LU85780A1 - Nouveaux esters enoliques precurseurs de medicaments et composition pharmaceutique les contenant - Google Patents

Nouveaux esters enoliques precurseurs de medicaments et composition pharmaceutique les contenant Download PDF

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Publication number
LU85780A1
LU85780A1 LU85780A LU85780A LU85780A1 LU 85780 A1 LU85780 A1 LU 85780A1 LU 85780 A LU85780 A LU 85780A LU 85780 A LU85780 A LU 85780A LU 85780 A1 LU85780 A1 LU 85780A1
Authority
LU
Luxembourg
Prior art keywords
methyl
carboxamide
dioxide
benzothiazine
pyridyl
Prior art date
Application number
LU85780A
Other languages
English (en)
French (fr)
Inventor
Joseph George Lombardino
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of LU85780A1 publication Critical patent/LU85780A1/fr

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • Rheumatology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
LU85780A 1984-02-23 1985-02-20 Nouveaux esters enoliques precurseurs de medicaments et composition pharmaceutique les contenant LU85780A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US58268484A 1984-02-23 1984-02-23
US58268484 1984-02-23

Publications (1)

Publication Number Publication Date
LU85780A1 true LU85780A1 (fr) 1985-12-11

Family

ID=24330094

Family Applications (1)

Application Number Title Priority Date Filing Date
LU85780A LU85780A1 (fr) 1984-02-23 1985-02-20 Nouveaux esters enoliques precurseurs de medicaments et composition pharmaceutique les contenant

Country Status (22)

Country Link
JP (1) JPS60184077A (de)
KR (1) KR850006198A (de)
AU (1) AU552478B2 (de)
BE (1) BE901783A (de)
DD (1) DD232045A5 (de)
DE (1) DE3505576A1 (de)
DK (1) DK81185A (de)
ES (1) ES8606312A1 (de)
FI (1) FI850742L (de)
FR (1) FR2565980A1 (de)
GB (1) GB2154585A (de)
GR (1) GR850442B (de)
HU (1) HUT37616A (de)
IL (1) IL74407A0 (de)
IT (1) IT1185514B (de)
LU (1) LU85780A1 (de)
NL (1) NL8500485A (de)
NO (1) NO850725L (de)
PL (1) PL252023A1 (de)
PT (1) PT79988B (de)
SE (1) SE8500889L (de)
ZA (1) ZA851317B (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4623486A (en) * 1985-05-29 1986-11-18 Pfizer Inc. [4-substituted benzoyloxy]-N-substituted-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxides having anti-arthritic activity
US4610982A (en) * 1985-06-03 1986-09-09 Pfizer Inc. Anti-inflammatory benzo- and thieno-1,2-thiazine-3-carboxamide 1,1-dioxide derivatives, compositions, and method of use therefor
US20090238763A1 (en) 2006-07-09 2009-09-24 Chongxi Yu High penetration compositions and uses thereof
US20090221703A1 (en) 2006-07-09 2009-09-03 Chongxi Yu High penetration composition and uses thereof
CN101522692A (zh) * 2006-10-11 2009-09-02 于崇曦 具有快速皮肤穿透速度的带正电荷的水溶性的昔康及其相关化合物的前药
WO2008149181A1 (en) 2007-06-04 2008-12-11 Techfields Inc Pro-drugs of nsaias with very high skin and membranes penetration rates and their new medicinal uses
RU2630577C2 (ru) 2008-12-04 2017-09-11 Чунси ЮЙ Композиции интенсивного проникновения и их применение

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3591574A (en) * 1968-05-29 1971-07-06 American Home Prod Tri-n-phenylglycyl derivatives of insulin
US3787324A (en) * 1971-03-01 1974-01-22 Warner Lambert Co 4-hydroxy-3-(3-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,dioxides and process for their production
US3704298A (en) * 1971-06-22 1972-11-28 Warner Lambert Co 4-acyloxy-3-(2-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,1-dioxides
AU518216B2 (en) * 1977-09-06 1981-09-17 Hafslund Nycomed Pharma Aktiengesellschaft Thienothiazine derivatives
JPS5714589A (en) * 1980-06-27 1982-01-25 Mitsui Toatsu Chem Inc Benzothiazine derivative, its preparation and drug composition
US4309427A (en) * 1981-01-15 1982-01-05 Pfizer Inc. Benzothiazine dioxide derivatives
IT8219486A0 (it) * 1982-02-05 1982-02-05 Chiesi Farma Spa Nuovi composti ad attivita'antiinfiammatoria, procedimento per la loro preparazione e relative composizioni farmaceutiche.
IT1206525B (it) * 1982-12-10 1989-04-27 Zionale S R L A Roma Preparato anti-infiammatorio nonsteroideo, per il trattamento delle affezioni artroreumatiche e metodo per la sua preparazione

Also Published As

Publication number Publication date
ES540590A0 (es) 1986-04-16
FR2565980A1 (fr) 1985-12-20
AU552478B2 (en) 1986-06-05
DK81185A (da) 1985-09-10
JPS60184077A (ja) 1985-09-19
SE8500889D0 (sv) 1985-02-22
FI850742A0 (fi) 1985-02-22
DE3505576A1 (de) 1985-09-05
IT1185514B (it) 1987-11-12
NO850725L (no) 1985-08-26
ZA851317B (en) 1986-10-29
IL74407A0 (en) 1985-05-31
GB2154585A (en) 1985-09-11
HUT37616A (en) 1986-01-23
IT8519585A1 (it) 1986-08-21
PT79988B (en) 1987-02-02
FI850742A7 (fi) 1985-08-24
GR850442B (de) 1985-06-19
KR850006198A (ko) 1985-10-02
IT8519585A0 (it) 1985-02-21
AU3906685A (en) 1985-09-05
GB8504355D0 (en) 1985-03-20
PL252023A1 (en) 1985-11-05
BE901783A (fr) 1985-08-21
NL8500485A (nl) 1985-09-16
ES8606312A1 (es) 1986-04-16
FI850742L (fi) 1985-08-24
SE8500889L (sv) 1985-08-24
DK81185D0 (da) 1985-02-22
PT79988A (en) 1985-03-01
DD232045A5 (de) 1986-01-15

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