B1 (fr)	2005-05-04	Derives de piperazine ayant une activite antagoniste sst1
US4447361A (en)	1984-05-08	Aryl substituted pyrido[1,4]benzodiazepines
US3732212A (en)	1973-05-08	1,2,3,10,11,11a-hexahydro-5h-pyrrolo(2,1-c)(1,4)benzodiazepine-5,11-diones
US4167570A (en)	1979-09-11	2-Methyl-6-alkyl-11-aminoalkyl-6,11-dihydro-5H-pyrido(2,3-B)(1,5)benzodiazepin-5-ones and salts thereof
US4311700A (en)	1982-01-19	Pyrimidobenzodiazepinones, their use and medicaments containing them
EP0107261B1 (fr)	1988-09-21	(2-((Nitropyridinyl)amino)phényl)arylméthanones et sels, leur utilisation en médecine, compositions pharmaceutiques les contenant et leur utilisation dans la préparation de (2-((aminopyridinyl)amino)phényl)arylméthanones et de pyrido(1,4)benzodiazépines
EP0076017B1 (fr)	1990-08-16	Pyrido(1,4)benzodiazépines substituées par un phényl et intermédiaires
US4556667A (en)	1985-12-03	Aryl substituted pyrido[1,4]benzodiazepines and their use as antidepressives
NZ199610A (en)	1985-05-31	Tricyclic pyrrole derivatives
US4495183A (en)	1985-01-22	Aryl substituted pyrido[1,4]benzodiazepines for treatment of depression
US4668675A (en)	1987-05-26	2-[(amino-pyridinyl)amine]phenyl]aryl methanones, their thioxomethyl, ketal or thioketal analogs
US4059584A (en)	1977-11-22	2-Acylamino-3-[3-(dialkylamino)propyl]imidazo[4,5-b]pyridines
JP2531678B2 (ja)	1996-09-04	トリアゾロピリダジン誘導体
US4558132A (en)	1985-12-10	Nitro, amino and aroylamino-N-phenylpyridinamines in a process for preparing pyrido[1,4]benzodiazepines
US4180573A (en)	1979-12-25	1-Piperazino-6-phenyl-4H-s-triazolo[3,4-c]thieno[2,3-e]1,4-diazepines
US4698430A (en)	1987-10-06	Nitro, amino and aroylamino-n-phenylpyridinamines
CA1199324A (fr)	1986-01-14	Derives de substitution phenyles de pyrido¬1,4\| benzodiazepines, et produits intermediaires
US4628100A (en)	1986-12-09	Intermediates for the preparation of aryl substituted pyrido[1,4]benzodiazepines
US4518603A (en)	1985-05-21	[2-[(Nitropyridinyl)amino]phenyl]arylmethanones in a process for preparing pyrido[1,4]benzodiazepines
NO872271L (no)	1983-03-25	(2-((aminopyridinyl)amino(fenyl)-arylmethanoner.
JPS634830B2 (fr)	1988-02-01
NO880084L (no)	1984-04-02	Utgangsmaterialer for fremstilling av pyrido(1,4)benzodiazepiner.
NO161175B (no)	1989-04-03	Pyrido(1,4)-benzodiazepiner.